Keywords: گیرنده های سیگما; Donepezil-flavonoid hybrids; Neurogenesis; Neuroprotection; Sigma receptors; Human acetylcholinesterase; Human 5-lipoxygenase; Human monoamine oxidases; AChE; acetylcholinesterase; AD; Alzheimer's disease; ATCh; acetylthiocholine; BBB; blood-brain barrier
مقالات ISI گیرنده های سیگما (ترجمه نشده)
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Keywords: گیرنده های سیگما; Glia; Neurodegeneration; Neurotoxicity; Sigma receptors;
Keywords: گیرنده های سیگما; Bn; bombesin; BnR; bombesin receptor; BR; biotin receptor; c(RGD-K); cyclic {Arginine-Glycine-Aspartic acid (RGD)} containing peptide; CA; cholic acid; DOX; doxorubicin; EGF; epidermal growth factor; EGFR; epidermal growth factor receptor; ETRB; endotheli
(+)-Pentazocine attenuates SH-SY5Y cell death, oxidative stress and microglial migration induced by conditioned medium from activated microglia
Keywords: گیرنده های سیگما; DTG; 1,3-di-(2-tolyl) guanidine; DTNB; 2,2-dithio-bis-nitrobenzoic acid; CNS; central nervous system; Hsp70; heat shock protein 70; IL-10; interleukin 10; NO; nitric oxide; LPS; lipopolysaccharide; PBS; phosphate buffered saline solution; ROS; reactive ox
Do spiroindolines have the potential to replace vesamicol as lead compound for the development of radioligands targeting the vesicular acetylcholine transporter?
Keywords: گیرنده های سیگما; YBQFMGUWXJJOBE-OWOJBTEDSA-N; UJLKLUQGBGSJOO-OWOJBTEDSA-N; DSSGEOKNTGYRDY-OWOJBTEDSA-N; RDXPBCTWNYFBFI-OWOJBTEDSA-N; MTENKAMVZFIDIJ-OWOJBTEDSA-N; WLWBMTWWXNCMJH-OWOJBTEDSA-N; VAChT; Vesamicol; Spiroindolines; PET; Sigma receptors;
Nanoencapsulation strategies for the delivery of novel bifunctional antioxidant/Ï1 selective ligands
Keywords: گیرنده های سیگما; ALA; alpha lipoic acid; BS; back scattering; Brij® 98; polyoxyethylene (20) oleyl ether, Oleth-20; Cutina CP; cetyl palmitate; Cryo-TEM; cryogenic transmission electron microscopy; Da; PDI after freeze-thawing; Db; PDI before freeze-thawing; DDAB; dime
Gaining in pan-affinity towards sigma 1 and sigma 2 receptors. SAR studies on arylalkylamines
Keywords: گیرنده های سیگما; Sigma receptors; Arylalkylamine; Pan-affinity; QSAR;
Development of sigma-1 (Ï1) receptor fluorescent ligands as versatile tools to study Ï1 receptors
Keywords: گیرنده های سیگما; Sigma receptors; Fluorescent ligand; DTG; 1,3-di-2-tolylguanidine; DMEM; Dulbecco's modified Eagle's medium; PBS; Phosphate buffered saline; SDS; Sodium dodecyl sulfate;
Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy)alkyl]- and N-{2-[2-(phenoxy)ethoxy]ethyl}aminoalkanols as anticonvulsant agents
Keywords: گیرنده های سیگما; VGGMLGZQRUZPAC-HQKYYOGZSA-N; SORDYQMTTXQNIQ-CQSZACIVSA-NAminoalkanols; Anticonvulsant activity; Seizures; Sigma receptors; 5-HT; MES; Metabolic stability; Mutagenicity; Vibrio harveyi; Pharmacokinetics
Computer-assisted design, synthesis, binding and cytotoxicity assessments of new 1-(4-(aryl(methyl)amino)butyl)-heterocyclic sigma 1 ligands
Keywords: گیرنده های سیگما; Sigma receptors; Binding affinity; Cytotoxicity; Molecular modeling;
Synthesis and pharmacological evaluation of 11C-labeled piperazine derivative as a PET probe for sigma-2 receptor imaging
