Keywords: N، N-دییزوپروپیلتیلامین; QPA; quaternary protoberberine alkaloid; TF; transcriptional factor; UC; ulcerative colitis; IEC-6; intestinal epithelial cell-6; XBP1; X-box-binding protein 1; MIC; minimal inhibitory concentration; SAR; structure-activity relationship; SASP; Sulfasalazi
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Keywords: N، N-دییزوپروپیلتیلامین; SI; supporting information; NBD-Cl; 4-chloro-7-nitrobenzofurazan; NBD-OH; 4-hydroxy-7-nitrobenzofurazan; DIC; N,Nâ²-diisopropylcarbodiimide; DMAP; 4-dimethylaminopyridine; DIEA; N,N-diisopropylethylamine; HATU; 1-[bis(dimethylamino)methylene]-1H-1,2,3-tr
Keywords: N، N-دییزوپروپیلتیلامین; Bub1; budding uninhibited by benzimidazoles 1; Cbz; benzyloxycarbonyl; CD69; a human transmembrane C-Type lectin protein; DAST; diethylaminosulfur trifluoride; dba; dibenzylideneacetone; DIPEA; N,N-diisopropylethylamine; DMAD; dimethyl acetylenedicarboxyl
Keywords: N، N-دییزوپروپیلتیلامین; Ac; acetyl; AcOH; acetic acid; AccQ; 6-aminoquinolyl-N-hydroxysuccinimidyl carbamate; AIDA; 1-aminoindan-1,5-dicarboxylic acid; aq.; aqueous; BA; butylamine; Boc; tert-butyloxycarbonyl; t-BuCQD; t-butylcarbamoylated quinidine-based CSP; t-BuCQN; t-butylca
Keywords: N، N-دییزوپروپیلتیلامین; AF-1; activation function-1; AF-2; activation function-2; AP-1; activator protein 1; dppp; 1,3-bis(diphenylphosphino)propane; DEX; dexamethasone; DIEA; N,N-diisopropylethylamine; FKBP5; FK506-binding protein 5; GR; glucocorticoid receptor; GRE; glucocorti
Keywords: N، N-دییزوپروپیلتیلامین; BS; brassinosteroids; DMAP; N,N-dimethylaminopyridine; EBl; 24-epibrassinolide; DIPEA; N,N-diisopropylethylamine; TBAF; tetra-n-butylammonium fluoride; TBAI; tetra-n-butylammonium iodide; TBSCl; tert-butyldimethylsilyl chloride; TFA; trifluoroacetic acid;
Keywords: N، N-دییزوپروپیلتیلامین; DAPI; 4â²,6-diamidino-2-phenylindole; DIC; diisopropylcarbodiimide; DMEM; Dulbecco's Modified Eagle's medium; EDIPA; N,N-diisopropylethylamine; FBS; fetal bovine serum; FITC; fluorescein isothiocyanate; GFP; green fluorescent protein; HaCaT; human kerati
Identification of highly selective and potent orexin receptor 1 antagonists derived from a dual orexin receptor 1/2 antagonist based on the structural framework of pyrazoylethylbenzamide
Keywords: N، N-دییزوپروپیلتیلامین; OX1R; orexin 1 receptor; OX2R; orexin 2 receptor; DORA; dual orexin receptor antagonist; SORA; selective orexin receptor antagonist; SI; selectivity index; BBB; blood-brain barrier; CNS; central nervous system; SAR; structure-activity relationship; Boc; t
Keywords: N، N-دییزوپروپیلتیلامین; Methyl oleate; Trimethyl chlorosilane; Acid binding agent; N,N-diisopropylethylamine; Lubricity; Silicon-based biological lubricating base oil;
Metal coordinated pyrrole-based macrocycles as contrast agents for magnetic resonance imaging technologies: Synthesis and applications
