Keywords: Glycopeptide; Isostere; Peptidomimetic; Deacetylation; Carbohydrate; Chemical biology
مقالات ISI (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: Benzocaine; Isostere; Methemoglobin; Methemoglobinemia; Rodenticide; Rat toxicant;
Keywords: Isostere; Purine; Triazine; Enzyme inhibitor; Anticancer; Antiviral
Pyrrolo[2,1-f][1,2,4]triazines: From C-nucleosides to kinases and back again, the remarkable journey of a versatile nitrogen heterocycle
Keywords: Kinase inhibitor; C-nucleoside; Pyrrolotriazine; Isostere; CNS;
Discovery of diazepane amide DORAs and 2-SORAs enabled by exploration of isosteric quinazoline replacements
Keywords: Orexin; Antagonists; Sleep; Isostere; Quinazoline;
Synthesis and PGE2 production inhibition of s-triazine derivatives as a novel scaffold in RAW 264.7 macrophage cells
Keywords: Inflammation; Prostaglandin E2; Cyanuric chloride; s-Triazine; Isostere; Docking study;
Discovery of acylurea isosteres of 2-acylaminothiadiazole in the azaxanthene series of glucocorticoid receptor agonists
Keywords: Acylurea; Imide; Isostere; Glucocorticoid receptor; Non-steroidal glucocorticoid receptor agonists;
Investigations of amide bond variation and biaryl modification in analogues of α7 nAChR agonist SEN12333
Keywords: α7 nicotinic receptors; Acetylcholine receptor; AChR; CNS; Structure–activity relationships; Tetrazole; Isostere
Synthesis and HDAC inhibitory activity of isosteric thiazoline-oxazole largazole analogs
Keywords: Largazole; HDAC; Oxazole; Isostere; Conformation;
Cis-Amide isosteric replacement in thienobenzoxepin inhibitors of PI3-kinase
Keywords: PI3-kinase; Isostere; Structure-based design; Property-guided design
Synthesis of novel histamine H4 receptor antagonists
Keywords: Histamine; Azaindole; Bicyclic; Amidine; Isostere;
Discovery of an orally-bioavailable CC Chemokine Receptor 2 antagonist derived from an acyclic diaminoalcohol backbone
Keywords: Chemokine; GPCR; CCR2; Isostere;
Synthesis and arylation of unprotected sulfonimidamides
Keywords: Sulfonimidamides; Arylation; Isostere; C-N coupling; Pd catalysis;
Identification of a sirtuin 3 inhibitor that displays selectivity over sirtuin 1 and 2
Keywords: Sirtuins; Histone deacetylase; Isostere; Rigid analogues; N-Unsubstituted-1,2,3-triazolyl pyridine
3-O-Arylmethylgalangin, a novel isostere for anti-HCV 1,3-diketoacids (DKAs)
Keywords: 3-O-Arylmethylgalangin; 1,3-Diketoacid; Isostere; Hepatitis C Virus (HCV)
Novel methylene-linked heterocyclic EP1 receptor antagonists
Keywords: EP1 antagonist; Pyrazole; Isostere; Heterocycle
Synthesis of leucine-enkephalin analogs containing α-amino squaric acid
Keywords: Squaric acid; Isostere; Enkephalin; Peptide; Amino acid;
Synthesis and evaluation of isosteres of N-methyl indolo[3,2-b]-quinoline (cryptolepine) as new antiinfective agents
Keywords: Antiinfective; Antifungal; Antibacterial; Antimalarial; Antileishmanial; Cryptolepine analog; Indoloquinoline; Indenoquinoline; Benzofuroquinoline; Benzothienoquinoline; Isostere; Fungal inhibition; Fungistatic agents
BACE-1 inhibition by a series of ψ[CH2NH] reduced amide isosteres
Keywords: β-Secretase; Reduced amide; Isostere
Discovery of novel biaryl heterocyclic EP1 receptor antagonists
Keywords: EP1 antagonist; Pain; Heterocycles; Cyclopentene; Isostere
Structure–activity relationships of 1,5-biaryl pyrroles as EP1 receptor antagonists
Keywords: EP1 antagonist; Pyrrole; Isostere; Pain; Established FCA