Keywords: فارنزیل ترانسفراز; DTT; dithiothreitol; Farnesyltransferase; Zinc protein; Ras protein; Farnesyl group;
مقالات ISI فارنزیل ترانسفراز (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: فارنزیل ترانسفراز; Farnesyltransferase; Phenothiazine; Cysteine; Methionine; Serine; Valine; CAAX inhibitor;
Keywords: فارنزیل ترانسفراز; FT; farnesyltransferase; SHR; spontaneously hypertensive rat; WKY; Wistar-Kyoto rat; FTI; farnesyltransferase inhibitor; ERK1/2; extracellular-signal regulated kinases 1/2; FPP; farnesyl pyrophosphate; MVA; mevalonate; TGF-β1; transforming growth factor-
Systemic or Forebrain Neuron-Specific Deficiency of Geranylgeranyltransferase-1 Impairs Synaptic Plasticity and Reduces Dendritic Spine Density
Keywords: فارنزیل ترانسفراز; ALS; amyotrophic lateral sclerosis; aCSF; artificial cerebrospinal fluid; AD; Alzheimer's disease; ANOVA; analysis of variance; AO; apical oblique; BS; basal shaft; CaMKII α; Ca2+/calmodulin-dependent protein kinase; CNS; central nervous system; Cre+;
Production of authentic geranylgeranylated KRAS4b using an engineered baculovirus system
Keywords: فارنزیل ترانسفراز; Prenylation; RAS; Geranylgeranylation; Protein production; Baculovirus; FNT; farnesyltransferase; GGTase; geranylgeranyltransferase; MBP; maltose-binding protein; FMe; farnesylated and methylated; GGMe; geranylgeranylated and methylated; GG; geranylgerany
Mammalian farnesyltransferase α subunit regulates vacuolar protein sorting-associated protein 4A (Vps4A) - dependent intracellular trafficking through recycling endosomes
Keywords: فارنزیل ترانسفراز; Farnesyltransferase; Oligomerization; Isoprenylation; Trafficking;
Antroquinonol blocks Ras and Rho signaling via the inhibition of protein isoprenyltransferase activity in cancer cells
Keywords: فارنزیل ترانسفراز; Antroquinonol; Ras; Farnesyltransferase; Prenylation; Autophagy
Peptidomimetic modification improves cell permeation of bivalent farnesyltransferase inhibitors
Keywords: فارنزیل ترانسفراز; Bivalent inhibitors; Farnesyltransferase; K-Ras4B; Protein-protein interaction; Whole cell activity;
αvβ3 Integrin and Fibroblast growth factor receptor 1 (FGFR1): Prognostic factors in a phase I-II clinical trial associating continuous administration of Tipifarnib with radiotherapy for patients with newly diagnosed glioblastoma
Keywords: فارنزیل ترانسفراز; Glioblastoma; Farnesyltransferase; FGFR1; ILK; Integrins; Radiotherapy; Phase II;
Role of protein farnesylation events in the ABA-mediated regulation of the Pinoresinol-Lariciresinol Reductase 1 (LuPLR1) gene expression and lignan biosynthesis in flax (Linum usitatissimum L.)
Keywords: فارنزیل ترانسفراز; Abscisic acid; Enhanced Response to Abscisic Acid 1 (ERA1); Farnesyltransferase; Lignan; Linum usitatissimum; Pinoresinol-lariciresinol reductase (PLR); (+)-Secoisolariciresinol;
Pharmacological modulation of geranylgeranyltransferase and farnesyltransferase attenuates opioid withdrawal in vivo and in vitro
Keywords: فارنزیل ترانسفراز; Morphine dependence; Withdrawal syndrome; GGTI-2133; FTI-276; Geranylgeranyl transferase; Farnesyltransferase
Inhibition of farnesyltransferase reduces angiogenesis by interrupting endothelial cell migration
Keywords: فارنزیل ترانسفراز; Farnesyltransferase; Angiogenesis; Migration; Endothelial cell; Microtubule;
Ras inhibition via direct Ras binding-is there a path forward?
