دانلود مقالات ISI درباره نخود + ترجمه فارسی

Discovery of benzothiazoles as antimycobacterial agents: Synthesis, structure-activity relationships and binding studies with Mycobacterium tuberculosis decaprenylphosphoryl-β-d-ribose 2′-oxidase

Keywords: نخود; TB; tuberculosis; Mtb; Mycobacterium tuberculosis; MIC; minimal inhibitory concentration; CYP; cytochrome P450; SAR; structure-activity relationships; MMIC; mammalian cytotoxicity; DprE1; decaprenylphosphoryl-β-d-ribose 2′-oxidase; TEA; triethylamine

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2015 سفارش ترجمه

Design, chemical synthesis and biological evaluation of 3-spiromorpholinone/3-spirocarbamate androsterone derivatives as inhibitors of 17β-hydroxysteroid dehydrogenase type 3

Keywords: نخود; ADT; androsterone; AR; androgen receptor; Ar; aryl group; DBD; DNA binding domain; DCM; dichloromethane; DHT; dihydrotestosterone; DIPEA; N,N-diisopropylethylamine; DMF; dimethylformamide; DMSO; dimethylsulfoxide; Δ4-dione; 4-androstene-3,17-dione; EtOAc

دانلود رایگان متن کامل مقاله ISI 43 صفحه سال انتشار : 2015 سفارش ترجمه

Structure-based design and synthesis of covalent-reversible inhibitors to overcome drug resistance in EGFR

Keywords: نخود; CRI; covalent reversible inhibitor; EDC·HCl; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide hydrochloride; HOBt; hydroxybenzotriazole; DIPEA; N,N-diisopropylethylamine; EGFR; epidermal growth factor receptor; NOE; nuclear Overhauser effect; NSCLC; non-sma

دانلود رایگان متن کامل مقاله ISI 48 صفحه سال انتشار : 2015 سفارش ترجمه

The synthesis of indolo[2,3-b]quinoline derivatives with a guanidine group: Highly selective cytotoxic agents

Keywords: نخود; Neocryptolepine; Antiproliferative activity; Antifungal activity; Biofilm; Guanidine group; Mechanism of action; Apoptosis; Hemolytic activity; Boc; tert-butyloxycarbonyl group; BSTU; N,N′-bis-Boc-thiourea; DIPEA; N,N-diisopropylethylamine; DMF; dimethy

دانلود رایگان متن کامل مقاله ISI 50 صفحه سال انتشار : 2015 سفارش ترجمه

Design and synthesis of novel small molecule CCR2 antagonists: Evaluation of 4-aminopiperidine derivatives

Keywords: نخود; AcOH; acetic acid; Boc; tert-butyloxycarbonyl; CCL2; chemokine ligand 2; CCR2; chemokine receptor 2; DCE; dichloroethane; DCM; dichloromethane; DIPEA; N,N-diisopropylethylamine; DMAP; N,N-dimethylaminopyridine; DMSO; dimethylsulfoxide; INCB3344; N-(2-(((3

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2014 سفارش ترجمه

Structure-activity relationships of non-opioid [des-Arg7]-dynorphin A analogues for bradykinin receptors

Keywords: نخود; BK; bradykinin; BR; bradykinin receptor; CNS; central nervous system; DALKD; [des-Arg10, Leu9]-kallidin; DIPEA; diisopropylethylamine; DMF; N,N-dimethylformamide; Dyn A; dynorphin A; Fmoc; 9-fluorenylcarboxy; HBTU; 2-(1H-benzotriazole-1-yl)-1,1,3,3-tetram

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2014 سفارش ترجمه

Potentiometric determination of dissociation constant and thermodynamic parameters of dissociation process of some newly synthesized pyrimidine derivatives in MeOH/DMF-water medium at different temperatures

Keywords: نخود; DCP; 2, 4-dichloropyrimidine; TMA; 4-((1H-1, 2, 4-triazol-1-yl) methyl)aniline; DIPEA; N, N-diisopropylethyl amine; DMF; N, N-dimethylformamide; A R; Analytical reagent; Dissociation constant; Pyrimidine derivative; Methanol; DMF; Thermodynamic parameter;