Keywords: N، N-دییزوپروپیلتیلامین; AAV9; adeno-associated serotype 9 viral vector; BODIPY; boron-dipyrromethene; BSA; bovine serum albumin; C60; Buckminsterfullerene; CCMV; cowpea chlorotic mottle virus; CD; β-cyclodextrin; Cell line H1299; human non-small cell lung carcinoma cell line; C
Keywords: N، N-دییزوپروپیلتیلامین; ABTS; 2,2â²-azino-bis(3-ethylbenzothiazoline-6-sulfonic acid)diammonium salt; BSA; bovine serum albumin; (bt)-VEGF165; biotinylated-VEGF165; 6-Cl·HOBt; 6-chloro-1-hydroxybenzotriazole dehydrate; DIPEA; N,N-diisopropylethylamine; ELISA; enzyme-linked imm
Keywords: N، N-دییزوپروپیلتیلامین; RNCGDQLZIATDOU-ZDRBWGSPSA-N; ICYPJNZJUFGALC-PDTBJYIYSA-N; PDRMAVOIWIVXKH-SFUSBHMVSA-N; ISADXJRTBSLWPX-ZDRBWGSPSA-N; NLBLLPROASDPSC-QWWZWVQMSA-N; XKMIKZDBUOHHDK-ZDRBWGSPSA-N; BTURADNXKHTWGA-IJOLSIAMSA-N; UEKHRDLXBMZMPD-ZYIYBEKCSA-N; UQCLCXDOXVZEOA-JARUQAPT
Keywords: N، N-دییزوپروپیلتیلامین; AA; amino acid; AcOH; acetic acid; 6-Cl-HOBt; 6-chloro-1-hydroxybenzotriazole; DCM; dichloromethane; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; Fmoc; 9-fluorenylmethoxycarbonyl; h; hour; HOBt; 1-hydroxybenzotriazole hydrate; HPLC; high-
Keywords: N، N-دییزوپروپیلتیلامین; Antisense oligonucleotides; PEGylation; Disulfide bioconjugates; Solid phase synthesis; Gene silencing; ON; oligonucleotide; PEG; polyethylene glycol; CPG; controlled pore glass; LCAA; long chain amino alkyl; TCEP; tris(2-carboxyethyl)phosphin; TBP; tri-n
Keywords: N، N-دییزوپروپیلتیلامین; SAMs; self-assembled monolayers; RG; reactive group; GOX; glucose oxidase; LOX; lactate oxidase; HAOX; hydroxyacid oxidase; BSA; bovine serum albumin; NHS; N-hydroxysuccinimide; TFAAD; trifluoroacetyl-protected 10-amino-1-decene; TFA; trifluoroacetyl; TFE
Keywords: N، N-دییزوپروپیلتیلامین; BPO; benzoyl peroxide; DCM; dichloromethane; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; DMSO; dimethyl sulfoxide; FaSSIF; fasted state simulated intestinal fluid; HATU; 1-[bis(dimethylamino)methylene]-1H-1,2,3-triazolo[4,5-b]pyridinium
Keywords: N، N-دییزوپروپیلتیلامین; ATX/NPP2; autotaxin; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; DMSO; dimethylsulfoxide; GPCR; G-protein coupled receptor; GRI; Genomic Research Institute; HBTU; O-(benzotriazol-1-yl)-N,N,Nâ²,Nâ²-tetramethyluronium hexafluorophosphate
Keywords: N، N-دییزوپروپیلتیلامین; Pro-apoptotic agents; Anticancer agents; Cyclic peptides; Peptidomimetics; Nur77; Tubulin; Bcl-2; NMR studies; Molecular modeling; Confocal microscopy; FACS analysis; ADT; AutoDock Tools; COSY; correlation spectroscopy; DBU; 1,8-Diazabicyclo[5.4.0]undec-7
Keywords: N، N-دییزوپروپیلتیلامین; Nitro compounds; Natural products; Pharmaceuticals; Stereoselective synthesis; Organocatalysis; Metal catalysis; Nitronates; Nitrile oxides; AIBN; azobisisobutyronitrile; AZADO; 2-azaadamantane-N-oxyl; 9-BBN; 9-borabicyclo[3.3.1]nonane; BINAP; 2,2â²-bis(
Keywords: N، N-دییزوپروپیلتیلامین; BBB; blood-brain barrier; Boc; tert-butyloxycarbonyl; cAMP; cyclic adenosine monophosphate; CNS; central nervous system; DAMGO; H-Tyr-d-Ala-Gly-NMePhe-Gly-ol; DCM; dichloromethane; DIEA; N,N-diisopropylethylamine; DOR; δ-opioid receptor; DPDPE; Tyr-c(d
