Keywords: nAChR، گیرنده استیل کولین نیکوتین; TSLP, thymic stromal lymphopoietin; AD, atopic dermatitis; MAPK, mitogen-activated protein kinase; NF-κB, nuclear factor-κB; ERK, extracellular signal-regulated kinase; nAChR, nicotinic acetylcholine receptor; PI3K, phosphoinositide 3-kinase; AMPK, AMP-ac
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Keywords: nAChR، گیرنده استیل کولین نیکوتین; NAChR, Nicotinic acetylcholine receptor; SSRI, selective serotonin reuptake inhibitor; NRI, selective norepinephrine reuptake inhibitor; FST, forced swim test; NSFT, novelty suppressed feeding test; NE, norepinephrine; TST, tail suspension testNicotinic r
Keywords: nAChR، گیرنده استیل کولین نیکوتین; ACh, Acetylcholine; E/I, excitatory-to-inhibitory; LTD, long-term depression; LTP, long-term potentiation; nAChR, nicotinic acetylcholine receptor; α7KO, α7-nAChR constitutive knockout mouse; O–LM, oriens–lacunosum moleculare; PV, parvalbumin; 5-HT3AR, se
Keywords: nAChR، گیرنده استیل کولین نیکوتین; AC, adenocarcinoma; HAEC, human airway epithelial cell; nAChR, nicotinic acetylcholine receptor; NSCLC, non-small cell lung carcinoma; SCC, squamous cell carcinomaNicotinic receptor; Proliferation; Invasion; Non-small cell lung cancer
Keywords: nAChR، گیرنده استیل کولین نیکوتین; Nicotinic receptor; Nicotine; Non-human primate; Rhesus; Cynomolgus; Macaqueα-CTx, α-conotoxin; GWAS, genome wide association study; NHP, non-human primate; nAChR, nicotinic acetylcholine receptor; SNP, single nucleotide polymorphism
Keywords: nAChR، گیرنده استیل کولین نیکوتین; Acetylcholine; Brain development; Chlorpyrifos; Nicotine; Organophosphate pesticidesACh, acetylcholine; ChAT, choline acetyltransferase; HC3, hemicholinium-3; nAChR, nicotinic acetylcholine receptor; PN, postnatal day
Keywords: nAChR، گیرنده استیل کولین نیکوتین; ACh, acetylcholine; nAChR, nicotinic acetylcholine receptor; PAMs, positive allosteric modulators; Ds, PNU-120596-sensitive desensitization; Di, PNU-120596-insensitive desensitizationSynaptic function; Signal transduction; Molecular biology; Electrophysio
Keywords: nAChR، گیرنده استیل کولین نیکوتین; nAChR, nicotinic acetylcholine receptor; B3LYP, Becke, three-parameter, Lee–Yang–Parr; D-PCM, dielectric polarizable continuum modelPiperazines; Conformational analysis; Computational chemistry
Nicotinic receptor blockade decreases fos immunoreactivity within orexin/hypocretin-expressing neurons of nicotine-exposed rats
Keywords: nAChR، گیرنده استیل کولین نیکوتین; CNS, central nervous system; DA, dopamine; ir, immunoreactivity; nAChR, nicotinic acetylcholine receptor; NAcc, nucleus accumbens; OxA, orexin-A; Ox1R, orexin receptor subtype 1; Ox2R, orexin receptor subtype 2; PBS, phosphate-buffered saline; VTA, ventra
Dissection of N,N-diethyl-N′-phenylpiperazines as α7 nicotinic receptor silent agonists
Keywords: nAChR، گیرنده استیل کولین نیکوتین; ACh, acetylcholine; AcOH, acetic acid; DiEPP, N,N-diethyl-N′-phenylpiperazinium; DiMPP, N,N-dimethyl-N′-phenylpiperazinium; PAM, positive allosteric modulator; PEP, N-phenyl-N′ethylpiperazine; nAChR, nicotinic acetylcholine receptor; TFAA, trifluoroacetic
Differential effects of co-administration of oxotremorine with SCH 23390 on impulsive choice in high-impulsive rats and low-impulsive rats