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2014 سفارش ترجمه

A total synthesis of a highly N-methylated cyclodepsipeptide [2S,3S-Hmp]-aureobasidin L using solid-phase methods

Keywords: نخود; Aureobasidin; N-Methylated cyclodepsipeptide; Depsidipeptide; Fmoc-based solid-phase peptide synthesis; Boc; tert-butyloxycarbonyl; BTC; bis-(trichloromethyl)-carbonate; 13C NMR; carbon-13 nuclear magnetic resonance; COSY; correlation spectroscopy; DBU; 1

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2014 سفارش ترجمه

The CuI-catalyzed alkyne-azide cycloaddition as direct conjugation/cyclization method of peptides to steroids

Keywords: نخود; Steroids; Peptide conjugates; Click chemistry; Peptidosteroids; Conjugation; Boc; tert-butoxycarbonyl; CuAAC; CuI-catalyzed alkyne-azide 1,3-dipolar cycloaddition; EDC; 1-(3-dimethylaminopropyl)-3-ethylcarbodiimide; DIPEA; N,N-di-iso-propyl-N-ethylamine

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2014 سفارش ترجمه

A site-selective, irreversible inhibitor of the DNA replication auxiliary factor proliferating cell nuclear antigen (PCNA)

Keywords: نخود; APC; allophycocyanin; ATR; ataxia telangiectasia mutated and rad3-related; BCA; bicinchoninic acid; Chk1; checkpoint kinase 1; CSK buffer; cytoskeleton buffer; DBU; 1,8-diazabicyclo[5.4.0]undec-7-ene; DCM; dichloromethane; DIPEA; N,N-diisopropylethylamine

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2014 سفارش ترجمه

Targeting (cellular) lysosomal acid ceramidase by B13: Design, synthesis and evaluation of novel DMG-B13 ester prodrugs

Keywords: نخود; B13; (1R,2R)-2-(tetradecanoylamino)-1-(4′-nitrophenyl)-1,3-propandiol; DMG; N,N-dimethyl glycine; LCL521; 1,3-O,O-DMG-B13 dihydrochloride; LCL522; 3-O-DMG-B13 hydrochloride; LCL596; 1-O-DMG-B13 hydrochloride; CX; stable mono-DMG-B13; ACDase; acid cerami

دانلود رایگان متن کامل مقاله ISI 12 صفحه سال انتشار : 2014 سفارش ترجمه

Tetrahedron report number 1022Recent developments of the Stille reaction as a revolutionized method in total synthesis

Keywords: نخود; Stille coupling; Natural product; Palladium; Total synthesis; Cross coupling; CuTC; copper(I) thiophene-2-carboxylate; DIBAL-H; diisobutylaluminum hydride; DIPEA; diisopropylethylamine; DMF; dimethylformamide; MOM; methoxymethyl; NMP; N-methylpyrrolidone;

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2014 سفارش ترجمه

Design, synthesis, and structure-activity relationships of a series of novel N-aryl-2-phenylcyclopropanecarboxamide that are potent and orally active orexin receptor antagonists

Keywords: نخود; OX1R; orexin 1 receptor; OX2R; orexin 2 receptor; THF; tetrahydrofuran; TBDPS; tert-butyldiphenylsilyl; DMF; N,N-dimethylformamide; DIAD; diisopropyl azodicarboxylate; TBAF; tetra-n-butylammonium fluoride; DMSO; dimethyl sulfoxide; TEA; triethylamine; DCM

دانلود رایگان متن کامل مقاله ISI 18 صفحه سال انتشار : 2014 سفارش ترجمه

Discovery and optimization of novel small-molecule HIV-1 entry inhibitors using field-based virtual screening and bioisosteric replacement

Keywords: نخود; ADME; absorption, distribution, metabolism, and excretion; AMLV; amphotropic murine leukemia virus; BBB; blood-brain barrier; BIF; bioisostere factor; CNS; central nervous system; DCM; dichloromethane; DiEA; diisopropylethylamine; DIPEA; N,N-diisopropyl