Keywords: N، N-دییزوپروپیلتیلامین; Cyclic peptides; Microwave assisted synthesis; Lactam-bridge cyclic peptides; SHU9119; MTII; MWA-SPPS; microwave-assisted solid phase peptide synthesis; MBHA; methylbenzhydryl; MCR; melanocortin receptors; NDP; [Nle4, DPhe7]-αMSH; MTII; melanotan-II; RP-
Keywords: N، N-دییزوپروپیلتیلامین; Abz; ortho-aminobenzoic acid; EDDnp; N-(2,4-dinitrophenyl)-ethylenediamine; FRET; fluorescence resonance energy transfer; hMIP; human mitochondrial intermediate peptidase; HOBt; hydroxybenzotriazole; TBTU; O-(benzotriazol-1-yl)-N,N,Nâ²,Nâ²-tetramethylur
Keywords: N، N-دییزوپروپیلتیلامین; Obesity; Diabetes; DGAT1; Inhibitor; Adamantane; DGAT; acyl CoA:diacylglycerol acyltransferase; TG; triglyceride; DIPEA; N,N-diisopropylethylamine; OLTT; oral lipid tolerance test; DIO; diet-induced obesity; EDCI; 1-ethyl-3-(3-dimethylaminopropyl)carbodii
Keywords: N، N-دییزوپروپیلتیلامین; AMPs; antimicrobial peptides; ATCC; American type culture collection; CD; circular dichroism; CFU; colony forming units; CLSI; Clinical and Laboratory Standards Institute; DIPEA; N,N-diisopropylethylamine; DMEM; Dulbecco's modified eagle's medium; DMF; N,
Keywords: N، N-دییزوپروپیلتیلامین; Peptidomimetic boronates; Proteasome inhibitors; Docking studies; ChT-L; chymotrypsin-like; T-L; trypsin-like; PGPH; post-glutamyl peptide hydrolyzing; DMSO; dimethyl sulfoxide; DMF; dimethylformamide; Pd2(dba)3; tris(benzylideneacetone)dipalladium; EDC;
Design, synthesis, in vitro and in vivo evaluation, and structure-activity relationship (SAR) discussion of novel dipeptidyl boronic acid proteasome inhibitors as orally available anti-cancer agents for the treatment of multiple myeloma and mechanism stud
Keywords: N، N-دییزوپروپیلتیلامین; SAR; structureactivity relationship; UPP; ubiquitinproteasome pathway; FDA; Food and Drug Administration; ATP; Adenosine triphosphate; CP; core particle; RP; regulatory proteasome; C-L; caspase-like; T-L; trypsin-like; CT-L; chymotrypsin-like; EDCI; 1-eth
DNA sequence-specific ligands. XVII. Synthesis, spectral properties, virological and biochemical studies of fluorescent dimeric bisbenzimidazoles DBA(n)
Keywords: N، N-دییزوپروپیلتیلامین; topo-I; DNA topoisomerase I; DMT; DNA methyltransferase; HSV-1; herpes simplex virus type 1; CMV; cytomegalovirus; scDNA; supercoiled DNA; b.p.; base pairs; MABs; monoclonal antibodies; ACV; acyclovir; PBS; phosphate buffered saline; PFU/cells; plaque for
Design and synthesis of alkyl substituted pyridino[2,3-D]pyrimidine compounds as PI3Kα/mTOR dual inhibitors with improved pharmacokinetic properties and potent in vivo antitumor activity
Keywords: N، N-دییزوپروپیلتیلامین; PI3K; phosphoinositide 3-kinase; mTOR; mammalian target of rapamycin; TSC; tuberous sclerosis; DDQ; 2,3-dicyano-5,6-dichlorobenzoquinone; THF; tetrahydrofuran; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; MRT; mean retention time; PI3Kα/
