Keywords: دگزوسی سیتیدین کیناز; Chemotherapy; Imaging; Pancreatic cancer; Pathology; Radiotherapy; Targeted therapy; 18FDG-PET; 18F-fluorodeoxyglucose-positron emission tomography; 5FU; 5-fluorouracil; α-SMA; α-smooth muscular actin; AA; amino acid; APA; adapted physical activity; ATP
مقالات ISI دگزوسی سیتیدین کیناز (ترجمه نشده)
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The 4-N-acyl and 4-N-alkyl gemcitabine analogues with silicon-fluoride-acceptor: Application to 18F-Radiolabeling
Keywords: دگزوسی سیتیدین کیناز; dFdC; 2â²,2â²-difluoro-2â²-deoxycytidine (Gemcitabine); hENT1; human equilibrative nucleoside transport protein 1; dCK; deoxycytidine kinase; dFdU; 2â²,2â²-difluorouridine; CDA; cytidine deaminase; [18F]FAC; 1-(2-deoxy-2-[18F]fluoro-β-d-arabinofuran
Nucleosidic DNA demethylating epigenetic drugs - A comprehensive review from discovery to clinic
Keywords: دگزوسی سیتیدین کیناز; ALL; Acute lymphoblastic leukemia; AML; Acute myeloid leukemia; AUC; Area under the curve; AZA; 5-azacytidine; 5-aza-CdR; 2â²-deoxy-5-azacytidine; 5-aza-CR; 5-azacytidine; AZN; Azanucleosides; BED; Biologically effective dose; BSC; Best supportive care;
All-trans retinoic acid enhances gemcitabine cytotoxicity in human pancreatic cancer cell line AsPC-1 by up-regulating protein expression of deoxycytidine kinase
Keywords: دگزوسی سیتیدین کیناز; ACEIs; angiotensin converting enzyme inhibitors; ANOVA; analysis of variance; ATRA; all-trans retinoic acid; dCK; deoxycytidine kinase; IC50; half-maximal (50%) inhibitory concentration; PFS; progression-free survival; RARs; retinoic acid receptors; RXRs;
Monophosphorylation by deoxycytidine kinase affects apparent cellular uptake of decitabine in HCT116 colon cancer cells
Keywords: دگزوسی سیتیدین کیناز; Equilibrative nucleoside transporter 1; Uridine; Decitabine; Deoxycytidine kinase; Monophosphorylation; Irinotecan; Etoposide; Cytarabine; Gemcitabine; Kinetics;
Sugar-modified poly(propylene imine) dendrimers as drug delivery agents for cytarabine to overcome drug resistance
Keywords: دگزوسی سیتیدین کیناز; ALL; acute lymphocytic leukemia; AML; acute myeloid leukemia; Ara-C; cytarabine; Ara-CTP; cytarabine triphosphate; CDD; cytidine deaminase; dCK; deoxycytidine kinase; DP; dipyridamole; FBS; fetal bovine serum; hENT1; human equilibrative nucleoside transpo
Acquisition of chemoresistance to gemcitabine is induced by a loss-of-function missense mutation of DCK
Keywords: دگزوسی سیتیدین کیناز; Gemcitabine; Deoxycytidine kinase; Chemoresistance; MKN28; TGBC1-TKB;
Protein phosphatase 2A regulates deoxycytidine kinase activity via Ser-74 dephosphorylation
Keywords: دگزوسی سیتیدین کیناز; dCK; deoxycytidine kinase; pSer-74-dCK; dCK phosphorylated at Ser-74; ATM; ataxia telangiectasia mutated; PP; Ser/Thr phosphatase; PP1; Ser/Thr protein phosphatase 1; PP1c; catalytic subunit of PP1; PP2A; Ser/Thr protein phosphatase 2A; PP2Ac; catalytic s
Facile method for determination of deoxycytidine kinase activity in biological milieus
Keywords: دگزوسی سیتیدین کیناز; Chemiluminescent assay; Deoxycytidine kinase; Gemcitabine
ReviewGemcitabine: Metabolism and molecular mechanisms of action, sensitivity and chemoresistance in pancreatic cancer
Keywords: دگزوسی سیتیدین کیناز; 5â²-NT; 5â²-nucleotidase; APE1/Ref1; Apurinic/apyrimidinic endonuclease 1/redox-factor-1; CDA; Cytidine deaminase; cN; Cytosolic 5â²-nucleotidase; CXCL12; C-X-C motif chemokine 12; CXCR4; C-X-C motif chemokine receptor 4; dCK; Deoxycytidine kinase; dCT
