Keywords: رابطه ساختار-فعالیت; Cholesterol cationic lipids; Structure-activity relationship; Intracellular uptake; Gene delivery;
مقالات ISI رابطه ساختار-فعالیت (ترجمه نشده)
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Keywords: رابطه ساختار-فعالیت; Dual specificity phosphatases; Virtual screening methods; Phosphatases of regenerating liver; Enzyme inhibitors; Thienopyridone; 2-Cyano-2-ene-esters; DIFMUP; 6,8-difluoro-4-methylumbelliferyl phosphate; DSP; dual specificity phosphatase; MTT; 3-(4,5-dime
Keywords: رابطه ساختار-فعالیت; ATP; adenosine triphosphate; ADP; adenosine diphosphate; Cer; ceramide; ERK-1/2; extra-cellular signal-regulated kinase 1/2; HDAC; histone deacetylase; LDH; lactate dehydrogenase; S1P; sphingosine-1-phosphate; SAR; structure-activity relationship; Sph;
Keywords: رابطه ساختار-فعالیت; Immune thrombocytopenia; Pyrazole derivatives; Phagocytosis inhibitors; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Sulfonylhydrazide; Indoleamine 2,3-dioxygenase; Structure-activity relationship; Molecular docking;
Keywords: رابطه ساختار-فعالیت; Toxoplasma gondii; 1-Deoxy-d-xylulose-5-phosphate reductoisomerase; Protein expression; Enzyme inhibition; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; CCK; cholecystokinin ligand; CCK1-R; cholecystokinin 1 receptor; CCK2-R; cholecystokinin 2 receptor; MSH; melanotropin ligand; SAR; structure-activity relationship; Trp; tryptophan; Met; methionine; Asp; aspartic acid; Phe; phenyl alanine; Nle; norleuci
Keywords: رابطه ساختار-فعالیت; EPM; elevated plus maze; Anxiolytic-like activity; Dipeptide; Aromatic amino acid; Tyrosyl leucine; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Strigolactones; Strigolactone analogues; Germination parasitic weeds; Structure-activity relationship; Mode of action; New plant hormones; Design and synthesis;
Keywords: رابطه ساختار-فعالیت; Phthalide; 2-Benzofuran-1(3H)-one; Monoamine oxidase; MAO-B; Reversible inhibition; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; SAR; structure-activity relationship; DPPH; 2,2-diphenyl-1-picrylhydrazyl; FRSA; free radical scavenging activity; Curcumin derivatives; Antitumor; Antioxidant activity; Aqueous solubility;
Keywords: رابطه ساختار-فعالیت; Caffeic acid; Matrix metalloproteinase; Tumor; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; Strobilurin-pyrimidine; Antiproliferative activity; Lung cancer; Leukemia; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; DCM; dichloromethane; LRR; loss of righting reflex; NMDA; N-methyl-d-aspartate; PWR; pedal withdrawal reflex score; Ketamine; Esters; Anaesthesia; Short-acting; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; CC50; concentration of inhibitor resulting in 50% parasite growth inhibition; DCM; dichloromethane; DMF; N,N-dimethylformamide; DMSO; dimethyl sulfoxide; EDC·HCl; 1-ethyl-3-(3-dimethyllaminopropyl)carbodiimide hydrochloride; Et3N; triethylamine; EtOH; et
Keywords: رابطه ساختار-فعالیت; Acrylamide formation; Antioxidants; Structure-activity relationship; Reaction conditions;
Keywords: رابطه ساختار-فعالیت; Prolactin-releasing peptide; G-protein-coupled receptor; Substituted cysteine accessibility method; Methanethiosulfonate; Structure-activity relationship;
