Keywords: UDP-گلوکورونوزیل ترانسفراز; Carcinogenesis; Chemoprevention; Chemotherapy; Oxidative stress; Nrf2; Phytochemicals; AKT; protein kinase B; AMPK; AMP-activated protein kinase; ARE; antioxidant response element; ATF-2; activating transcriptional factor; BBN; N-butyl-N-(4-hydroxybutyl)n
مقالات ISI UDP-گلوکورونوزیل ترانسفراز (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: UDP-گلوکورونوزیل ترانسفراز; Therapeutic drug monitoring; Antipsychotic; Antidepressant; Psychopharmacology; Psychiatry; Psychopharmacotherapy; Pharmacokinetics; HPLC; Mass spectrometry; LC-MS/MS; ABCB1; ATP-binding cassette sub-family B member 1; AGNP; Arbeitsgemeinschaft für Neuro
Keywords: UDP-گلوکورونوزیل ترانسفراز; Thyroid hormones; Isotope tracer; On-line SPE LC-MS/MS; Turnover rate; Thyroidectomy; Deiodinases; UDP-glucuronosyltransferases; Sulfotransferases
Keywords: UDP-گلوکورونوزیل ترانسفراز; AhR; aryl hydrocarbon receptor; ARNT; aryl hydrocarbon receptor nuclear translocator; BT; β-tubulin; CYP; cytochrome P450 monooxygenase enzymes; EF; elongation factor; GAPDH; glyceraldehyde 3-phosphate dehudrogenase; GR; glucocorticoid receptor; HSP; hea
Keywords: UDP-گلوکورونوزیل ترانسفراز; AD; Alzheimer's disease; Aβ; β amyloid peptide; ERT; estrogen replacement therapy; ESR; estrogen receptor; E1; estrone; E2; estradiol; E3; estriol; CYP; cytochrome P450; CYP11A1; cytochrome P450 cholesterol side chain cleavage enzyme; HSD-3β; 3β-hydro
Amentoflavone is a potent broad-spectrum inhibitor of human UDP-glucuronosyltransferases
Keywords: UDP-گلوکورونوزیل ترانسفراز; Amentoflavone; UDP-Glucuronosyltransferases; Broad-spectrum inhibitor; Herb-drug interactions (HDIs);
Shikonin upregulates the expression of drug-metabolizing enzymes and drug transporters in primary rat hepatocytes
Keywords: UDP-گلوکورونوزیل ترانسفراز; AhR; aryl hydrocarbon receptor; AP1; activating protein 1; ARE; antioxidant-response element; CAR; constitutive androstane receptor; CYP; cytochrome P450; DREs; dioxin-responsive elements; EMSA; electromobility gel shift assay; FBS; fetal bovine serum; GS
Resveratrol represses estrogen-induced mammary carcinogenesis through NRF2-UGT1A8-estrogen metabolic axis activation
Keywords: UDP-گلوکورونوزیل ترانسفراز; 2-MeOE1/E2; 4-MeOE1/E2, methoxyestrogens; 2-OHE1/E2; 4-OHE1/E2, hydroxyestrogens; 53BP1; tumor protein p53 binding protein 1; DMBA; 7,12-dimethylbenz(a)anthracene; DSBs; DNA double-strand breaks; E1; estrone; E2; estradiol; E2-3G; E2-3-glucuronide; E2-17G
Inefficient UGT-conjugation of adrenal 11β-hydroxyandrostenedione metabolites highlights C11-oxy C19 steroids as the predominant androgens in prostate cancer
Keywords: UDP-گلوکورونوزیل ترانسفراز; UDP; uridine diphosphate; UGT; UDP-glucuronosyltransferases; 17βHSD; 17β-hydroxysteroid dehydrogenase; AKR1C3; 17β-hydroxysteroid dehydrogenase type 5; 11βHSD2; 11β-hydroxysteroid dehydrogenase type 2; SRD5A; 5α-reductase; SRD5A1; 5α-reductase type
Development of a LC-MS/MS method to investigate the interference of pharmacokinetics of the main constituents in Saxifraga stolonifera: Involvement of drug metabolism enzymes
Keywords: UDP-گلوکورونوزیل ترانسفراز; Saxifraga stolonifera; Pharmacokinetics; Metabolism; UDP-glucuronosyltransferases; Catechol-O- methyltransferase;
Design and optimization of the cocktail assay for rapid assessment of the activity of UGT enzymes in human and rat liver microsomes
Keywords: UDP-گلوکورونوزیل ترانسفراز; Estradiol (PubChem CID: 5757); Chenodeoxycholic acid (PubChem CID: 10133); Serotonin (PubChem CID: 5202); Propofol (PubChem CID: 4943); Zidovudine (PubChem CID: 35370); CYP; cytochrome P450; UGT; UDP-glucuronosyltransferases; DDI; drug-drug interactions;
