Keywords: Antileishmanial; Antimicrobial; Antiplasmodial; Antitrypanosomal; Drug discovery; Eleusine indica; Macaranga barteri;
مقالات ISI (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: Azole; Antitrypanosomal; Antiplasmodial; Antileishmanial; Antifungal; CYP51; In vivo studies; NTDs; neglected tropical diseases; CYP51; sterol 14α-demethylase; Ph; phenyl; Py; 1-pyrrolyl; Tb; Trypanosoma brucei rhodesiense; Tc; Trypanosoma cruzi; Ld; Le
Keywords: Antiplasmodial; Antimalarial; Quinolone; Fluoroquinolone; Structure-activity relationship;
Keywords: Fusidic acid; Malaria; Antiplasmodial;
Keywords: Bioorganometallic chemistry; Ferrocene; Antiplasmodial; Heterobimetallic; Water-soluble complexes
Keywords: Antimalarial; Antiplasmodial; Arylamino alcohol; Plasmepsin II enzyme; Hemozoin inhibition; Mannich reaction;
Keywords: PM; plasmepsin; SPP; signal peptide peptidase; HIV; human immunodeficiency virus; SAR; structure-activity relationships; BACE; beta-site APP cleaving enzyme 1 or beta-secretase; TCAMS; Tres Cantos Antimalarial Set; RBC; red blood cells; CatD; cathepsin
Keywords: Indoloquinoline alkaloid; Azide rearrangement; Isocryptolepine; Antiplasmodial; Antiproliferative; Cytotoxicity;
Keywords: Antiplasmodial; Alpha-glucosidase; Epoxidation; Virtual screening; Dihydroxylation
Keywords: Synthesis; Antiplasmodial; Tryptanthrin derivatives; Gametocytes; Malaria
Keywords: Pantothenamides; Antibacterial; Antiplasmodial; Baker's yeast; Coenzyme A;
Keywords: 2-Amino-4-(2-pyridyl)thiazoles; Antimycobacterial; Antiplasmodial; Structure-activity relationship; Hit optimisation;
Keywords: Marine natural products; Isonitriles; Plasmodium falciparum; Heme detoxification; Antiplasmodial
Antiplasmodial alkaloids from bulbs of Amaryllis belladonna Steud.
Keywords: Amaryllis belladonna; Crinane; Lycorine; Antiplasmodial; Bioassay-guided; OFVVOKYDPLAWBU-TUXNIGETSA-N; FNYADSSSNOZMIA-KDOFPFPSSA-N; DZXAUWNEDZVVNU-FDPQUTSJSA-N; QAHZAHIPKNLGAS-MUPGEQOCSA-N; SEWQEQSXDGJDGG-ZTFGCOKTSA-N; DONUVZIVKLIMJU-UHFFFAOYSA-N;
seco-Tiaminic acids B and C: Identification of two novel 3,4-seco-tirucallane triterpenoids isolated from the root of Entandrophragma congoënse (Meliaceae)
Keywords: Entandrophragma congoënse; Tirucallane; Triterpenes; Antiplasmodial; Cytotoxicity;
The genus Psiadia: Review of traditional uses, phytochemistry and pharmacology
Keywords: Psiadia; Terpenoids; Flavonoids; Antiplasmodial; Antimicrobial;
Biological activities of plant extracts from Ficus elastica and Selaginella vogelli: An antimalarial, antitrypanosomal and cytotoxity evaluation
Keywords: Antiplasmodial; Antitrypanosomal; Cytotoxicity; Ficus elastica; Selaginella vogelii;
Secondary metabolites and biological activity of Pentas species: A minireview
Keywords: Pentas; Lanceolata; Rubiaceae; Anthraquinone; Iridoid; Antiplasmodial; Healing;
In vitro antiplasmodial efficacy of synthetic coumarin-triazole analogs
Keywords: Coumarin; Plasmodium falciparum; Antiplasmodial; DNA gyrase;
Structure-activity relationship of new antimalarial 1-aryl-3-susbtituted propanol derivatives: Synthesis, preliminary toxicity profiling, parasite life cycle stage studies, target exploration, and targeted delivery
Keywords: Antiplasmodial; Antimalarial; Arylamino alcohol; Multi-stage activity; Hsp90; Enantiomer separation;
Isolation, structure elucidation, and synthesis of antiplasmodial quinolones from Crinum firmifolium
