Keywords: شاخص انتخابی; Anticancer activity; Cytotoxicity; Fluorescent cyanine; Pentamethinium salt; Recognition; Sulfated polysaccharides; A549; cells of lung adenocarcinoma; AIDS; acquired immune deficiency syndrome; BJ; human fibroblasts (non-malignant cell line); BrdU; 5-bro
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Keywords: شاخص انتخابی; Vero; verda reno; MEM; Eagle minimum essential medium; ROS; Reactive Oxygen Species; MRSA; Methicillin-resistant Staphylococcus aureus; BHT; butylated hydroxytoluene; TBHQ; tertbutylhydroquinone; EO; essential oil; ST1; vegetative stage; ST2; full floweri
Keywords: شاخص انتخابی; HOBt; hydroxybenzotriazole; EDCl; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide; DMF; N-N-dimethyl formamide; s; singlet; 5-FU; 5-fluorouracil; P. falciparum; Plasmodium falciparum; SI; Selectivity Index; TLC; Thin Layer Chromatography; IR; infra-red; NMR
Keywords: شاخص انتخابی; Plasmodium falciparum; Plasmodium berghei ANKA; Terpenes; Experimental cerebral malaria; Protein isoprenylation; Cytokines; [3H]-FPP; [1-(n)-3H]farnesyl pyrophosphate triammonium salt; [3H]-GGPP; [1-(n)-3H]geranylgeranyl pyrophosphate triammonium salt; CB
Keywords: شاخص انتخابی; ATCC; American Type Culture Collection, Manassas, Virginia, USA; CC; Cell Controls; CC50; 50% Cytostatic/Cytotoxic Concentration; CPE; CytoPathic Effect; CRF; Chirang Reserve Forest; DMSO; DiMethyl SulphOxide; EC50; 50% Effective Concentration; EC90; 90%
Keywords: شاخص انتخابی; ATCC; American Type Culture Collection; LC50; 50% lethal concentration; MEM; minimal essential medium; MIC; minimum inhibitory concentration; MTT; 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide; PBS; phosphate buffered saline; SI; selectivit
Identification of highly selective and potent orexin receptor 1 antagonists derived from a dual orexin receptor 1/2 antagonist based on the structural framework of pyrazoylethylbenzamide
Keywords: شاخص انتخابی; OX1R; orexin 1 receptor; OX2R; orexin 2 receptor; DORA; dual orexin receptor antagonist; SORA; selective orexin receptor antagonist; SI; selectivity index; BBB; blood-brain barrier; CNS; central nervous system; SAR; structure-activity relationship; Boc; t
meso-Dihydroguaiaretic acid derivatives with antibacterial and antimycobacterial activity
Keywords: شاخص انتخابی; meso-Dihydroguaiaretic acid; Lignans; Antimycobacterial; Antibacterial; Selectivity index;
Synthesis of readily available fluorophenylalanine derivatives and investigation of their biological activity
Keywords: شاخص انتخابی; AChE; acetylcholinesterase; BAC; bacitracin; BChE; butyrylcholinesterase; ChE; cholinesterases; DMAP; 4-(dimethylamino)pyridine; EDC; N-(3-dimethylaminopropyl)-Nâ²-ethylcarbodiimide hydrochloride; ESBL; extended-spectrum β-lactamase; FLU; fluconazole; m
Keywords: شاخص انتخابی; Oxadiazole-benzohydrazone hybrids; Leishmaniasis; SAR study; Molecular docking studies; DFT; Selectivity index;
Keywords: شاخص انتخابی; 5-Nitro-2-aminothiazoles; Type I nitroreductase; Antitrypanosomal agents; Chagas disease; Leishmania; MZSRZQZBRGCXDO-UHFFFAOYSA-N; NTD; Neglected tropical diseases; T. brucei; Trypanosoma brucei; HAT; human African trypanosomiasis; T. cruzi; Trypanosoma
Keywords: شاخص انتخابی; Nitrotriazoles; Type I nitroreductase; Chagas disease; HAT disease; Leishmania; NTD; Neglected tropical diseases; T. brucei; Trypanosoma brucei; HAT; human African trypanosomiasis; T. cruzi; Trypanosoma cruzi; Bnz; benznidazole (N-benzyl-2-(2-nitro-1H-i