دانلود رایگان متن کامل مقاله ISI 26 صفحه سال انتشار : 2014 سفارش ترجمه

Intramolecular Diels-Alder reaction as a key step in tandem or sequential processes: a versatile tool for the synthesis of fused and bridged bicyclic or polycyclic compounds

Keywords: نخود; Diels-Alder; Natural product; One-pot; Sequential; Tandem; IMDA; intramolecular Diels-Alder; IMHDA; intramolecular hetero Diels-Alder; DA; Diels-Alder; IEDDA; intramolecular inverse-electron-demand Diels-Alder; DAIB or DIB; diacetoxyiodobenzene;

دانلود رایگان متن کامل مقاله ISI 32 صفحه سال انتشار : 2014 سفارش ترجمه

Antiprotozoal activity and DNA binding of N-substituted N-phenylbenzamide and 1,3-diphenylurea bisguanidines

Keywords: نخود; Trypanosoma brucei; Plasmodium falciparum; Parasite chemotherapy; Guanidine; Minor groove binder; surface plasmon resonance (SPR) biosensor; BBB; blood-brain barrier; CNS; central nervous system; DIPEA; diisopropylethylamine; EDAC; 1-ethyl-3-(3-dimethyl

دانلود رایگان متن کامل مقاله ISI 66 صفحه سال انتشار : 2014 سفارش ترجمه

Backbone cyclic helix mimetic of chemokine (C-C motif) receptor 2: A rational approach for inhibiting dimerization of G protein-coupled receptors

Keywords: نخود; ACN; acetonitrile allocallyloxycarbonyl; BBB; blood brain barrier; Boc; t-butyloxycarbonyl; BTC; bis(trichloromethyl)carbonate; CCR2; chemokine (C-C motif) receptor 2; CCR5; chemokine (C-C motif) receptor 5; CNS; central nervous system; DIPEA; diisopr

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2013 سفارش ترجمه

Discovery of pyrazole as C-terminus of selective BACE1 inhibitors

Keywords: نخود; Alzheimer's disease; BACE1; C-terminus; Click chemistry; In situ screening assay; Pyrazole; EDCl; N-(3-dimethylaminopropyl)-N′-ethylcarbodiimide hydrochloride; HOBt; N-hydroxybenzotriazole; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; E

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2013 سفارش ترجمه

Design, synthesis, and biological activities of novel hexahydropyrazino[1,2-a]indole derivatives as potent inhibitors of apoptosis (IAP) proteins antagonists with improved membrane permeability across MDR1 expressing cells

Keywords: نخود; HATU; O-(7-azabenzotriazol-1-yl)-N,N,N′,N′-tetramethyluronium hexafluorophosphate; DIPEA; N-ethyldiisopropylamine; Ac; acetyl; CDCl3; deuteratedchloroform; DMF; N,N-dimethylformamide; DMSO; dimethyl sulfoxide; DMT-MM; 4-(4,6-dimethoxy-1,3,5-triazin-2-

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2013 سفارش ترجمه

Linear and cyclic glycopeptide as HIV protease inhibitors

Keywords: نخود; HIV-1 protease; Linear and cyclic glycopeptides; Solid and solution peptide synthesis; Molecular docking; AIDS; acquired immunodeficiency syndrome; CTC; 2-chlorotrityl chloride; DCM; dichloromethane; DIPEA; N,N-diisopropyl ethylamine; DMF; N,N-dimethylfor

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2013 سفارش ترجمه

Novel TIPP (H-Tyr-Tic-Phe-Phe-OH) analogues displaying a wide range of efficacies at the δ opioid receptor. Discovery of two highly potent and selective δ opioid agonists

Keywords: نخود; Boc; tert-butyloxycarbonyl; Cl-HOBt; 6-chloro-1-hydroxybenzotriazole; DAMGO; H-Tyr-d-Ala-Gly-Phe(NMe)-Gly-ol; DIC; 1,3-diisopropylcarbodiimide; DIPEA; N,N-diisopropylethylamine; DPDPE; H-Tyr-c[d-Pen-Gly-Phe-D-Pen]OH; DSLET; H-Tyr-d-Ser-Gly-Phe-Leu-Thr-OH;

