Keywords: افزایش تابش; Cyclodextrin nanosponge; DPC; PMDA; Curcumin; Solubility enhancement; Nanocarrier;
مقالات ISI افزایش تابش (ترجمه نشده)
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Keywords: افزایش تابش; Solid dispersion; Cardiovascular effects; Quercetin; Polyvinylpyrrolidone; Solubility enhancement; Injectable aqueous solution;
Keywords: افزایش تابش; Milk protein; Solubility enhancement; Ethanol; Hydrophobic compounds; Drug delivery; Sodium caseinate;
Keywords: افزایش تابش; Camptothecin; Heterolipid E1E; Self-microemulsifying drug delivery system; Solubility enhancement; Anti-tumor activity; Molecular simulation;
Keywords: افزایش تابش; Quercetin (PubChem CID: 5280343); hydroxypropylmethylcellulose acetate succinate (PubChem CID: 121950); polyvinylpyrrolidone (PubChem CID: 6917); ASD; amorphous solid dispersion; CCAB; carboxycellulose acetate butyrate; CASub; cellulose acetate suberate;
Keywords: افزایش تابش; Amorphous drug; Solid dispersion; Solubility enhancement; Spray-drying; Wet-granulation; Nilvadipine;
Keywords: افزایش تابش; Oligopyridine; Nanoemulsions; Solubility enhancement; Biomimetic media; Preclinical studies;
Keywords: افزایش تابش; Surfactant; Solid dispersion; Plasticizers; Stability; Supersaturation; Solubility enhancement;
Keywords: افزایش تابش; Taylor Dispersion Analysis; Peptide prodrug; Aggregation; Cyclodextrin; Solubility enhancement; Formulation;
Keywords: افزایش تابش; Erlotinib; Tyrosine kinase inhibitor; Pancreatic cancer; Phospholipid complex; Solubility enhancement; Oral bioavailability;
Keywords: افزایش تابش; ASD; amorphous solid dispersion; AUC; area under the curve; BCS; biopharmaceutics classification system; C; supersaturated drug concentration; CSat; drug saturation solubility; CFX; cefuroxime; CIP; ciprofloxacin; DLS; dynamic light scattering; DXT; dextr
Keywords: افزایش تابش; solubility; polymers; poorly soluble drugs; Flory-Huggins; shake-flask method; amorphous solid dispersion; solubility enhancement; thermal analysis;
Keywords: افزایش تابش; BSC class II drugs; Porous materials; Spray drying; Physisorption studies; Solubility enhancement; Oral drug delivery
Keywords: افزایش تابش; Solubility; Amorphous; Liquid-liquid phase separation; Membrane transport rate; Solubility enhancement; Absorption;
Keywords: افزایش تابش; Resistance maltodextrin; Polyphenols; Naringin; Spray-drying; Encapsulation; Solubility enhancement;
Keywords: افزایش تابش; Resveratrol; Anticancer; Nanoformulation; Targeting; Solubility enhancement;
Keywords: افزایش تابش; Hot-melt extrusion; Orally disintegrating tablets; Solid dispersion; Solubility enhancement; Taste masking effect; Molecular interaction
Keywords: افزایش تابش; Factorial design; Amorphous solid dispersion; Spray drying; EUDRAGIT® E PO; Solvent casting; Solubility enhancement;
Keywords: افزایش تابش; Amorphous solid dispersion; Quality by Design; Solubility enhancement; Selection of polymer; Spray drying
Keywords: افزایش تابش; Low-molecular-weight succinoglycans; Sinorhizobium meliloti; Pindolol; Solubility enhancement; Cyclodextrin; Complexation
Keywords: افزایش تابش; Elementary osmotic pump; Carbamazepine; Solubility enhancement; Taguchi orthogonal design; Zero order
Keywords: افزایش تابش; Particle technology; Drug solubility; Poorly water soluble drug; Solubility enhancement; Dissolution
Solubility and dissolution rate enhancement of ibuprofen by co-milling with polymeric excipients
Keywords: افزایش تابش; PM; physical mixture; mPM; milled physical mixture; A; absorbance; Poor soluble drugs; Ball milling; Solubility enhancement; Dissolution rate; Particle size; Amorphous content;
Poly(methyl vinyl ether-co-maleic acid) for enhancement of solubility, oral bioavailability and anti-osteoporotic effects of raloxifene hydrochloride
Keywords: افزایش تابش; Electrospray; Raloxifene; Solubility enhancement; Poly(methyl vinyl ether maleic acid); Oral delivery; Ovariectomized rats;