Keywords: Antiplasmodial; Quinolone; Crinum; Amaryllidaceae;
4-Aminoquinoline-chalcone/-N-acetylpyrazoline conjugates: Synthesis and antiplasmodial evaluation
Keywords: 4-Aminoquinoline; Chalcone; N-acetylpyrazoline; Click chemistry; Antiplasmodial;
Medicinal plants for in vitro antiplasmodial activities: A systematic review of literature
Keywords: IC50; Half-maximal inhibitory concentration; NP; Natural products; Traditional herbs; Systematic review; Antiplasmodial; In vitro; IC50;
In vitro antiplasmodial and antioxidant activities of bisbenzylisoquinoline alkaloids from Alseodaphne corneri Kosterm
Keywords: Bisbenzylisoquinoline; Laurotetanine; Norstephasubine; Antiplasmodial; Antioxidant; Oxidative stress
The changes in morphogenesis and bioactivity of Tetradenia riparia, Mondia whitei and Cyanoptis speciosa by an aeroponic system
Keywords: Aeroponic; Antibacterial; Antiplasmodial; Large-scale cultivation; Medicinal plant
Synthesis, characterization and antimicrobial evaluation of mono- and polynuclear ferrocenyl-derived amino and imino complexes
Keywords: Bioorganometallic chemistry; Ferrocene; Polyamines; Antimycobacterial; Antiplasmodial; Dendrimer
Composés á structure imidazopyridinyl-arylpropénone, nouveaux agents anti-infectieux potentiels
Keywords: Imidazopyridine; Arylpropenone; Antiplasmodial; Nematicidal; Anti-Candida albicans; Imidazopyridine; Arylpropénone; Antiplasmodial; Nématocide; Anticandidosique;
Mono- and polynuclear ferrocenylthiosemicarbazones: Synthesis, characterisation and antimicrobial evaluation
Keywords: Ferrocene; Thiosemicarbazones; Polyamines; Antimycobacterial; Antiplasmodial; Metallodendrimer
Antimalarial actions of Lawsonia inermis, Tithonia diversifolia and Chromolaena odorata in combination
Keywords: Lawsonia inermis; Tithonia diversifolia; Chromolaena odorata; Antiplasmodial; Combination
Identification of β-Amino alcohol grafted 1,4,5 trisubstituted 1,2,3-triazoles as potent antimalarial agents
Keywords: β-aminoalcohol; Antiplasmodial; Antimalarial; Pharmacokinetics; p53 protein upregulation
Apocynaceae species with antiproliferative and/or antiplasmodial properties: a review of ten genera
Keywords: Apocynaceae; antiproliferative; antiplasmodial; herbal medicine review;
Antiplasmodial constituents from the stem bark of Polyalthia longifolia var pendula
Keywords: Clerodane; Diterpenes; Antiplasmodial; Polyalthia longifolia; Bisclerodane imide;
Minor secondary metabolites from the bark of Entandrophragma congoënse (Meliaceae)
Keywords: Entandrophragma congoënse; Meliaceae; Triterpenoids; Antiplasmodial; Cytotoxicity
Antivascular and anti-parasite activities of natural and hemisynthetic flavonoids from New Caledonian Gardenia species (Rubiaceae)
Keywords: Flavonoids; Antivascular agents; Endothelial cells; Antiplasmodial; Trypanocidal; Antileishmanial
In vitro antiplasmodial activity of triazole-linked chloroquinoline derivatives synthesized from 7-chloro-N-(prop-2-yn-1-yl)quinolin-4-amine
Keywords: Antiplasmodial; 4-Aminoquinoline; CuAAC click chemistry; Triazole linkers; Resistance reversal;
Antiproliferative and antiplasmodial compounds from selected Streptomyces species
Keywords: Streptomyces; Antiproliferative; Antiplasmodial; Dereplication; Structure elucidation; Nuclear Magnetic Resonance;
