Keywords: Ac; acetyl; AD-mix; asymmetric dihydroxylation mix; ATP; adenosine triphosphate; Bn; benzyl; Boc; tert-butyloxycarbonyl; Bu; butyl (n-Bu, n-butyl; I; isobutyl; sec-Bu; sec-butyl; t-Bu; tert-butyl); Bz; benzoyl; CAL-B; Candida antartcia lipase-B; CAN; ceri
مقالات ISI (ترجمه نشده)
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Keywords: CD; circular dichroism; CPE; cytopathic effect; DMF; dimethylformamide; FBS; fetal bovine serum; Fmoc; 9-fluorenylmethoxycarbonyl; HBTU; O-benzotriazole-N,N,Nâ²,Nâ²-tetramethyl-uronium-hexafluorophosphate; HOBt; N-hydroxybenzotriazole; HPLC; high perfor
Keywords: Nitro compounds; Natural products; Pharmaceuticals; Stereoselective synthesis; Organocatalysis; Metal catalysis; Nitronates; Nitrile oxides; AIBN; azobisisobutyronitrile; AZADO; 2-azaadamantane-N-oxyl; 9-BBN; 9-borabicyclo[3.3.1]nonane; BINAP; 2,2â²-bis(
Keywords: MeCN; acetonitrile; CL; clearance; Dess-Martin periodinane; 1,1,1-tris(acetyloxy)-1,1-dihydro-1,2-benziodoxol-3-(1H)-one; DIBALH; diisobutylaluminum hydride; DMF; N,N-dimethylformamide; EtOAc; ethyl acetate; HBTU; N,N,Nâ²,Nâ²-tetramethyl-O-(1H-benzotr
Keywords: Abz; ortho-aminobenzoic acid; EDDnp; N-(2,4-dinitrophenyl)-ethylenediamine; FRET; fluorescence resonance energy transfer; hMIP; human mitochondrial intermediate peptidase; HOBt; hydroxybenzotriazole; TBTU; O-(benzotriazol-1-yl)-N,N,Nâ²,Nâ²-tetramethylur
Keywords: AIBN; α,αâ²-azoisobutyronitrile; AmP-MCF; amino-functionalized mesocellular foam; AP-SiO2; silica functionalized with 3-aminopropyl groups; BCL; Burkholderia cepacia lipase; Bz; benzyl; CAL-A; Candida antarctica lipase A; CAL-B; Candida antarctica lipa
Keywords: SERT; serotonin transporter; NET; norepinephrine transporter; DAT; dopamine transporter; NSS; neurotransmitter/sodium (Na+/Clâ) symporter; SSRI; selective serotonin reuptake inhibitor; NBD; nitrobenzoxadiazolealanine; NMM; N-methylmorpholine; NHS; N-hyd
DNA sequence-specific ligands. XVII. Synthesis, spectral properties, virological and biochemical studies of fluorescent dimeric bisbenzimidazoles DBA(n)
Keywords: topo-I; DNA topoisomerase I; DMT; DNA methyltransferase; HSV-1; herpes simplex virus type 1; CMV; cytomegalovirus; scDNA; supercoiled DNA; b.p.; base pairs; MABs; monoclonal antibodies; ACV; acyclovir; PBS; phosphate buffered saline; PFU/cells; plaque for
Continuous assays for meprin alpha and beta using prolyl tripeptidyl aminopeptidase (PtP) from Porphyromonas gingivalis
Keywords: Astacins; Auxiliary enzyme; Continuous assay; Meprin α/β; Prolyl tripeptidyl aminopeptidase (PtP); AMC; 7-amido-4-methylcoumarin; Boc; tert-butyloxycarbonyl; DCM; dichloromethane; DMF; dimethylformamide; DTE; Dithioerythritol; HIC-EBA; hydrophobic inter
New N-phenylpyrrolamide DNA gyrase B inhibitors: Optimization of efficacy and antibacterial activity
Keywords: Antibacterial; DNA gyrase; GyrB; Inhibitor; N-phenylpyrrolamide; ParE; Topoisomerase IV; ATCC; American type culture collection; ATR; attenuated total reflectance; CDI; 1,1â²-carbonyldiimidazole; CFU; colony-forming unit; CLSI; Clinical and Laboratory St
Substituted α-mercaptoketones, new types of specific neprilysin inhibitors
Keywords: BTFA; boron trifluoroacetate; DIEA; diisopropylethylamine; EtOH; ethanol; HPLC; High Performance Liquid Chromatography; LC/MS; Liquid Chromatography/Mass Spectroscopy; LDA; lithium diisopropyl amide; NEP; neprilysin; NMM; N-methylmorpholine; PMBSH; para-m
Bivalent SIRT1 inhibitors
Keywords: β-NAD+; β-nicotinamide adenine dinucleotide; NAM; nicotinamide; 2â²-O-AADPR; 2â²-O-acyl-ADP-ribose; RP-HPLC; reversed-phase high performance liquid chromatography; HRMS; high-resolution mass spectrometry; EDC-MeI; 1-(3-dimethylaminopropyl)-3-ethylcarb
Cyclic peptide-based potent and selective SIRT1/2 dual inhibitors harboring Nε-thioacetyl-lysine
