Keywords: پریازولوپیریمیدین; 8-Aminoquinoline; Pyrazolopyrimidine; Plasmodium falciparum; Structure activity relationship; Hybridization;
مقالات ISI پریازولوپیریمیدین (ترجمه نشده)
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Discovery of pyrazolopyrimidine derivatives as novel inhibitors of ataxia telangiectasia and rad3 related protein (ATR)
Keywords: پریازولوپیریمیدین; ATR; Pyrazolopyrimidine; DNA damage; PI3K; HTS;
A novel solid-phase synthetic method for production of N-alkyl-4-alkylamino-1-aryl-1H-pyrazolo[3,4-d]pyrimidine-6-carboxamide library
Keywords: پریازولوپیریمیدین; Screening library; Privileged structure; Heterocycle; Pyrazolopyrimidine; Solid-phase organic synthesis;
New structure–activity relationships of N-acetamide substituted pyrazolopyrimidines as pharmacological ligands of TSPO
Keywords: پریازولوپیریمیدین; FXXXIMZIANBQLJ-UHFFFAOYSA-NTSPO; Pyrazolopyrimidine; SAR; Cancer; Precision medicine
Identification of novel GLUT inhibitors
Keywords: پریازولوپیریمیدین; DXJIXNIYGMNIFL-UHFFFAOYSA-NGLUT1 inhibitor; Pyrazolopyrimidine; Warburg effect; Structure–activity relationships (SAR); In vitro pharmacokinetics (PK)
Synthesis and mechanistic aspects of 2-anilinonicotinyl-pyrazolo[1,5-a]pyrimidine conjugates that regulate cell proliferation in MCF-7 cells via estrogen signaling
Keywords: پریازولوپیریمیدین; Estrogen receptors; Cell cycle; Cyclin D1; Bcl-2; Pyrazolopyrimidine;
Discovery of pyrazolopyrimidine phosphodiesterase 10A inhibitors for the treatment of schizophrenia
Keywords: پریازولوپیریمیدین; Schizophrenia; Antipsychotic activity; Cognitive improvement; Phosphodiesterase 10A; Fragment-based drug discovery; Pyrazolopyrimidine; Rational design; Positron emission tomography
Development of small molecules targeting the pseudokinase Her3
Keywords: پریازولوپیریمیدین; Her3; Pseudokinase; Hydrophobic tagging; Cancer; Pyrazolopyrimidine;
The discovery of potent, orally bioavailable pyrazolo and triazolopyrimidine CXCR2 receptor antagonists
Keywords: پریازولوپیریمیدین; CXCR2; Chemokines; Pyrazolopyrimidine; Triazolopyrimidine; Neutrophils; COPD;
Diphenylpyrroles: Novel p53 activators
Keywords: پریازولوپیریمیدین; Pyrroles; Triazolopyrimidine; Benzimidazopyrimidine; Pyrazolopyrimidine; p53-specific ubiquitin E3 ligase HDM2
Development of potent and selective Plasmodium falciparum calcium-dependent protein kinase 4 (PfCDPK4) inhibitors that block the transmission of malaria to mosquitoes
Keywords: پریازولوپیریمیدین; Plasmodium falciparum; PfCDPK4; PfCDPK1; Pyrazolopyrimidine; Exflagellation; ACT; artemisinin combination therapy; ATP; adenosine triphosphate; Boc; tert-butyloxycarbonyl; CAMKII; Ca2+/calmodulin-dependent protein kinase II; CDPK1; calcium-dependent prote
Synergistic effect of Wnt modulatory small molecules and an osteoinductive ceramic on C2C12 cell osteogenic differentiation
Keywords: پریازولوپیریمیدین; ALP; alkaline phosphatase; hMSC; human mesenchymal stem cell; TCP; tricalcium phosphate; THQ; tetrahydroquinoline; PP; pyrazolopyrimidine; Ph; phenyl; C2C12; Mesenchymal stromal cells; Tricalcium phosphate ceramic; Small molecules; Wnt; Osteogenesis;
Sc(OTf)3 promoted multicomponent synthesis of fluorescent imidazo[1,2-c]pyrazolo[3,4-d]pyrimidine
Keywords: پریازولوپیریمیدین; Multicomponent reactions (MCRs); Scandium triflate; Pyrazolopyrimidine; Imidazo[12-c]pyrazolo[3,4-d]pyrimidine; Fluorescent probes;
A scalable approach to diaminopyrazoles using flow chemistry
Keywords: پریازولوپیریمیدین; Flow chemistry; Sequential flow process; Aminopyrazole; Pyrazolopyrimidine; Single mode microwave;
Design and evaluation of a series of pyrazolopyrimidines as p70S6K inhibitors
Keywords: پریازولوپیریمیدین; p70S6K inhibitor; Pyrazolopyrimidine; PI3K pathway; Cancer
Pyrazolopyrimidines as dual Akt/p70S6K inhibitors
