Keywords: OCT، حمل و نقل کاتیونی آلی; BCRP, breast cancer related protein; CML, chronic myeloid leukemia; IMA, Imatinib; P-gP, P-glycoprotein; OCT, organic cation transporter; TKI, tirosine kinase inhibitorCML; Imatinib resistance; Therapeutic interruptions; Membrane drug transporters; P-glyc
مقالات ISI OCT، حمل و نقل کاتیونی آلی (ترجمه نشده)
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Keywords: OCT، حمل و نقل کاتیونی آلی; pharamcokinetics; drug interaction; intestinal absorption; peptide transporters; renal excretion; organic anion transporters; DDIs, drug-drug interactions; PEPT, H+/peptide transporter; OAT, organic anion transporter; OCT, organic cation transporter; ACEI
Involvement of organic cation transporter 1 and CYP3A4 in retrorsine-induced toxicity
Keywords: OCT، حمل و نقل کاتیونی آلی; PAs, pyrrolizidine alkaloids; RTS, retrorsine; CYP, cytochrome P450; OCT, organic cation transporter; MDCK, Madin–Darby canine kidney; PCRH, primary cultured rat hepatocytes; SLC, solute carrier; MATE, multidrug and toxin extrusion; P-gp/MDR1, P-glycoprot
In-cell Western™ detection of organic cation transporters in bronchial epithelial cell layers cultured at an air–liquid interface on Transwell® inserts
Keywords: OCT، حمل و نقل کاتیونی آلی; ICW, in-cell Western™; NIR, near infra-red; OCT, organic cation transporter; ALI, air liquid interface; NHBE, normal human bronchial epithelial; FBS, foetal bovine serum; PFA, paraformaldehyde; BSA, bovine serum albumin; GAPDH, glyceraldehyde-3-phosphate
Transfer of metformin across the rat placenta is mediated by organic cation transporter 3 (OCT3/SLC22A3) and multidrug and toxin extrusion 1 (MATE1/SLC47A1) protein
Keywords: OCT، حمل و نقل کاتیونی آلی; GDM, gestational diabetes mellitus; MATE, multidrug and toxin extrusion proteins; MPP+, 1-methyl-4-phenylpyridinium iodide; OCT, organic cation transporter; SLC, solute carrierMetformin; Organic cation transporter 3; Multidrug and toxin extrusion 1; Place
Enhancement effect of P-gp inhibitors on the intestinal absorption and antiproliferative activity of bestatin
Keywords: OCT، حمل و نقل کاتیونی آلی; P-gp; Bestatin; Intestinal absorption; Antiproliferative activityDDI, drug–drug interaction; P-gp, P-glycoprotein; PEPT, H+/peptide transporter; OAT, organic anion transporter; OCT, organic cation transporter; MRP2, multidrug resistance-associated protein
Cisplatin-induced ototoxicity: Transporters playing a role in cisplatin toxicity
Keywords: OCT، حمل و نقل کاتیونی آلی; NF-kB, nuclear transcription factor-kappa B; TNF-α, tumour necrosis factor-α; Ctr, copper transporter; Atox1, anti-oxidant 1; OCT, organic cation transporter; SLC, solute carrier; TRP, transient receptor potential; IP3R, inositol trisphosphate receptor; M
Organic cation transporter OCT/SLC22A and H+/organic cation antiporter MATE/SLC47A are key molecules for nephrotoxicity of platinum agents
Keywords: OCT، حمل و نقل کاتیونی آلی; OCT, organic cation transporter; MATE, multidrug and toxin extrusion; Ctr1, copper transporter 1; DACH, diaminocyclohexaneCisplatin; Renal handling; Pharmacokinetics; Drug transporter; Copper transporter Ctr1
Unfaithful neurotransmitter transporters: Focus on serotonin uptake and implications for antidepressant efficacy
Keywords: OCT، حمل و نقل کاتیونی آلی; DA, dopamine; DAT, dopamine transporter; KO, knockout; MDMA, 3,4-methylenedioxymethamphetamine; NE, norepinephrine; NET, norepinephrine transporter; OCT, organic cation transporter; PMAT, plasma monoamine transporter; SSRI, selective serotonin reuptake in
Increase in P-glycoprotein accompanied by activation of protein kinase Cα and NF-κB p65 in the livers of rats with streptozotocin-induced diabetes
Keywords: OCT، حمل و نقل کاتیونی آلی; ABC, ATP-binding cassette; MDR, multidrug resistance; P-gp, P-glycoprotein; STZ, streptozotocin; MRP, multidrug resistance-associated protein; OAT, organic anion transporter; OCT, organic cation transporter; PKC, protein kinase C; NF-κB, nuclear factor κB
Physiological and pharmacokinetic roles of H+/organic cation antiporters (MATE/SLC47A)
Keywords: OCT، حمل و نقل کاتیونی آلی; MATE, multidrug and toxin extrusion; MPP, 1-methyl-4-phenylpyridinium; NMN, N1-methylnicotinamide; OCT, organic cation transporter; OCTN, novel organic cation transporter; SLC, solute carrier; SNP, single nucleotide polymorphism; TEA, tetraethylammoniumH+
In vivo relevance of Mrp2-mediated biliary excretion of the Amanita mushroom toxin demethylphalloin
Keywords: OCT، حمل و نقل کاتیونی آلی; DIDS, diisothiocyanostilbenedisulfonat; DMP, Demethylphalloin; OATP/Oatp, human/rat Organic anion transporting polypeptide; Oct, Organic cation transporter; Oat, Organic anion transporter; MRP/Mrp, human/rat multidrug resistance-associated protein; Mdr1,
Comparison of permeation enhancing strategies for an oral factor Xa inhibitor using the Caco-2 cell monolayer model
Keywords: OCT، حمل و نقل کاتیونی آلی; Papp, apparent permeability; P-gp, P-glycoprotein; OCT, organic cation transporter; BCS, Biopharmaceutics Classification System; PSA, polar surface area; MCGs, medium chain glycerides; ABC, ATP-binding cassette; CTS, chitosan; TEER, transepithelial electr
Expression of transporters potentially involved in the targeting of cytostatic bile acid derivatives to colon cancer and polyps
Keywords: OCT، حمل و نقل کاتیونی آلی; ASBT, apical sodium-dependent bile salt transporter; MDR, multidrug resistance protein; MRP, multidrug resistance-associated protein; OATP, organic anion transporting polypeptide; OCT, organic cation transporter; OST, organic solute transporter; TC, tauro
Alterations in transporter expression in liver, kidney, and duodenum after targeted disruption of the transcription factor HNF1α
Keywords: OCT، حمل و نقل کاتیونی آلی; Cyp, cytochrome P450; HNF, hepatocyte nuclear factor; MODY-3, maturity onset diabetes of the young type 3; Mrp, multidrug resistance-associated protein; Mdr, multidrug resistance protein; Oat, organic anion transporter; Oct, organic cation transporter; NI
Drug and Bile Acid Transporters in Rosuvastatin Hepatic Uptake: Function, Expression, and Pharmacogenetics
Keywords: OCT، حمل و نقل کاتیونی آلی; HMG-CoA, 3-hydroxy-3-methylglutaryl coenzyme A; NTCP, sodium-dependent taurocholate cotransporting polypeptide; OATP, organic anion transporting polypeptide; OCT, organic cation transporter; SNP, single nucleotide polymorphism.