Keywords: nAChR، گیرنده استیل کولین نیکوتین; HI rat, High-impulsive rat; LI rat, Low-impulsive rat; ACh, Acetylcholine; mAChR, Muscarinic acetylcholine receptor; nAChR, Nicotinic acetylcholine receptor; DA, Dopamine; mPFC, Medial prefrontal cortexOxotremorine; SCH 23390; Impulsive choice; Delay disc
Anxiolytic- and antidepressant-like effects of the methadone metabolite 2-ethyl-5-methyl-3,3-diphenyl-1-pyrroline (EMDP)
Keywords: nAChR، گیرنده استیل کولین نیکوتین; Anxiety; Depression; Nicotinic acetylcholine receptor; Behavior; Rodent; OpiateFST, forced swim task; nAChR, nicotinic acetylcholine receptor; EMDP, 2-ethyl-5-methyl-3,3-diphenyl-1-pyrroline; EDDP, 2-ethylidene-1,5-dimethyl-3,3-diphenylpyrrolidine2-ethyl-
Two mutations in nAChR beta subunit is associated with imidacloprid resistance in the Aphis gossypii
Keywords: nAChR، گیرنده استیل کولین نیکوتین; nAChR, nicotinic acetylcholine receptor; P450, cytochrome P450; ABC transporter, ATP binding cassette transporter; GST, glutathione S-transferase; UGT, UDP-glucuronosyltransferase; NGS, next generation sequencing; 2DE, two-dimentional electrophoresis; IEF
Methadone’s effect on nAChRs—a link between methadone use and smoking?
Keywords: nAChR، گیرنده استیل کولین نیکوتین; αBTX, α-bungarotoxin; DA, dopamine; IPN, interpeduncular nucleus; MHb, medial habenula; nAChR, nicotinic acetylcholine receptor; NRT, nicotine replacement therapy; NAcc, nucleus accumbens; VTA, ventral tegmental areaNicotine; Methadone; Nicotinic acetylch
αS-conotoxin GVIIIB potently and selectively blocks α9α10 nicotinic acetylcholine receptors
Keywords: nAChR، گیرنده استیل کولین نیکوتین; nAChR, nicotinic acetylcholine receptor; ACh, acetylcholine; HPLC, high performance liquid chromatography; SEC, size-exclusion chromatography; TFA, trifluoroacetic acid.Protein purification; Oocyte; Nicotinic receptor; Alpha9 alpha10; Conotoxin
Alpha7 nicotinic receptors as therapeutic targets for Parkinson's disease
Keywords: nAChR، گیرنده استیل کولین نیکوتین; Bcl, B-cell lymphoma; α-BTX, α-bungarotoxin; DMXB, 3-[2,4-dimethoxybenzylidene]anabaseine; LIDs, l-dopa-induced dyskinesias; MLA, methyllycaconitine; nAChR, nicotinic acetylcholine receptor; PC, pheochromocytoma; *, indicates the possible presence of othe
α-conotoxin MrIC is a biased agonist at α7 nicotinic acetylcholine receptors
Keywords: nAChR، گیرنده استیل کولین نیکوتین; nAChR, nicotinic Acetylcholine receptor; PNU120596, N-(5-Chloro-2,4-dimethoxyphenyl)-N′-(5-methyl-3-isoxazolyl)-urea; EDTA, Ethylenediaminetetraacetic acid; HEPES, 4-(2-Hydroxyethyl)piperazine-1-ethanesulfonic acid, N-(2-Hydroxyethyl)piperazine-N′-(2-etha
Reducing inflammation and rescuing FTD-related behavioral deficits in progranulin-deficient mice with α7 nicotinic acetylcholine receptor agonists
Keywords: nAChR، گیرنده استیل کولین نیکوتین; nAChR, nicotinic acetylcholine receptor; FTD, frontotemporal dementia; PGRN, progranulin; LPS, lipopolysaccharide; PFA, paraformaldehyde; IP, intraperitoneal; DAB, 3,3'-diaminobenzidine; GM-CSF, granulocyte macrophage colony-stimulating factorFrontotempor
Combined effect between CHRNB3–CHRNA6 region gene variant (rs6474412) and smoking in psoriasis vulgaris severity
