Keywords: مهار کننده های آنزیم; Urease; Nickel delivery; Drug screening; Protein-protein interactions; Enzyme inhibitors; Helicobacter pylori;
مقالات ISI مهار کننده های آنزیم (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: مهار کننده های آنزیم; Antioxidant; Enzyme inhibitors; Ethnic wheat; North Dakota Common Emmer; Phenolics; Type 2 diabetes;
Keywords: مهار کننده های آنزیم; Teas and herbal infusions; Melatonin; Phenolic compounds; Enzyme inhibitors; Antioxidant capacity;
Keywords: مهار کننده های آنزیم; Enzyme inhibitors; Antibiotic; Biotin protein ligase; Azide-alkyne cycloaddition; Staphylococcus aureus;
Keywords: مهار کننده های آنزیم; Morita-Baylis-Hillman bromides; Palladium-catalyzed coupling; Phosphonic acids; Enzyme inhibitors; Structure-activity relationship;
Keywords: مهار کننده های آنزیم; Sphingolipid; Lipopolysaccharide; Lung injury; Ceramide; Inflammation; Enzyme inhibitors; ARDS; Acute respiratory distress syndrome; LPS; lipopolyssacharide; ASM; acid sphingomyelinase; NSM; neutral sphingomyelinase; SPT; serine palmitoyl transferase; DS;
Keywords: مهار کننده های آنزیم; Human carbonic anhydrase; Enzyme inhibitors; Sulfonamides
Keywords: مهار کننده های آنزیم; Nanoparticles; Metal nanoparticles; Antibacterial activity; Enzyme inhibitors;
Keywords: مهار کننده های آنزیم; Lignocellulose; Food industry waste; Pre-treatment; Enzyme inhibitors; Renewable resources;
Keywords: مهار کننده های آنزیم; Pretreatment; Saccharification; Enzyme inhibitors; Lignin; Thermotolerant yeast
Keywords: مهار کننده های آنزیم; Antimicrobials; Antioxidants; Bioautography; Drug discovery; Enzyme inhibitors; Thin-layer chromatography;
Keywords: مهار کننده های آنزیم; Thiazole; Antimicrobials; Anti-cancer; Antioxidants; Anti-inflammatory; Anticonvulsants; Enzyme inhibitors; Lead compounds;
Keywords: مهار کننده های آنزیم; Drug design; Enzyme inhibitors; Proteases; Reversible covalent inhibitors; Virtual screening
Keywords: مهار کننده های آنزیم; Serine hydrolase inhibitors; Enzyme inhibitors; Screening library; Fatty acid amide hydrolase;
Keywords: مهار کننده های آنزیم; Dual specificity phosphatases; Virtual screening methods; Phosphatases of regenerating liver; Enzyme inhibitors; Thienopyridone; 2-Cyano-2-ene-esters; DIFMUP; 6,8-difluoro-4-methylumbelliferyl phosphate; DSP; dual specificity phosphatase; MTT; 3-(4,5-dime
Keywords: مهار کننده های آنزیم; Aldose reductase; Enzyme inhibitors; Anti-inflammatory agents; Molecular modelling; 5-Arylidene-4-thiazolidinone derivatives; 5-(carbamoylmethoxy)benzylidene-2-oxo/thioxo-4-thiazolidinone derivatives; AGEs; advanced glycation-end products; AR; aldose redu
Keywords: مهار کننده های آنزیم; Algal drugs; Enzyme inhibitors; Dementia; Diabetes; Drug likeness; Inflammation; Structure activity relationship
Keywords: مهار کننده های آنزیم; Fatty acid amide hydrolase (FAAH); Enzyme inhibitors; Solubility; Cannabinoid system; Drug disposition properties;
Keywords: مهار کننده های آنزیم; Drug discovery; Enzyme inhibitors; Dynamic combinatorial chemistry; Ligand separation; Imine formation
Keywords: مهار کننده های آنزیم; enzyme inhibitors; ethnic vegetables; flavonoids; polyphenols
Thiazolo[3,2-a]pyrimidin-5-one derivatives as a novel class of 11β-hydroxysteroid dehydrogenase inhibitors
Keywords: مهار کننده های آنزیم; Thiazolo[3,2-a]pyrimidine derivatives; 11β-Hydroxysteroid dehydrogenase; Enzyme inhibitors; Molecular docking;
A novel derivatives of thiazol-4(5H)-one and their activity in the inhibition of 11β-hydroxysteroid dehydrogenase type 1
Keywords: مهار کننده های آنزیم; Thiazolone derivatives; 11β-Hydroxysteroid dehydrogenase; Enzyme inhibitors; Synthesis; Molecular docking;
HPLC-MS/MS-based metabolic profiling and pharmacological properties of extracts and infusion obtained from Amelanchier parviflora var. dentata
Keywords: مهار کننده های آنزیم; Amelanchier parviflora; Antioxidants; Chemical fingerprints; Enzyme inhibitors; Phenolics; Anthocyanins;
