Keywords: ALT; alanine aminotransferase; ANOVA; analysis of variance; CCl4; carbon tetrachloride; COX-2; cyclooxygenase-2; DLS; dynamic light scattering; ESI; electrospray ionization; GI; gastrointestinal; 6G; 6-gingerol; 8G; 8-gingerol; GE; ginger extract; HPMC; h
مقالات ISI (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: AOT; dioctyl sulfoccinate; CEH; cholesteryl ester hydrolase; CPP; cell penetrating peptide; DL; drug load; EE; encapsulation efficiency; FA; Fatty Acid; GI; Gastrointestinal; GSH; reduced glutathione; HIP; hydrophobic ion pairing; HPH; high pressure homog
Keywords: C; chitosan; CCMV; cowpea chlorotic mottle virus; CPMV; cowpea mosaic virus; CF; cystic fibrosis; LC; long chain; MC; medium chain; NAC; N-acetylcysteine; NL; no lipids; PLGA; poly(lactic-co-glycolic acid); PCL; periciliary layer; PGA; 6 phosphoglucuronic
Keywords: BCA; bicinchoninic acid; BRO; bromelain; CYS; cysteine; DNA; deoxyribonucleic acid; EDAC; ethyl-dimethylaminopropyl-carbodiimide; LMWH; low molecular weight heparin; MCS; mucolytic carrier system; MECS; mucolytic enzyme decorated carrier systems; NHS; N-h
Keywords: Drug delivery; Lipid carrier; Nanotechnology; Nanocarrier; Controlled release; NEMS; Nano electromechanical systems; MEMS; Micro-electromechanical systems; NE; Nanoemulsions; NPs; Nanoparticles; QD; Quantum dots; PLA; Polylactic acid; PGA; Polyglycolic ac
Keywords: SEDDS; Vaginal application; Curcumin; Mucus interaction; Spreading; Mucus permeation;
Keywords: Liquisolid; Dissolution enhancement; Leflunomide; SEDDS; BCS class II;
Keywords: Trypsin; α-Chymotrypsin; Pemulen; Carbopol Ultrez; Emulsifier; SEDDS;
Keywords: Self-emulsification; SEDDS; Solidification; Adsorption; Granulation; Spray drying;
Keywords: i.v; Nanocrystals; Nanosuspension; High fat diet; Oil formulation; s.c.; SEDDS;
Keywords: Drug delivery; In vitro digestion; Lipase; Lipids; Lipolysis; o/w emulsions; CEH; pancreatic carboxyl ester hydrolase; GI; gastrointestinal; GL; gastric lipase; LBF; lipid-based formulation; LC; long chain acylglycerols; MC; medium chain acylglycerols; P
Keywords: ABC; ATP-binding cassette; BCS; Biopharmaceutics Classification System; BDDCS; Biopharmaceutics Drug Disposition Classification System; EPAR; European Public Assessment Report; FDA; Food and Drug Administration Agency; SEDDS; Self Emulsifying Drug Deliver
Keywords: Hydrogel system; Lovastatin; SEDDS; Lipids; Factorial design;
Keywords: SEDDS; SMEDDS; Lipid formulations; Medium chain mono- and glycerides; Poorly water-soluble compounds
Keywords: LFCS Consortium; lipid-based drug delivery systems; SEDDS; drug solubilization; in vitro digestion testing; solubility; bioavailability; in vitro models; precipitation; supersaturation;
Design and evaluation of SEDDS exhibiting high emulsifying properties
Keywords: Self-emulsifying drug delivery systems; SEDDS; Emulsifying properties; Log D SEDDS/Water; Emulsification time;
Mucus permeating self-emulsifying drug delivery systems (SEDDS): About the impact of mucolytic enzymes
Keywords: Mucolytic enzymes; Bromelain; Papain; Trypsin; Mucus permeation; SEDDS;
Do drug release studies from SEDDS make any sense?
