The discovery of novel benzofuran-2-carboxylic acids as potent Pim-1 inhibitors
Keywords: شیمی دارویی; Enzyme, Kinase; Inhibitor; Benzofuran; X-ray structure; Structure based design; Salt-bridge; Hydrogen bond interaction; Synthesis; Carboxylic acid; Amine; Basicity; SPR; Medicinal chemistry; Fragment screening