Keywords: nAChR، گیرنده استیل کولین نیکوتین; PV, psoriasis vulgaris; GWAS, genome-wide association studies; PASI, Psoriasis Area and Severity Index; IL13, interleukin-13; nAChR, nicotinic acetylcholine receptor; BMI, body mass index; WHO, World Health Organization; OR, odds ratios; CI, confidence in
α7 nicotinic acetylcholine receptors control cytochrome c release from isolated mitochondria through kinase-mediated pathways
Keywords: nAChR، گیرنده استیل کولین نیکوتین; ACh, acetylcholine; nAChR, nicotinic acetylcholine receptor; cyt c, cytochrome c; MLA, methyllicaconitine; MPTP, mitochondria permeability transition pore; ROS, reactive oxygen species; CaMKII, calcium-calmodulin-dependent kinase; PKC, protein kinase C; P
Synthesis and biological evaluation of both enantiomers of [18F]flubatine, promising radiotracers with fast kinetics for the imaging of α4β2-nicotinic acetylcholine receptors
Keywords: nAChR، گیرنده استیل کولین نیکوتین; AD, Alzheimers’s disease; nAChR, nicotinic acetylcholine receptor; 2-[18F]FA, 2-[18F]fluoro-3-(2(S)-azetidinylmethoxy)pyridine; PET, positron emission tomography; 5-[123I]IA, 5-[123I]-5-iodo-3-(2(S)-azetidinylmethoxy)pyridine; HPLC, high performance liqui
Gymnopilins, a product of a hallucinogenic mushroom, inhibit the nicotinic acetylcholine receptor
Keywords: nAChR، گیرنده استیل کولین نیکوتین; Gymnopilin; Mushroom poisoning; Nicotinic acetylcholine receptor; PC12 cellACh, acetylcholine; DMPP, 1,1-Dimethyl-4-phenylpiperazinium iodide; NGF, nerve growth factor; nAChR, nicotinic acetylcholine receptor; VGCC, voltage-gated Ca2+ channel; cAMP, cycli
Hydrophobic residues at position 10 of α-conotoxin PnIA influence subtype selectivity between α7 and α3β2 neuronal nicotinic acetylcholine receptors
Keywords: nAChR، گیرنده استیل کولین نیکوتین; nAChR, nicotinic acetylcholine receptor; α-Ctxα, -conotoxin; AChBP, acetylcholine binding protein; Abu, aminobuteric acid; Nva, norvaline; Nle, norleucine; Aha, aminoheptanoic acid; Aoa, aminooctanoic acid; Cha, cyclohexylalanine; Nal, naphthylalanine; Bo
Modulation of immune functions in polymorphonuclear neutrophils induced by physostigmine, but not neostigmine, independent of cholinergic neurons
Keywords: nAChR، گیرنده استیل کولین نیکوتین; CAP, cholinergic-anti-inflammatory-pathway; CD11b, Mac-1; CD62l, L-selectin; Ch-I, cholinesterase inhibitors; DHR, dihydrorhodamine; FITC, fluoresceinisothiocyanate; fMLP, n-formyl-methionyl-leucylphenylalanine; nAChR, nicotinic acetylcholine receptor; PI
Investigating nicotinic acetylcholine receptor expression in neonicotinoid resistant Myzus persicae FRC
Keywords: nAChR، گیرنده استیل کولین نیکوتین; nAChR, nicotinic acetylcholine receptor; NNIC, neonicotinoid; IMD, imidacloprid; TMX, thiamethoxam; MLA, methyllycaconitine; SCO, succinate cytochrome C oxidase; ER, endoplasmic reticulum; ‘laboratory control Myzuspersicae’, clone 4106A lab reared since 2
Three-finger toxins, a deadly weapon of elapid venom – Milestones of discovery
Keywords: nAChR، گیرنده استیل کولین نیکوتین; Three-fingered toxins; α-Neurotoxins; Isolation; Structure; Activity; Snake venomα-Bgt, α-bungarotoxin; mAChR, muscarinic acetylcholine receptor; nAChR, nicotinic acetylcholine receptor; TFT, three-finger toxin