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2012 سفارش ترجمه

Activity based subcellular resolution imaging of lipases

Keywords: نخود; ABP; activity based probe; ACN; acetonitrile; ATGL; adipose triglyceride lipase; CuAAC; copper (I) catalyzed azide alkyne [3+2] cycloaddition; DIPEA; diisopropylethylamine; FA; formic acid; HSL; hormone sensitive lipase; MGL; monoglyceride lipase; TGH1; t

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2012 سفارش ترجمه

Synthesis of [11C]uric acid, using [11C]phosgene, as a possible biomarker in PET imaging for diagnosis of gout

Keywords: نخود; PET; positron emission tomography; DMPU; N,N′-dimethylpropyleneurea; DIPEA; N,N-diisopropylethylamine; [11C]uric acid; Positron emission tomography (PET); [11C]phosgene; Hyperuricemia; Gout;

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2012 سفارش ترجمه

Handling a tricycle: Orthogonal versus random oxidation of the tricyclic inhibitor cystine knotted peptide gurmarin

Keywords: نخود; 4-PDS; 4,4-dithiodipyridine; Acm; acetamidomethyl; DIPEA; diisopropylethylamine; DMSO; dimethylsulfoxide; EDT; ethanedithiol; ICK; inhibitor cystine knot; NMP; N-methylpyrrolidone; Pyr; pyroglutamic acid; StBu; tert-Butylthio; TFA; trifluoroacetic acid; T

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2012 سفارش ترجمه

Design and synthesis of novel amphiphilic Janus dendrimers for bone-targeted drug delivery

Keywords: نخود; Janus dendrimer; Amphiphilic; Bone-targeting; Drug delivery; DIPEA; N,N-diisopropylethylamine; DMAP; dimethylamino pyridine; EDCI·HCl; 1-(3-dimethylaminopropyl)-3-ethylcarbodiimide hydrochloride; IBCF; isobutyl chloroformate; HBTU; o-benzotriazol-1-yl-N,

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2012 سفارش ترجمه

Discovery of novel A3 adenosine receptor ligands based on chromone scaffold

Keywords: نخود; [3H]CCPA; [3H](2R,3R,4S,5R)-2-[2-chloro-6-(cyclopentylamino)purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol; [3H]HEMADO; [3H] 2-(1-Hexynyl)-N6-methyladenosine; [3H]NECA; [3H]adenosine-5′-(N-ethylcarboxamide); AR; Adenosine receptor; Arg; arginine; Asn; as

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2012 سفارش ترجمه

Orthogonal ligation to spherical polymeric microparticles: Modular approaches for surface tailoring

Keywords: نخود; AIBN; azo-bis-isobutyronitrile; ATR; attenuated total reflectance; ATRP; atom transfer radical polymerization; Con A; Concanavalin A; CRP; controlled radical polymerization; CuAAC; copper-catalyzed azide alkyne cycloaddition; DIPEA; diisopropylethylamine;

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2012 سفارش ترجمه

Cellular uptake and biophysical properties of galactose and/or tryptophan containing cell-penetrating peptides

Keywords: نخود; ATR Spectroscopy; Attenuated Total Reflection Spectroscopy; CPP; cell-penetrating peptide; CHO; Chinese hamster ovary; DIPEA; diisopropylethylamine; DMF; dimethylformamide; DMPC; dimyristoylphosphatidylcholine; DMPG; dimyristoylphosphatidylglycine; DSC; d

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2012 سفارش ترجمه

Synthesis, anticonvulsant activity, and neuropathic pain-attenuating activity of N-benzyl 2-amino-2-(hetero)aromatic acetamides