Keywords: شاخص انتخابی; Hybrid molecules; Anti-fungal; Anti-tubercular; Anti-malarial; anti-inflammatory; ACTs; artemesinin based combination therapy; CQ; chloroquine; CC50; concentration required to reduce growth by 50%; EC50; half maximal effective concentration; Fqa; ferroqui
Keywords: شاخص انتخابی; SCLC; small cell lung cancer; NSCLC; non-small-cell lung cancer; LNCaP; human prostate adenocarcinoma; DU-145; human prostate carcinoma; MDA-MB-231; human breast adenocarcinoma; BGC-823; human gastric cancer; SI; selectivity index; SAR; structure-activi
Keywords: شاخص انتخابی; Asc; ascaridole; Car; carvacrol; Caryo; caryophyllene oxide; DMPO; 5,5-dimethyl-1-pyrroline-N-oxide; DMSO; dimethyl sulfoxide; DPPH; 2,2-diphenyl-1-picrylhydrazyl; EO; essential oil; ESR; electron spin resonance; FIC; fractional inhibitory concentration;
Keywords: شاخص انتخابی; AVS; adrenal vein sampling; IVC; inferior vena cava; SI; selectivity index;
Keywords: شاخص انتخابی; CC50; concentration of the compound required to reduce cell viability by 50%; CSF; classical swine fever; CSFV; classical swine fever virus; Ct; cycle threshold; ER; endoplasmic reticulum; GTs; glycosyltransferases; IC50; concentration of the compound req
Keywords: شاخص انتخابی; Nitrotriazoles; Nitroimidazoles; Heteroarylamides; Heteroarylsulfonamides; Chagas disease; Antitrypanosomal agents; NTD; neglected tropical diseases; T. cruzi; Trypanosoma cruzi; T. brucei; Trypanosoma brucei; HAT; human African trypanosomiasis; Nfx; ni
Keywords: شاخص انتخابی; Antitubercular activity; Isoniazid derivatives; Mycobacterium tuberculosis; Resistance; QSARs; Synthesis; AE; average error; AAE; absolute average error; ASNNs; associative neural networks; BCG; Bacillus Calmette-Guérin; CCC; concordance correlation co
Keywords: شاخص انتخابی; Veronica americana; Acylated iridoids; Cytotoxicity; Selectivity index;
Keywords: شاخص انتخابی; JTLGJFBDQUBICH-UHFFFAOYSA-N; FEBATDALCUAQCM-UHFFFAOYSA-N; KZASLSLPFQAZRC-UHFFFAOYSA-N; APTXIDCPFDQWLD-UHFFFAOYSA-N; ZPMMPPBRCTWMHF-UHFFFAOYSA-N; LYXYENKXUDZGBB-UHFFFAOYSA-N; JKJRTNOOSNWMJV-UHFFFAOYSA-N; REFAZYLZAXUBGI-UHFFFAOYSA-N; RONHWZKWQSMGNP-UHFFFAOY
Keywords: شاخص انتخابی; AVS; Adrenal Vein Sampling; ACTH; Adrenocorticotropin Hormone; APA; Aldosterone Producing Adenoma; BAH; Bilateral Adrenal Hyperplasia; BC; British Columbia; IVC; Inferior Vena Cava; LAV; Left Adrenal Vein; LI; Lateralization Index; LL; LifeLabs; PA; Prima
In vitro antiplasmodial activity and identification, using tandem LC-MS, of alkaloids from Aspidosperma excelsum, a plant used to treat malaria in Amazonia
Keywords: شاخص انتخابی; Ae-Alk; Total alkaloids obtained directly from trunk bark powder; APCI; Atmospheric Pressure Chemical Ionization; DAD; Diode-Array Detector; ELAe; Lyophilized tincture (hydroethanolic extract) of Aspidosperma excelsum trunk bark; ELAe-Alk; Total alkaloids
Polynuclear copper(II) complexes with nalidixic acid hydrazones: Antiproliferative activity and selectivity assessment over a panel of tumor cells
Keywords: شاخص انتخابی; Complex 1A or [Cu2(h2imi)Cl4]; Copper(II) complex synthesized from CuCl2 and 2-imidazolyl hydrazone; Complex 1B or [Cu3Cl4(h2imiâ)2H2O]; Crystal structure of the copper(II) complex synthesized from CuCl2 and 2-imidazolyl hydrazone; Complex 2A or [Cu3(h4