Keywords: Self-emulsifying drug delivery systems; SEDDS; Drug release; Partition coefficient;
Glyceryl ester surfactants: Promising excipients to enhance the cell permeating properties of SEDDS
Keywords: Cell permeation enhancer; Cell uptake; Glycerol ester surfactants; SEDDS; Curcumin;
Development of self-emulsifying drug delivery systems (SEDDS) for ciprofloxacin with improved mucus permeating properties
Keywords: SEDDS; Ciprofloxacin; Pulmonary infections; Cystic fibrosis sputum; Mucus permeation; Particle tracking; Minimal inhibitory concentration;
Oral Delivery of Highly Lipophilic, Poorly Water-Soluble Drugs: Self-Emulsifying Drug Delivery Systems to Improve Oral Absorption and Enable High-Dose Toxicology Studies of a Cholesteryl Ester Transfer Protein Inhibitor in Preclinical Species
Keywords: solubility; absorption; bioavailability; lipid-based formulations; self-emulsifying; preclinical species; AUC; area under the curve; GI tract; gastrointestinal tract; ND; not determined; IV; intravenous; SEDDS; self-emulsifying drug delivery systems; SMED
Assessment of cell viability and permeation enhancement in presence of lipid-based self-emulsifying drug delivery systems using Caco-2 cell model: Polysorbate 80 as the surfactant
Keywords: LBDDS; lipid-based drug delivery system; LBSEDDS; lipid-based self-emulsifying drug delivery system; SEDDS; self-emulsifying drug delivery system; SMEDDS; self-microemulsifying drug delivery system; MTT; 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazoliu
Development of solid SEDDS, VI: Effect of precoating of Neusilin® US2 with PVP on drug release from adsorbed self-emulsifying lipid-based formulations
Keywords: SEDDS; Solid dosage forms; Silicates; Lipid based formulations; PVP; Pore size distribution; NCE's; new chemical entities; GI; gastro-intestinal; SEDDS; self-emulsifying drug delivery systems; SMEDDS; self-microemulsifying drug delivery systems;
Cytotoxicity assessment of lipid-based self-emulsifying drug delivery system with Caco-2 cell model: Cremophor EL as the surfactant
Keywords: LBDDS; Lipid-based drug delivery system; LBSEDDS; Lipid-based self-emulsifying drug delivery system; SEDDS; Self-emulsifying drug delivery system; SMEDDS; Self-microemulsifying drug delivery system; MTT; (3-(4.5-Dimethylthiazol-2-yl)-2.5-diphenyltetrazoli
Self-emulsifying phospholipid pre-concentrates (SEPPs) for improved oral delivery of the anti-cancer genistein: Development, appraisal and ex-vivo intestinal permeation
Keywords: GEN; genistein; SEPP; self-emulsifying phospholipid pre-concentrate; SNEDDS; self-nanoemulsifying drug delivery system; SEDDS; self-emulsifying drug delivery system; S/CO; surfactant/co-surfactant mixture; PC; phosphatidylcholine; Genistein; Self-emulsify
50Â years of oral lipid-based formulations: Provenance, progress and future perspectives
Keywords: AP; Aqueous phase; API; Active pharmaceutical ingredient; b-r-o-5; Beyond rule-of-five; BS; Bile salt; DG; Diglyceride; FA; Fatty acid; GIT; Gastrointestinal tract; IL; Ionic liquid; LBF; Lipid based formulation; LCT; Long chain triglyceride; LFCS; Lipid
Using in situ Raman spectroscopy to study the drug precipitation inhibition and supersaturation mechanism of Vitamin E TPGS from self-emulsifying drug delivery systems (SEDDS)
Keywords: SEDDS; Raman spectroscopy; Indomethacin; Vitamin E TPGS; Probucol;
Role of solid carriers in pharmaceutical performance of solid supersaturable SEDDS of celecoxib
Keywords: SEDDS; Solid carrier; Silicon dioxide; Porosity; Surface area; Hydrophobicity-hydrophilicity; In vitro drug release;
A novel approach for the development and optimization of self emulsifying drug delivery system using HLB and response surface methodology: Application to fenofibrate encapsulation
Keywords: SEDDS; HLB; Box-Behnken; Optimization; Fenofibrate;
Novel semisolid SNEDDS based on PEG-30-dipolyhydroxystearate: Development and characterization
Keywords: %T; percentage transmittance; 1H NMR; proton nuclear magnetic resonance; aN; hyperfine coupling constant; D2O; deuterium oxide; dB; decibel; d-DMSO; deuterated dimethyl sulfoxide; DLS; dynamic light scattering; DPHS; Cithrol® DPHS; DSC; differential scan
Choice of Nonionic Surfactant Used to Formulate Type IIIA Self-Emulsifying Drug Delivery Systems and the Physicochemical Properties of the Drug Have a Pronounced Influence on the Degree of Drug Supersaturation that Develops During In Vitro Digestion
