Keywords: مهار کننده رقابت; Xanthine oxidase; Genistein; Competitive inhibitor; Inhibition mechanism; Multispectroscopic methods; Molecular simulation
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Keywords: مهار کننده رقابت; Lipoxygenase inhibitors; Alkyl protocatechuates; Slow-binding inhibitor; Competitive inhibitor;
Keywords: مهار کننده رقابت; CO; competitive inhibitor; [D]; molar concentration of antipsychotics in the extracellular fluid; DAT; dopamine transporter; D2R; dopamine D2 receptor; D2H; high-affinity D2R; D2L; low-affinity D2R; EC50; half-maximal effective concentration; Kd; dissocia
Inhibition of Leishmania amazonensis arginase by fucogalactan isolated from Agrocybe aegerita mushroom
Keywords: مهار کننده رقابت; Agrocybe aegerita; Fucogalactan; Chemical structure; Leishmania amazonensis; Arginase; Competitive inhibitor;
A broad spectrum amperometric pesticide biosensor based on glutathione S-transferase immobilized on graphene oxide-gelatin matrix
Keywords: مهار کننده رقابت; GST; CDNB; Pesticide biosensors; Substrate specificity; Dinocap; Competitive inhibitor;
Selective inhibition of monoamine oxidase A by purpurin, an anthraquinone
Keywords: مهار کننده رقابت; Purpurin; Monoamine oxidase A; Selective inhibitor; Competitive inhibitor; Molecular docking;
Mechanism of inhibition of botulinum neurotoxin type A light chain by two quinolinol compounds
Keywords: مهار کننده رقابت; Botulinum; Neurotoxin; Quinolinol; Competitive inhibitor; FRET peptide; Fluorescence quenching;
Pyrrole-indolinone SU11652 targets the nucleoside diphosphate kinase from Leishmania parasites
Keywords: مهار کننده رقابت; Nucleoside diphosphate kinase; Purine-salvage pathway; Leishmania; Pyrrole-indolinone compounds; Competitive inhibitor; Biophysical characterization; NDK; Nucleoside Diphosphate Kinase; LmNDK; NDK from Leishmania major; DSF; Differential Scanning Fluoresc
Competitive protein tyrosine phosphatase 1B (PTP1B) inhibitors, prenylated caged xanthones from Garcinia hanburyi and their inhibitory mechanism
Keywords: مهار کننده رقابت; PTP1B; protein tyrosine phosphatase 1B; IC50; the inhibitor concentration leading 50% activity loss; Ki; inhibition constant; Kiapp; apparent Ki; Vmax; maximum velocity; Km; Michaelis-Menten constant; Kobs; apparent first-order rate constant for the trans
Azachalcones: A new class of potent polyphenol oxidase inhibitors
Keywords: مهار کننده رقابت; PPO; Tyrosinase; Azachalcone; Competitive inhibitor
Blocking the entrance of AMP pocket results in hormetic stimulation of imidazolium-based ionic liquids to firefly luciferase
Keywords: مهار کننده رقابت; Ionic liquid; Hormetic concentration response; Molecular dynamics simulation; Competitive inhibitor; Luciferase;
Inhibition of chrysin on xanthine oxidase activity and its inhibition mechanism
Keywords: مهار کننده رقابت; Xanthine oxidase; Chrysin; Competitive inhibitor; Inhibition mechanism; Multispectroscopic methods; Molecular simulation;
Salicylic acid inhibits enzymatic browning of fresh-cut Chinese chestnut (Castanea mollissima) by competitively inhibiting polyphenol oxidase
Keywords: مهار کننده رقابت; Chinese chestnut; Competitive inhibitor; Enzymatic browning; Peroxidase; Polyphenol oxidase; Salicylic acid; Salicylic acid (PubChem CID: 338);
Alt a 1 from Alternaria interacts with PR5 thaumatin-like proteins
Keywords: مهار کننده رقابت; Alt a 1; PR5-thaumatin-like protein; Kiwi-PR5; Competitive inhibitor; Alternaria; Kiwi;
Inhibitory effects of celastrol on rat liver cytochrome P450 1A2, 2C11, 2D6, 2E1 and 3A2 activity
Keywords: مهار کننده رقابت; Celastrol; Cytochrome P450 (CYP); Competitive inhibitor; Mixed-type inhibitor