Keywords: رابطه ساختار-فعالیت; DAPI; 4â²,6-diamidino-2-phenylindole; DCC; dicyclohexylcarbodiimide; EDC; N-(3-dimethylaminopropyl)-Nâ²-ethyl-carbodiimide; FITC; fluorescein isothiocyanate; NBT/BCIP; nitro-blue tetrazolium chloride and 5-bromo-4-chloro-3â²-indolyphosphate p-toluidine
Keywords: رابطه ساختار-فعالیت; Quaternary phosphonium salts; Pyridoxine; Structure-activity relationship; Lipophilicity; Antibacterial activity;
Keywords: رابطه ساختار-فعالیت; Olfactory system; Olfactory stimulus-problem; Structure-activity relationship; Structure-odor relationship; Odor perception; Spatial coding; Olfactory receptors; Topography; Hedonics; Basic odors; Vertebrate olfaction; Insect olfaction;
Keywords: رابطه ساختار-فعالیت; AMP; Anti-microbial peptide; APA; Amino pentanoic acid; CD; Circular dichroism; CHO; Chinese hamster ovary; CPP; Cell-penetrating peptide; DLS; Dynamic Light Scattering; DMPC; Dimyristoyl phosphatidylcholine; DMPG; Dimyristoyl phosphatidylglycerol; DOPC;
Keywords: رابطه ساختار-فعالیت; 1,3-Dipolar-cycloaddition; Fatty acid; Mode of action; MR; molar refractivity; MW; molecular weight; MV; molecular volume; PASS; predicted activity spectrum of substances; PSA; polar surface area; SAR; structure-activity relationship; MIC; minimal inhib
Keywords: رابطه ساختار-فعالیت; NAM; negative allosteric modulator; nAChRs; neuronal nicotinic acetylcholine receptors; HBK; HEPES-buffered Krebs; LBVS; ligand-based virtual screening; SBVS; structure-based virtual screening; SAR; structure-activity relationship; nh; Hill coefficient;
Keywords: رابطه ساختار-فعالیت; MYCTYVPWNJZLME-UHFFFAOYSA-N; YVZSXHDGUKDVQB-QHCPKHFHSA-N; QACWKSJESHQSRJ-DEOSSOPVSA-N; ZPDZEKYMDZYYJD-NRFANRHFSA-N; BZDDMQPTXGUOMI-QFIPXVFZSA-N; BYIRXFDIJRLJDH-QFIPXVFZSA-N; QWODNELMNXBHBK-NRFANRHFSA-N; VLRQDEYLMBEMCJ-NRFANRHFSA-N; IQBKUUJAQQSHJY-NRFANRHF
Keywords: رابطه ساختار-فعالیت; DENV; dengue virus; WNV; West Nile virus; YFV; yellow fever virus; TBEV; tick-borne encephalitis virus; HCV; hepatitis C virus; WEEV; Western equine encephalitis virus; VSV; vesicular stomatitis virus; HBV; hepatitis B virus; HIV; human immunodeficiency v
In vivo anti-hyperuricemic and xanthine oxidase inhibitory properties of tuna protein hydrolysates and its isolated fractions
Keywords: رابطه ساختار-فعالیت; Hyperuricemic mice; Xanthine oxidase inhibition; Structure-activity relationship; Di-/tri-peptide; Molecular docking;
Site-specific effect of polar functional group-modification in lipids of TLR2 ligands for modulating the ligand immunostimulatory activity
Keywords: رابطه ساختار-فعالیت; Toll-like receptor 2; Pam2CSK4; Structure-activity relationship; Lipopeptide;
Synthesis of novel (â)-epicatechin derivatives as potential endothelial GPER agonists: Evaluation of biological effects
Keywords: رابطه ساختار-فعالیت; Epi; (â)-epicatechin; eNOS; endothelial nitric oxide synthase; NO; nitric oxide; GPER; G-protein coupled estrogen receptor; BCAEC; bovine coronary artery endothelial cells; GPCRs; G-protein coupled receptors; EPI-COLUMN; affinity column with Epi covalen
An efficient synthesis and biological evaluation of novel analogues of natural product Cephalandole A: A new class of antimicrobial and antiplatelet agents
Keywords: رابطه ساختار-فعالیت; Cephalandole A; Antimicrobial; Antibacterial; Antifungal; Antiplatelet activity; Structure-activity relationship;
Design, synthesis and biological evaluation of pyrazolyl-thiazolinone derivatives as potential EGFR and HER-2 kinase inhibitors
