Keywords: نخود; COSY; correlation spectroscopy; DIPEA; diisopropylethylamine; DS; degree of substitution; DMSO; dimethylsulfoxide; GlcA; glucuronic acid; GlcNAc; N-acetylglucosamine; HA; hyaluronan; h; hour; HSQC; hetero nuclear single quantum coherence; IPA; isopropyl a
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Keywords: نخود; Bub1; budding uninhibited by benzimidazoles 1; Cbz; benzyloxycarbonyl; CD69; a human transmembrane C-Type lectin protein; DAST; diethylaminosulfur trifluoride; dba; dibenzylideneacetone; DIPEA; N,N-diisopropylethylamine; DMAD; dimethyl acetylenedicarboxyl
Keywords: نخود; Acac; acetylacetone; Ar; aryl; BDPP; 2,4-bis(diphenylphosphino)pentane; BINAP; 2,2â²-bis(diphenylphosphino)-1,1â²-binaphthyl; BINOL; 1,1â²-bi-2-naphthol; Bn; benzyl; Boc; tert-butoxycarbonyl; Bz; benzoyl; Cbz; benzyloxycarbonyl; Cy; cyclohexyl; DCE; 1,
Keywords: نخود; Ac; acetyl; AD-mix; asymmetric dihydroxylation mix; ATP; adenosine triphosphate; Bn; benzyl; Boc; tert-butyloxycarbonyl; Bu; butyl (n-Bu, n-butyl; I; isobutyl; sec-Bu; sec-butyl; t-Bu; tert-butyl); Bz; benzoyl; CAL-B; Candida antartcia lipase-B; CAN; ceri
Keywords: نخود; Ac; acetyl; AcOH; acetic acid; AccQ; 6-aminoquinolyl-N-hydroxysuccinimidyl carbamate; AIDA; 1-aminoindan-1,5-dicarboxylic acid; aq.; aqueous; BA; butylamine; Boc; tert-butyloxycarbonyl; t-BuCQD; t-butylcarbamoylated quinidine-based CSP; t-BuCQN; t-butylca
Keywords: نخود; BS; brassinosteroids; DMAP; N,N-dimethylaminopyridine; EBl; 24-epibrassinolide; DIPEA; N,N-diisopropylethylamine; TBAF; tetra-n-butylammonium fluoride; TBAI; tetra-n-butylammonium iodide; TBSCl; tert-butyldimethylsilyl chloride; TFA; trifluoroacetic acid;
Identification of highly selective and potent orexin receptor 1 antagonists derived from a dual orexin receptor 1/2 antagonist based on the structural framework of pyrazoylethylbenzamide
Keywords: نخود; OX1R; orexin 1 receptor; OX2R; orexin 2 receptor; DORA; dual orexin receptor antagonist; SORA; selective orexin receptor antagonist; SI; selectivity index; BBB; blood-brain barrier; CNS; central nervous system; SAR; structure-activity relationship; Boc; t
Design, selection, and development of cyclic peptide ligands for human erythropoietin
Keywords: نخود; AC; affinity chromatography; BSA; bovine serum albumin; CHAPS; 3-[(3-cholamidopropyl) dimethylammonio]-1-propanesulfonate; CHO; Chinese hamster ovary; DCM; dichloromethane; DCR; divide couple re-combine; DIPEA; diisopropylethylamine; DMF; N,N-dimethylform
Keywords: نخود; ADMET; adsorption distribution metabolism excretion and toxicity; CtD; complexity-to-diversity; DCC; N,Nâ²-dicyclohexylcarbodiimide; DCE; 1,2-dichloroethane; DIPEA; N,Nâ²-diisopropylethylamine; DMAP; 4-dimethylaminopyridine; DMF; N,Nâ²-dimethylformamid
Keywords: نخود; BBB; blood brain barrier; BK; bradykinin; Boc; t-butyloxycarbonyl; BR; bradykinin receptor; CNS; central nervous system; DALKD; [des-Arg10, Leu9]-kallidin; DIPEA; diisopropylethylamine; DMF; N,N-dimethylformamide; Dyn A; dynorphin A; Fmoc; fluorenylmethyl
Keywords: نخود; ABTS; 2,2â²-azino-bis(3-ethylbenzothiazoline-6-sulfonic acid)diammonium salt; BSA; bovine serum albumin; (bt)-VEGF165; biotinylated-VEGF165; 6-Cl·HOBt; 6-chloro-1-hydroxybenzotriazole dehydrate; DIPEA; N,N-diisopropylethylamine; ELISA; enzyme-linked imm