Keywords: گیرنده های سیگما; Sigma receptors; Sigma-2; PET; Imaging; Carbon-11; Cancer
Haloperidol metabolite II prodrug: Asymmetric synthesis and biological evaluation on rat C6 glioma cells
Keywords: گیرنده های سیگما; Glioma; HDAC; Sigma receptors; Inhibitors; Medicinal chemistry
Carboline- and phenothiazine-derivated heterocycles as potent SIGMA-1 protein ligands
Keywords: گیرنده های سیگما; Sigma receptors; Carboline; Tetrahydrobenzofuropyridine; Phenoxazine; PhenothiazineER, endoplasmic reticulum; MAM, mitochondrion associated endoplasmic reticulum membrane; S1R, sigma 1 receptors; S2R, sigma 2 receptors; BiP, immunoglobulin heavy-chain bin
Ether modifications to 1-[2-(3,4-dimethoxyphenyl)ethyl]-4-(3-phenylpropyl)piperazine (SA4503): Effects on binding affinity and selectivity for sigma receptors and monoamine transporters
Keywords: گیرنده های سیگما; Sigma receptors; Dopamine transporter; Serotonin transporter; In vitro binding;
New systematically modified vesamicol analogs and their affinity and selectivity for the vesicular acetylcholine transporter – A critical examination of the lead structure
Keywords: گیرنده های سیگما; VAChT; Vesamicol; PET; Sigma receptors
Pharmacological evaluation of SN79, a sigma (σ) receptor ligand, against methamphetamine-induced neurotoxicity in vivo
Keywords: گیرنده های سیگما; Dopamine; Hyperthermia; Methamphetamine; Neurotoxicity; Serotonin; Sigma receptors
7-Azabicyclo[2.2.1]heptane as a scaffold for the development of selective sigma-2 (Ï2) receptor ligands
Keywords: گیرنده های سیگما; Azanorbornanes; Pyrrolidines; Sigma receptors; CNS; Structure-activity relationships;
A Ï1 receptor pharmacophore derived from a series of N-substituted 4-azahexacyclo[5.4.1.02,6.03,10.05,9.08,11]dodecan-3-ols (AHDs)
Keywords: گیرنده های سیگما; Trishomocubanes; Sigma receptors; CNS; Structure-activity relationships;
Neuroprotective effects of high affinity sigma 1 receptor selective compounds
Keywords: گیرنده های سیگما; Sigma receptors; Sigma 1 receptors; Neuroprotection;
Sigma-1 receptor agonists provide neuroprotection against gp120 via a change in bcl-2 expression in mouse neuronal cultures
Keywords: گیرنده های سیگما; Dementia; Neuroprotection; Glycoprotein 120; Sigma receptors; Human immunodeficiency virus;
Synthesis, radioiodination and in vitro and in vivo sigma receptor studies of N-1-allyl-N´-4-phenethylpiperazine analogs
Keywords: گیرنده های سیگما; Sigma receptors; I-125; Allylpiperazines;
Trishomocubane as a scaffold for the development of selective dopamine transporter (DAT) ligands
Keywords: گیرنده های سیگما; Trishomocubanes; Monoamine transporters; Sigma receptors; CNS; Structure-activity relationships;
Effects of linker elongation in a series of N-(2-benzofuranylmethyl)-N′-(methoxyphenylalkyl)piperazine σ1 receptor ligands
Keywords: گیرنده های سیگما; Piperazines; Sigma receptors; CNS; Structure–affinity relationships
Synthesis and in vivo evaluation of [18F]N-(2-benzofuranylmethyl)-N′-[4-(2-fluoroethoxy)benzyl]piperazine, a novel σ1 receptor PET imaging agent
Keywords: گیرنده های سیگما; Piperazines; Sigma receptors; Positron emission tomography; Fluorine-18
N-Arylalkyl-2-azaadamantanes as cage-expanded polycarbocyclic sigma (Ï) receptor ligands