Identification of tagitinin C from Tithonia diversifolia as antitrypanosomal compound using bioactivity-guided fractionation
Keywords: شاخص انتخابی; 1D and 2D NMR; One and two-dimensional nuclear magnetic resonance; BALB//3T3; Mouse fibroblasts; CH2Cl2/MeOH; Methylene chloride/Methanol; DMSO; Dimethylsulfoxide; HAT; Human African Trypanosomiasis; NTDs; Neglected tropical diseases; SAR; Structure-activ
Chemical composition of Ocimum canum Sims. essential oil and the antimicrobial, antiprotozoal and ultrastructural alterations it induces in Leishmania amazonensis promastigotes
Keywords: شاخص انتخابی; OCEO; Ocimum canum essential oil; DMSO; dimethyl sufoxide; CG/MS; gas chromatography-mass spectrometry; MIC; minimum inhibitory concentration; MTT; 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide; IC50; 50% inhibition of parasite growth; CC
In vitro activity of new N-benzyl-1H-benzimidazol-2-amine derivatives against cutaneous, mucocutaneous and visceral Leishmania species
Keywords: شاخص انتخابی; Benzimidazole derivatives; Antileishmanial activity; Selectivity Index; Arginase;
The potential use of leaf extracts of two Newtonia (Fabaceae) species to treat diarrhoea
Keywords: شاخص انتخابی; AchEI; acetylcholinesterase inhibitors; MIC; minimum inhibitory concentration; DPPH; 2,2â²-diphenyl-1-picrylhydrazyl; ABTS; 2,2-azino-bis (3-ethylbenzothiazoline-6-sulfonic acid) diammonium salt; MTT; 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium
1,3,5-triazaspiro[5.5]undeca-2,4-dienes as selective Mycobacterium tuberculosis dihydrofolate reductase inhibitors with potent whole cell activity
Keywords: شاخص انتخابی; Dihydrofolate reductase (DHFR); Antimycobacterial agent; Tuberculosis (TB); 1,3,5-triazaspiro[5.5]undeca-2,4-diene; DHFR; dihydrofolate reductase; DMPK; drug metabolism and pharmacokinetics; FRLM; female rat liver microsomes; HBA; hydrogen bond acceptors;
Novel indanone derivatives as MAO B/H3R dual-targeting ligands for treatment of Parkinson's disease
Keywords: شاخص انتخابی; Multi-targeting; Neurodegenerative diseases; Histamine H3 receptor antagonist; Monoamine oxidase inhibitor; Neurotransmitter dysregulation; Parkinson's disease; AChE; acetylcholinesterase; anal. calc.; elementary analysis calculated; BuChE; butyrylcholine
Anti-Mycobacterium tuberculosis activity of essential oil and 6,7-dehydroroyleanone isolated from leaves of Tetradenia riparia (Hochst.) Codd (Lamiaceae)
Keywords: شاخص انتخابی; Mycobacterium tuberculosis; Tetradenia riparia; Essential oil; Antimycobacterial activity; Cytotoxicity; TB; Tuberculosis; HIV; human immunodeficiency virus; MDR; multidrug-resistant; XDR; extensively drug-resistant; TrEO; Tetradenia riparia essential oil
Pharmacokinetics and cytotoxic study of euphol from Euphorbia umbellata (Bruyns) Pax latex
Keywords: شاخص انتخابی; Euphol; Cell culture; Cytotoxic activity; UHPLC-MS; Euphorbia; Pharmacokinetics; 1D and 2D NMR; one and two dimension nuclear magnetic resonance spectroscopy; ACN; acetonitrile; ATCC; american type culture collection; CDCl3; deuterated chloroform; CDK; cy
Metabolic profiling and correlation analysis for the determination of killer compounds of proliferating and clonogenic HRT-18 colon cancer cells from Lafoensia pacari