Keywords: نخود; RNCGDQLZIATDOU-ZDRBWGSPSA-N; ICYPJNZJUFGALC-PDTBJYIYSA-N; PDRMAVOIWIVXKH-SFUSBHMVSA-N; ISADXJRTBSLWPX-ZDRBWGSPSA-N; NLBLLPROASDPSC-QWWZWVQMSA-N; XKMIKZDBUOHHDK-ZDRBWGSPSA-N; BTURADNXKHTWGA-IJOLSIAMSA-N; UEKHRDLXBMZMPD-ZYIYBEKCSA-N; UQCLCXDOXVZEOA-JARUQAPT
Keywords: نخود; AA; amino acid; AcOH; acetic acid; 6-Cl-HOBt; 6-chloro-1-hydroxybenzotriazole; DCM; dichloromethane; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; Fmoc; 9-fluorenylmethoxycarbonyl; h; hour; HOBt; 1-hydroxybenzotriazole hydrate; HPLC; high-
Keywords: نخود; SAMs; self-assembled monolayers; RG; reactive group; GOX; glucose oxidase; LOX; lactate oxidase; HAOX; hydroxyacid oxidase; BSA; bovine serum albumin; NHS; N-hydroxysuccinimide; TFAAD; trifluoroacetyl-protected 10-amino-1-decene; TFA; trifluoroacetyl; TFE
Keywords: نخود; Antisense oligonucleotides; PEGylation; Disulfide bioconjugates; Solid phase synthesis; Gene silencing; ON; oligonucleotide; PEG; polyethylene glycol; CPG; controlled pore glass; LCAA; long chain amino alkyl; TCEP; tris(2-carboxyethyl)phosphin; TBP; tri-n
Keywords: نخود; BPO; benzoyl peroxide; DCM; dichloromethane; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; DMSO; dimethyl sulfoxide; FaSSIF; fasted state simulated intestinal fluid; HATU; 1-[bis(dimethylamino)methylene]-1H-1,2,3-triazolo[4,5-b]pyridinium
Keywords: نخود; Sulfatase; Enzyme; Inhibitor; Estrogen; Cancer; SERM; ALP; alkaline phosphatase; DEA; diethylamine; DHEA; dehydroepiandrosterone; DHEAS; dehydroepiandrosterone sulfate; 5-diol; 5-androstene-3β,17β-diol; DIPEA; diisopropylamine; E1; estrone; E1S; estrone
Keywords: نخود; ATX/NPP2; autotaxin; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; DMSO; dimethylsulfoxide; GPCR; G-protein coupled receptor; GRI; Genomic Research Institute; HBTU; O-(benzotriazol-1-yl)-N,N,Nâ²,Nâ²-tetramethyluronium hexafluorophosphate
Keywords: نخود; Pro-apoptotic agents; Anticancer agents; Cyclic peptides; Peptidomimetics; Nur77; Tubulin; Bcl-2; NMR studies; Molecular modeling; Confocal microscopy; FACS analysis; ADT; AutoDock Tools; COSY; correlation spectroscopy; DBU; 1,8-Diazabicyclo[5.4.0]undec-7
Keywords: نخود; Ac; acetyl; ALS; acetolactate synthase; aq; aqueous; BzCl; benzoyl chloride; cat.; catalytic; DBU; 1,8-diazabicyclo[5.4.0]undec-7-ene; DIPEA; diisopropylethylamine; DMA; dimethylacetamide; DME; dimethoxyethane; DMF; dimethylformamide; equiv; equivalent; F
Keywords: نخود; Nitro compounds; Natural products; Pharmaceuticals; Stereoselective synthesis; Organocatalysis; Metal catalysis; Nitronates; Nitrile oxides; AIBN; azobisisobutyronitrile; AZADO; 2-azaadamantane-N-oxyl; 9-BBN; 9-borabicyclo[3.3.1]nonane; BINAP; 2,2â²-bis(
Keywords: نخود; SPPS; solid phase peptide synthesis; DMF; dimethyl formamide; DIPEA; diisopropylethylamine; DIPC; diisopropylcarbodiimide; HOBt; 1-hydroxybenzotriazole; Fmoc; 9-fluorenylmethyloxycarbonyl; HFIP; 1,1,1,3,3,3-hexafluoropropan-2-ol; TFA; trifluoroacetic acid
Keywords: نخود; Abz; ortho-aminobenzoic acid; EDDnp; N-(2,4-dinitrophenyl)-ethylenediamine; FRET; fluorescence resonance energy transfer; hMIP; human mitochondrial intermediate peptidase; HOBt; hydroxybenzotriazole; TBTU; O-(benzotriazol-1-yl)-N,N,Nâ²,Nâ²-tetramethylur
