Synthesis and evaluation of prodrugs of corticotropin-releasing factor-1 (CRF1) receptor antagonist BMS-665053 leading to improved oral bioavailability

Synthesis and evaluation of prodrugs of corticotropin-releasing factor-1 (CRF1) receptor antagonist BMS-665053 leading to improved oral bioavailability

Database: Elsevier - ScienceDirect (ساینس دایرکت)
Journal: Bioorganic & Medicinal Chemistry Letters - Volume 27, Issue 6, 15 March 2017, Pages 1360-1363

Richard A. Hartz, Vivekananda M. Vrudhula, Vijay T. Ahuja, James E. Grace, Nicholas J. Lodge, Joanne J. Bronson, John E. Macor,