Keywords: گیرنده های سیگما; Adamantanes; Polycarbocyclic; Sigma receptors; CNS; Structure-activity relationships;
Molecular hybridization of 4-azahexacyclo[5.4.1.02,6.03,10.05,9.08,11]dodecane-3-ol with sigma (σ) receptor ligands modulates off-target activity and subtype selectivity
Keywords: گیرنده های سیگما; Trishomocubanes; Sigma receptors; CNS; Structure–activity relationships
Antiproliferative activity of phenylbutyrate ester of haloperidol metabolite II [(±)-MRJF4] in prostate cancer cells
Keywords: گیرنده های سیگما; Histone deacetylase; Inhibitors; LNCaP; PC3; Sigma receptors;
SA 4503 attenuates cocaine-induced hyperactivity and enhances methamphetamine substitution for a cocaine discriminative stimulus
Keywords: گیرنده های سیگما; Sigma receptors; Cocaine; Locomotor activity; Drug discrimination
Effect of structural modification in the amine portion of substituted aminobutyl-benzamides as ligands for binding Ï1 and Ï2 receptors
Keywords: گیرنده های سیگما; Sigma receptors; Structure-activity relationships; Aminobutyl-benzamides;
Effects of the selective sigma receptor ligand, 1-(2-phenethyl)piperidine oxalate (AC927), on the behavioral and toxic effects of cocaine
Keywords: گیرنده های سیگما; Cocaine; Conditioned place preference; Drug discrimination; Locomotor activity; Self-administration; Sigma receptors
The sigma receptor agonist SA4503 both attenuates and enhances the effects of methamphetamine
Keywords: گیرنده های سیگما; Sigma receptors; Methamphetamine; Dopamine release; Locomotor activity; Drug discrimination;
Sigma Receptor Agonists: Receptor Binding and Effects on Mesolimbic Dopamine Neurotransmission Assessed by Microdialysis
Keywords: گیرنده های سیگما; Abuse liability; addiction; cocaine; dopamine microdialysis; nucleus accumbens; reinforcing effects; sigma receptors
ASIC1a channels are activated by endogenous protons during ischemia and contribute to synergistic potentiation of intracellular Ca2+ overload during ischemia and acidosis
Keywords: گیرنده های سیگما; Sigma receptors; Ischemia; Acidosis; Neurotransmission; Calcium; Neurons; Stroke;
Delayed treatments for stroke influence neuronal death in rat organotypic slice cultures subjected to oxygen glucose deprivation
Keywords: گیرنده های سیگما; ischemia; inflammation; neuroprotection; sigma receptors; human umbilical cord blood cellsDAF-FM, 4-amino-5-methylamino-2′,7′-difluorofluorescein; DMEM, Dulbecco's modified Eagles medium; DTG, 1,3-di-o-tolylguanidine; HUCBC, human umbilical cord blood cel
Screening of anti-glioma effects induced by sigma-1 receptor ligands: Potential new use for old anti-psychiatric medicines
Keywords: گیرنده های سیگما; Cell migration; Cell proliferation; Chemotherapy; Donepezil; Glioblastoma; Mitotic arrest; Sigma receptors
Behavioural effects of trishomocubanes in rats with unilateral 6-hydroxydopamine lesions
Keywords: گیرنده های سیگما; Rat; Medial forebrain bundle; Sigma receptors; Locomotor behaviour; Tyrosine hydroxylase; Anxiety; Sedation
On the mechanism of antidepressant-like action of berberine chloride
Keywords: گیرنده های سیگما; Berberine chloride; Antidepressant; Nitric oxide; Sigma receptors; Monoamines