Keywords: شاخص انتخابی; LC-DAD-MS; Liquid chromatography coupled to Diode Array Detector and Mass spectrometry; MAC; extract obtained by maceration; DEC; extract obtained by decoction; S-CPC; Spot Chromatography Partition Centrifuge; LC-ESI-QqTOF-MS; Liquid chromatography couple
Tatanan A from the Acorus calamus L. root inhibited dengue virus proliferation and infections
Keywords: شاخص انتخابی; Acorus calamus l; Tatanan A; Dengue; DENV2 infection; CC; column chromatography; CC50; half maximal cytotoxicity concentration; CPE; cytopathic effect; DENV; dengue virus; DENV2; dengue virus type 2; DEPT; distortionless enhancement by polarization transf
An appraisal on synthetic and pharmaceutical perspectives of pyrazolo[4,3-d]pyrimidine scaffold
Keywords: شاخص انتخابی; A. flavus; Aspergillus flavus; C. albicans; Candida albicans; cAMP; cyclic adenosine monophosphate; CDK; cyclin-dependent kinase; CNS; central nervous system; COX; cyclooxygenase; CRF; corticotropin-releasing hormone; CRK; cdc2-related kinase; CYC6; cycli
Tacrine derivatives stimulate human glioma SF295 cell death and alter important proteins related to disease development: An old drug for new targets
Keywords: شاخص انتخابی; TMZ; temozolomide; GBM; glioblastoma multiforme; CNS; central nervous system; ROS; reactive oxygen species; BBB; blood-brain barrier; CC50; 50% cytotoxic concentration; TEM; transmission electron microscopy; SI; selectivity index; âÏm; mitochondrial me
Acridone alkaloids from the stem bark of Citrus aurantium display selective cytotoxicity against breast, liver, lung and prostate human carcinoma cells
Keywords: شاخص انتخابی; A549; human lung adenocarcinoma; ANOVA; one-way analysis of variance; ATCC; American type culture collection; CDCl3; chloroform; DMSO; dimethyl sulfoxide; ECACC; European collection of authenticated cell cultures; HepG2; human liver adenocarcinoma; HPLC;
Synthesis and biological evaluation of a library of hybrid derivatives as inhibitors of influenza virus PA-PB1 interaction
Keywords: شاخص انتخابی; Anti-Influenza; PA-PB1; RdRp; Amino acid coupling; SPPS; Diphenyl-pyridine; AcOEt; Ethyl acetate; CC50; Half maximal cytotoxic concentration; cRNA; complementar RNA; DCM; dichloromethane; DDQ; 2,3-Dichloro-5,6-dicyano-1,4-benzoquinone; DIPEA; N,N-Diisopro
Substituted 1,5-naphthyridine derivatives as novel antileishmanial agents. Synthesis and biological evaluation
Keywords: شاخص انتخابی; Leishmania; Naphthyridines; DNA-topoisomerase; VL; Visceral Leishmaniasis; TopIB; Type IB DNA Topoisomerase; IRFP; Infra Red Fluorescent Protein; FCS; Fetal Calf Serum; DMSO; Dimethyl sulfoxide; SI; Selectivity Index; CPT; camptothecin; CPTs; camptothecin
Metabolomic profile of Schinopsis brasiliensis via UPLC-QTOF-MS for identification of biomarkers and evaluation of its cytotoxic potential
Keywords: شاخص انتخابی; Medicinal plants; Northeastern Brazil; Dereplication; LC-MS; Selectivity index; Flavanols;
Efficacy of 2-hydroxy-3-phenylsulfanylmethyl-[1,4]-naphthoquinone derivatives against different Trypanosoma cruzi discrete type units: Identification of a promising hit compound
Keywords: شاخص انتخابی; Trypanosoma cruzi; Naphthoquinones; Trypanocidal activity; Chemotherapy; CD; Chagas disease; Bz; Benznidazole; Nif; Nifurtimox; ROS; Reactive oxygen species; CC50; Concentration of compound that reduces 50% of mammalian cell viability; IC50; Concentration
Structure-activity relationship studies of lipophilic teicoplanin pseudoaglycon derivatives as new anti-influenza virus agents