Keywords: فارنزیل ترانسفراز; ATP; adenosine triphosphate; FTase; farnesyltransferase; FTmap; fourier transform correlation mapping; GAP; GTPase activating protein; GDP; guanosine diphosphate; GEF; guanine-nucleotide exchange factor; GST; glutathione s-transferase; GTP; guanosine trip
Chemical and biological explorations of the electrophilic reactivity of the bioactive marine natural product halenaquinone with biomimetic nucleophiles
Keywords: فارنزیل ترانسفراز; Marine natural product; Electrophilic; PLA2; Farnesyltransferase; Plasmodium falciparum
Thiazole- and imidazole-containing peptidomimetic inhibitors of protein farnesyltransferase
Keywords: فارنزیل ترانسفراز; Farnesyltransferase; Peptidomimetic inhibitors; Antiproliferative agents; Antitumors; Prenylation inihibitors;
Design, synthesis, and characterization of piperazinedione-based dual protein inhibitors for both farnesyltransferase and geranylgeranyltransferase-I
Keywords: فارنزیل ترانسفراز; Piperazinedione; Farnesyltransferase; Geranylgeranyltransferase; Cancer; Dual protein inhibitor;
Computer-aided drug design and ADMET predictions for identification and evaluation of novel potential farnesyltransferase inhibitors in cancer therapy
Keywords: فارنزیل ترانسفراز; Farnesyltransferase; Cancer; Drug design; Virtual screening; ADMET predictions
A versatile photoactivatable probe designed to label the diphosphate binding site of farnesyl diphosphate utilizing enzymes
Keywords: فارنزیل ترانسفراز; Benzophenone; Farnesyltransferase; Farnesyl diphosphate synthase; Sesquiterpene cyclase; Photoaffinity labeling
High glucose induced endothelial cell growth inhibition is associated with an increase in TGFβ1 secretion and inhibition of Ras prenylation via suppression of the mevalonate pathway
Keywords: فارنزیل ترانسفراز; Ras; Prenylation; TGFβ1; High glucose; Farnesyltransferase;
Peptidomimetic inhibitors of farnesyltransferase with high in vitro activity and significant cellular potency
Keywords: فارنزیل ترانسفراز; Farnesyltransferase; Peptidomimetic inhibitors; Antiproliferative agents; Antitumors
Resistance mutations at the lipid substrate binding site of Plasmodium falciparum protein farnesyltransferase
Keywords: فارنزیل ترانسفراز; Plasmodium; Falciparum; Farnesyltransferase; PFT; Drug resistance; Malaria;
Pharmacophore mapping of diverse classes of farnesyltransferase inhibitors
Keywords: فارنزیل ترانسفراز; Cytotoxic agents; Farnesyltransferase; Pharmacophore model; Inhibitors; QSAR
Farnesyltransferase pharmacophore model derived from diverse classes of inhibitors
Keywords: فارنزیل ترانسفراز; Farnesyltransferase; Inhibitor; Anticancer; Pharmacophore model; QSAR
Design, synthesis and biological evaluation of substituted dioxodibenzothiazepines and dibenzocycloheptanes as farnesyltransferase inhibitors
Keywords: فارنزیل ترانسفراز; Farnesyltransferase; Cytotoxicity; Cancer; Dioxodibenzothiazepine; Dibenzocycloheptane
Modulation of host metabolism as a target of new antivirals
Keywords: فارنزیل ترانسفراز; HCV; hepatitis C virus; CH; chronic hepatitis; HCC; hepatocellular carcinoma; IFN; interferon; SVR; sustained virological response; PEG-IFN; pegylated-IFN; GBV-B; GB virus B; uPA-SCID; urokinase plasminogen activator-severe combined immunodeficiency; NS;
Guiding farnesyltransferase inhibitors from an ECLiPS® library to the catalytic zinc
Keywords: فارنزیل ترانسفراز; Anti-cancer; Catalytic zinc; Farnesyltransferase; Rational drug design; Solution-phase synthesis; X-ray crystallography;
Farnesyltransferase inhibitors
Keywords: فارنزیل ترانسفراز; Farnesyltransferase; Prenylation; Lonafarnib; Tipifarnib; Ras; Rho; G-proteins; HDJ-2
Solid-phase synthesis and pharmacological evaluation of a library of peptidomimetics as potential farnesyltransferase inhibitors: an approach to new lead compounds
Keywords: فارنزیل ترانسفراز; Farnesyltransferase; Inhibitors; Peptidomimetics; Solid phase synthesis;
Modeling of farnesyltransferase inhibition by some thiol and non-thiol peptidomimetic inhibitors using genetic neural networks and RDF approaches
Keywords: فارنزیل ترانسفراز; Farnesyltransferase; Neural networks; Genetic algorithm; Enzyme inhibition; QSAR;
A multinomial Phase II study of lonafarnib (SCH 66336) in patients with refractory urothelial cancer
Keywords: فارنزیل ترانسفراز; Bladder neoplasms; Drug therapy; Farnesyltransferase; Lonafarnib;
Dominant negative FTase (DNFTα) inhibits ERK5, MEF2C and CREB activation in adipogenesis
Keywords: فارنزیل ترانسفراز; Farnesyltransferase; ERK5; CREB; Insulin; Adipogenesis; Differentiation;
Design, synthesis, and evaluation of potent and selective benzoyleneurea-based inhibitors of protein geranylgeranyltransferase-I
Keywords: فارنزیل ترانسفراز; Geranylgeranyltransferase-I; Peptidomimetics; Farnesyltransferase; Antitumor agents;
Molecular targets for altering radiosensitivity: Lessons from Ras as a pre-clinical and clinical model
Keywords: فارنزیل ترانسفراز; PTI; prenyltransferase inhibitors; FTase; farnesyltransferase; GGTase; Geranylgeranyl transferase; FTI; FTase inhibitor; GGTI; GGTase inhibitor; MAPK; mitogen activated protein kinase; PI3K; phosphatidylinositol 3â²-kinase; RTK; receptor tyrosine kinase;