Potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors based on the benzoisoxazole moiety: application of a bioisosteric scaffold hopping approach to flufenamic acid

Potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors based on the benzoisoxazole moiety: application of a bioisosteric scaffold hopping approach to flufenamic acid

Database: Elsevier - ScienceDirect (ساینس دایرکت)
Journal: European Journal of Medicinal Chemistry - Volume 150, 25 April 2018, Pages 930-945

Agnese Chiara Pippione, Irene Maria Carnovale, Davide Bonanni, Marcella Sini, Parveen Goyal, Elisabetta Marini, Klaus Pors, Salvatore Adinolfi, Daniele Zonari, Claudio Festuccia, Weixiao Yuan Wahlgren, Rosmarie Friemann, Renzo Bagnati, Donatella Boschi,