Efflux transport of estrogen glucuronides by human MRP2, MRP3, MRP4 and BCRP
Keywords: UDP-گلوکورونوزیل ترانسفراز; E1-S; estrone sulfate; E1-G; estrone glucuronide; E2-3G; estradiol-3-glucuronide; E2-17G; estradiol-17β-glucuronide; E3-3G; estriol-3-glucuronide; E3-16G; estriol-16α-glucuronide; BCRP, ABCG2; breast cancer resistance protein; MRP, ABCC; multidrug resis
Molecular and functional characterization of UDP-glucuronosyltransferase 1A in cynomolgus macaques
Keywords: UDP-گلوکورونوزیل ترانسفراز; Cynomolgus monkey; Drug metabolism; Gene; Genome; UDP-glucuronosyltransferases;
Inhibition of UDP-glucuronosyltransferase (UGT)-mediated glycyrrhetinic acid 3-O-glucuronidation by polyphenols and triterpenoids
Keywords: UDP-گلوکورونوزیل ترانسفراز; UDP-Glucuronosyltransferase; UGT; Licorice; Glycyrrhetinic acid; Glycyrrhizin; Glucuronidation; Glucuronide; Natural medicine; Adverse reaction; Pseudohyperaldosteronism; DMSO; dimethyl sulfoxide; GA; Glycyrrhetinic acid; HPLC; high-performance liquid chr
Characterization of oxycodone in vitro metabolism by human cytochromes P450 and UDP-glucuronosyltransferases
Keywords: UDP-گلوکورونوزیل ترانسفراز; Oxycodone; Cytochromes P450; UDP-glucuronosyltransferases; In vitro metabolism;
Direct comparison of UDP-glucuronosyltransferase and cytochrome P450 activities in human liver microsomes, plated and suspended primary human hepatocytes from five liver donors
Keywords: UDP-گلوکورونوزیل ترانسفراز; UDPGA; 5â²-diphosphoglucuronic acid; CRMs; chemically reactive metabolites; CYP; cytochrome P450; HLM; human liver microsomes; PHH; primary human hepatocytes; UGTs; UDP-glucuronosyltransferases; β-estradiol (PubChem CID:5757); Chenodeoxycholic acid (Pub
Identification and characterization of human UDP-glucuronosyltransferases responsible for the in vitro glucuronidation of ursolic acid
Keywords: UDP-گلوکورونوزیل ترانسفراز; Ursolic acid; UDP-glucuronosyltransferases; Metabolism pathway; Metabolism characterization; UA; ursolic acid; HLMs; human liver microsomes; HIMs; human intestinal microsomes; UGTs; UDP-glucuronosyltransferases; DDI; drug-drug interactions; RILD; Resear
The inhibitory effects of nor-oleanane triterpenoid saponins from Stauntonia brachyanthera towards UDP-glucuronosyltransferases
Keywords: UDP-گلوکورونوزیل ترانسفراز; Herb-drug interaction; Nor-oleanane triterpenoid saponins; UDP-glucuronosyltransferases
Glucuronidation of bavachinin by human tissues and expressed UGT enzymes: Identification of UGT1A1 and UGT1A8 as the major contributing enzymes
Keywords: UDP-گلوکورونوزیل ترانسفراز; Bavachinin; UDP-glucuronosyltransferases; UGT1A1; UGT1A8; Glucuronidation; Human tissues
Diethylstilbestrol can effectively accelerate estradiol-17-O-glucuronidation, while potently inhibiting estradiol-3-O-glucuronidation
Keywords: UDP-گلوکورونوزیل ترانسفراز; DES; diethylstilbestrol; UGT; UDP-glucuronosyltransferases; HLM; human liver microsomes; DLM; liver microsomes from beagle dog; RbtLM; liver microsomes from New Zealand rabbits; RLM; liver microsomes from Sprague-Dawley rats; MLM; liver microsomes from
Tissue and species differences in the glucuronidation of glabridin with UDP-glucuronosyltransferases
Keywords: UDP-گلوکورونوزیل ترانسفراز; GA; glabridin; UGT; UDP-glucuronosyltransferases; HLM and HIM; liver and intestinal microsomes from humans, respectively; RLM and RIM; liver and intestinal microsomes from rats, respectively; CyLM and DLM; liver microsomes from cynomolgus monkeys and beag