Keywords: نخود; Diosgenin; Thioureas; Selenoureas; Antioxidant; ROS scavenger; Antiproliferative agent; BHT; butylated hydroxytoluene, 2,6-di-tert-butyl-4-methylphenol; CM-H2DCFDA; 5-(and-6) chloromethyl-2â²,7â²-dichlorodihydrofluorescein diacetate acetyl ester; CuAAC;
Keywords: نخود; Obesity; Diabetes; DGAT1; Inhibitor; Adamantane; DGAT; acyl CoA:diacylglycerol acyltransferase; TG; triglyceride; DIPEA; N,N-diisopropylethylamine; OLTT; oral lipid tolerance test; DIO; diet-induced obesity; EDCI; 1-ethyl-3-(3-dimethylaminopropyl)carbodii
Keywords: نخود; AA; arachidonic acid; AD; Alzheimer disease; AdA; adrenic acid; ALA; α-linolenic acid; AMPP; N-(4-aminomethylphenyl)pyridinium; APCI; atmospheric pressure chemical ionization; aSAH; aneurysmal subarachnoid hemorrhage; BHT; butylated hydroxytoluene; BSTFA
Keywords: نخود; Phthalocyanines; Carbohydrates; Glycophthalocyanines; Water-solubility; Photodiagnosis; Photodynamic therapy (PDT); Cel; cellobiose; CH; carbohydrate; DBU; 1,8-diazabicyclo[5.4.0]undec-7-ene; Diglyme; diglycol methyl ether; DIPEA; N,Nâ²-diisopropylethyla
Keywords: نخود; AMPs; antimicrobial peptides; ATCC; American type culture collection; CD; circular dichroism; CFU; colony forming units; CLSI; Clinical and Laboratory Standards Institute; DIPEA; N,N-diisopropylethylamine; DMEM; Dulbecco's modified eagle's medium; DMF; N,
Keywords: نخود; Peptidomimetic boronates; Proteasome inhibitors; Docking studies; ChT-L; chymotrypsin-like; T-L; trypsin-like; PGPH; post-glutamyl peptide hydrolyzing; DMSO; dimethyl sulfoxide; DMF; dimethylformamide; Pd2(dba)3; tris(benzylideneacetone)dipalladium; EDC;
Design, synthesis, in vitro and in vivo evaluation, and structure-activity relationship (SAR) discussion of novel dipeptidyl boronic acid proteasome inhibitors as orally available anti-cancer agents for the treatment of multiple myeloma and mechanism stud
Keywords: نخود; SAR; structureactivity relationship; UPP; ubiquitinproteasome pathway; FDA; Food and Drug Administration; ATP; Adenosine triphosphate; CP; core particle; RP; regulatory proteasome; C-L; caspase-like; T-L; trypsin-like; CT-L; chymotrypsin-like; EDCI; 1-eth
DNA sequence-specific ligands. XVII. Synthesis, spectral properties, virological and biochemical studies of fluorescent dimeric bisbenzimidazoles DBA(n)
Keywords: نخود; topo-I; DNA topoisomerase I; DMT; DNA methyltransferase; HSV-1; herpes simplex virus type 1; CMV; cytomegalovirus; scDNA; supercoiled DNA; b.p.; base pairs; MABs; monoclonal antibodies; ACV; acyclovir; PBS; phosphate buffered saline; PFU/cells; plaque for
Microcystins: Synthesis and structure-activity relationship studies toward PP1 and PP2A
Keywords: نخود; Adda; (2S,3S,8S,9S)-3-amino-9-methoxy-2,6,8-trimethyl-10-phenyldeca-4,6-dienoic acid; Amba; (2S,3S)-3-amino-2-methylbutanoic acid; Boc; tert-butoxycarbonyl; BOP; benzotriazol-1-yloxy-tris-dimethylaminophosphoniumhexafluoro phosphate; Cbz; carboxybenzyl; D
Cathepsin B inhibitors: Further exploration of the nitroxoline core
Keywords: نخود; Abz; 2-aminobenzoyl; AMC; 7-amido-4-methylcoumarin; catB; cathepsin B; DIPEA; N,N-diisopropylethylamine; DMSO; dimethyl sulfoxide; ECM; extracellular matrix; EDC; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide; HATU; 1-[bis(dimethylamino)methylene]-1H-1,2,
