کد مقاله کد نشریه سال انتشار مقاله انگلیسی نسخه تمام متن
1366067 981580 2007 4 صفحه PDF دانلود رایگان
عنوان انگلیسی مقاله ISI
Synthesis and structure–activity relationship of RXR antagonists based on the diazepinylbenzoic acid structure
کلمات کلیدی
موضوعات مرتبط
مهندسی و علوم پایه شیمی شیمی آلی
پیش نمایش صفحه اول مقاله
Synthesis and structure–activity relationship of RXR antagonists based on the diazepinylbenzoic acid structure
چکیده انگلیسی

Synthesis and structure–activity relationship of RXR antagonists employing a diazepinylbenzoic acid scaffold are described. Of those antagonists, sulfonamide derivatives (6v and 6w) reveal a high antagonistic activity and good pharmacokinetic properties.

Synthesis and structure–activity relationship of RXR antagonists employing a diazepinylbenzoic acid scaffold are described. The sulfonamide derivatives were found to reveal a high antagonistic activity and good pharmacokinetic properties.Figure optionsDownload as PowerPoint slide

ناشر
Database: Elsevier - ScienceDirect (ساینس دایرکت)
Journal: Bioorganic & Medicinal Chemistry Letters - Volume 17, Issue 17, 1 September 2007, Pages 4808–4811
نویسندگان
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