Formulation of olanzapine nanosuspension based orally disintegrating tablets (ODT); comparative evaluation of lyophilization and electrospraying process as solidification techniques
Keywords: افزایش تابش; Nanosuspension; Electrospraying; Lyophilization; Orally disintegrating tablets; Solubility enhancement; Psychological disorders;
Study on effect of L-arginine on solubility and dissolution of Zaltoprofen: Preparation and characterization of binary and ternary cyclodextrin inclusion complexes
Keywords: افزایش تابش; Ternary complex; Cyclodextrin; Dissolution enhancement; Inclusion complex; Solubility enhancement;
Interactions of dimethylaminoethyl methacrylate copolymer with non-acidic drugs demonstrated high solubilization in vitro and pronounced sustained release in vivo
Keywords: افزایش تابش; Solubility enhancement; Polymer drug interaction; Oral bioavailability; Sustained release;
Development of controlled release amorphous solid dispersions (CRASD) using polyvinyl acetate-based release retarding materials: Effect of dosage form design
Keywords: افزایش تابش; ASD; amorphous solid dispersion; ATR; attenuated total reflectance; AUC; area under the curve; BCS; Biopharmaceutic Classification System; CEL; celecoxib; Cmax; maximum concentration, or peak kinetic solubility; CR; controlled release; CRASD; controlled r
Host-guest interaction study of Efavirenz with hydroxypropylâβâcyclodextrin and lâarginine by computational simulation studies: Preparation and characterization of supramolecular complexes
Keywords: افزایش تابش; Efavirenz; Solubility enhancement; Inclusion complex;
Antibacterial and antioxidant electrospun materials from poly(3-hydroxybutyrate) and polyvinylpyrrolidone containing caffeic acid phenethyl ester - “in” and “on” strategies for enhanced solubility
Keywords: افزایش تابش; Caffeic acid phenethyl ester; Poly(3-hydroxybutyrate); Polyvinylpyrrolidone; Electrospinning; Solubility enhancement; Antibacterial activity; Antioxidant capacity;
Solid dispersions to enhance the delivery of a potential drug candidate LPSF/FZ4 for the treatment of schistosomiasis
Keywords: افزایش تابش; Schistosomiasis; Solid dispersions; Solubility enhancement; Drug candidate; Supersaturation; Bioavailability;
A bird's eye view of nanoparticles prepared by electrospraying: advancements in drug delivery field
Keywords: افزایش تابش; Electrospraying; Nanoparticles; Electrohydrodynamic atomization; Controlled release; Solubility enhancement; Surface morphology; AA; Acetic Acid; BD; Beclomethasone Dipropionate; BSA; Bovine Serum Albumin; C; Critical Polymer concentration; CD; Circular D
Inclusion complex of chrysin with sulfobutyl ether-β-cyclodextrin (Captisol®): Preparation, characterization, molecular modelling and in vitro anticancer activity
Keywords: افزایش تابش; Polyphenols; Cancer; Solubility enhancement; Sulfobutyl ether-beta-cyclodextrin; Chrysin; Inclusion complexation;
Application of miscibility analysis and determination of Soluplus solubility map for development of carvedilol-loaded nanofibers
Keywords: افزایش تابش; Poorly soluble drugs; Solvent mapping; Electrospinning; Solid dispersions; Solubility enhancement; Interaction parameter;
A two-step synthetic strategy to obtain a water-soluble derivative of curcumin with improved antioxidant capacity and in vitro cytotoxicity in C6 glioma cells
Keywords: افزایش تابش; Curcumin; Polyester dendrons; Solubility enhancement; Antioxidant capacity;
Hybridization of polyvinylpyrrolidone to a binary composite of curcumin/α-glucosyl stevia improves both oral absorption and photochemical stability of curcumin
Keywords: افزایش تابش; CUR; curcumin; DSC; differential scanning calorimetry; Hesperidin-G; α-glucosyl hesperidin; PM; physical mixture; PVP; polyvinylpyrrolidone; PXRD; powder X-ray diffraction; RH; relative humidity; Rutin-G; α-glucosyl rutin; Stevia-G; α-glucosyl stevia;
Effect of polymer type and drug dose on the in vitro and in vivo behavior of amorphous solid dispersions