Attenuation of methamphetamine-induced effects through the antagonism of sigma (σ) receptors: Evidence from in vivo and in vitro studies
Keywords: گیرنده های سیگما; Dopamine; Dopamine transporter; Hyperthermia; Locomotor activity; Methamphetamine; NG108-15 cells; Sigma receptors; Striatum
(+)-Morphine and (−)-morphine stereoselectively attenuate the (−)-morphine-produced tail-flick inhibition via the naloxone-sensitive sigma receptor in the ventral periaqueductal gray of the rat
Keywords: گیرنده های سیگما; Sigma receptors; Analgesia; Opioid; Morphine; Periaqueductal gray; (Rat)
Involvement of dopamine (DA)/serotonin (5-HT)/sigma (σ) receptor modulation in mediating the antidepressant action of ropinirole hydrochloride, a D2/D3 dopamine receptor agonist
Keywords: گیرنده های سیگما; Ropinirole; Forced swim test (FST); Tail suspension test (TST); Dopaminergic modulation; Serotonergic modulation; Sigma receptors
Inhibition of hyperpolarization-activated cation currents by phencyclidine and some sigma ligands in rat hippocampal CA1 pyramidal neurons in vitro
Keywords: گیرنده های سیگما; Ih channels; PCP; Sigma receptors; NMDA; ExcitabilityIh, hyperpolarization-activated cation currents; PCP, phencyclidine; CPP, d-3-(2-Carboxypiperazin-4-yl)-propyl-1-phosphonic acid; NE-100, N,N-dipropyl-2-[4-methoxy-3-(2-phenylethoxy)-phenyl]-ethylamine
Design, synthesis, and SAR analysis of novel selective σ1 ligands
Keywords: گیرنده های سیگما; Arylalkylamines; Sigma receptors; Molecular modeling; SAR studies
The sigma-2 receptor agonist PB28 inhibits calcium release from the endoplasmic reticulum of SK-N-SH neuroblastoma cells
Keywords: گیرنده های سیگما; Caffeine; Carbachol; Fura-2; PB28; Sigma receptors
Effect of haloperidol on transient outward potassium current in rat ventricular myocytes
Keywords: گیرنده های سیگما; Haloperidol; Transient outward current; Sigma receptors; Rat ventricular myocytes; Whole-cell patch clamp; Quantitative model
Synthesis and characterization of selective dopamine D2 receptor antagonists
Keywords: گیرنده های سیگما; Indoles; D2-like dopamine receptors; Sigma receptors; Dopamine receptor antagonists
Synthesis and in vivo evaluation of a new PET radioligand for studying sigma-2 receptors
Keywords: گیرنده های سیگما; Sigma receptors; Radioligand; Carbon-11; PET
In vitro characterization of radioiodinated (+)-2-[4-(4-iodophenyl) piperidino]cyclohexanol [(+)-pIV] as a sigma-1 receptor ligand
Keywords: گیرنده های سیگما; (+)-pIV; Vesamicol; Sigma receptors; Radioligand;
In vivo evaluation of [123I]-3-(4-iodobenzyl)-1,2,3,4-tetrahydro-8-hydroxychromeno[3,4-c]pyridin-5-one: a presumed dopamine D4 receptor ligand for SPECT studies
Keywords: گیرنده های سیگما; Sigma receptors; Dopamine D4 receptors; SPECT; 123I;
Involvement of sigma (Ï) receptors in the acute actions of methamphetamine: Receptor binding and behavioral studies
Keywords: گیرنده های سیگما; Antisense; BD1063; BD1047; Locomotor; Methamphetamine; Sigma receptors;
In vivo evaluation of [123I]-4-iodo-N-(4-(4-(2-methoxyphenyl)-piperazin-1-yl)butyl)-benzamide: a potential sigma receptor ligand for SPECT studies
Keywords: گیرنده های سیگما; Sigma receptors; Dopamine D3 receptors SPECT; 123I;