Keywords: 5-HT; 5-Hydroxytryptamine or serotonin; AA-5-HT; N-arachidonoyl-serotonin; ACEA; arachidonoyl 2â²-chloroethylamide; AEA; N-arachidonoylethanolamine; 2-AG; 2-arachidonoylglycerol; AM251; N-(piperidin-1-yl)-5-(4-iodophenyl)-1-(2,4-dichlorophenyl)-4-methyl-
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SGIP1 alters internalization and modulates signaling of activated cannabinoid receptor 1 in a biased manner
Keywords: Seven transmembrane receptors; G-protein coupled receptors; Cannabinoid receptor 1; Protein-protein interactions; Bias signaling; Receptor endocytosis; SGIP1; src homology 3-domain growth factor receptor-bound 2-like (endophilin) interacting protein 1; CC
Cannabinoid receptor interacting protein (CRIP1a) attenuates CB1R signaling in neuronal cells
Keywords: 2-AG; 2-arachidonoylglycerol; BSA; bovine serum albumin; CB1; cannabinoid receptor; CP55940; (â)-cis-3-[2-Hydroxy-4-(1,1-dimethylÂheptyl)phenyl]-trans-4-(3-hydroxypropyl)cyclohexanol; CRIP1a; Cannabinoid Receptor Interacting Protein 1a; DAGL; diacylgly
The interaction of cannabinoid receptor agonists, CP55940 and WIN55212-2 with membranes using solid state 2H NMR
Keywords: Cannabinoid receptor agonist; Win55212-2; CP55940; THC; Lipid membrane phase transition; Drug membrane interaction; Lipid domain; Solid state NMR;
In vitro and in vivo pharmacological characterization of two novel selective cannabinoid CB2 receptor inverse agonists
Keywords: THCÎ; 9-tetrahydrocannabinol; BSA; bovine serum albumin; CHO; Chinese hamster ovary; CP55940; (â)-cis-3-[2-hydroxy-4-(1,1-dimethylheptyl)phenyl]-trans-4-(3-hydroxypropyl)cyclohexanol; DMSO; dimethyl sulphoxide; JTE-907; N-(1,3-benzodioxol-5-ylmethyl)-1
Cannabinoid receptor-mediated translocation of NO-sensitive guanylyl cyclase and production of cyclic GMP in neuronal cells
Keywords: CB1 cannabinoid receptor; CP55940; cyclic GMP; Gene expression; G-protein coupled receptors; G-proteins; NO-sensitive guanylyl cyclase; Protein translocation; Real-time polymerase chain reaction; Rimonabant (SR141716); WIN55212-2;
Interactions between endocannabinoids and stress-induced decreased sensitivity to natural reward
Keywords: AEA, N-arachidonylethanolamine; 2-AG, 2-arachidonylglycerol; CB1, Central cannabinoid receptor; FAAH, Fatty acid amide hydrolase; ANOVA, Analysis of variance.Allostasis; Cannabinoid; CB1 receptor; CP55940; Fatty acid amide hydrolase; Rimonabant; URB597
Identification and characterisation of a novel splice variant of the human CB1 receptor
Keywords: 2-AG; 2-arachidonoylglycerol; CP55940; (â)-cis-3-[2-hydroxy-4-(1,1-dimethylheptyl)phenyl]-trans-4-(3-hydroxypropyl)cyclohexanol; WIN55,212-2; R(_)-[2,3-di-hydro-5-methyl-3-[(morpholinyl)methyl]pyrrolo[1,2,3-de]-1,4-benz-oxazinyl]-(1-naphthalenyl)-methan