
Synthesis and biological evaluation of bivalent cannabinoid receptor ligands based on hCB2R selective benzimidazoles reveal unexpected intrinsic properties
Keywords: Ag, measuring in agonism mode; Ant, measuring in antagonism mode; atm., atmosphere; CDI, 1,1′-carbonyldiimidazole; DMF, N,N-dimethylformamide; DMSO, dimethyl sulfoxide; EC50, half maximal effective concentration (potency); ECS, endocannabinoid system; Ema