Keywords: mGlu4; GRM4; α-Subunit of the GABAA; GABRA1; Gene expression; TCN 238; Hippocampus
مقالات ISI (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Pharmacological activation of mGlu4 and mGlu7 receptors, by LSP2-9166, reduces ethanol consumption and relapse in rat
Keywords: Operant ethanol self-administration; LSP2-9166; mGlu4; mGlu7; Rat; Relapse;
mGlu4 allosteric modulation for treating Parkinson's disease
Keywords: Parkinson's disease; Dyskinesia; Glutamate; Dopamine; mGlu4; 6-OHDA; 6-hydroxydopamine; ADX88178; 4-methyl-N-[5-methyl-4-(1H-pyrazol-4-yl)-1,3-thiazol-2-yl]pyrimidin-2-amine; AIM; abnormal involuntary movements; CODA-RET; complemented donor acceptor reson
Discovery of 3-aminopicolinamides as metabotropic glutamate receptor subtype 4 (mGlu4) positive allosteric modulator warheads engendering CNS exposure and in vivo efficacy
Keywords: mGlu4; Metabotropic glutamate receptor; Positive allosteric modulator (PAM); Parkinson's disease; Structure-activity relationship (SAR);
Functional modulation of G-protein coupled receptors during Parkinson disease-like neurodegeneration
Keywords: Metabotropic glutamate receptor; mGlu4; mGlu5; Parkinson's disease; Positron emission tomography; Pharmacological magnetic resonance imaging;
Co-operative binding assay for the characterization of mGlu4 allosteric modulators
Keywords: Metabotropic glutamate receptor; Parkinson disease; mGlu4; Binding affinity;
Related functions of mGlu4 and mGlu8
Keywords: mGlu4; mGlu8; Open field; Zero maze; Fear conditioning; Body weight;
Synthesis and SAR of a novel metabotropic glutamate receptor 4 (mGlu4) antagonist: Unexpected ‘molecular switch’ from a closely related mGlu4 positive allosteric modulator
Keywords: Metabotropic glutamate receptor 4; mGlu4; Molecular switch; Antagonist
An orally bioavailable positive allosteric modulator of the mGlu4 receptor with efficacy in an animal model of motor dysfunction
Keywords: Allosteric modulator; mGlu4; Parkinson’s disease; Styryl pyrimidinyl amines
Metabotropic glutamate receptor 4 novel agonist LSP1-2111 with anxiolytic, but not antidepressant-like activity, mediated by serotonergic and GABAergic systems
Keywords: Metabotropic glutamate receptors; Anxiety; LSP1-2111; mGlu4
Design and synthesis of APTCs (aminopyrrolidinetricarboxylic acids): Identification of a new group III metabotropic glutamate receptor selective agonist
Keywords: Metabotropic glutamate receptor; mGlu4; Excitatory amino acids
Modulation of retino-collicular transmission by Group III metabotropic glutamate receptors at different ages during development
Keywords: Superior colliculus; mGlu4; mGlu8; mGlu7; Retino-collicular transmission; L-AP4; Development; Presynaptic receptors; Metabotropic glutamate receptors;