Synthesis, biological evaluation and molecular modeling of a novel series of 7-azaindole based tri-heterocyclic compounds as potent CDK2/Cyclin E inhibitors
Keywords: Cyclin-dependent kinase 2; Kinase inhibitors; Anti-tumor agent; 1H-pyrrolo[2,3-b]pyridine; [3Â +Â 2] cycloaddition; 1,4-Triazole; 1,5-Triazole; 3D-QSAR CoMFA; CCR2; CC chemokine receptor 2; CCL2; CC chemokine ligand 2; CCR5; CC chemokine receptor 5;