Kojic acid derived hydroxypyridinone-chloroquine hybrids: Synthesis, crystal structure, antiplasmodial activity and β-haematin inhibition
Keywords: IDOOIPQTVCLXSY-UHFFFAOYSA-N; LIOLOYTVLKUEJJ-UHFFFAOYSA-N; Hydroxypyridinone; Kojic acid; Haematin inhibition; Antiplasmodial; Hybrids;
Indolosesquiterpene alkaloids from the Cameroonian medicinal plant Polyalthia oliveri (Annonaceae)
Keywords: Polyalthia oliveri; Annonaceae; Indolosesquiterpenes; Absolute configuration; High resolution mass spectrometry; Antiplasmodial; Cytotoxicity;
Research PaperHPLC-based activity profiling for antiplasmodial compounds in the traditional Indonesian medicinal plant Carica papaya L
Keywords: Carica papaya; Antiplasmodial; HPLC-based activity profiling; Piperidine alkaloid; Carpaine; Flavonol;
Isolation and relative stereochemistry of lippialactone, a new antimalarial compound from Lippia javanica
Keywords: Antiplasmodial; Lippialactone; Malaria; Verbenaceae; Lippia javanica;
Voulkensin C-E, new 11-oxocassane-type diterpenoids and a steroid glycoside from Caesalpinia volkensii stem bark and their antiplasmodial activities
Keywords: Caesalpinia volkensii; 11-Oxocassane-type diterpenoids; 3-O-[β-Glucopyranosyl(1â2)-O-β-xylopyranosyl]-stigmasterol; Antiplasmodial;
Tetrazole-based deoxyamodiaquines: Synthesis, ADME/PK profiling and pharmacological evaluation as potential antimalarial agents
Keywords: ADME; absorption distribution metabolism excretion; HPLC; High pressure liquid chromatography; LC-MS; Liquid chromatography mass spectrometry; LORA; Low Oxygen Recovery Assay; MABA; Microplate Alamar Blue Assay; TMSN3; trimethylsilyl azide; Antiplasmodi
Botany, uses, phytochemistry and pharmacology of Vallaris: A short review
Keywords: Antiproliferative; Antiplasmodial; Antimicrobial; Analgesic; Anti-inflammatory;
Isolation and identification of β-hematin inhibitors from Flacourtia indica as promising antiplasmodial agents
Keywords: Flacourtia indica; Phenolic glycoside; Phenylpropanoid catechin; Antiplasmodial; β-Hematin; Hydrogen peroxide-mediated hemin degradation
Monoterpenes with antibacterial activities from a Cameroonian medicinal plant Canthium Multiflorum (Rubiaceae)
Keywords: Canthium multiflorum; Rubiaceae; Iridoids; Antibacterial; Antiplasmodial
Synthesis and antiprotozoal activities of benzyl phenyl ether diamidine derivatives
Keywords: Diamidines; Prodrugs; Benzyl phenyl ether derivatives; Antiprotozoal; Antitrypanosomal; Antiplasmodial; AntileishmanialATMS, artemisinin; BPE, benzyl phenyl ether; CQ, chloroquine; FMD, furamidine; HAT, human African trypanosomiasis; IC50, 50% inhibition
Flavonoids with antiplasmodial and cytotoxic activities of Macaranga triloba
Keywords: Euphorbiaceae; Macaranga triloba; Flavonoids; Malaysianone A; Antiplasmodial; Cytotoxic
Benzoheterocyclic amodiaquine analogues with potent antiplasmodial activity: Synthesis and pharmacological evaluation
Keywords: Benzothiazole; Benzoxazole; Amodiaquine; Benzoheterocyclic; Antiplasmodial; Reactive metabolite; Quinone imine
Flavonoids from Friesodielsia discolor
Keywords: Friesodielsia discolor; Annonaceae; Flavonoids; Antimycobacterial; Antiplasmodial; Cytotoxicity;
Antiparasitic compounds from Cornus florida L. with activities against Plasmodium falciparum and Leishmania tarentolae
Keywords: Cornus; Antiplasmodial; Antileishmanial; Malaria; Cytotoxicity; Triterpene; Betulinic acid;