Role of cytochrome P450 and UDP-glucuronosyltransferases in metabolic pathway of homoegonol in human liver microsomes
Keywords: UDP-گلوکورونوزیل ترانسفراز; Homoegonol; 4-O-demethylation; Glucuronidation; Human liver microsomes; Cytochrome P450s; UDP-Glucuronosyltransferases
Tissue-, sex- and development-specific transcription profiles of eight UDP-glucuronosyltransferase genes in zebrafish (Danio rerio) and their regulation by activator of aryl hydrocarbon receptor
Keywords: UDP-گلوکورونوزیل ترانسفراز; Ugt; UDP-Glucuronosyltransferases; Phase II enzymes; Zebrafish; Transcription profile; Developmental expression; Aryl hydrocarbon receptor
Regioselective glucuronidation of the isoflavone calycosin by human liver microsomes and recombinant human UDP-glucuronosyltransferases
Keywords: UDP-گلوکورونوزیل ترانسفراز; HLMs; human liver microsomes; UGTs; UDP-glucuronosyltransferases; SGR; Structure-glucuronidation relationship; HPLC; high performance liquid chromatography; NADPH; nicotinamide adenine dinucleotide phosphate reduced; CYP450s; cytochrome P450s; PAPS; 3â
Hepatic expression patterns of aryl hydrocarbon receptor, pregnane X receptor, two cytochrome P450s and five phase II metabolism genes responsive to 17alpha-methyltestosterone in rare minnow Gobiocypris rarus
Keywords: UDP-گلوکورونوزیل ترانسفراز; AHR; aryl hydrocarbon receptor; PXR; pregnane X receptor; CYP; cytochrome P450; SULT; sulfotransferase; UGT; UDP-glucuronosyltransferases; AHR2; PXR; Cytochrome P450; Sulfotransferase; UDP-glucuronosyltransferases; 17Alpha-methyltestosterone;
Coupling ultra-high-pressure liquid chromatography with mass spectrometry for in-vitro drug-metabolism studies
Keywords: UDP-گلوکورونوزیل ترانسفراز; ADC; Analog-to-digital converter; ADMET; Absorption, distribution, metabolism, excretion and toxicity; APCI; Atmospheric pressure chemical ionization; CYP; Cytochrome P450; DDI; Drug-drug interaction; DMPK; Drug metabolism and pharmacokinetics; DT; Dwell
Relevance of UDP-glucuronosyltransferase polymorphisms for drug dosing: A quantitative systematic review
Keywords: UDP-گلوکورونوزیل ترانسفراز; UDP-glucuronosyltransferases; Pharmacogenetics; Polymorphism; Pharmacogenetics-based dose adjustments; Drug metabolism; UGT1A1A, Adenine; Afr, Africans; As, Asians; AUC, area under the curve; C, Cytosine; Cauc./Cau, Caucasians; Cl, Clearance; ClHet, Clear
Stilbene glucoside inhibits the glucuronidation of emodin in rats through the down-regulation of UDP-glucuronosyltransferases 1A8: Application to a drug-drug interaction study in Radix Polygoni Multiflori
Keywords: UDP-گلوکورونوزیل ترانسفراز; Radix Polygoni Multiflori; Stilbene glucoside; Emodin; Drug-drug interactions; Pharmacokinetics; UDP-glucuronosyltransferases;
Human UDP-glucuronosyltransferases: Feedback loops between substrates and ligands of their transcription factors
Keywords: UDP-گلوکورونوزیل ترانسفراز; AhR; Ah receptor; CAR; constitutive androstane receptor; CYP; cytochrome P450; FXR; farnesoid receptor; GST; glutathione S-transferase; HETE; hydroxyeicosatetraenoic acid; LATF; ligand-activated transcription factor; LTB4; leucotriene B4; PPAR; peroxisome
Absorption and metabolism of milk thistle flavanolignans in humans
Keywords: UDP-گلوکورونوزیل ترانسفراز; HCV; hepatitis C virus; ESI; electrospray interface; MRM; multiple reaction monitoring; UDP; uridine diphosphate; UGTs; UDP-glucuronosyltransferases; SULTs; sulphotransferases; EHR; entero-hepatic recirculation; amu; atomic mass unit; Flavanolignans; Urin