Identification of 3-acyl-2-phenylamino-1,4-dihydroquinolin-4-one derivatives as inhibitors of the phosphatase SerB653 in Porphyromonas gingivalis, implicated in periodontitis
Keywords: مهار کننده رقابت; IC50; half-maximal inhibitory concentration; MIC; minimum inhibitory concentration; IL-8; interleukin-8; PMSF; phenylmethylsulfonyl fluoride; DMSO; dimethyl sulfoxide; MAPK; mitogen-activated protein kinase; Periodontitis; Gram-negative anaerobe; Haloacid
Bergamottin is a competitive inhibitor of CYP1A1 and is antimutagenic in the Ames test
Keywords: مهار کننده رقابت; Antimutagenesis; Grape fruit juice; Bergamottin; Salmonella typhimurium; Competitive inhibitor;
Exploration of α-aminophosphonate N-derivatives as novel, potent and selective inhibitors of protein tyrosine phosphatases
Keywords: مهار کننده رقابت; α-Aminophosphonate; Protein tyrosine phosphatases; Competitive inhibitor; Selective inhibitor; Cell viability; ApoptosisDMEM, Dulbecco's modified Eagle's medium; EA, elemental analysis; ESI-MS, electrospray ionization mass spectrometry; FBS, fetal bovine
Probing the binding pocket of the active site of aromatase with 2-phenylaliphatic androsta-1,4-diene-3,17-dione steroids
Keywords: مهار کننده رقابت; Aromatase; Competitive inhibitor; Androsta-1,4-diene-3,17-dione; 2-Phenylaliphatic substituent; Suicide substrate; Breast cancer
Effect of the axial ligands on the structure and reactivity of tin verdoheme in the ring opening process
Keywords: مهار کننده رقابت; Heme degradation; Tin porphyrin; Ring opening; Axial ligand; Competitive inhibitor; DFT;
How tin metal prevents verdoheme ring opening? Comparative study of various nucleophiles
Keywords: مهار کننده رقابت; Heme degradation; Tin verdoheme; Ring opening; Tin porphyrin; Competitive inhibitor; Nucleophilic addition;
Synthesis and biological evaluation of helicid analogues as mushroom tyrosinase inhibitors
Keywords: مهار کننده رقابت; Helicid analogues; Tyrosinase inhibitors; Competitive inhibitor; Inhibition kinetics; Circular dichroism
Aminoethyl chitooligosaccharides inhibit the activity of angiotensin converting enzyme
Keywords: مهار کننده رقابت; Chitooligosaccharides (COS); Aminoethyl COS; Competitive inhibitor; Angiotensin I converting enzyme (ACE); Chitosan; Chitin
Lithospermic acid as a novel xanthine oxidase inhibitor has anti-inflammatory and hypouricemic effects in rats
Keywords: مهار کننده رقابت; Lithospermic acid; Xanthine oxidase; Superoxide scavenging; Competitive inhibitor; Neutrophilis; Gouty arthritis
X-ray absorption analysis of the active site of Streptomyces antibioticus Tyrosinase upon binding of transition state analogue inhibitors
Keywords: مهار کننده رقابت; Tyrosinase; Streptomyces; X-ray absorption spectroscopy; Competitive inhibitor; Kojic acid; MXAN; Reaction center; Crystal structure
Synthesis of 5-deoxy-5-phospho-d-ribonohydroxamic acid: a new competitive and selective inhibitor of type B ribose-5-phosphate isomerase from Mycobacterium tuberculosis
Keywords: مهار کننده رقابت; Competitive inhibitor; Phosphate sugar; 5-Phosphate d-ribose isomerase; 6-Phosphate d-allose isomerase; RpiB;
Improvement of ACE inhibitory activity of chitooligosaccharides (COS) by carboxyl modification
Keywords: مهار کننده رقابت; Chitooligosaccharides (COS); Angiotensin I converting enzyme (ACE); Carboxylated COS; Quartenized amino COS; Competitive inhibitor
Structure-activity relationships of 2-, 4-, or 6-substituted estrogens as aromatase inhibitors
Keywords: مهار کننده رقابت; Aromatase inhibition; 2-Halogeno estrogens; 6-Alkyl estrogens; 6-Aryl estrogens; Structure-activity relationship; Competitive inhibitor;
A combination formula of Michaelis-Menten-Monod type
Keywords: مهار کننده رقابت; Michaelis-Menten; Monod; Competitive inhibitor; Noncompetitive inhibitor; Huxley's allometric law;