Stearoyl gemcitabine nanoparticles overcome resistance related to the over-expression of ribonucleotide reductase subunit M1
Keywords: دگزوسی سیتیدین کیناز; Cytotoxicity; In vivo anti-tumor activity; Proteomics; Nucleoside transporter; Deoxycytidine kinase; siRNA
Phosphorylation of deoxycytidine kinase on Ser-74: Impact on kinetic properties and nucleoside analog activation in cancer cells
Keywords: دگزوسی سیتیدین کیناز; CLL; dCTP; Deoxycytidine kinase; Nucleoside analogs; Ser-74 phosphorylation;
Levels of Gemcitabine Transport and Metabolism Proteins Predict Survival Times of Patients Treated With Gemcitabine for Pancreatic Adenocarcinoma
Keywords: دگزوسی سیتیدین کیناز; Nucleoside Transporters; Drug Metabolism; Pancreatic Cancer; Biomarker; CI; confidence interval; dCK; deoxycytidine kinase; hENT1; human equilibrative nucleoside transporter 1; HR; hazard ratio; OS; overall survival; PDAC; pancreatic ductal adenocarcinoma
Cladribine inhibits cytokine secretion by T cells independently of deoxycytidine kinase activity
Keywords: دگزوسی سیتیدین کیناز; Cladribine; Deoxycytidine kinase; Immunomodulation; Multiple sclerosis; Purine nucleoside; T cells;
Identification of genes associated to 2â²,2â²-difluorodeoxycytidine resistance in HeLa cells with a lentiviral short-hairpin RNA library
Keywords: دگزوسی سیتیدین کیناز; araC; 1-β-arabinofuranocylcytosine; dCK; deoxycytidine kinase; dFdC; 2â²,2â²-difluorodeoxycytidine; 5-FdUrd; 5-fluorodeoxyuridine; RNAi; RNA interference; shRNA; short-hairpin RNA; siRNA; short-interfering RNA; SFPQ; splicing factor proline/glutamine-r
Evaluation of a UCMK/dCK fusion enzyme for gemcitabine-mediated cytotoxicity
Keywords: دگزوسی سیتیدین کیناز; Gemcitabine; Deoxycytidine kinase; Uridine/cytidine monophosphate kinase; Pathway engineering; Fusion protein; Gene therapy
3-Deazauridine enhances the antileukemic action of 5-aza-2′-deoxycytidine and targets drug-resistance due to deficiency in deoxycytidine kinase
Keywords: دگزوسی سیتیدین کیناز; 5-Aza-2′-deoxycytidine; 3-Deazauridine; Epigenetic therapy; Synergy; Drug-resistance; Deoxycytidine kinase; Acute lymphoblastic leukemia
Regulation by degradation, a cellular defense against deoxyribonucleotide pool imbalances
Keywords: دگزوسی سیتیدین کیناز; ADA; adenosine deaminase; 5BU; 5-Bromo uracil; AdR; deoxyadenosine; cdN; cytosolic 5â²-deoxynucleotidase; cNI; cytosolic 5â²-nucleotidase I; cNII; cytosolic 5â²-nucleotidase II; cpm; counts per minute; dCK; deoxycytidine kinase; dGK; deoxyguanosine kin
Casein kinase 1δ activates human recombinant deoxycytidine kinase by Ser-74 phosphorylation, but is not involved in the in vivo regulation of its activity
Keywords: دگزوسی سیتیدین کیناز; Deoxycytidine kinase; Ser-74 phosphorylation; Casein kinase 1δ; Post-translational modification; Nucleoside analogue; B-CLL cells
Evaluation of the role of three candidate human kinases in the conversion of the hepatitis C virus inhibitor 2′-C-methyl-cytidine to its 5′-monophosphate metabolite
Keywords: دگزوسی سیتیدین کیناز; Antiviral drugs; siRNA; Nucleoside/nucleotide derivatives; Metabolism and activation; Uridine–cytidine kinase; Deoxycytidine kinase
Gene Expression Levels as Predictive Markers of Outcome in Pancreatic Cancer after Gemcitabine-Based Adjuvant Chemotherapy