Keywords: شاخص انتخابی; Teicoplanin; Lipoglycopeptide; Maleimide; Sulfonamide; Influenza virus inhibitor; Coronavirus; DCM; dichloromethane; DMF; dimethylformamide; CPE; cytopathic effect; Et3N; triethylamine; Galp; galactopyranose; HA; hemagglutinin; HIV; human immunodeficiency
β-Lapachone and its iodine derivatives cause cell cycle arrest at G2/M phase and reactive oxygen species-mediated apoptosis in human oral squamous cell carcinoma cells
Keywords: شاخص انتخابی; ctDNA; Calf thymus DNA; CTL; Negative control; DAF-FM diacetate; 4-amino-5-methylamino-2'-,7'-difluofluorescein diacetate; DCF-DA; 2',7'-dichlorodihydrofluorescein diacetate; DMSO; Dimethyl sulfoxide; DOX; Doxorubicin; FBS; Fetal bovine serum; FSC; Fo
Tithonia diversifolia (Hemsl.) A. Gray as a medicinal plant: A comprehensive review of its ethnopharmacology, phytochemistry, pharmacotoxicology and clinical relevance
Keywords: شاخص انتخابی; ABTS; 2,2â²-Azinobis (3-ethylbenzothiazoline-6-sulphonate); Ach; acetyl choline; ALP; alkaline phosphatase; ALT; alanine aminotransferase; AMPK; 5' adenosine monophosphate-activated protein kinase; AST; Aspartate transaminase; CAs; chlorogenic acids; CC5
In vitro antiplasmodial activity of Withania frutescens-Solanaceae
Keywords: شاخص انتخابی; Antiplasmodial activity; Withania frutescens; Plasmodium falciparum; Cytotoxicity; Selectivity index;
New hydrazine and hydrazide quinoxaline 1,4-di-N-oxide derivatives: In silico ADMET, antiplasmodial and antileishmanial activity
Keywords: شاخص انتخابی; ACTs; artemisinin-based combination therapies; QdNO; quinoxaline 1,4-di-N-oxide; SAR; structure-activity relationship; VL; virtual library; SI; selectivity index; TPSA; topological polar surface area; %ABS; human intestinal absorption; Malaria; Leishmania
Pharmacological properties of extracts from six South African medicinal plants used to treat sexually transmitted infections (STIs) and related infections
Keywords: شاخص انتخابی; MIC; minimum inhibitory concentration; SI; selectivity index; IC50; extract concentration that inhibited 50% of cell growth; Antimicrobial; Cytotoxicity; Medicinal plants; Selectivity index; Sexually transmitted infections; Synergistic effect;
In vitro and in vivo cysticidal activity of extracts and isolated flavanone from the bark of Prunus serotina: A bio-guided study
Keywords: شاخص انتخابی; Prunus serotina; Taenia crassiceps cysts; Cysticidal activity; Selectivity index; 2,3-Dihydro-5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-1-benzopyran-4-one [naringenin];
Isolation, structural characterization and neuraminidase inhibitory activities of polyphenolic constituents from Flos caryophylli
Keywords: شاخص انتخابی; NA; neuraminidase; HA; haemagglutinin; MUNANA; methylumbelliferyl-α-d-N-acetylneuraminate; MDCK; Madin-Darby canine kidney; MNCC; maximal non-cytotoxic concentration; HHDP; hexahydroxydiphenoyl; MTT; 3-[4,5-dimethyl-thiazol-2-yl]-2,5- diphenyl tetrazoliu
Pyrrolizines: Design, synthesis, anticancer evaluation and investigation of the potential mechanism of action
Keywords: شاخص انتخابی; ALK1; activin receptor-like kinase; CDCl3; deuterated chloroform; MTT; 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyl tetrazolium bromide; DSV; discovery studio visualizer; DYRK3; dual specificity tyrosine phosphorylation-regulated kinase; CDK2; cyclin-depende