Keywords: نخود; AED; antiepileptic drug; ASP; Anticonvulsant Screening Program; B:P; brain-to-plasma; Cbz; carboxybenzyl; DBU; 1,8-diazabicycloundec-7-ene; DIPEA; N,N-diisopropylethylamine; DMTMM; 4-(4,6-dimethoxy-1,3,5-triazin-2-yl)-4-methylmorpholinium chloride; ED50;

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2012 سفارش ترجمه

Weight loss effects of quaternary salts of 5-amino-1-(chloromethyl)-1,2-dihydro-3H-benz[e]indoles; structure-activity relationships

Keywords: نخود; AIBN; 2,2′-azobis[isobutyronitrile]; CBI; seco-1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indol-4-one; CSA; camphorsulfonic acid; DIPEA; diisopropylethylamine; DMA; dimethylacetamide; DMAP; 4-dimethylaminopyridine; EDCI·HCl; N-ethyl-N′-(3-dimethylaminopr

دانلود رایگان متن کامل مقاله ISI 16 صفحه سال انتشار : 2012 سفارش ترجمه

The discovery and synthesis of JNJ 31020028, a small molecule antagonist of the Neuropeptide Y Y2 receptor

Keywords: نخود; DCM; dichloromethane; HOBt; 1-hydroxy-benzotriazole; EDCI; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide; BOC; butoxycarbonyl; MeOH; methanol; K2CO3; potassium carbonate; Na2CO3; sodium carbonate; DMF; dimethylformamide; Et3N; triethylamine; Et2O; ether;

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2011 سفارش ترجمه

Biological and conformational evaluation of angiotensin II lactam bridge containing analogues

Keywords: نخود; AAA; Amino acid analysis; ACN; Acetonitrile; AII; angiotensin II; BOP; (Benzotriazol-1-yl-oxy)tris(dimethylamino)phosphonium hexafluorophosphate; BSA; bovine serum albumin; CD; Circular Dichroism; CE; Capillary Electrophoresis; CHO; Chinese hamster ovary;

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2011 سفارش ترجمه

N-alkylated cyclen cobalt(III) complexes of 1-(chloromethyl)-3-(5,6,7-trimethoxyindol-2-ylcarbonyl)-2,3-dihydro-1H-pyrrolo[3,2-f]quinolin-5-ol DNA alkylating agent as hypoxia-activated prodrugs

Keywords: نخود; Cancer therapy; Hypoxia; Prodrug; Cobalt(III) complex; Pyrrolo[3,2-f]quinolin-5-ol; Cyclen; Cytotoxicity; 8-QOH; 8-hydroxyquinoline; Bn; benzyl; CBI; seco-1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indol-4-one; Cbz; benzyloxycarbonyl; cyclen; 1,4,7,10-tetraaz

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2011 سفارش ترجمه

Bi- and trivalent glycopeptide mannopyranosides as inhibitors of type 1 fimbriae-mediated bacterial adhesion: variation of valency, aglycon and scaffolding

Keywords: نخود; Fmoc; fluorenylmethoxycarbonyl; Gly; l-glycine; Ser; l-serine; Lys; l-lysine; DPr; l-diaminopropionic acid; Ala; l-alanine; HATU; O-(7-azabenzotriazol-1-yl)-N,N,N',N'-tetramethyluronium hexafluorophosphate; DIPEA; N-ethyl-N-diisopropylamine; GFP; gree

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2011 سفارش ترجمه

Novel analogues of the therapeutic complement inhibitor compstatin with significantly improved affinity and potency

Keywords: نخود; Ac; acetyl group; DCM; dichloromethane; DIC; 1,3-diisopropylcarbodiimide; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; ESI; electrospray ionization; Fmoc; 9-fluorenylmethoxycarbonyl; HOAt; 1-hydroxy-7-aza-benzotriazole; ITC; isothermal ti

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2011 سفارش ترجمه

Substrate specificity of kallikrein-related peptidase 13 activated by salts or glycosaminoglycans and a search for natural substrate candidates

Keywords: نخود; Kinin; Protease; Histatins; Kosmotropic salts; Myelin basic protein; Q-EDDP; (glutamyl-N-[ethylenediamine] 2,4-dinitrophenyl); Abz; ortho-aminobenzoic acid; HOBt; N hydroxybenzotriazole; TBTU; 2-(1H-benzotriazole-1-yl)-1,1,3,3-tetramethylaminium tetrafluo