Keywords: رابطه ساختار-فعالیت; Pyrazolyl-thiazolidinone; EGFR; HER-2; Antitumor; Structure-activity relationship;
Correlation between synthesis pH, structure and Cu/MgO/Al2O3 heterogeneous catalyst activity and selectivity in CO2 hydrogenation to methanol
Keywords: رابطه ساختار-فعالیت; Co-precipitation material preparation; Metallic copper dispersion; Magnesium oxide phases; Carbon dioxide conversion; Added-value chemical production; Structure-activity relationship;
Targeting phosphatases of regenerating liver (PRLs) in cancer
Keywords: رابطه ساختار-فعالیت; Protein tyrosine phosphatase; Metastasis; Theinopyridone; Structure; CBS; cystathionine-beta-synthase; CHO; Chinese hamster ovary; CNNM; magnesium transporters of cyclin M; EMT; epithelial-mesenchymal transition; HMVEC; human microvascular endothelial c
The evaluation of potent antitumor activities of shikonin coumarin-carboxylic acid, PMMB232 through HIF-1α-mediated apoptosis
Keywords: رابطه ساختار-فعالیت; HIF-1α; hypoxia-inducible factor alpha 1; DMAP; 4 dimethyamino- pyridine; DCC; N, N' dicyclohexylcarbodiimide; DMEM; Dulbecco's modified Eagle's medium; MTT; 3-(4 5-dimethyl-2-thiazolyl)-2 5-diphenyl-2-H-tetrazolium bromide; IC50; Half of maximal i
Design and synthesis of 1-(1-benzothiophen-7-yl)-1H-pyrazole, a novel series of G protein-coupled receptor 52 (GPR52) agonists
Keywords: رابطه ساختار-فعالیت; GPR52; G protein-coupled receptor 52; SAR; structure-activity relationship; cAMP; 3â²,5â²-cyclic adenosine monophosphate; EC50; half maximal effective concentration; MAP; methamphetamine; NMDA; N-methyl-d-aspartate; PK; pharmacokinetic; CHO; Chinese h
Synthesis of jaspine B regioisomers through palladium-catalyzed stereoselective tetrahydrofuran formation: Insight into the ligand recognition of sphingosine kinases
Keywords: رابطه ساختار-فعالیت; Palladium; Sphingosine kinase; Kinase inhibitor; Jaspine B; Structure-activity relationship;
Natural products as sources of new fungicides (V): Design and synthesis of acetophenone derivatives against phytopathogenic fungi in vitro and in vivo
Keywords: رابطه ساختار-فعالیت; Natural products; Acetophenone derivatives; Antifungal activity; Structure-activity relationship;
Identification of novel quinazolinedione derivatives as RORγt inverse agonist
Keywords: رابطه ساختار-فعالیت; AUC; area under the plasma concentration-time curve; BA; bioavailability; EAE; experimental autoimmune encephalomyelitis; LBD; ligand-binding domain; RORγt; retinoic acid receptor-related orphan receptor-gamma t; SAR; structure-activity relationship; T
Structure-activity relationship of eight high content flavonoids analyzed with a preliminary assign-score method and their contribution to antioxidant ability of flavonoids-rich extract from Scutellaria baicalensis shoots
Keywords: رابطه ساختار-فعالیت; Scutellaria baicalensis shoots; UPLC-Q-TOF-MS; Primary flavonoids; Antioxidant activity; Structure-activity relationship; A preliminary assign-score method;
Fragment-growing guided design of Keap1-Nrf2 protein-protein interaction inhibitors for targeting myocarditis
Keywords: رابطه ساختار-فعالیت; ROS; reactive oxygen species; NQO-1; NADPH:quinone oxidoreductase 1; HO-1; heme oxygenase-1; ARE; antioxidant response element; Nrf2; nuclear factor erythroid 2-related factor 2; Keap1; Kelch-like ECH-associated protein 1; DMF; dimethyl fumarate; CDDO-Me;