Cathepsin B inhibitors: Further exploration of the nitroxoline core
Keywords: N، N-دییزوپروپیلتیلامین; Abz; 2-aminobenzoyl; AMC; 7-amido-4-methylcoumarin; catB; cathepsin B; DIPEA; N,N-diisopropylethylamine; DMSO; dimethyl sulfoxide; ECM; extracellular matrix; EDC; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide; HATU; 1-[bis(dimethylamino)methylene]-1H-1,2,
Novel aromatic sulfonyl naphthalene-based boronates as 20S proteasome inhibitors
Keywords: N، N-دییزوپروپیلتیلامین; TEA; triethylamine; THF; tetrahydrofuran; Py; pyridine; DIPEA; N,N-diisopropylethylamine; TBTU; 2-(1H-benzotriazole-1-yl)-1,1,3,3-tetramethyluronium tetrafluoroborate; DCM; dichloromethane; TPLM; (1R)-(S)-pinanediol-1-ammonium trifluoroacetate-3-methylbut
Optimization of permeability in a series of pyrrolotriazine inhibitors of IRAK4
Keywords: N، N-دییزوپروپیلتیلامین; ABC; Activated B Cell-like; BTK; Bruton's Tyrosine Kinase; CD79; Cluster of Differentiation 79; CDK; Cyclin Dependent Kinase; CLK; CDC-Like Kinase; DCM; dichloromethane; DDQ; 2,3-Dichloro-5,6-DicyanobenzoQuinone; DIPEA; N,N-diisopropylethylamine; DLBCL;
Design, synthesis, and evaluation of carboxyl-modified oseltamivir derivatives with improved lipophilicity as neuraminidase inhibitors
Keywords: N، N-دییزوپروپیلتیلامین; NA; neuraminidase; OS; oseltamivir; OC; oseltamivir carboxylate; TFA; trifluor-oacetic acid; HATU; 1-[bis(dimethylamino)methylene]-1H-1,2,3-triazolo[4,5-b]pyr-idinium 3-oxid hexafluorophosphate; DIPEA; N,N-diisopropylethylamine; PDB; protein data bank; In
Scaffold hopping identifies 6,8-disubstituted purines as novel anaplastic lymphoma kinase inhibitors
Keywords: N، N-دییزوپروپیلتیلامین; ALK; anaplastic lymphoma kinase; cMet; hepatocyte growth factor receptor; DIPEA; N,N-Diisopropylethylamine; DMF; N,N-Dimethylformamide; EML4; echinoderm microtubule-associated protein-like 4; FDA; food and drug administration; gk; gatekeeper; μW; micro w
Discovery of benzimidazole derivatives as orally active renin inhibitors: Optimization of 3,5-disubstituted piperidine to improve pharmacokinetic profile
Keywords: N، N-دییزوپروپیلتیلامین; BA; bioavailability; RAAS; renin-angiotensin-aldosterone system; BP; blood pressure; Ang I; angiotensin I; ACE; Angiotensin-converting enzyme; Ang II; angiotensin II; AT1; Ang II type I receptor; DRI; direct renin inhibitor; TPSA; topological polar surfac
Branched pentapeptides as potent inhibitors of the vascular endothelial growth factor 165 binding to Neuropilin-1: Design, synthesis and biological activity
Keywords: N، N-دییزوپروپیلتیلامین; Neuropilin-1; VEGF165; Neuropilin/VEGF165 binding inhibition; Structure-activity relationship; Peptide biostability; ABTS; 2,2â²-azino-bis(3-ethylbenzothiazoline-6-sulfonic acid) diammonium salt; Ahp; 7-aminoheptanoic acid; Aun; 11-aminoundecanoic acid;
Development of potent and proteolytically stable human neuromedin U receptor agonists