The effects of lobeline on α4β2* nicotinic acetylcholine receptor binding and uptake of [18F]nifene in rats
Keywords: nAChR، گیرنده استیل کولین نیکوتین; BBB, blood–brain barrier; B/F, bound-to-free ratio; nAChR, nicotinic acetylcholine receptor; PET, positron emission tomography; 1TCM, one tissue compartment model[18F]nifene; Nicotinic acetylcholine receptor; PET; lobeline; BBB amine transporter; Smoking
The role of estrogen receptor β and nicotinic cholinergic receptors in postpartum depression
Keywords: nAChR، گیرنده استیل کولین نیکوتین; PPD, postpartum depression; ER, estrogen receptor; nAChR, nicotinic acetylcholine receptor; HPA, hypothalamic-pituitary-adrenal; CRH, corticotropin-releasing hormone; PVN, paraventricular nucleus; ACTH, adrenocorticotropic hormone; ERE, estrogen response
Genetic matters: Thirty years of progress using mouse models in nicotinic research
Keywords: nAChR، گیرنده استیل کولین نیکوتین; nAChR, nicotinic acetylcholine receptor; LS, long sleep mice; SS, Short sleep mice; Chrna, genes encoding α subunits of the nAChR; Chrnb, genes encoding β subunits of the nAChRNicotine; Mouse genetics; Knockout mice; Nicotinic acetylcholine receptors; Mut
Isolation and characterization of α-conotoxin LsIA with potent activity at nicotinic acetylcholine receptors
Keywords: nAChR، گیرنده استیل کولین نیکوتین; nAChR, nicotinic acetylcholine receptor; RP-HPLC, reverse phase-high performance liquid chromatography; NMR, nuclear magnetic resonance; ACh, acetylcholine; GPCR, G protein-coupled receptor; FLIPR, fluorometric imaging plate reader; IC50, half-maximal inh
Transcriptional regulation by nicotine in dopaminergic neurons
Keywords: nAChR، گیرنده استیل کولین نیکوتین; DAVID, Database for Annotation, Visualization and Integrated Discovery; ER, endoplasmic reticulum; FPKM, fragments per kilobase per million mapped reads; IPA, Ingenuity Pathway Analysis; nAChR, nicotinic acetylcholine receptor; PD, Parkinson's disease; SN
Multiple CNS nicotinic receptors mediate l-dopa-induced dyskinesias: Studies with parkinsonian nicotinic receptor knockout mice
Keywords: nAChR، گیرنده استیل کولین نیکوتین; α-CtxMII, α-conotoxinMII; nAChR, nicotinic acetylcholine receptor; *, the possible presence of other subunits in the receptor complexDyskinesias; Nicotine; Nicotinic receptors; Parkinson's disease; Striatum
Dendritic spine alterations in the hippocampus and parietal cortex of alpha7 nicotinic acetylcholine receptor knockout mice
Keywords: nAChR، گیرنده استیل کولین نیکوتین; AD, Alzheimer’s disease; BTNRH, Boys Town National Research Hospital; MLA, methyllycaconitine; nAChR, nicotinic acetylcholine receptor; SEM, standard error of the meanalpha7 nicotinic receptor; hippocampus; dendrite; CA1 region; parietal cortex; cognition
Prenatal dexamethasone augments the sex-selective developmental neurotoxicity of chlorpyrifos: Implications for vulnerability after pharmacotherapy for preterm labor
Keywords: nAChR، گیرنده استیل کولین نیکوتین; ACh, acetylcholine; ANOVA, analysis of variance; ChAT, choline acetyltransferase; GD, gestational day; HC3, hemicholinium-3; nAChR, nicotinic acetylcholine receptor; PN, postnatal dayChlorpyrifos; Cholinergic neurotransmission; Dexamethasone; Glucocortico
