Keywords: شیمی دارویی; Natural products; Salinomycin; Molecular editing; Coordination chemistry; Cancer; Cancer stem cells; Iron; Fenton chemistry; Medicinal chemistry; Chemical biology;
مقالات ISI شیمی دارویی (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: شیمی دارویی; Chlorins; Conjugate; PDT; Targeted delivery; Water-solubility; Medicinal chemistry;
Keywords: شیمی دارویی; Phenazine; Antibacterials; Biofilms; Medicinal chemistry;
Keywords: شیمی دارویی; Oxazole; Biological activity; Medicinal chemistry;
Keywords: شیمی دارویی; Flow synthesis; Microreactors; Heterocycles; Thiadiazoles; Medicinal chemistry;
Keywords: شیمی دارویی; Antimicrobial resistance; Nitrofuran isoxazoline; MRSA; Medicinal chemistry; Antibacterial activity; Structure activity relationship;
Keywords: شیمی دارویی; Medicinal chemistry; Pharmaceutical sciences; Teaching assistant; Performance enhancing drugs; Sports pharmacy;
Keywords: شیمی دارویی; TPH1; Peripheral serotonin; 5-HT; Medicinal chemistry; Acyl guanidine;
Keywords: شیمی دارویی; ER stress; Endoplasmic reticulum; Drug discovery; Small molecules; Medicinal chemistry
Keywords: شیمی دارویی; Peroxide chemistry; Antimalarial; Reductive amination; Chemoselective reduction; Medicinal chemistry;
Keywords: شیمی دارویی; 2-Aminothiazole; Thiazole; Review; Bioactive; Drugs; Medicinal chemistry; Pharmacological activityPYOHXOCYLWZLHG-POBNSRABSA-N; PJIYRYGHRUYOKC-UHFFFAOYSA-N; CLLVHNSKSXYNSO-UHFFFAOYSA-N
Keywords: شیمی دارویی; Screening; Protein; Medicinal chemistry; Structure-based drug design;
Keywords: شیمی دارویی; Cisplatin; Metallodrugs; Bioinorganic chemistry; Medicinal chemistry; Antitumor agents; Platinum; Platinated proteinsa.u., asymmetric unit; Atox-1, a copper chaperone protein; ATP7A, Menkes’ disease protein; ATP7B, Wilson's disease protein; beSOD, superox
Keywords: شیمی دارویی; Seven-membered rings; Azepane; Oxepane; Diazocarbonyl; Medicinal chemistry;
Keywords: شیمی دارویی; Therapeutic peptides; Passive permeability; Physicochemical properties; Medicinal chemistry; Macrocyclic peptides; Protein–protein interactions
Keywords: شیمی دارویی; Fluorine; C-F bond activation; Catalysis; Medicinal chemistry;
Keywords: شیمی دارویی; Plasmodium falciparum; Malaria; Medicinal chemistry; Phenotypic hit; DMPK; drug metabolism and pharmacokinetics; SAR; structure-activity relationship; WHO; World Health Organisation; WHO-TDR; World Health Organisation Programme for Research and Training i
Keywords: شیمی دارویی; Boron clusters; Carbohydrate; Carbohydrate mimetics; Cancer therapy; Glycoconjugates; Medicinal chemistry;
Keywords: شیمی دارویی; Neurodegenerative disease; Parkinson disease; MALDI-TOF imaging; Biological screening; Medicinal chemistry; Quinoxaline
Keywords: شیمی دارویی; AAT; alpha-1 antitrypsin (alpha-1 proteinase inhibitor, α-1 PI); AATD; alpha-1 antitrypsin deficiency; ALI; acute lung injury; ARDS; acute respiratory distress syndrome; BE; bronchiectasis; CF; cystic fibrosis; COPD; chronic obstructive pulmonary disease
Keywords: شیمی دارویی; ADME; absorption, distribution, metabolism, excretion; BBB; blood-brain barrier; CEV; California encephalitis virus; CNS; central nervous system; CPE; cytopathic effect; ECMV; encephalomyocarditis virus; fLUC; firefly luciferase; FMV; Fort Morgan virus;
Keywords: شیمی دارویی; Aromatase inhibitors; Breast cancer; Medicinal chemistry; Molecular modeling; Ring substituted androstanes; Steroids;
Keywords: شیمی دارویی; Molecular database; Undergraduate pharmacy education; Medicinal chemistry; Respiratory pharmacology; Visualization
Keywords: شیمی دارویی; Click chemistry; Azides; Alkynes; Medicinal chemistry; Cycloadditions;
Keywords: شیمی دارویی; Medicinal chemistry; Video; Structure–activity relationships; MOE
3-Hydroxy-1,5-dihydro-2H-pyrrol-2-ones as novel antibacterial scaffolds against methicillin-resistant Staphylococcus aureus
Keywords: شیمی دارویی; Natural products; Antibiotics; Heterocycles; Cyclization; Medicinal chemistry;
A new target for Alzheimer's disease: A small molecule SERCA activator is neuroprotective in vitro and improves memory and cognition in APP/PS1 mice
Keywords: شیمی دارویی; Alzheimer's disease; ER stress; SERCA; Drug discovery; Small molecules; Medicinal chemistry; Neurodegeneration;
Case-based studies in teaching medicinal chemistry in PharmD curriculum: Perspectives of students, faculty, and pharmacists from academia
Keywords: شیمی دارویی; Medicinal chemistry; Curriculum; Case studies; Therapeutic decision-making;
Synthesis of cis- and trans-(±)-3-mercaptoproline and pipecolic acid derivatives via thio-Michael addition
Keywords: شیمی دارویی; Thio-Michael addition; Proline derivatives; Pipecolic acid derivatives; Cysteine derivatives; Medicinal chemistry;
Small molecule SUMOylation activators are novel neuroprotective agents