Keywords: N، N-دییزوپروپیلتیلامین; Neuromedin U (NMU); NMU-8; Neuromedin U receptor agonists; Plasma stability; 1â²Nal; 1â²-naphtylalanine; 2â²Nal; 2â²-naphtylalanine; 7-OH-Tic; 7-hydroxy-L-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid; ACN; acetonitrile; AUC; area under the curve;
Remarkable differences and similarities between the isomeric Mn(II)-cis- and trans-1,2-diaminocyclohexane-N,N,Nâ²,Nâ²-tetraacetate complexes
Keywords: N، N-دییزوپروپیلتیلامین; MRI; magnetic resonance imaging; DFT; Density Functional Theory; APC; aminopolycarboxylate; CA; contrast agent; dtpa; diethylenetriaminepentaacetic acid; dota; 1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid; NSF; nephrogenic systemic fibrosis; e
The 4-N-acyl and 4-N-alkyl gemcitabine analogues with silicon-fluoride-acceptor: Application to 18F-Radiolabeling
Keywords: N، N-دییزوپروپیلتیلامین; dFdC; 2â²,2â²-difluoro-2â²-deoxycytidine (Gemcitabine); hENT1; human equilibrative nucleoside transport protein 1; dCK; deoxycytidine kinase; dFdU; 2â²,2â²-difluorouridine; CDA; cytidine deaminase; [18F]FAC; 1-(2-deoxy-2-[18F]fluoro-β-d-arabinofuran
Fragment-growing guided design of Keap1-Nrf2 protein-protein interaction inhibitors for targeting myocarditis
Keywords: N، N-دییزوپروپیلتیلامین; ROS; reactive oxygen species; NQO-1; NADPH:quinone oxidoreductase 1; HO-1; heme oxygenase-1; ARE; antioxidant response element; Nrf2; nuclear factor erythroid 2-related factor 2; Keap1; Kelch-like ECH-associated protein 1; DMF; dimethyl fumarate; CDDO-Me;
Synthesis and biological evaluation of a library of hybrid derivatives as inhibitors of influenza virus PA-PB1 interaction
Keywords: N، N-دییزوپروپیلتیلامین; Anti-Influenza; PA-PB1; RdRp; Amino acid coupling; SPPS; Diphenyl-pyridine; AcOEt; Ethyl acetate; CC50; Half maximal cytotoxic concentration; cRNA; complementar RNA; DCM; dichloromethane; DDQ; 2,3-Dichloro-5,6-dicyano-1,4-benzoquinone; DIPEA; N,N-Diisopro
Evaluation of a novel GRPR antagonist for prostate cancer PET imaging: [64Cu]-DOTHA2-PEG-RM26
Keywords: N، N-دییزوپروپیلتیلامین; BBN; bombesin; BFCs; bifunctional chelates; BSA; bovine serum albumin; CB-TE2A; 4,11-bis(carboxymethyl)-1,4,8,11-tetraazabicyclo[6.6.2]hexadecane; CH3CN; acetonitrile; C-NE3TA; 4-carboxymethyl-7-[2-(carboxymethyl-amino)-3-(4-nitro-phenyl)-propyl]-[1,4,7]t
Design, synthesis, and structure-activity-relationship of a novel series of CXCR4 antagonists
Keywords: N، N-دییزوپروپیلتیلامین; Chemokine; CXCR4; Antagonist; GPCR; Scaffold hybridization; Therapy; APC; allophycocyanin; BPO; benzoyl peroxide; CCD; charge coupled device; CYP; cytochrome P450; DC; dendritic cells; DCE; 1,2-dichloroethane; DIPEA; N,N-diisopropylethylamine; DMEM; Dulbe
Development of novel oxazolo[5,4-d]pyrimidines as competitive CB2 neutral antagonists based on scaffold hopping
Keywords: N، N-دییزوپروپیلتیلامین; Cannabinoid; CB2 receptor; Neutral antagonist; oxazolo[5,4-d]pyrimidine; Boc; tert-butyloxycarbonyl; cAMP; cyclic adenosine monophosphate; CHO; Chinese hamster ovary cells; CHO-CB2; Chinese hamster ovary cells expressing CB2 receptors; CHO-WT; Chinese ham