A comparative study of the effects of ABT-418 and methylphenidate on spatial memory in an animal model of ADHD
Keywords: nAChR، گیرنده استیل کولین نیکوتین; ADHD, attention deficit hyperactivity disorder; nAChR, nicotinic acetylcholine receptor; MPH, methylphenidate; SHRs, spontaneously hypertensive rats; ABT-418 hydrochloride, 3-methyl-5-[(2S)-1-methyl-2-pyrrolidinyl]isoxazole hydrochlorideAttention deficit
Cholinergic signalling in gut immunity
Keywords: nAChR، گیرنده استیل کولین نیکوتین; ACh, acetylcholine; nAChR, nicotinic acetylcholine receptor; mAChR, muscarinic acetylcholine receptor; TJ, tight junction; ENS, enteric nervous system; LPS, lipopolysaccharide; ChAT, choline acetyltransferase; CrAT, carnitine O-acetyltransferase; AChE, ac
Intrathecal α-conotoxins Vc1.1, AuIB and MII acting on distinct nicotinic receptor subtypes reverse signs of neuropathic pain
Keywords: nAChR، گیرنده استیل کولین نیکوتین; Conotoxin; Pain; Nicotinic; nAChR; Allodynia; IntrathecalAUC, area under curve; eEPSC, evoked excitatory post-synaptic current; nAChR, nicotinic acetylcholine receptor; PNL, partial nerve ligation; PWT, paw withdrawal threshold
Differential metabolism of sulfoximine and neonicotinoid insecticides by Drosophila melanogaster monooxygenase CYP6G1
Keywords: nAChR، گیرنده استیل کولین نیکوتین; SAR, structure activity relationship; CLSFX, chloropyridine-analog of sulfoxaflor; nAChR, nicotinic acetylcholine receptor; IPM, integrated pest managementSulfoximine; Sulfoxaflor; Neonicotinoid; CYP6G1; Insecticide resistance and metabolism; Homology mod
RegIIA: An α4/7-conotoxin from the venom of Conus regius that potently blocks α3β4 nAChRs
Keywords: nAChR، گیرنده استیل کولین نیکوتین; AChBP, acetylcholine-binding protein; CNS, central nervous system; DMSO, dimethyl sulfoxide; DTT, dithiothreitol; EST, expressed sequence tag; GABABR, γ-aminobutyric acid type B receptor; IAM, iodoacetamide; nAChR, nicotinic acetylcholine receptor; PCR, p
Feasibility of [18F]-2-Fluoro-A85380-PET Imaging of Human Vascular Nicotinic Acetylcholine Receptors In Vivo
Keywords: nAChR، گیرنده استیل کولین نیکوتین; arteries; multiple system atrophy; nicotinic acetylcholine receptors; Parkinson's disease; positron emission tomographyCT, computed tomography; JV, jugular vein; MSA, multiple system atrophy; nAChR, nicotinic acetylcholine receptor; PAS, percent active se
Functional expression of the α7 and α4-containing nicotinic acetylcholine receptors on the neonatal rat carotid body
Keywords: nAChR، گیرنده استیل کولین نیکوتین; CB, carotid body; ACh, acetylcholine; nAChR, nicotinic acetylcholine receptor; CA, catecholamineCarotid body; Acetylcholine; Nicotinic acetylcholine receptors; Catecholamines
Changes in glycine receptor subunit expression in forebrain regions of the Wistar rat over development
Keywords: nAChR، گیرنده استیل کولین نیکوتین; ACTB, beta-actin; DA, dopamine; FC, frontal cortex; GAPDH, glyceraldehyde 3-phosphate dehydrogenase; GlyR, glycine receptor; IHC, immunohistochemistry; nAc, nucleus accumbens; nAChR, nicotinic acetylcholine receptor; PFC, prefrontal cortex; qPCR, quantita