C19-Diterpenoid alkaloid arabinosides from an aqueous extract of the lateral root of Aconitum carmichaelii and their analgesic activities
Keywords: رابطه ساختار-فعالیت; Ranunculaceae; Aconitum carmichaelii; C19-diterpenoid alkaloid; Arabinoside; Aconicarmichosides EâL; Analgesic effect; Structure-activity relationship;
Discovery and characterization of a potent Wnt and hedgehog signaling pathways dual inhibitor
Keywords: رابطه ساختار-فعالیت; Wnt signaling pathway; Hedgehog signaling pathway; Porcupine; Smoothened; Antagonist; Stem cell; Cancer therapy; AUC; area under the plasma time-concentration curve; BCC; basal cell carcinoma; BPO; benzoyl peroxide; CL; clearance; CSC; cancer stem cells;
Potential therapeutic applications of the genus Annona: Local and traditional uses and pharmacology
Keywords: رابطه ساختار-فعالیت; ABTS; 2,2-Azinobis-3-Ethylbenzothizoline-6-Sulphonate; ACGs; Acetogenins; AEF; Acetogenin-Enriched Fraction; ATP; Adenosine Triphosphate; COX; Cyclooxygenase; CYP; Cytochrome P450; DNA; Deoxyribonucleic Acid; DPPH; 1,1-Diphenyl-2-Picrylhydrazyl; EC50; Eff
Novel 12N-substituted matrinanes as potential anti-coxsackievirus agents
Keywords: رابطه ساختار-فعالیت; Matrinane; Structure-activity relationship; Coxsakievirus; Broad-spectrum; Druglike;
Cytotoxic activity, apoptosis induction and structure-activity relationship of 8-OR-2-aryl-3,4-dihydroisoquinolin-2-ium salts as promising anticancer agents
Keywords: رابطه ساختار-فعالیت; Isoquinoline; Benzo[c]phenanthridine alkaloid; Cytotoxicity; Apoptosis induction; Structure-activity relationship;
Identification of selective inhibitors of sphingosine kinases 1 and 2 through a structure-activity relationship study of 4-epi-jaspine B
Keywords: رابطه ساختار-فعالیت; Sphingosine kinase; Kinase inhibitor; Jaspine B; Structure-activity relationship;
Optically active stereoisomers of 5-(1-iodoethyl)-4-(4â²-isopropylphenyl)dihydrofuran-2-one: The effect of the configuration of stereocenters on apoptosis induction in canine cancer cell lines
Keywords: رابطه ساختار-فعالیت; Structure-activity relationship; β-Aryl-δ-iodo-γ-lactones; Apoptosis; Canine cancers; Canine cancer cell lines;
COx-free hydrogen generation via decomposition of ammonia over copper and zinc-based catalysts
Keywords: رابطه ساختار-فعالیت; Hydrogen production; Catalytic ammonia conversion; Cu/Zn/Al2O3; Metal dispersion and acid-base character; Structure-activity relationship;
Novel anti-inflammatory agents targeting CXCR4: Design, synthesis, biological evaluation and preliminary pharmacokinetic study
Keywords: رابطه ساختار-فعالیت; CXCR4; Amide-sulfamide; Inflammation; Structure-activity relationship; Pharmacokinetic study; KBWXKIUGGGUTOE-UHFFFAOYSA-N;
Development of a novel series of non-natural triaryl agonists and antagonists of the Pseudomonas aeruginosa LasR quorum sensing receptor
Keywords: رابطه ساختار-فعالیت; Anti-virulence; Pseudomonas aeruginosa; Structure-activity relationship; Computational modeling; Quorum sensing;
5-Bromo-2-aryl benzimidazole derivatives as non-cytotoxic potential dual inhibitors of α-glucosidase and urease enzymes
Keywords: رابطه ساختار-فعالیت; Benzimidazole; In vitro; Urease; α-glucosidase; Dual inhibitor; Structure-activity relationship; Thiourea; Cytotoxicity; In silico;