Design and synthesis of alkyl substituted pyridino[2,3-D]pyrimidine compounds as PI3Kα/mTOR dual inhibitors with improved pharmacokinetic properties and potent in vivo antitumor activity
Keywords: نخود; PI3K; phosphoinositide 3-kinase; mTOR; mammalian target of rapamycin; TSC; tuberous sclerosis; DDQ; 2,3-dicyano-5,6-dichlorobenzoquinone; THF; tetrahydrofuran; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; MRT; mean retention time; PI3Kα/
Novel aromatic sulfonyl naphthalene-based boronates as 20S proteasome inhibitors
Keywords: نخود; TEA; triethylamine; THF; tetrahydrofuran; Py; pyridine; DIPEA; N,N-diisopropylethylamine; TBTU; 2-(1H-benzotriazole-1-yl)-1,1,3,3-tetramethyluronium tetrafluoroborate; DCM; dichloromethane; TPLM; (1R)-(S)-pinanediol-1-ammonium trifluoroacetate-3-methylbut
Optimization of permeability in a series of pyrrolotriazine inhibitors of IRAK4
Keywords: نخود; ABC; Activated B Cell-like; BTK; Bruton's Tyrosine Kinase; CD79; Cluster of Differentiation 79; CDK; Cyclin Dependent Kinase; CLK; CDC-Like Kinase; DCM; dichloromethane; DDQ; 2,3-Dichloro-5,6-DicyanobenzoQuinone; DIPEA; N,N-diisopropylethylamine; DLBCL;
Design, synthesis, and evaluation of carboxyl-modified oseltamivir derivatives with improved lipophilicity as neuraminidase inhibitors
Keywords: نخود; NA; neuraminidase; OS; oseltamivir; OC; oseltamivir carboxylate; TFA; trifluor-oacetic acid; HATU; 1-[bis(dimethylamino)methylene]-1H-1,2,3-triazolo[4,5-b]pyr-idinium 3-oxid hexafluorophosphate; DIPEA; N,N-diisopropylethylamine; PDB; protein data bank; In
Scaffold hopping identifies 6,8-disubstituted purines as novel anaplastic lymphoma kinase inhibitors
Keywords: نخود; ALK; anaplastic lymphoma kinase; cMet; hepatocyte growth factor receptor; DIPEA; N,N-Diisopropylethylamine; DMF; N,N-Dimethylformamide; EML4; echinoderm microtubule-associated protein-like 4; FDA; food and drug administration; gk; gatekeeper; μW; micro w
Branched pentapeptides as potent inhibitors of the vascular endothelial growth factor 165 binding to Neuropilin-1: Design, synthesis and biological activity
Keywords: نخود; Neuropilin-1; VEGF165; Neuropilin/VEGF165 binding inhibition; Structure-activity relationship; Peptide biostability; ABTS; 2,2â²-azino-bis(3-ethylbenzothiazoline-6-sulfonic acid) diammonium salt; Ahp; 7-aminoheptanoic acid; Aun; 11-aminoundecanoic acid;
Development of potent and proteolytically stable human neuromedin U receptor agonists
Keywords: نخود; Neuromedin U (NMU); NMU-8; Neuromedin U receptor agonists; Plasma stability; 1â²Nal; 1â²-naphtylalanine; 2â²Nal; 2â²-naphtylalanine; 7-OH-Tic; 7-hydroxy-L-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid; ACN; acetonitrile; AUC; area under the curve;
Remarkable differences and similarities between the isomeric Mn(II)-cis- and trans-1,2-diaminocyclohexane-N,N,Nâ²,Nâ²-tetraacetate complexes
Keywords: نخود; MRI; magnetic resonance imaging; DFT; Density Functional Theory; APC; aminopolycarboxylate; CA; contrast agent; dtpa; diethylenetriaminepentaacetic acid; dota; 1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid; NSF; nephrogenic systemic fibrosis; e
The 4-N-acyl and 4-N-alkyl gemcitabine analogues with silicon-fluoride-acceptor: Application to 18F-Radiolabeling