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2011 سفارش ترجمه

The effect of sulfonate leaving groups on the hypoxia-selective toxicity of nitro analogs of the duocarmycins

Keywords: نخود; CBI; seco-1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indol-4-one; DIPEA; diisopropylethylamine; DMA; dimethylacetamide; EDCI·HCl; N-ethyl-N′-(3-dimethylaminopropyl)carbodiimide hydrochloride; HCR; hypoxic cytotoxicity ratio; TMI; 5,6,7-trimethoxyindole; Cy

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2011 سفارش ترجمه

Oxidized and nitrated oleic acid in biological systems: Analysis by GC-MS/MS and LC-MS/MS, and biological significance

Keywords: نخود; BSTFA; N,O-bis(trimethylsilyl)trifluoroacetamide; CID; collision-induced dissociation; DIPEA; N,N-diisopropylethylamine; ECNICI; electron capture negative-ion chemical ionization; EI; electron ionization; cis-EpOA; cis-9,10-epoxyoctadecanoic acid; ESI; el

دانلود رایگان متن کامل مقاله ISI 12 صفحه سال انتشار : 2011 سفارش ترجمه

Separation of fluorinated amino acids and oligopeptides from their non-fluorinated counterparts using high-performance liquid chromatography

Keywords: نخود; Cys; cysteine; DCM; dichloromethane; DIC; N,N′-diisopropylcarbodiimide; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; EtOH; ethanol; F%wt; fluorine weight percentage in an analyte or a solvent; Fmoc; fluorenylmethoxycarbonyl; HFIP; hexaf

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2010 سفارش ترجمه

Rational conversion of noncontinuous active region in proteins into a small orally bioavailable macrocyclic drug-like molecule: The HIV-1 CD4:gp120 paradigm

Keywords: نخود; AcOH; acetic acid; Alloc; allyloxycarbonyl; Boc; t-butoxycarbonyl; BTC; bis(trichloromethyl)carbonate; DBU; 1,8-diazabicyclo[5.4.0]undec-7-ene; DCM; methylene chloride; DIC; N,N′-diisopropylcarbodiimide; DIPEA; diisopropylethylamine; DMAP; dimethylamino

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2010 سفارش ترجمه

Solid-phase peptide head-to-side chain cyclodimerization: Discovery of C2-symmetric cyclic lactam hybrid α-melanocyte-stimulating hormone (MSH)/agouti-signaling protein (ASIP) analogues with potent activities at the human melanocortin receptors

Keywords: نخود; All; allyl; AgRP; Agouti-related protein; ASIP; agouti-signaling protein; Boc; tert-butyloxycarbonyl; Fmoc; fluorenylmethoxycarbonyl; CH3CN; acetonitrile; Cl-HOBt; 1-hydroxy-6-chlorobenzotriazole; DCM; dichloromethane; DIPEA; diisopropylethylamine; DMF; N

دانلود رایگان متن کامل مقاله ISI 12 صفحه سال انتشار : 2010 سفارش ترجمه

Tetrahedron report number 922Homocoupling reactions of alkynes, alkenes and alkyl compounds

Keywords: نخود; DABCO; 1,4-diazabicyclo[2.2.2]octane; DBA; dibenzylidenoacetone; DBU; 1,8-diazabicyclo[5.4.0]undec-7-ene; DIPEA; diisopropylethylamine; DMAP; N,N-4-dimethylaminopyridine; DMF; N,N-dimethylformamide; DMI; 1,3-dimethyl-2-Imidazolidinone; DMSO; dimethylsulph

دانلود رایگان متن کامل مقاله ISI 48 صفحه سال انتشار : 2010 سفارش ترجمه

A novel non-phosphorylated potential antitumoral peptide inhibits STAT3 biological activity