Keywords: supersaturation; precipitation; SEDDS; poorly water-soluble drugs; LFCS; lipids; surfactants; in vitro models; SRM;
Interactions between human multidrug resistance related protein (MRP2; ABCC2) and excipients commonly used in self-emulsifying drug delivery systems (SEDDS)
Keywords: Excipients; MRP2; Caco-2; Membrane vesicles transport assay; SEDDS;
Novel self-emulsifying formulation of quercetin for improved in vivo antioxidant potential: Implications for drug-induced cardiotoxicity and nephrotoxicity
Keywords: QT; quercetin; CyA; cyclosporin A; Dox; doxorubicin; SEDDS; self-emulsifying drug delivery system; PDI; polydispersity index; MTT; 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide; DPPH; 1,1-diphenyl-2-picrylhydrazyl; QT-SEDDS; quercetin-loade
A novel lipid-based solid dispersion for enhancing oral bioavailability of Lycopene – In vivo evaluation using a pig model
Keywords: Lycopene bioavailability; Lipid-based formulation; SEDDS; Solid dispersions; Gelucire 44/14; Pig model
Optimized nanoemulsifying systems with enhanced bioavailability of carvedilol
Keywords: SEDDS; Bioavailability; Formulation by design (FbD); SNEOFs; In situ single pass intestinal perfusion; IVIVC
Formulation design and in vivo antimalarial evaluation of lipid-based drug delivery systems for oral delivery of β-arteether
Keywords: β-Arteether; SEDDS; Oral administration; Antimalarial efficacy; Plasmodium berghei
Molecular modelling and multisimplex optimization of tocotrienol-rich Self Emulsified Drug Delivery Systems
Keywords: Surfactants; Nanoemulsions; Physical characterization; Tocotrienol; Multisimplex®; SEDDS;
Toward the Establishment of Standardized In Vitro Tests for Lipid-Based Formulations, Part 1: Method Parameterization and Comparison of In Vitro Digestion Profiles Across a Range of Representative Formulations
Keywords: LFCS Consortium; lipid-based drug delivery systems; SEDDS; drug solubilization; in vitro digestion testing; Solubility; Biopharmaceutics classification system (BCS); Bioavailability; In vitro models; Precipitation
A formulationâenabled preclinical efficacy assessment of a farnesoid X receptor agonist, GW4064, in hamsters and cynomolgus monkeys
Keywords: FXR agonist; efficacy; SEDDS; oral bioavailability; salt form; poorly soluble drug;
Recent advances of discrete coordination complexes and coordination polymers in drug delivery
Keywords: ADMET; absorption, distribution, metabolism, excretion, and toxicity; AL; ancillary ligand; API; active pharmaceutical ingredient; ASP; aspirin and copper(II)-aspirinate complexes; BBB; blood-brain barrier; BCS; Biopharmaceutics Classification System;
Impact of emulsion-based drug delivery systems on intestinal permeability and drug release kinetics
Keywords: Oil-in-water emulsions; Effect of formulation parameters; Self-emulsifying drug delivery systems; SEDDS; Experimental design
Design of Lipid-Based Formulations for Oral Administration of Poorly Water-Soluble Drugs: Precipitation of Drug after Dispersion of Formulations in Aqueous Solution
Keywords: lipid formulation classification system; self-emulsifying systems; self-emulsifying drug delivery systems; SEDDS; SMEDDS; drug precipitation; oral drug delivery;
Formulation and in vivo evaluation of chlorpropham (CIPC) oral formulations
Keywords: chloropropham; SEDDS; bioavailability; pharmacokinetics; solubility; oral drug delivery; formulation;
Formulation and in vitro and in vivo characterization of a phenytoin self-emulsifying drug delivery system (SEDDS)
Keywords: SEDDS; Phenytoin; Emulsions; Zeta potential; Improving dissolution; In vivo testing
Comparison between lipolysis and compendial dissolution as alternative techniques for the in vitro characterization of α-tocopherol self-emulsified drug delivery systems (SEDDS)
Keywords: Lipolysis; SEDDS; Griseofulvin; Dissolution; Optimization
Stable drug encapsulation in micelles and microemulsions
Keywords: Bioavailability; Hydrophobic drugs; Micelles; Microemulsions; Precipitation; SEDDS; SMEDDS; Self-emulsifying; Solubilization; Self-microemulsifying
Effect of combined use of nonionic surfactant on formation of oil-in-water microemulsions
Keywords: Surfactant; Microemulsions; Preconcentrate; Flurbiprofen; SMEDDS; SEDDS;