Keywords: نخود; dFdC; 2â²,2â²-difluoro-2â²-deoxycytidine (Gemcitabine); hENT1; human equilibrative nucleoside transport protein 1; dCK; deoxycytidine kinase; dFdU; 2â²,2â²-difluorouridine; CDA; cytidine deaminase; [18F]FAC; 1-(2-deoxy-2-[18F]fluoro-β-d-arabinofuran
Fragment-growing guided design of Keap1-Nrf2 protein-protein interaction inhibitors for targeting myocarditis
Keywords: نخود; ROS; reactive oxygen species; NQO-1; NADPH:quinone oxidoreductase 1; HO-1; heme oxygenase-1; ARE; antioxidant response element; Nrf2; nuclear factor erythroid 2-related factor 2; Keap1; Kelch-like ECH-associated protein 1; DMF; dimethyl fumarate; CDDO-Me;
Synthesis and biological evaluation of a library of hybrid derivatives as inhibitors of influenza virus PA-PB1 interaction
Keywords: نخود; Anti-Influenza; PA-PB1; RdRp; Amino acid coupling; SPPS; Diphenyl-pyridine; AcOEt; Ethyl acetate; CC50; Half maximal cytotoxic concentration; cRNA; complementar RNA; DCM; dichloromethane; DDQ; 2,3-Dichloro-5,6-dicyano-1,4-benzoquinone; DIPEA; N,N-Diisopro
Design, synthesis, and structure-activity-relationship of a novel series of CXCR4 antagonists
Keywords: نخود; Chemokine; CXCR4; Antagonist; GPCR; Scaffold hybridization; Therapy; APC; allophycocyanin; BPO; benzoyl peroxide; CCD; charge coupled device; CYP; cytochrome P450; DC; dendritic cells; DCE; 1,2-dichloroethane; DIPEA; N,N-diisopropylethylamine; DMEM; Dulbe
Synthesis and evaluation of a novel urea-based 68Ga-complex for imaging PSMA binding in tumor
Keywords: نخود; SPECT; single photon emission computer tomography; PET; positron emission tomography; HPLC; High performance liquid chromatography; HRMS; High-resolution mass spectrometry; PBS; phosphate buffered saline; SPE; solid-phase extraction; GMP; good manufacturi
Synthesis and biological evaluation of novel thiazole- VX-809 hybrid derivatives as F508del correctors by QSAR-based filtering tools
Keywords: نخود; Aminoarylthiazole; Corrector; QSAR; Cystic fibrosis; CFTR; VX809; CF; cystic fibrosis; CFTR; CF transmembrane conductance regulator; AATs; aminoarylthiazoles; HS-YFP; halide-sensitive yellow fluorescent protein; QSAR; quantitative-structure activity relat
Discovery and evaluation of Cav3.1-selective T-type calcium channel blockers
Keywords: نخود; AcOH; acetic acid; 9-BBN; 9-borabicyclo(3.3.1)nonane; DAST; diethylaminosulfur trifluoride; DIPEA; N,N-diisopropylethylamine; DMAP; 4-(dimethylamino)pyridine; DMF; N,N-dimethylformamide; EDC·HCl; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide hydrochlorid
Phenylglycine racemization in Fmoc-based solid-phase peptide synthesis: Stereochemical stability is achieved by choice of reaction conditions
Keywords: نخود; COMU; (1-cyano-2-ethoxy-2-oxoethylidenaminooxy)dimethylaminomorpholinocarbenium hexafluorophosphate; DBU; 1,8-diazabicyclo[5.4.0]undec-7-ene; DEPBT; 3-diethoxyphosphoryloxy)-1,2,3-benzotriazin-4(3H)-one; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethyl
Discovery and evaluation of Cav3.2-selective T-type calcium channel blockers
Keywords: نخود; AcOH; acetic acid; Boc; tert-butylocycarbonyl; DIPEA; N,N-diisopropylethylamine; DMAP; 4-(dimethylamino)pyridine; DMF; N,N-dimethylformamide; EDC·HCl; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide hydrochloride; HOBt; hydroxybenzotriazole; KHMDS; potassi