New insights about the peculiar role of the 28-38 C-terminal segment and some selected residues in PACAP for signaling and neuroprotection
Keywords: N، N-دییزوپروپیلتیلامین; ACN; acetonitrile; BBB; bloodbrain barrier; Bip; biphenylalanine; Boc; tert-butoxycarbonyl; BOP; (benzotriazol-1-yloxy)tris(dimethylamino) phosphonium hexafluorophosphate; BRET; bioluminescence resonance energy transfer; CHO cells; Chinese hamster ovary c
Synthesis and biological evaluation of novel thiazole- VX-809 hybrid derivatives as F508del correctors by QSAR-based filtering tools
Keywords: N، N-دییزوپروپیلتیلامین; Aminoarylthiazole; Corrector; QSAR; Cystic fibrosis; CFTR; VX809; CF; cystic fibrosis; CFTR; CF transmembrane conductance regulator; AATs; aminoarylthiazoles; HS-YFP; halide-sensitive yellow fluorescent protein; QSAR; quantitative-structure activity relat
Discovery and evaluation of Cav3.1-selective T-type calcium channel blockers
Keywords: N، N-دییزوپروپیلتیلامین; AcOH; acetic acid; 9-BBN; 9-borabicyclo(3.3.1)nonane; DAST; diethylaminosulfur trifluoride; DIPEA; N,N-diisopropylethylamine; DMAP; 4-(dimethylamino)pyridine; DMF; N,N-dimethylformamide; EDC·HCl; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide hydrochlorid
Formation of platinum (II) as a six member ring for sustained polymeric delivery
Keywords: N، N-دییزوپروپیلتیلامین; Hyaluronic acid; Cisplatin chemotherapy; Lysine; Homo-lysine; Five-membered ring; Six-membered ring; HA; hyaluronic acid; PPG; photoremovable protecting group; pHP; p-hydroxyphenacyl; Fmoc; fluorenylmethoxy-carbonyl; HATU; 2-(1H-7-azabenzotriazol-1-yl)-1,
Phenylglycine racemization in Fmoc-based solid-phase peptide synthesis: Stereochemical stability is achieved by choice of reaction conditions
Keywords: N، N-دییزوپروپیلتیلامین; COMU; (1-cyano-2-ethoxy-2-oxoethylidenaminooxy)dimethylaminomorpholinocarbenium hexafluorophosphate; DBU; 1,8-diazabicyclo[5.4.0]undec-7-ene; DEPBT; 3-diethoxyphosphoryloxy)-1,2,3-benzotriazin-4(3H)-one; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethyl
Discovery and evaluation of Cav3.2-selective T-type calcium channel blockers
Keywords: N، N-دییزوپروپیلتیلامین; AcOH; acetic acid; Boc; tert-butylocycarbonyl; DIPEA; N,N-diisopropylethylamine; DMAP; 4-(dimethylamino)pyridine; DMF; N,N-dimethylformamide; EDC·HCl; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide hydrochloride; HOBt; hydroxybenzotriazole; KHMDS; potassi
Structure-activity relationship study of tetrapeptide inhibitors of the Vascular Endothelial Growth Factor A binding to Neuropilin-1
Keywords: N، N-دییزوپروپیلتیلامین; ABTS; 2,2â²-azino-bis(3-ethylbenzothiazoline-6-sulfonic acid) diammonium salt; ACN; acetonitrile; BSA; bovine serum albumin; Dab; L-2,4-diaminobutyric acid; Dap; L-2,3-diaminopropionic acid; DIPEA; N,N-diisopropylethylamine; EC; endothelial cells; ELISA;