Keywords: شیمی دارویی; SUMO; Small ubiquitin-like modifier; Drug discovery; Small molecules; Medicinal chemistry; Neurodegeneration;
Discovery of 2,4-dimethoxypyridines as novel autophagy inhibitors
Keywords: شیمی دارویی; Autophagy; Phenotypic screening; High-throughput screening; Natural products; Medicinal chemistry;
Microcystins: Synthesis and structure-activity relationship studies toward PP1 and PP2A
Keywords: شیمی دارویی; Adda; (2S,3S,8S,9S)-3-amino-9-methoxy-2,6,8-trimethyl-10-phenyldeca-4,6-dienoic acid; Amba; (2S,3S)-3-amino-2-methylbutanoic acid; Boc; tert-butoxycarbonyl; BOP; benzotriazol-1-yloxy-tris-dimethylaminophosphoniumhexafluoro phosphate; Cbz; carboxybenzyl; D
New insights in Au-NHCs complexes as anticancer agents
Keywords: شیمی دارویی; Medicinal chemistry; Antitumor agents; N-heterocyclic carbenes; Azolium salts; Gold(I); Gold(III);
Chloro(triphenylphosphine)gold(I) a forefront reagent in gold chemistry as apoptotic agent for cancer cells
Keywords: شیمی دارویی; Medicinal chemistry; Metallotherapeutic; Gold(I) complexes; Breast cancer cells; Pnictogen; Apoptosis;
Diterpenoid lead stevioside and its hydrolysis products steviol and isosteviol: Biological activity and structural modification
Keywords: شیمی دارویی; Stevioside; Steviol; Isosteviol; Medicinal chemistry; Lead exploration;
Meeting report: Third Summer School on Innovative Approaches for Identification of Antiviral Agents (IAAASS)
Keywords: شیمی دارویی; Antiviral therapies; Summer school; Emerging infections; Antiviral drugs; Medicinal chemistry;
NMR strategies to support medicinal chemistry workflows for primary structure determination
Keywords: شیمی دارویی; NMR methods; Medicinal chemistry; Primary structure; Regioisomers; Rotamers;
A pilot study assessing the value of 3D printed molecular modelling tools for pharmacy student education
Keywords: شیمی دارویی; 3D; three-dimensional; ABS; acrylonitrile butadiene styrene; CAD; computer-aided design; PDB; protein data bank; PLA; polylactic acid; RCSB; Research Collaboratory for Structural Bioinformatics; 3D printing; Education; Medicinal chemistry; Molecular model
Synthesis of heterocycles from arylacetonitriles: Powerful tools for medicinal chemists
Keywords: شیمی دارویی; Arylacetonitriles; Heterocycles; Medicinal chemistry;
Discovering novel 7-azaindole-based series as potent AXL kinase inhibitors
Keywords: شیمی دارویی; AXL; 7-Azaindole; Receptor tyrosine kinase; Kinase inhibitor; Modeling study; Medicinal chemistry;
Improving the throughput of batch photochemical reactions using flow: Dual photoredox and nickel catalysis in flow for C(sp2)C(sp3) cross-coupling
Keywords: شیمی دارویی; Photoredox; Dual catalysis; Flow chemistry; C(sp2)C(sp3) cross-coupling; Medicinal chemistry;
A new target for Parkinson's disease: Small molecule SERCA activator CDN1163 ameliorates dyskinesia in 6-OHDA-lesioned rats
Keywords: شیمی دارویی; Parkinson's disease; ER stress; Endoplasmic reticulum; Drug discovery; Small molecules; Medicinal chemistry;
The discovery of benzoxazine sulfonamide inhibitors of NaV1.7: Tools that bridge efficacy and target engagement
Keywords: شیمی دارویی; NaV1.7; voltage gated sodium channel 1.7; SCN9A; sodium voltage-gated channel alpha subunit 9; TM; transmembrane; VSD; voltage sensing domain; CLu; unbound clearance; HLM; human liver microsome; RLM; rat liver microsome; PX; patch express; LLE; ligand lip
African trypanosomiasis: Synthesis & SAR enabling novel drug discovery of ubiquinol mimics for trypanosome alternative oxidase
Keywords: شیمی دارویی; Antiprotozoal agents; Oxidoreductase; Medicinal chemistry; Synthesis design;
Medicinal chemistry and biological potential of Cyperus rotundus Linn.: An overview to discover elite chemotype(s) for industrial use
Keywords: شیمی دارویی; Cyperus rotundus; Medicinal chemistry; Biological properties; Chemotype(s); Natural product;
Medicinal chemistry of antischistosomal drugs: Praziquantel and oxamniquine
Keywords: شیمی دارویی; Schistosomiasis; Praziquantel; Oxamniquine; Medicinal chemistry;
The medicinal chemistry of Chikungunya virus
Keywords: شیمی دارویی; Chikungunya; Medicinal chemistry; Synthesis; Natural products; In silico;
Thiosemicarbazones and 4-thiazolidinones indole-based derivatives: Synthesis, evaluation of antiproliferative activity, cell death mechanisms and topoisomerase inhibition assay
Keywords: شیمی دارویی; Medicinal chemistry; Anticancer therapy; Cellular death; DNA interaction; Topoisomerase inhibition;
Synthesis of novel, functionalised tricycles utilising the interrupted Pummerer reaction
Keywords: شیمی دارویی; Interrupted Pummerer; Cyclisation; Heterocycle; Drug discovery; Medicinal chemistry;
C-H activation reactions as useful tools for medicinal chemists
Keywords: شیمی دارویی; C-H activation; Heterocycles; Pharmaceuticals; Drug discovery; Medicinal chemistry;