Keywords: رابطه ساختار-فعالیت; Structure-activity relationship; Beta-carboline; Haspin; Kinase; Inhibitor;
مقالات ISI رابطه ساختار-فعالیت (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: رابطه ساختار-فعالیت; Advanced glycation end products; Procyanidins; Inhibitory mechanism; Molecular docking; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Nannocystin; Structure-activity relationship; Anticancer; Eukaryotic elongation factor 1A;
Keywords: رابطه ساختار-فعالیت; Cinnamic acid ester; Acaricidal activity; Psoroptes cuniculi; Psoroptic disease; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; TMV; tobacco mosaic virus; CMV; cucumber mosaic virus; TMV-CP; tobacco mosaic virus coat protein; 1H NMR; 1H nuclear magnetic resonance; 13C NMR; 13C nuclear magnetic resonance; EC50; 50% effective concentration; HRMS; high-resolution mass spectrometry; S
Keywords: رابطه ساختار-فعالیت; Natural products-based pesticide; Fraxinellone; Pesticidal activity; Pyrazole ring; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; TMV; tobacco mosaic virus; 1H NMR; 1H nuclear magnetic resonance; 13C NMR; 13C nuclear magnetic resonance; HRMS; high-resolution mass spectrometer; EC50; half-maximal effective concentration; MST; microscale thermophoresis; SAR; structure-activity relat
Keywords: رابطه ساختار-فعالیت; SAR; structure-activity relationship; UDP-GlcNAc; UDP-N-acetylglucosamine; Peptidoglycan; MurA enzyme; Antibacterial agents; Quinazolinones;
Isatin hybrids and their anti-tuberculosis activity
Keywords: رابطه ساختار-فعالیت; Isatin hybrids; Mycobacterium tuberculosis; Quinolone; Structure-activity relationship; Review;
Keywords: رابطه ساختار-فعالیت; TMV; tobacco mosaic virus; 1H NMR; 1H nuclear magnetic resonance; 13C NMR; 13C nuclear magnetic resonance; IR; infrared spectroscopy; EC50; 50% effective concentration; HRMS; high-resolution mass spectrometry; SAR; structure-activity relationship; TMV-C
Keywords: رابطه ساختار-فعالیت; Benzothiazepine derivatives; Pyridine; 1,3-Dipolar cycloaddition; Antiviral activity; YYRNVXFTRZVMRS-UHFFFAOYSA-N; KIZODVVVLZAAEP-UHFFFAOYSA-N; AMCKYOLBFWMGPW-UHFFFAOYSA-N; RZWVFWUINNLNNM-UHFFFAOYSA-N; ITSYQYKUGUDNGM-UHFFFAOYSA-N; CHCMHFYRPUYOKD-UHFFFAOYS
Keywords: رابطه ساختار-فعالیت; Extremely randomized trees; Decision trees; Structure-activity relationship; Molecular modeling; Antimalarials; Dihydrofolate reductase; Trimethoprim; Pyrimethamine; Cycloguanil; Hydrophobic feature;
Keywords: رابطه ساختار-فعالیت; CC; carbon-carbon double bond; COOH; carboxyl; Cy; cyanidin; Dp; delphinidin; E; trans; GC; p-coumaryl-glucose unit; Mv; malvidin; OH; hydroxyl; Pg; pelargonidin; pKH; hydration constant; Pn; peonidin; Pt; petunidin; SAR; structure-activity relationsh
Keywords: رابطه ساختار-فعالیت; BBB; blood brain barrier; BK; bradykinin; Boc; t-butyloxycarbonyl; BR; bradykinin receptor; CNS; central nervous system; DALKD; [des-Arg10, Leu9]-kallidin; DIPEA; diisopropylethylamine; DMF; N,N-dimethylformamide; Dyn A; dynorphin A; Fmoc; fluorenylmethyl
Keywords: رابطه ساختار-فعالیت; Proteasome inhibitors; Phthalazinone; Triphenylphosphine; Drug design; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Drug discovery; Anticancer; Structure-activity relationship; Benzoxaborole;
Keywords: رابطه ساختار-فعالیت; BIZZGWUOKSACNS-UHFFFAOYSA-N; KGNZBIBLGJECSF-UHFFFAOYSA-N; HRDVUEQUGMWEGF-UHFFFAOYSA-N; FFJOJEQDLDDOIX-UHFFFAOYSA-N; XYEJZBSKDAHDQC-UHFFFAOYSA-N; PCNDTEOUGMJGJW-UHFFFAOYSA-N; XKJGEJQMWFNIOY-UHFFFAOYSA-N; GVJFGKNQHQKCSX-UHFFFAOYSA-N; WPXHEEXWLXFRBU-UHFFFAOY