Keywords: افزایش تابش; Non-sink dissolution; Amorphous solid dispersion; Bioavailability; Dose-dependence; Polymers; In vitro; In vivo; IVIVC; Supersaturation; Poorly soluble drugs; Solubility enhancement; Celecoxib; PVP; HPMC; PVA
Development and characterisation of sustained release solid dispersion oral tablets containing the poorly water soluble drug disulfiram
Keywords: افزایش تابش; Sustained release; Solid dispersion; Solubility enhancement; Hot melt; Disulfiram;
Novel pimozide-β-cyclodextrin-polyvinylpyrrolidone inclusion complexes for Tourette syndrome treatment
Keywords: افزایش تابش; Pimozide; Inclusion complex; Solubility enhancement;
Potential of erlotinib cyclodextrin nanosponge complex to enhance solubility, dissolution rate, in vitro cytotoxicity and oral bioavailability
Keywords: افزایش تابش; Erlotinib; Tyrosine kinase inhibitor; Nanosponge; Solubility enhancement; In vitro cytotoxicity; Oral bioavailabilityErlotinib hydrochloride (PubChem CID: 176871); β-Cyclodextrin (PubChem CID: 444041); Ammonium acetate (PubChem CID: 517165); Atorvastatin
Enhanced in vitro dissolution of Iloperidone using Caesalpinia Pulcherrima mucoadhesive microspheres
Keywords: افزایش تابش; Iloperidone; Caesalpinia pulcherrima mucilage; Spray drying; Mucoadhesive microspheres; Solubility enhancement
Synthesis of large-ring cyclodextrin from tapioca starch by amylomaltase and complex formation with vitamin E acetate for solubility enhancement
Keywords: افزایش تابش; Large-ring cyclodextrin; Amylomaltase; Tapioca starch; Vitamin E acetate; Solubility enhancement
Inclusion complex of erlotinib with sulfobutyl ether-β-cyclodextrin: Preparation, characterization, in silico, in vitro and in vivo evaluation
Keywords: افزایش تابش; Erlotinib; Tyrosine kinase inhibitor; Pancreatic cancer; Cyclodextrin; Sulfobutyl ether β-cyclodextrin; Solubility enhancement; Erlotinib hydrocholide (PubChem CID: 176871); α-Cyclodextrin (PubChem CID: 444913); β-Cyclodextrin (PubChem CID: 444041); γ
A new combination approach of CI jet and QESD to formulate pH-susceptible amorphous solid dispersions
Keywords: افزایش تابش; ASDs; Amorphous solid dispersions; BCS; Biopharmaceutics classification system; BI; Boehringer Ingelheim Pharmaceuticals; CIJ; Confined impinging jet; CQAs; Critical quality attributes; DCM; Dicholoromethane; HP-55; Hydroxypropyl methylcellulose phthalate
Water soluble binary and ternary complexes of diosmin with β-cyclodextrin: Spectroscopic characterization, release studies and anti-oxidant activity
Keywords: افزایش تابش; Diosmin; β-Cyclodextrin; Complexation; Solubility enhancement; Antioxidant activity;
A comparative study on solubilizing and taste-masking capacities of hydroxypropyl-β-cyclodextrin and maltodextrins with high amylose content
Keywords: افزایش تابش; Taste-masking; Solubility enhancement; Electronic taste sensing; Electronic tongue; Maltodextrin; Hydroxypropyl-β-cyclodextrin
Preparation and characterisation of Kolliphor® P 188 and P 237 solid dispersion oral tablets containing the poorly water soluble drug disulfiram
Keywords: افزایش تابش; Solid dispersion; Solubility enhancement; Solvent evaporation; Hot melt; Disulfiram
Statistical approaches to maximize recombinant protein expression in Escherichia coli: A general review
Keywords: افزایش تابش; Solubility enhancement; Statistically designed experiments; Recombinant protein; Escherichia coli; Response surface methodology (RSM); Fractional factorial
Ultra fine super self-nanoemulsifying drug delivery system (SNEDDS) enhanced solubility and dissolution of indomethacin
Keywords: افزایش تابش; Self-nanoemulsifying drug delivery system; Indomethacin; Dissolution; Solubility enhancement;
Cyclodextrin-water soluble polymer ternary complexes enhance the solubility and dissolution behaviour of poorly soluble drugs. Case example: Itraconazole
Keywords: افزایش تابش; Ternary cyclodextrin complexes; Solubility enhancement; Transfer experiments; Intestinal drug precipitation; PBPK modelling; IVIVC