Keywords: فالسیپین-2; Phthalimides; Plasmodium falciparum; Piperazine; Docking; Falcipain-2
مقالات ISI فالسیپین-2 (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Docking, synthesis and antimalarial activity of novel 4-anilinoquinoline derivatives
Keywords: فالسیپین-2; Malaria; Plasmodium falciparum; Falcipain-2; Cysteine protease; 4-Anilinoquinoline triazine; β-Haematin;
Synthesis and structure–activity-relationship studies of thiazolidinediones as antiplasmodial inhibitors of the Plasmodium falciparum cysteine protease falcipain-2
Keywords: فالسیپین-2; Antiplasmodial agents; Thiazolidinone; Falcipain-2
Dietary flavonoids fisetin and myricetin: Dual inhibitors of Plasmodium falciparum falcipain-2 and plasmepsin II
Keywords: فالسیپین-2; Dietary flavonoids; Falcipain-2; Plasmepsin II; Dual inhibitor;
Falcipain-2 inhibition by suramin and suramin analogues
Keywords: فالسیپین-2; FP-2; falcipain-2; Suramin; 8,8â²-[carbonylbis[imino-3,1-phenylenecarbonylimino(4-methyl-3,1-phenylene)carbonylimino]]bis-1,3,5-naphthalenetrisulfonic acid; AMC; 7-amino-4-methyl coumarin; NF037; 8,8â²-[carbonylbis[imino-3,1-phenylenecarbonylimino-3,1-p
Design and synthesis of small molecular dual inhibitor of falcipain-2 and dihydrofolate reductase as antimalarial agent
Keywords: فالسیپین-2; Falcipain-2; Dihydrofolate reductase; Dual inhibitor; Antimalarial drug; SAR; Molecular docking;
High-level expression of Falcipain-2 in Escherichia coli by codon optimization and auto-induction
Keywords: فالسیپین-2; Falcipain-2; Plasmodium falciparum; Synthetic gene; Codon optimization; Auto-induction;
Design and synthesis of protein-protein interaction mimics as Plasmodium falciparum cysteine protease, falcipain-2 inhibitors
Keywords: فالسیپین-2; Malaria; Falcipain-2; Cystatin; Protein-protein interaction mimics; DCM; dichloromethane; DIPEA; diisopropylethylamine; DMF; N,N-dimethylformamide; DMSO; dimethyl sulfoxide; DTT; dithiothreitol; EDTA; ethylenediaminetetraacetic acid; Fmoc; fluorenylmeth
Synthesis and in vitro evaluation of gold(I) thiosemicarbazone complexes for antimalarial activity
Keywords: فالسیپین-2; Falcipain-2; Gold(I) complexes; P. falciparum; Thiosemicarbazones
Design and synthesis of novel 2-pyridone peptidomimetic falcipain 2/3 inhibitors
Keywords: فالسیپین-2; Malaria; Plasmodium falciparum; Cysteine protease; Falcipain-2; Peptidomimetic
Is dihydrolipoic acid among the reductive activators of parasite CysHis proteases?
Keywords: فالسیپین-2; DHLA; dihydrolipoic acid (reduced disulfhydryl); LA(S-S); lipoic acid disulfide (oxidized disulfide); LA; lipoic acid (unspecified redox state); Falcipain-2; Cathepsin B; Iron redox; Malaria parasites; Plasmodium falciparum; Trypanosoma cruzi;
Design, synthesis, and antimalarial activity of structural chimeras of thiosemicarbazone and ferroquine analogues
Keywords: فالسیپین-2; Malaria; Antimalarial agents; Chimeras; Ferroquine; Thiosemicarbazones; Falcipain-2; Bioorganometallics
Synthesis and biological evaluation of phenolic Mannich bases of benzaldehyde and (thio)semicarbazone derivatives against the cysteine protease falcipain-2 and a chloroquine resistant strain of Plasmodium falciparum
Keywords: فالسیپین-2; Malaria; Antimalarial agents; Mannich bases; Thiosemicarbazones; Cysteine proteases; Falcipain-2
Dipeptide vinyl sultams: Synthesis via the Wittig–Horner reaction and activity against papain, falcipain-2 and Plasmodium falciparum
Keywords: فالسیپین-2; Wittig–Horner reaction; Vinyl sultams; Papain; Antimalarials; Cysteine proteases; Falcipain-2; Plasmodium falciparum; Molecular modelling
Application of multicomponent reactions to antimalarial drug discovery. Part 2: New antiplasmodial and antitrypanosomal 4-aminoquinoline γ- and δ-lactams via a ‘catch and release’ protocol
Keywords: فالسیپین-2; Parallel synthesis; Multicomponent reaction; Ugi reaction; Polymer-supported reagents; 4-Aminoquinolines; Lactams; Antimalarial activity; Falcipain-2; Antitrypanosomal activity
A role of falcipain-2, principal cysteine proteases of Plasmodium falciparum in merozoite egression
Keywords: فالسیپین-2; Plasmodium falciparum; RNA interference; siRNA; Falcipain-2; Merozoite egress; Erythrocyte membrane rupture;
Biosynthesis, localization, and processing of falcipain cysteine proteases of Plasmodium falciparum
Keywords: فالسیپین-2; FP-1; Falcipain-1; FP-2; Falcipain-2; FP-3; Falcipain-3; Mu-Leu-Hph-VSPh; Morpholine urea-leucine-homophenylalanine-phenyl vinyl sulfone; BFA; Brefeldin-A; E-64; N-(trans-epoxysuccinyl)-l-leucine 4 guanidobutylaminde; E-64d; (2S,3S)-trans-epoxysuccinyl-l-
Design, synthesis and anti-plasmodial evaluation in vitro of new 4-aminoquinoline isatin derivatives
Keywords: فالسیپین-2; Isatins; Aminoquinolines; Plasmodium falciparum; Malaria; Anti-plasmodial activity; Falcipain-2; Mannich bases; Thiosemicarbazones