Keywords: مطالعات تکاملی مولکولی; Oxadiazole-benzohydrazone hybrids; Leishmaniasis; SAR study; Molecular docking studies; DFT; Selectivity index;
مقالات ISI مطالعات تکاملی مولکولی (ترجمه نشده)
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Keywords: مطالعات تکاملی مولکولی; Thiobarbituric acid; Synthesis; Urease inhibition; Molecular docking studies
Keywords: مطالعات تکاملی مولکولی; 3,4-Methylenedioxycyanostilbenes; 3,4-Ethylenedioxycyanostilbenes; Synthesis of cyanostilbenes; Anti-cancer activity; Molecular docking studies
Keywords: مطالعات تکاملی مولکولی; Jack-Bean Urease; Dithiocarbamates; Molecular docking studies;
Keywords: مطالعات تکاملی مولکولی; Quinoline-pyrazole hybrids; SC-XRD analysis; Antitubercular activity; Antibacterial activity; Cytotoxicity; Molecular docking studies;
Keywords: مطالعات تکاملی مولکولی; Chalcones; 1D and 2D NMR spectroscopy; Tyrosinase inhibitors; Flavokawain A; Flavokawain B; Molecular docking studies
Keywords: مطالعات تکاملی مولکولی; 6-Methyl nicotinate; 1,3,4-Oxadiazole; Antimicrobial studies; Antioxidant studies; Molecular docking studies;
4-Aminopyridine based amide derivatives as dual inhibitors of tissue non-specific alkaline phosphatase and ecto-5â²-nucleotidase with potential anticancer activity
Keywords: مطالعات تکاملی مولکولی; Ecto-5â²-nucleotidase (e5â²NT); Alkaline phosphatases (APs); 4-aminopyridinederivatives; Mechanism of action; Molecular docking studies;
Synthesis, in vitro urease inhibitory activity, and molecular docking studies of thiourea and urea derivatives
Keywords: مطالعات تکاملی مولکولی; Synthesis; Urea; Thiourea; In vitro urease activity; Structure-activity relationship; Molecular docking studies;
Synthesis, structure-activity relationship and molecular docking studies of 3-O-flavonol glycosides as cholinesterase inhibitors
Keywords: مطالعات تکاملی مولکولی; Flavonoids; Flavonols; 3-Hydroxyflavones; Glycosides; Cholinesterases; AChE/BChE inhibitors; Molecular docking studies;
Copper(II) complexes of bidentate mixed ligands as artificial nucleases: Synthesis, crystal structure, characterization and evaluation of biological properties
Keywords: مطالعات تکاملی مولکولی; Mixed ligand complexes; single crystal; ctDNA binding studies; Molecular Docking studies; Nuclease activity;
Synthesis, characterization, stereochemistry and biological investigation of certain N-dichloroacetyl-bis(2-chlorophenyl)piperidin-4-ones
Keywords: مطالعات تکاملی مولکولی; N-Dichloroacetyl-bis(2-chlorophenyl)piperidin-4-one; NMR spectra; Twist boat conformation; X-ray structure; Molecular docking studies; Antimicrobial activity; Antioxidant activity;
Synthesis, structure-activity relationship and molecular docking of 3-oxoaurones and 3-thioaurones as acetylcholinesterase and butyrylcholinesterase inhibitors
Keywords: مطالعات تکاملی مولکولی; Flavonoids; Aurones; 3-Thioaurones; Lawesson's reagent; AChE/BChE inhibitors; Molecular docking studies;
Design, synthesis and biological evaluation of 1,3-diphenylbenzo[f][1,7]naphthyrdines
Keywords: مطالعات تکاملی مولکولی; 1,3-Diphenylbenzo[f][1,7]benzonaphthyrdines; Human Topoisomerase IIα inhibitors; Cytotoxic agents; Molecular docking studies; Imino Diels-Alder reaction;
Synthesis, structural, spectroscopic and docking studies of new 5C-substituted 2,4-diamino-5H-chromeno[2,3-b]pyridine-3-carbonitriles
Keywords: مطالعات تکاملی مولکولی; chromeno[2,3-b]pyridines; Multicomponent reactions; Spectroscopic studies; Powder XRD; Keto-enol equilibrium; Molecular docking studies; FCSZJXMCXHPBGY-MHQSUUTLSA-N;
Synthesis, in vitro β-glucuronidase inhibitory potential and molecular docking studies of quinolines
Keywords: مطالعات تکاملی مولکولی; β-Glucuronidase; Quinoline; Sulfonamide; Sulfonate; Molecular docking studies;