Keywords: رابطه ساختار-فعالیت; Diphenylamine derivatives; Intermediate Derivatization Methods; Fungicidal activity; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Phosphoramide mustard prodrug; Prostate-specific antigen; Site-specific activation; Self-immolative linker; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; MTT; 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide; DPPH; 2,2-diphenyl-1-picrylhydrazyl; EDTA; ethylenediaminetetraacetic acid; ERK1/2; extracellular signal-regulated kinase; mTOR; mammalian target of rapamycin; AMPKα; 5â² adenosine monop
Keywords: رابطه ساختار-فعالیت; Asperphenamate; Dipeptide analog; Synthesis; Anticancer activity; Structure-activity relationship; Inducing autophagy;
Keywords: رابطه ساختار-فعالیت; 4,5-Dihydro-1,2,4-triazin-3(2H)-one; Pymetrozine; Insecticidal activity; Aphid; Synergistic effect; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; 1,5-Disubstituted tetrazoles; COX-2 inhibitors; COX-1 inhibitors; Molecular docking; Structure-activity relationship; Methylsulfonyl; Aminosulfonyl;
Keywords: رابطه ساختار-فعالیت; Adipose triglyceride lipase (ATGL); Atglistatin; Inhibitors; Structure-activity relationship; Lipolysis; Adipocytes;
Keywords: رابطه ساختار-فعالیت; DHLA; dihydrolipoic acid; DMEM; Dulbecco's Modified Eagle's Medium; EDTA; ethylenediaminetetraacetic acid; FBS; foetal bovine serum; GPx; glutathione peroxidase; GSH; glutathione; GSSG; glutathione disulphide; HPLC; high performance liquid chromatogra
Keywords: رابطه ساختار-فعالیت; SCLC; small cell lung cancer; NSCLC; non-small-cell lung cancer; LNCaP; human prostate adenocarcinoma; DU-145; human prostate carcinoma; MDA-MB-231; human breast adenocarcinoma; BGC-823; human gastric cancer; SI; selectivity index; SAR; structure-activi
Keywords: رابطه ساختار-فعالیت; ATX/NPP2; autotaxin; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; DMSO; dimethylsulfoxide; GPCR; G-protein coupled receptor; GRI; Genomic Research Institute; HBTU; O-(benzotriazol-1-yl)-N,N,Nâ²,Nâ²-tetramethyluronium hexafluorophosphate
Keywords: رابطه ساختار-فعالیت; Monobactam; Siderophore; Structure-activity relationship; Antibacterial activity; Click chemistry; AZN; Aztreonam; MDR; multidrug-resistant; SAR; structureâactivity relationship; PIH; pyridoxal isonicotinoyl hydrazone; Trt; triphenylmethyl; Boc; t-but
Keywords: رابطه ساختار-فعالیت; SAR; structure-activity relationship; ACT; artemisinin combination therapy; DMAP; 4-dimethylaminopyridine; EDC; N-(3-dimethylaminopropyl)-Nâ²-ethylcarbodiimide hydrochloride; Antimalarial chemotherapy; Trioxane dimer esters; Single oral dose ACT; Oral
Keywords: رابطه ساختار-فعالیت; 1,2,4-Oxadiazoles; Structure-activity relationship; Antibiotics;
Keywords: رابطه ساختار-فعالیت; Nitrogen mustard sophoridinic acid derivatives; Antitumor activity; Structure-activity relationship; Molecular docking;
Keywords: رابطه ساختار-فعالیت; Ultrasound; Five-component reaction (5-CR); Pyrimidine; Antibacterial activity; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; [6,6,5] tricyclic core structure; Structure-activity relationship; Antibacterial activity; Liver microsomal stability;
Keywords: رابطه ساختار-فعالیت; DX; Derek Nexus; LS; Leadscope; SVM; Support Vector Machine; FN; false negatives; TN; true negatives; TP; true positives; NPV; negative predictive value; PPV; positive predictive value; GTI; genotoxic impurity; SAR; structure-activity relationship; IH;