Keywords: دگزوسی سیتیدین کیناز; 5â²-NT; 5â²-nucleotidase; AC; adjuvant chemotherapy; CDA; cytidine deaminase; dCK; deoxycytidine kinase; DFS; disease-free survival; EUS-FNA; endoscopic ultrasound-guided fine needle aspiration; FFPE; formalin-fixed paraffin-embedded; hENT1; human equil
5-Fluorocytosine derivatives as inhibitors of deoxycytidine kinase
Keywords: دگزوسی سیتیدین کیناز; Immunology; Virology; Cancer; Deoxycytidine kinase; Pharmacokinetics
Lead optimization and structure-based design of potent and bioavailable deoxycytidine kinase inhibitors
Keywords: دگزوسی سیتیدین کیناز; Immunology; Virology; Cancer; Deoxycytidine kinase; Pharmacokinetics
Mimicking phosphorylation of Ser-74 on human deoxycytidine kinase selectively increases catalytic activity for dC and dC analogues
Keywords: دگزوسی سیتیدین کیناز; Deoxycytidine kinase; Nucleoside analogues; Prodrug phosphorylation; Protein phosphorylation; Subcellular localisation
Positive regulation of deoxycytidine kinase activity by phosphorylation of Ser-74 in B-cell chronic lymphocytic leukaemia lymphocytes
Keywords: دگزوسی سیتیدین کیناز; B-CLL lymphocytes; Deoxycytidine kinase; Immunocytochemistry; Nucleoside analogues; Ser-74 phosphorylation
Cell cycle effect on the activity of deoxynucleoside analogue metabolising enzymes
Keywords: دگزوسی سیتیدین کیناز; Deoxycytidine kinase; Deoxyguanosine kinase; Cell proliferation; 5′-Nucleotidase; Deoxynucleoside analogue; Resistance
The pattern of deoxycytidine- and deoxyguanosine kinase activity in relation to messenger RNA expression in blood cells from untreated patients with B-cell chronic lymphocytic leukemia
Keywords: دگزوسی سیتیدین کیناز; Purine analogues; Deoxycytidine kinase; Deoxyguanosine kinase; Chronic lymphocytic leukemia
Increased expression of mRNA specific for thymidine kinase, deoxycytidine kinase or thymidine phosphorylase in human papillary thyroid carcinoma
Keywords: دگزوسی سیتیدین کیناز; Human papillary thyroid carcinoma; Thymidine kinase 1; Deoxycytidine kinase; Thymidine phosphorylase; mRNA expression;
Docking simulation with a purine nucleoside specific homology model of deoxycytidine kinase, a target enzyme for anticancer and antiviral therapy
Keywords: دگزوسی سیتیدین کیناز; Deoxycytidine kinase; Computer aided molecular design; Docking simulation; Homology modeling; Antiviral and anticancer therapyAra-C, cytarabine; aa, amino acid; CAMD, computer aided molecular design; c, crystal; CdA, cladribine; Cyd, cytidine; dCKc, human
Activation of deoxycytidine kinase by deoxyadenosine: Implications in deoxyadenosine-mediated cytotoxicity
Keywords: دگزوسی سیتیدین کیناز; Deoxycytidine kinase; Cytotoxicity; 2-Chlorodeoxyadenosine; Adenosine deaminase; Tyrosine kinase inhibitors; Limited trypsinolysis; MAP kinase signalling;
Activity profiles of deoxynucleoside kinases and 5â²-nucleotidases in cultured adipocytes and myoblastic cells: insights into mitochondrial toxicity of nucleoside analogs
Keywords: دگزوسی سیتیدین کیناز; AZT; 3â²-azido-2â²,3â²-dideoxythymidine; cN-1b; cytosolic 5â²-nucleotidase 1b; cN-2; cytosolic 5â²-nucleotidase; dCK; deoxycytidine kinase; dGK; deoxyguanosine kinase; DMEM; Dubelcco's modified Eagle's medium; DNC; deoxynucleotide carrier; dNK; deoxy
The 5â²-nucleotidases as regulators of nucleotide and drug metabolism
Keywords: دگزوسی سیتیدین کیناز; 2,3-BPG; 2,3-bisphosphoglycerate; 3TCMP; 2â²-deoxy-3â²-thiacytidine monophosphate; 5-EddU; 5-ethynyl-dideoxyuridine; 5â²-NT; 5â²-nucleotidase; ADA; adenosine deaminase; AK; adenosine kinase; ALL; acute lymphoblastic leukemia; AML; acute myeloid leukem