Resistance and cross-resistance to the spinosyns – A review and analysis
Keywords: nAChR، گیرنده استیل کولین نیکوتین; IPM, integrated pest management; IRM, insect resistance management; nAChR, nicotinic acetylcholine receptor; RR, resistance ratio; OP, organophosphorus insecticide; MAC, molt accelerating compound; Kdr, knockdown resistanceSpinosyns; Insecticide resistanc
Neuronal nicotinic receptor antagonist reduces anxiety-like behavior in mice
Keywords: nAChR، گیرنده استیل کولین نیکوتین; ACh, acetylcholine; EPM, elevated plus-maze; HPA, hypothalamic–pituitary–adrenal; nAChR, nicotinic acetylcholine receptor; NMDA, N-methyl-d-aspartic acid; OFT, open-field testNicotinic receptor; Anxiety; Lobeline; Mecamylamine; Elevated plus-maze; Mice; M
Structural characterization and agonist binding to human α4β2 nicotinic receptors
Keywords: nAChR، گیرنده استیل کولین نیکوتین; Carb, carbamylcholine; Chol, cholesterol; nAChR, nicotinic acetylcholine receptor; PA, 1,2-diacyl-sn-glycero-3-phosphate; PC, 1,2-diacyl-sn-glycero-3-phosphocholineHuman nicotinic acetylcholine receptors; Torpedo; Structure; Agonist binding; Thermal stabi
Structure–function relationship of conotoxin lt14a, a potential analgesic with low cytotoxicity
Keywords: nAChR، گیرنده استیل کولین نیکوتین; nAChR, nicotinic acetylcholine receptor; DMF, N,N-dimethylformamide; TFA, trifluoroacetic acid; HBTU, 2-(1H-benzotriazol-l-yl) 1,1,3,3-tetrametyluronium hexafluorophosphate; DIPEA, N,N-diisopropylethylamine; MTT, 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenylt
Src family kinase potentiates the activity of nicotinic acetylcholine receptor in rat autonomic ganglion innervating urinary bladder
Keywords: nAChR، گیرنده استیل کولین نیکوتین; SFKs, Src kinases; PTK, protein tyrosine kinase; ACh, acetylcholine; MPG, major pelvic ganglion; nAChR, nicotinic acetylcholine receptor; [Ca2+]i, intracellular calcium ion concentrationMajor pelvic ganglia; Nicotinic acetylcholine receptor; Src family ki
An extracellular RRR motif flanking the M1 transmembrane domain governs the biogenesis of homomeric neuronal nicotinic acetylcholine receptors
Keywords: nAChR، گیرنده استیل کولین نیکوتین; ACh, acetylcholine; α3RRR, α3L210R; β4RRR, β4K208R/K210R; Bgtx, bungarotoxin; EB, epibatidine; ERAD, endoplasmic reticulum associated degradation; LGIC, ligand-gated ion channel; nAChR, nicotinic acetylcholine receptor; PCR, polymerase chain reaction; WT,
Effect of co-administration of varenicline and antidepressants on extracellular monoamine concentrations in rat prefrontal cortex
Keywords: nAChR، گیرنده استیل کولین نیکوتین; aCSF, artificial cerebrospinal fluid; DA, dopamine; MAO-I, monoamine oxidase inhibitor; mPFC, medial prefrontal cortex; MRM, multiple-reaction-monitoring; nAChR, nicotinic acetylcholine receptor; NE, norepinephrine; SSRI, selective serotonin reuptake inhi
Acute in vivo nicotine administration enhances synchrony among dopamine neurons
Keywords: nAChR، گیرنده استیل کولین نیکوتین; ACh, acetylcholine; DHβE, dihydro-β-erythroidine; DA, dopamine; ISI, interspike interval; nAChR, nicotinic acetylcholine receptor; NAc, nucleus accumbens; SNc, substantia nigra compacta; VTA, ventral tegmental areaNicotinic acetylcholine receptors; Mesoli