The effects of modified atmosphere packaging and enzyme inhibitors on protein oxidation of tilapia muscle during iced storage
Keywords: مهار کننده های آنزیم; Tilapia; Modified atmosphere packaging; Enzyme inhibitors; Protein oxidation;
Structure-activity relationships of rationally designed AMACR 1A inhibitors
Keywords: مهار کننده های آنزیم; α-Methylacyl-CoA racemase (AMACR, P504S); Drug lipophilicity; Enzyme inhibitors; Rational drug design; Structure-activity relationships; AMACR; α-methylacyl-CoA racemase; CDI; carbonyldiimidazole; DAST; (Diethylamino)sulfur trifluoride; DCC; Dicyclohexy
Discovery of 5-((5-chloro-2-methoxyphenyl)sulfonamido)nicotinamide (SBI-425), a potent and orally bioavailable tissue-nonspecific alkaline phosphatase (TNAP) inhibitor
Keywords: مهار کننده های آنزیم; Enzyme inhibitors; Inhibitors; TNAP; Tissue nonspecific alkaline phosphatase; Calcification;
2-Benzylpiperazine: A new scaffold for potent human carbonic anhydrase inhibitors. Synthesis, enzyme inhibition, enantioselectivity, computational and crystallographic studies and in vivo activity for a new class of intraocular pressure lowering agents
Keywords: مهار کننده های آنزیم; Carbonic anhydrase; Enzyme inhibitors; Piperazine; Enantioselectivity; Glaucoma;
In vitro and in silico evaluation of Centaurea saligna (K.Koch) Wagenitz-An endemic folk medicinal plant
Keywords: مهار کننده های آنزیم; Centaurea saligna; Folk medicine; Enzyme inhibitors; Bioactive compounds; Antioxidants;
Multidirectional investigations on different parts of Allium scorodoprasum L. subsp. rotundum (L.) Stearn: Phenolic components, in vitro biological, and in silico propensities
Keywords: مهار کننده های آنزیم; Allium; Phenolics; Antioxidants; Enzyme inhibitors; Natural agents;
Novel spiroindoline HDAC inhibitors: Synthesis, molecular modelling and biological studies
Keywords: مهار کننده های آنزیم; Antitumor agents; Bioinformatics; Drug design; Enzyme inhibitors; Epigenetics; HDAC;
Comparative in vitro studies of the biological potential and chemical composition of stems, leaves and berries Aronia melanocarpa's extracts obtained by subcritical water extraction
Keywords: مهار کننده های آنزیم; Subcritical water extraction; Aronia; HPLC; Antioxidants; Enzyme inhibitors; Cytotoxicity; Antimicrobial activity;
Plant-derived mPGES-1 inhibitors or suppressors: A new emerging trend in the search for small molecules to combat inflammation
Keywords: مهار کننده های آنزیم; Anti-inflammatory; Anti-rheumatism; mPGES-1; Enzyme inhibitors; Plant-derived compounds;
Potential drug targets in the Mycobacterium tuberculosis cytochrome P450 system
Keywords: مهار کننده های آنزیم; Mycobacterium tuberculosis; Cytochrome P450; Cholesterol degradation; Azole drugs; Enzyme inhibitors;
Quinazoline-1-deoxynojirimycin hybrids as high active dual inhibitors of EGFR and α-glucosidase
Keywords: مهار کننده های آنزیم; Quinazoline; 1-Deoxynojirimycin; Hybrids; Epidermal growth factor receptor (EGFR); α-Glucosidase; Enzyme inhibitors;
Design and examination of potent pseudosubstrate-based oligonucleotide inhibitors against bacterial topoisomerase IV
Keywords: مهار کننده های آنزیم; Topoisomerase IV; Enzyme inhibitors; Oligonucleotides; Pseudosubstrates; Antibiotics;
Development and crystallographic evaluation of histone H3 peptide with N-terminal serine substitution as a potent inhibitor of lysine-specific demethylase 1
Keywords: مهار کننده های آنزیم; Crystal structure; Enzyme inhibitors; Epigenetics; Peptides; Protein structure;
Addition of thiols to the double bond of dipeptide C-terminal dehydroalanine as a source of new inhibitors of cathepsin C
Keywords: مهار کننده های آنزیم; Dehydropeptides; Thiol addition; Cathepsin C; Enzyme inhibitors;
ReviewEffect of extrusion on the anti-nutritional factors of food products: An overview
Keywords: مهار کننده های آنزیم; Extrusion; Anti-nutritional factors; Legumes; Cereals; Phytate; Tannins; Enzyme inhibitors;
Isoniazid inhibits human erythroid 5-aminolevulinate synthase: Molecular mechanism and tolerance study with four X-linked protoporphyria patients
