Keywords: نفوذ مغز; Blood-brain barrier; Brain tumors; Drug delivery; Brain penetration; Nanoparticles;
مقالات ISI نفوذ مغز (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: نفوذ مغز; Brain/plasma-ratio; In vivo; Steady state; Brain penetration; Drug discovery; Loading dose; Rat; 3Rs-benefit; AUC; area under the plasma concentration curve; BBB; blood-brain-barrier; B/P-ratio; brain/plasma-ratio of drug concentration; CNS; central ner
Keywords: نفوذ مغز; Carbapenems; Pharmacokinetics; Brain penetration
P-glycoprotein (MDR1/ABCB1) and Breast Cancer Resistance Protein (BCRP/ABCG2) affect brain accumulation and intestinal disposition of encorafenib in mice
Keywords: نفوذ مغز; ABCB1; ABCG2; CYP3A enzymes; Encorafenib; Brain penetration;
Generation-6 hydroxyl PAMAM dendrimers improve CNS penetration from intravenous administration in a large animal brain injury model
Keywords: نفوذ مغز; Dendrimer; Hypothermic circulatory arrest; Canine model; Brain penetration; CSF/serum ratio; Biodistribution;
Cyclic AC253, a novel amylin receptor antagonist, improves cognitive deficits in a mouse model of Alzheimer's disease
Keywords: نفوذ مغز; Amylin receptor; AC253 peptide; Alzheimer's disease; Amyloid β; In vivo imaging; Brain penetration;
Discovery of novel potent imidazo[1,2-b]pyridazine PDE10a inhibitors
Keywords: نفوذ مغز; PDE10a inhibitor; Insulin secretagogues; Type 2 diabetes; GPCR; GSIS; Brain penetration;
Synthesis and biological evaluation of novel imidazol-1-ylacetic acid derivatives as non-brain penetrant bombesin receptor subtype-3 (BRS-3) agonists
Keywords: نفوذ مغز; Anti-obesity; Antedrug; Bombesin receptor subtype-3 (BRS-3); Brain penetration; Imidazole;
Basic neuroscienceIn vivo real time non invasive monitoring of brain penetration of chemicals with near-infrared spectroscopy: Concomitant PK/PD analysis
Keywords: نفوذ مغز; NIRS; HbO2; Hb; O2; CO2; Rat brain; In vivo; Non invasive; PK/PD; Brain penetration;
Comparative biodistribution and safety profiling of olmesartan medoxomil oil-in-water oral nanoemulsion
Keywords: نفوذ مغز; Olmesartan nanoemulsion; Tissue distribution; Sub-chronic toxicity; Hematological parameters; Histopathological characteristics; Brain penetration;
Synthesis and biological evaluation of novel chiral diazepine derivatives as bombesin receptor subtype-3 (BRS-3) agonists incorporating an antedrug approach
Keywords: نفوذ مغز; Anti-obesity; Antedrug; Bombesin receptor subtype-3 (BRS-3); Brain penetration; Diazepine;
Discovery of novel chiral diazepines as bombesin receptor subtype-3 (BRS-3) agonists with low brain penetration
Keywords: نفوذ مغز; Bombesin receptor subtype-3 (BRS-3) agonists; Diazepine; Brain penetration;
Sildenafil is not a useful modulator of ABCB1 and ABCG2 mediated drug resistance in vivo
Keywords: نفوذ مغز; Multidrug resistance; P-glycoprotein; BCRP protein; Brain penetration; Sildenafil; Docetaxel; Topotecan; Doxorubicin;
Indolyl and dihydroindolyl N-glycinamides as potent and in vivo active NPY5 antagonists
Keywords: نفوذ مغز; Indolyl glycinamide; Dihydroindolyl glycinamide; PGP efflux; Brain penetration
Research reportVerification of brain penetration of the unbound fraction of a novel HER2/EGFR dual kinase inhibitor (TAK-285) by microdialysis in rats
Keywords: نفوذ مغز; Brain and blood microdialysis; Brain penetration; TAK-285; Adsorption to outflow tubing; Perfusion with BSA;
N-Heteroaryl glycinamides and glycinamines as potent NPY5 antagonists
Keywords: نفوذ مغز; NPY5; N-Aryl glycinamide; Microsomal stability; Brain penetration;
Discovery of 3,9-diazabicyclo[4.2.1]nonanes as potent dual orexin receptor antagonists with sleep-promoting activity in the rat
Keywords: نفوذ مغز; Sleep; Insomnia; Diazepane; GPCR antagonist; Brain penetration; Orexin; Receptor;
Brain penetration of local anaesthetics in the rat: Implications for experimental neuroscience
Keywords: نفوذ مغز; Local anaesthetic; Anaesthesia; Brain exposure; Brain penetration; Brain tissue binding; fMRI; Electrophysiology;
Quantitative microdialysis using modified ultraslow microdialysis: Direct rapid and reliable determination of free brain concentrations with the MetaQuant technique
Keywords: نفوذ مغز; Quantitative; Microdialysis; Ultraslow; Recovery; Brain; Brain penetration; In vivo
CNS penetration of small molecules following local inflammation, widespread systemic inflammation or direct injury to the nervous system
Keywords: نفوذ مغز; Blood–brain barrier; Blood–spinal cord barrier; Brain penetration; Nerve injury; Pain; Oxycodone; Morphine; Atenolol
In vivo evaluation of P-glycoprotein and breast cancer resistance protein modulation in the brain using [11C]gefitinib
Keywords: نفوذ مغز; P-gp; BCRP; [11C]Gefitinib; GF120918; Cyclosporin A; Brain penetration
N-Glycine-sulfonamides as potent dual orexin 1/orexin 2 receptor antagonists
Keywords: نفوذ مغز; Orexin; Dual orexin antagonist; N-Glycine-sulfonamide; Oral bioavailability; Brain penetration
Discovery of brain penetrant, soluble, pyrazole amide EP1 receptor antagonists
Keywords: نفوذ مغز; Non-acidic EP1 antagonist; Amide EP1 antagonist; Brain penetration; CNS penetration; Solubility; Improved solubility; Oral exposure; Oral absorption
3,4-Dihydro-2H-benzo[1,4]oxazine derivatives as 5-HT6 receptor antagonists
Keywords: نفوذ مغز; 5-HT6 antagonist; Benzoxazine; Brain penetration; hERG; Lipophilicity
Preformulation studies and estimation of brain penetration for two alpidem analogues having anticonvulsant activity
Keywords: نفوذ مغز; Alpidem analogues; Solubility; Stability; Microdialysis; Brain penetration; Received 7 February 2005, accepted for publication 12 April 2005;