Antileishmanial activity of novel indolyl–coumarin hybrids: Design, synthesis, biological evaluation, molecular docking study and in silico ADME prediction
Keywords: مطالعات تکاملی مولکولی; Indolyl–coumarin hybrids; Ho3+ doped CoFe2O4 nanoparticles; Antileishmanial; Antioxidant; Molecular docking studies
Synthesis and biological evaluation of enantiomerically pure glyceric acid derivatives as LpxC inhibitors
Keywords: مطالعات تکاملی مولکولی; LpxC inhibitors; Structure–activity relationships; Glyceric acid derivatives; Chiral pool synthesis; Enantioselective desymmetrization; Molecular docking studies
Anti-uropathogenic activity, drug likeness, physicochemical and molecular docking assessment of (E-)-N′-(substituted-benzylidene)-2-(quinolin-8-yloxy) acetohydrazide
Keywords: مطالعات تکاملی مولکولی; Anti-uropathogenic; Bioactivity score; Physicochemical properties synthesis; Molecular docking studies
1-Benzyl-2-methyl-3-indolylmethylene barbituric acid derivatives: Anti-cancer agents that target nucleophosmin 1 (NPM1)
Keywords: مطالعات تکاملی مولکولی; 1-Benzyl-2-methyl-3-indolyl barbituric acid; Anticancer activity; Nucleophosmin 1; Anti-leukemic activity; Molecular docking studies; NPM1 oligomerization;
Antihormonal potential of selected D-homo and D-seco estratriene derivatives
Keywords: مطالعات تکاملی مولکولی; Molecular docking studies; D-homo-estratriene derivatives; 16,17-Seco-estratriene derivatives; Antiestrogens; Steroidogenesis enzymes inhibitors and activators; X-ray (XRD)
Synthesis, spectroscopic characterization and in vitro studies of new heteroleptic copper (II) complexes derived from 2-hydroxy napthaldehyde Schiff's bases and N, N donor ligands: Antimicrobial, DNA binding and cytotoxic investigations
Keywords: مطالعات تکاملی مولکولی; Copper (II) complexes; DNA binding; DNA cleavage; Molecular docking studies; Antimicrobial and cytotoxicity;
Synthesis, biological evaluation and molecular docking studies of benzyloxyacetohydroxamic acids as LpxC inhibitors
Keywords: مطالعات تکاملی مولکولی; LpxC inhibitors; Antibacterials; Enantioselective synthesis; Phenylethylene glycol derivatives; Molecular docking studies;
In vitro DNA binding, pBR322 plasmid cleavage and molecular modeling study of chiral benzothiazole Schiff-base-valine Cu(II) and Zn(II) complexes to evaluate their enantiomeric biological disposition for molecular target DNA
Keywords: مطالعات تکاملی مولکولی; Chiral Cu(II)/Zn(II) benzothiazole-valine complexes; Enantiomeric discrimination with DNA; Binding studies; Molecular docking studies; UV-vis; UV-visible; CT DNA; Calf thymus DNA; Tris; Tris(hydroxymethyl)aminomethane; EB; ethidium bromide;
Synthesis, crystal structure and antiproliferative activity of Cu(II) nalidixic acid-DACH conjugate: Comparative in vitro DNA/RNA binding profile, cleavage activity and molecular docking studies
Keywords: مطالعات تکاملی مولکولی; Nalidixic acid; pBR322 DNA cleavage; Topo-II inhibition assay; U2OS cells; Molecular docking studies; UV-vis; UV-visible; ct-DNA; Calf thymus DNA; Topo II; Topoisomerase II; U2OS; Human osteoblastoma cell line;
Flavanocoumarins from Guazuma ulmifolia bark and evaluation of their affinity for STAT1
Keywords: مطالعات تکاملی مولکولی; Guazuma ulmifolia; Flavanocoumarins; STAT1; Surface Plasmon Resonance; Molecular docking studies;
Molecular docking studies of some new imidazole derivatives for antimicrobial properties
Keywords: مطالعات تکاملی مولکولی; Molecular docking studies; Imidazoles; Pyrazoles; Antibacterial studies
Withanolides, a new class of natural cholinesterase inhibitors with calcium antagonistic properties
Keywords: مطالعات تکاملی مولکولی; Withanolides; Ajuga bracteosa; Withania somnifera; Acetylcholinesterase; Butyrylcholinesterase; Molecular docking studies; Enzyme inhibition; Calcium antagonist;