Keywords: مهار کننده های آنزیم; ALA; 5-aminolevulinic acid; ALAS1; non-specific isoform of 5-aminolevulinate synthase; ALAS2; erythroid-specific isoform of 5-aminolevulinate synthase; mALAS2; erythroid-specific isoform of murine 5-aminolevulinate synthase; ÎmALAS2; erythroid-specific i
Design and optimization of aspartate N-acetyltransferase inhibitors for the potential treatment of Canavan disease
Keywords: مهار کننده های آنزیم; ANAT; aspartate N-acetyltransferase; CD; Canavan disease; DCM; dichloromethane; DTNB; dithionitrobenzoate; EDCl; 1-ethyl-3-(3-(dimethylamino)propyl)carbodiimide; HEPES; 4-(2-hydroxyethyl)piperazine-1-ethanesulfonic acid; IPTG; isopropyl-β-thiogalactoside
Synthesis and characterization of oxidovanadium complexes as enzyme inhibitors targeting dipeptidyl peptidase IV
Keywords: مهار کننده های آنزیم; DPP-IV; dipeptidyl peptidase IV; mg V·kgâ 1; mg Vanadium injected/weight of mice in kg; GLP-1; glucagon-like peptide-1; GIP; glucose-dependent insulinotropic peptide; BEOV; bis(ethylmaltolato)oxovanadium(IV); PTP1B; protein tyrosine phosphatase 1B; P
Phenolic antioxidant-linked anti-hyperglycemic properties of rye cultivars grown under conventional and organic production systems
Keywords: مهار کننده های آنزیم; Antioxidant; Anti-hyperglycemia; Enzyme inhibitors; Phenolic bioactives;
Novel organophosphorus scaffolds of urease inhibitors obtained by substitution of Morita-Baylis-Hillman adducts with phosphorus nucleophiles
Keywords: مهار کننده های آنزیم; Phosphonic and phosphinic acids; Substitution of allyl acetates; Enzyme inhibitors; Structure-activity relationship; Binding mode;
Discovery of 4-[(5-arylidene-4-oxothiazolidin-3-yl)methyl]benzoic acid derivatives active as novel potent allosteric inhibitors of protein tyrosine phosphatase 1B: In silico studies and in vitro evaluation as insulinomimetic and anti-inflammatory agents
Keywords: مهار کننده های آنزیم; Protein tyrosine phosphatases; Enzyme inhibitors; Insulinomimetic effects; Anti-inflammatory activity; Molecular docking; 5-Arylidene-4-thiazolidinone derivatives; COX; cyclooxygenase; DM; diabetes mellitus; EI; enzyme-inhibitor complex; ESI; enzyme-subst
Structural basis of the lack of endo-glucanase inhibitory activity of Lupinus albus γ-conglutin
Keywords: مهار کننده های آنزیم; Seed proteins; Enzyme inhibitors; Mutagenesis; Plant defenceDLS, dynamic light scattering; GH, glycosyl hydrolase; PTM, post-translational modification; s.i., sequence identity; γ-c, seed-extracted γ-conglutin; rγc, recombinant γ-conglutin; rγcMu, recombi
Mechanism-based candidate inhibitors of uridine diphosphate galactopyranose mutase (UGM) †
Keywords: مهار کننده های آنزیم; Enzyme inhibitors; Mycobacterium tuberculosis; Synthesis; Transition-state analogues; UDP-galactopyranose mutase; UGM
Identification of novel scaffolds for potential anti-Helicobacter pylori agents based on the crystal structure of H. pylori 3-deoxy-d-manno-octulosonate 8-phosphate synthase (HpKDO8PS)
Keywords: مهار کننده های آنزیم; Structure-based virtual screening; Docking simulation; Enzyme inhibitors; X-ray crystallography; NMR spectroscopyKDO8PS, 3-deoxy-d-manno-octulosonate-8-phosphate synthase; PEP, phosphoenolpyruvate; A5P, d-arabinose-5-phosphate; HpKDO8PS, KDO8PS from Helic
Radiolabeled enzyme inhibitors and binding agents targeting PSMA: Effective theranostic tools for imaging and therapy of prostate cancer
Keywords: مهار کننده های آنزیم; Enzyme inhibitors; Gallium-68; Lutetium-177; Prostate cancer; Prostate-specific membrane antigen; Targeted radionuclide therapy
Iminopyrimidinones: A novel pharmacophore for the development of orally active renin inhibitors
Keywords: مهار کننده های آنزیم; Renin inhibitors; BACE1; Hypertension; Structure-based drug design; Enzyme inhibitors
Inhibition of bacterial mevalonate diphosphate decarboxylase by eriochrome compounds
Keywords: مهار کننده های آنزیم; Mevalonate diphosphate decarboxylase; Mevalonate pathway; Isoprenoid biosynthesis; Enzyme inhibitors;