Keywords: β-NAD+; β-nicotinamide adenine dinucleotide; MBHA; 4-methylbenzhydrylamine; SPPS; solid phase peptide synthesis; DMF; N,N-dimethylformamide; TFA; trifluoroacetic acid; DCM; dichloromethane; HBTU; 2-(1H-benzotriazole-1-yl)-1,1,3,3-tetramethylaminium hexa
Development of BPPO-based anion exchange membranes for electrodialysis desalination applications
Keywords: BPPO; N-methylmorpholine; Ion exchange capacity; Anion exchange membrane; Electrodialysis;
Novel double prodrugs of the iron chelator N,Nâ²-bis(2-hydroxybenzyl)ethylenediamine-N,Nâ²-diacetic acid (HBED): Synthesis, characterization, and investigation of activation by chemical hydrolysis and oxidation
Keywords: Iron; Double prodrug; Prochelator; Oxidative stress; Boronic acid; Chelation therapy; ROS; reactive oxygen species; DFO; desferrioxamine B; HBED; N,Nâ²-bis(2-hydroxybenzyl)ethylenediamine-N,Nâ²-diacetic acid; NMM; N-methylmorpholine; EDTA; ethylenediami
Development, synthesis and structure-activity-relationships of inhibitors of the macrophage infectivity potentiator (Mip) proteins of Legionella pneumophila and Burkholderia pseudomallei
Keywords: Mip; macrophage infectivity potentiator; PPIase; peptidyl-prolyl cis/trans isomerase; LpMip; L. pneumophila Mip; BpMip; B. pseudomallei Mip; SAR; structure-activity relationship; HSQC; Heteronuclear Single Quantum Coherence; NMM; N-methylmorpholine; DIP
Structure-activity relationship study using peptide arrays to optimize Api137 for an increased antimicrobial activity against Pseudomonas aeruginosa
Keywords: Apidaecin; Gram-negative bacterium; Proline-rich antimicrobial peptide (PrAMP); Pseudomonas aeruginosa; SPOT synthesis; AMP; antimicrobial peptide; DIC; N,Nâ²-diisopropylcarbodiimide; DIPEA; N-ethyldiisopropylamine; DMAP; 4-dimethylaminopyridine; gu; N,N
Structure-kinetics relationships of Capadenoson derivatives as adenosine A1 receptor agonists
Keywords: Residence time; Structure-affinity relationships; Structure-kinetics relationships; Adenosine A1 receptor; Extracellular loops; ADA; adenosine deaminase; Ac; acetyl; BCA; bicinchoninic acid; BEDROC; Boltzmann-enhanced discrimination of receiver-operating
Blood-brain transfer and antinociception of linear and cyclic N-methyl-guanidine and thiourea-enkephalins
Keywords: Blood-brain barrier (BBB) transport (influx/efflux); Antinociceptive activity; Linear/cyclic enkephalin analogs; In vivo mouse models; AUC; area under the curve; Alloc; allyloxycarbonyl; BBB; blood-brain barrier; Boc; tertButyloxycarbonyl; BSA; bovine
Chimeric derivatives of functionalized amino acids and α-aminoamides: Compounds with anticonvulsant activity in seizure models and inhibitory actions on central, peripheral, and cardiac isoforms of voltage-gated sodium channels
Keywords: AAA; α-aminoamide; ASD; antiseizure drug; ASP; Anticonvulsant Screening Program; CAD; catecholamine A-differentiated; CNS; central nervous system; ED50; effective dose (50%); FAA; functionalized amino acid; IBCF; isobutyl chloroformate; IC50; concentrati
Synthetic tripeptides as alternate substrates of murein peptide ligase (Mpl)
Keywords: Escherichia coli; Mpl; Murein peptide ligase; Peptidoglycan recycling; Tripeptide substrates; Abu; 2-aminobutyric acid; AcOH; acetic acid; Apm; 2-aminopimelic acid; A2pm; 2,6-diaminopimelic acid; Bn; benzyl; Boc; t-butyloxycarbonyl; DCC; N,Nâ²-dicyclohex
New α-adrenergic property for synthetic MTβ and CM-3 three-finger fold toxins from black mamba
Keywords: Muscarinic toxin; Muscarinic receptor; Adrenergic toxin; Adrenoceptor; Three-finger fold toxin; GPCRs; GPCR; G-protein coupled receptor; mAChRs; muscarinic acetylcholine receptors; MTs; muscarinic toxins; NMS; N-methylscopolamine; HCTU; 2-(6-Chloro-1H-ben
The pro-apoptotic action of new analogs of the insect gonadoinhibiting peptide Neb-colloostatin: Synthesis and structure-activity studies
Keywords: Ach; 1-aminocyclohexane-1-carboxylic acid; Acp; 1-aminocyclopentane-1-carboxylic acid; CD; circular dichroism; DMF; dimethylformamide; EDT; 1,2-ethanedithiol; Fmoc; 9-fluorenylmethoxycarbonyl; HBTU; O-benzotriazole-N,N,Nâ²,Nâ²-tetramethyl-uronium-hexafl