Keywords: پریازولوپیریمیدین; p70S6K inhibitor; Akt inhibitor; Pyrazolopyrimidine; PI3K pathway; Cancer
Synthesis, SAR and biological evaluation of 1,6-disubstituted-1H-pyrazolo[3,4-d]pyrimidines as dual inhibitors of Aurora kinases and CDK1
Keywords: پریازولوپیریمیدین; Aurora kinase; Cyclin dependent kinase; Cell cycle arrest; Pyrazolopyrimidine; Cytotoxicity;
One-pot synthesis of 2-alkyl-7-amino-5-aryl-pyrazolo[1,5-a]pyrimidine-6-carbonitriles via a domino three-component condensation-oxidation reaction
Keywords: پریازولوپیریمیدین; Pyrazolopyrimidine; 3-aminopyrazole; Malononitrile; Domino reaction
2-Substituted 5,6-dimethyl-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines: New series of highly potent and specific serotonin 5-HT6 receptor antagonists
Keywords: پریازولوپیریمیدین; Phenylsulfonyl; Pyrazolopyrimidine; 5-HT6 receptor antagonist; SAR5-HT6R, serotonin 5-HT6 receptor; 5-HT2BR, serotonin 5-HT2B receptor; DMPSPP, 5,7-dimethyl-3-phenylsulfonyl-pyrazolo [1,5-a] pyrimidine; TPSA, topological polar surface area; CNS, central n
Synthesis and antimicrobial activity of novel pyrazolo[3,4-d]pyrimidin derivatives
Keywords: پریازولوپیریمیدین; Pyrazolopyrimidine; Antimicrobial activity; Agar diffusion method
Synthesis and antimicrobial activities of some new thiazole and pyrazole derivatives based on 4,5,6,7-tetrahydrobenzothiophene moiety
Keywords: پریازولوپیریمیدین; Thiophene; Thiazole; Triazine; Pyrazolopyrimidine; Antimicrobial evaluation
Assessment of the putative binding conformation of a pyrazolopyridine class of inhibitors of MAPKAPK2 using computational studies
Keywords: پریازولوپیریمیدین; MAPKAPK2 (MK2); Kinase; Pyrazolopyridines; Pyrazolopyrimidine;
Synthesis of [125I]iodoDPA-713: A new probe for imaging inflammation
Keywords: پریازولوپیریمیدین; TSPO; translocator protein; [125I]iodoDPA-713; N,N-diethyl-2-[2-(3-[125I]iodo-4-methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl]acetamide; PK11195; N-butan-2-yl-1-(2-chlorophenyl)-N-methylisoquinoline-3-carboxamide; SPECT; single photon emission
EGF promotes invasion by PANC-1 cells through Rac1/ROS-dependent secretion and activation of MMP-2
Keywords: پریازولوپیریمیدین; DPI; diphenyleneiodonium; EGF; epidermal growth factor; EGFR; EGF receptor; MMP; matrix metalloproteinase; NADPH; nicotinamide adenine dinucleotide phosphate; PI3K; phosphatidylinositol 3-kinase; PP2; pyrazolopyrimidine; ROS; reactive oxygen species; PANC
One-pot synthesis and antibacterial activities of pyrazolo[4′,3′:5,6]pyrido[2,3-d]pyrimidine-dione derivatives
Keywords: پریازولوپیریمیدین; 1H-Pyrazol-5-amines; Barbituric acid; Pyrimidopyrimidine; Thiobarbituric acid; Pyrazolopyrimidine
Synthesis of disazo pyrazolo[1,5-a]pyrimidines
Keywords: پریازولوپیریمیدین; Pyrazolopyrimidine; Disazo; Intermolecular cyclization; Diazo-coupling reaction; Condensation reaction
3D-QSAR and molecular docking studies on pyrazolopyrimidine derivatives as glycogen synthase kinase-3β inhibitors
Keywords: پریازولوپیریمیدین; Glycogen synthase kinase-3 (GSK-3); Diabetes mellitus; Pyrazolopyrimidine; 3D-QSAR; CoMFA; CoMSIA; Molecular docking
Pyrazolo[1,5-a]pyrimidin-7-yl phenyl amides as novel anti-proliferative agents: parallel synthesis for lead optimization of amide region
Keywords: پریازولوپیریمیدین; Pyrazolopyrimidine; Anti-proliferative agents; Anti-cancer agents; Parallel synthesis;
Synthesis and in vivo evaluation of a novel peripheral benzodiazepine receptor PET radioligand
Keywords: پریازولوپیریمیدین; Pyrazolopyrimidine; Peripheral benzodiazepine receptor; Carbon-11; PET
Bombesin and angiotensin II rapidly stimulate Src phosphorylation at Tyr-418 in fibroblasts and intestinal epithelial cells through a PP2-insensitive pathway
Keywords: پریازولوپیریمیدین; Autophosphorylation; Tyrosine kinase; G protein-coupled receptor; Pyrazolopyrimidine; Intestinal epithelial cells; Fibroblasts; FAK;