Keywords: نخود; STAT3; Peptide inhibitor; Immunofluorescence; Cellular effects; Ahx; 6-amino hexanoic acid; Antp; Antennapedia sequence; BOP; (benzotriazol-1-yloxy)tris(dimethylamino)phosphonium hexafluorophosphate; DIPEA; diisopropylethylamine; GPK; GMP-protein dependan

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2009 سفارش ترجمه

The Barton ester free-radical reaction: a brief review of applications

Keywords: نخود; Radical reaction; Barton ester; Thiohydroxamate ester; Decarboxylation; Ac; acetyl; AIBN; 2,2′-azobisisobutyronitrile; DCC; dicyclohexylcarbodiimide; DIPEA; diisopropylethylamine; DMAP; N,N-4-dimethylaminopyridine; DME; ethylene glycol dimethyl ether; D

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2009 سفارش ترجمه

Synthesis of diamino-furostan sapogenins and their use as scaffolds for positioning peptides in a preorganized form

Keywords: نخود; Steroids; Steroidal sapogenins; Furostanes; Peptides; Cyclopeptides; Boc; tert-butoxycarbonyl; EDC; 1-(3-dimethylaminopropyl)-3-ethylcarbodiimide; DCC; N,N′-dicyclohexylcarbodiimide; DIC; N,N′-diisopropylcarbodiimide; DIPEA; N,N-di-iso-propyl-N-ethyla

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2008 سفارش ترجمه

Synthesis, SAR and in vitro evaluation of new cyclic Arg-Gly-Asp pseudopentapeptides containing a s-cis peptide bond as integrin αvβ3 and αvβ5 ligands

Keywords: نخود; All; allyl; DIC; N,N′-diisopropylcarbodiimide; DIPEA; N,N-diisopropylethylamine; DMAP; 4-dimethylaminopyridine; DMF; N,N-dimethylformamide; Fmoc; 9H-fluoren-9-yl-methyloxycarbonyl; HOBt; 1-hydroxybenzotriazole; NMM; N-methylmorpholine; Pbf; 2,2,4,6,7-pe

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2008 سفارش ترجمه

Halovinyl aldehydes: useful tools in organic synthesis

Keywords: نخود; Ac; acetyl; Ar; aryl; Bn; benzyl; Bu; butyl; DCM; dichloromethane; DDQ; dichloro dicyano quinone; TMEDA; tetramethylethylenediamine; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; DMSO; dimethylsulfoxide; ee; enantiomeric excess; Et; ethyl;

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2008 سفارش ترجمه

Synthesis and evaluation of chloromethyl sulfoxides as a new class of selective irreversible cysteine protease inhibitors

Keywords: نخود; ESI-MS; electrospray ionization mass spectrometry; Boc; tert-butyloxycarbonyl; BOP; (1H-benzotriazol-1-yloxy)tris(dimethylamino)phosphonium hexafluorophosphate; DBU; 1,8-diazabicyclo[5.4.0]undec-7-ene; DTT, dithiothreitol; DiPEA; N,N-diisopropylethylamine

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2007 سفارش ترجمه

PS-IIDQ: a supported coupling reagent for efficient and general amide bond formation

Keywords: نخود; Coupling reagent; Polymer-supported reagent; Immobilized reagent; IIDQ; Parallel synthesis; Amide bond formation; Amidation; Amide; BOP; benzotriazolyl-N-oxytrisdimethylaminophosphonium hexafluorophosphate; BOP-Cl; N,N′-bis(2-oxo-3-oxazolidinyl)-phosphi

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2007 سفارش ترجمه

Application of hydrolytic kinetic resolution (HKR) in the synthesis of bioactive compounds

Keywords: نخود; Hydrolytic kinetic resolution; Terminal epoxides; Bis-epoxides; meso-Epoxides; Natural products; Synthesis; Biological activity; Ac; acetyl; AD; asymmetric dihydroxylation; AE; asymmetric epoxidation; Bn; benzyl; NBS; N-bromosuccinimide; Boc; t-butoxycarb

دانلود رایگان متن کامل مقاله ISI 41 صفحه سال انتشار : 2007 سفارش ترجمه