Linear and cyclic glycopeptide as HIV protease inhibitors
Keywords: HIV-1 protease; Linear and cyclic glycopeptides; Solid and solution peptide synthesis; Molecular docking; AIDS; acquired immunodeficiency syndrome; CTC; 2-chlorotrityl chloride; DCM; dichloromethane; DIPEA; N,N-diisopropyl ethylamine; DMF; N,N-dimethylfor
Proteasome inhibitors for cancer therapy
Keywords: BOP; (benzotriazol-1-yloxy)tris(dimethylamino)phosphonium hexafluorophosphate; DMSO; dimethyl sulfoxide; HMPA; hexamethyl phosphoramide; HOBt; 1-hydroxybenzotriazole; NMM; N-methylmorpholine; DMF; N,N-dimethyformamide; LDA; lithium diisopropylamide; THF;
An efficient route to VEGF-like peptide porphyrin conjugates via microwave-assisted 'click-chemistry'
Keywords: Porphyrins; Angiogenesis; Click-chemistry; Microwaves; PDT; Cyclic peptide; Abs301; absorbance at 301Â nm; AcOH; acetic acid; All; allyl; Boc; tert-butoxycarbonyl; Da; dalton; DIEA; N,N-diisopropylethylamine; DMAc; N,N-dimethylacetamide; DMF; N,N-dimethyl
Synthesis of chiral threefold and sixfold functionalized macrocyclic imidazole peptides
Keywords: Amino acids; Cyclization; Imidazoles; Macrocycles; Peptidomimetics; Bn; benzyl; Boc; tert-butyloxycarbonyl; DCM; dichloromethane; DMF; N,N-dimethylformamide; NMM; N-methylmorpholine; PhtN; phthalimido; PyBOP; benzotriazole-1-yloxytrispyrrolidinophosphoniu
Densities, viscosities, and excess properties of (N-methylmorpholine + cyclohexane, + benzene, and + toluene) at T = (298.15, 303.15, 313.15, 323.15) K
Keywords: Density; Viscosity; N-Methylmorpholine; Excess molar volumes; Viscosity deviation; Binary mixtures
Synthesis, SAR and in vitro evaluation of new cyclic Arg-Gly-Asp pseudopentapeptides containing a s-cis peptide bond as integrin αvβ3 and αvβ5 ligands
Keywords: All; allyl; DIC; N,Nâ²-diisopropylcarbodiimide; DIPEA; N,N-diisopropylethylamine; DMAP; 4-dimethylaminopyridine; DMF; N,N-dimethylformamide; Fmoc; 9H-fluoren-9-yl-methyloxycarbonyl; HOBt; 1-hydroxybenzotriazole; NMM; N-methylmorpholine; Pbf; 2,2,4,6,7-pe
Synthesis of thiol-modified peptide nucleic acids designed for post-assembly conjugation reactions
Keywords: Peptide nucleic acid; Conjugation; Solid-phase synthesis; Boc; t-butyloxycarbonyl; Bhoc; benzhydryloxycarbonyl; DTT; dithiothreitol; Fmoc; 9-fluorenylmethyloxycarbonyl; PMB; para-methoxybenzyl; EDC; N-(3-dimethylaminopropyl)-Nâ²-ethylcarbodiimide hydroch
Aspartame analogues containing 1-amino-2-phenylcyclohexanecarboxylic acids (c6Phe). Part 2
Keywords: Strecker; Cyclohexanes; Constrained phenylalanines; Aspartame analogues; Computer-assisted methods; Chiral stationary phase; HPLC resolution; TEA; triethylamine; Cbz; benzyloxycarbonyl; EtOAc; ethyl acetate; MeOH; methanol; NMM; N-Methylmorpholine; OtBu;
Development of resin-to-resin transfer reactions (RRTR) using Sonogashira chemistry
Keywords: Solid-phase organic synthesis; Resin-to-resin transfer reactions; Sonogashira coupling; AIBN; 2,2â²-azobisisobutyronitrile; DIAD; diisopropylazadicarboxylate; DIEA; N,N-diisopropylethylamine; DIPCDI; N,Nâ²-diisopropylcarbodiimide; DMAP; 4-(N,N-dimethyla
Strategies for the efficient synthesis of stimuli-responsive ss-DNA bioconjugates for capture and transfection of plasmid DNA
Keywords: AIBN; 2,2-azoisobutyronitrile; AML; affinity macroligand; Boc; tert. butoxycarbonyl; CHO; Chinese hamster ovary (cells); CST; critical solution temperature; DCM; dichloromethane; DMF; dimethylformamide; Ds; double stranded; EGFP; enhanced green fluorescin
Synthetic approaches to the 2012 new drugs
Keywords: 1,2-DAP; 1,2-diaminopropane; 1,2-DCE; 1,2-dichloroethane; Ac; acetyl; aq; aqueous; B2(pin)2; bis(pinacolato)diboron; BINAP; 2,2â²-bis(diphenylphosphino)-1,1â²-binaphthyl; BOP; benzotriazol-1-yloxytris(dimethylamino)phosphonium hexafluorophospate; CDI; N