Keywords: رابطه ساختار-فعالیت; AcOH; acetic acid; Ach; acetylcholine; AChE; acetylcholinesterase; ASCh; acetylthiocholine; BChE or BuChE; butyrylcholinesterase; BSCh; butyrylthiocholine; CNS; central nervous system; DMF; N,N-dimethylformamide; DMSO; dimethylsulfoxide; DTNB; 5,5â²-dith
Keywords: رابطه ساختار-فعالیت; EC50; half-maximal effective concentration; 1H NMR; 1H nuclear magnetic resonance; 13C NMR; 13C nuclear magnetic resonance; MS; mass spectroscopy; TMV; tobacco mosaic virus; SAR; structure-activity relationship; 4-Amino-2-methylpyrimidine moiety; 1,3,4-
Keywords: رابطه ساختار-فعالیت; Mitochondrial uncoupling; Anti-obesity drugs; Metabolic diseases; Quinolinecarboxylate; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Ac; Aplysia californica; CH-IMI; nitromethylene analogue of imidacloprid; IMI; imidacloprid; LBD; ligand-binding domain; Ls; Lymnaea stagnalis; nAChR; nicotinic acetylcholine receptor; NIA; propargyl propyl phenylphosphonate (Niagara 16388); QSAR; quantit
Keywords: رابطه ساختار-فعالیت; ADME; absorption/distribution/metabolism/excretion; BBB; blood-brain barrier; CD3OD; tetradeuteromethanol; CDCl3; deuterochloroform; CH2Cl2; dichloromethane; C log D; distribution coefficient; C log P; calculated partition coefficient; CNS; central
Keywords: رابطه ساختار-فعالیت; Tubulin polymerization inhibitors; Pyrazoline; Molecular docking; CA-4; combretastatin A-4; SAR; structure-activity relationship; IC50; half maximal inhibitory concentration; MTT; 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide;
Keywords: رابطه ساختار-فعالیت; Diversity-oriented synthesis; Imidazoheterocyclic; Groebke-Blackburn-Bienayme reaction; Fused imidazole; Lewis acid; Ugi type; Ac; acetyl; Aq; aqueous; Ar; aryl; Bn; benzyl; Boc; tert-butoxycarbonyl; BDMS; bromodimethylsulfonium bromide; CDK; cyclin-d
Keywords: رابطه ساختار-فعالیت; ADME; absorption, distribution, metabolism, excretion; BBB; blood-brain barrier; CEV; California encephalitis virus; CNS; central nervous system; CPE; cytopathic effect; ECMV; encephalomyocarditis virus; fLUC; firefly luciferase; FMV; Fort Morgan virus;
Keywords: رابطه ساختار-فعالیت; Xoo; Xanthomonas oryzae pv. oryzae; Xoc; Xanthomonas oryzae pv. oryzicolaby; EC50; half-maximal effective concentration; 1H NMR; 1H nuclear magnetic resonance; 13C NMR; 13C nuclear magnetic resonance; IR; infrared spectroscopy; SAR; structure-activity r
Keywords: رابطه ساختار-فعالیت; SAR; structure-activity relationship; ACT; artemisinin combination therapy; HPLC; high performance liquid chromatography; DMAP; 4-dimethylaminopyridine; Py; pyridine; Antimalarial chemotherapy; Trioxane dimers; Single oral dose ACT; Oral bioavailability
Keywords: رابطه ساختار-فعالیت; Curcumin; BACE1; Alzheimer's disease; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Wall teichoic acids; MRSA; Ticlopidine; Clopidogrel; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; 2-Amino-4-(2-pyridyl)thiazoles; Antimycobacterial; Antiplasmodial; Structure-activity relationship; Hit optimisation;
Keywords: رابطه ساختار-فعالیت; Cantharidin; Acaricidal activity; Insecticidal activity; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Armillaria mellea; Physalacriaceae; Natural product characterization; Sesquiterpene aryl ester; Melleolide; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Cholesterol cationic lipids; Structure-activity relationship; Intracellular uptake; Gene delivery;