Effect of oxidative stress on UDP-glucuronosyltransferases in rat astrocytes
Keywords: UDP-گلوکورونوزیل ترانسفراز; UDP-glucuronosyltransferase; Astrocytes; Oxidative stress; NADPH:cytochrome P450 reductase; NAD(P)H:quinone oxidoreductase 1; 1-NP; 1-naphthol; ARE; antioxidant response element; DMSO; dimethyl sulfoxyde; FeHQ; FeCl3/8-hydroxyquinoline; FITC; fluorescein
Coupling of UDP-glucuronosyltransferases and multidrug resistance-associated proteins is responsible for the intestinal disposition and poor bioavailability of emodin
Keywords: UDP-گلوکورونوزیل ترانسفراز; AIC; Akaike's information criterion; UGT; UDP-glucuronosyltransferase; UDPGA; uridine diphosphoglucuronic acid; LTC4; leukotriene C4; NTP; National Toxicology Program; SD; Sprague-Dawley; DMEM; Dulbecco's modified Eagle's medium; AP; apical; BL; basolat
Modulation of biotransformation and elimination systems by BM-21, an aqueous ethanolic extract from Thalassia testudinum, and thalassiolin B on human hepatocytes
Keywords: UDP-گلوکورونوزیل ترانسفراز; Thalassia testudinum; Thalassiolin B; Polyphenols; Cytochrome P450; UDP-glucuronosyltransferases; P-glycoprotein; Human hepatocytesBM-21, aqueous ethanolic extract from Thalassia testudinum marine plant; TB, thalassiolin B; P450, cythocrome P450; UGT, UDP
Reliability and Robustness of Simultaneous Absolute Quantification of Drug Transporters, Cytochrome P450 Enzymes, and Udp-Glucuronosyltransferases in Human Liver Tissue by Multiplexed MRM/Selected Reaction Monitoring Mode Tandem Mass Spectrometry with Nan
Keywords: UDP-گلوکورونوزیل ترانسفراز; multiplexed MRM quantification of proteins; transporters; membrane transporter; cytochrome P450; UDP-glucuronosyltransferases; nano-LC; LC–MS/MS; mass spectrometry; proteomics
Haplotypes in the UGT1A1 gene and their role as genetic determinants of bilirubin concentration in healthy German volunteers
Keywords: UDP-گلوکورونوزیل ترانسفراز; UDP-glucuronosyltransferases; Haplotypes; Bilirubin; Caucasians
Endocrine alteration and other biochemical responses in juvenile turbot exposed to the Prestige fuel oil
Keywords: UDP-گلوکورونوزیل ترانسفراز; Prestige fuel oil; Juvenile turbot; EROD activity; FACs in bile; Plasmatic testosterone; UDP-glucuronosyltransferases
The human UDP-glucuronosyltransferase UGT1A3 is highly selective towards N2 in the tetrazole ring of losartan, candesartan, and zolarsartan
Keywords: UDP-گلوکورونوزیل ترانسفراز; Losartan; Candesartan; Zolarsartan (GR117289); UDP-glucuronosyltransferases; Substrate specificity; Tetrazole
Acute effects of novel selenazolidines on murine chemoprotective enzymes
Keywords: UDP-گلوکورونوزیل ترانسفراز; Selenium; Selenocysteine prodrugs; Selenazolidines; Mouse; mRNA; Thioredoxin reductase; Glutathione peroxidase; NAD(P)H-quinone oxidoreductase; Glutathione transferases; UDP-glucuronosyltransferases; Microsomal epoxide hydrolase
Rapid simultaneous determination of metabolic clearance of multiple compounds catalyzed in vitro by recombinant human UDP-glucuronosyltransferases
Keywords: UDP-گلوکورونوزیل ترانسفراز; UDP-glucuronosyltransferases; LC/ESI/MS/MS; n-in-one cocktails; Intrinsic clearance;
Toxicogenomic analysis of gene expression changes in rat liver after a 28-day oral benzene exposure
Keywords: UDP-گلوکورونوزیل ترانسفراز; Ah; aryl hydrocarbon; Alas2; aminolevulinic acid synthase 2; CO; control; Cyp; cytochrome P450 enzyme; G6pc; glucose-6-phosphatase; G6pd; glucose-6-phosphate dehydrogenase; GSH; glutathione; Gst; glutathione-S-transferase; Hnf; hepatic nuclear factor; Hnf