Keywords: Monobactam; Siderophore; Structure-activity relationship; Antibacterial activity; Click chemistry; AZN; Aztreonam; MDR; multidrug-resistant; SAR; structureâactivity relationship; PIH; pyridoxal isonicotinoyl hydrazone; Trt; triphenylmethyl; Boc; t-but
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Keywords: Ac; acetyl; ACTH; adrenocorticotropic hormone; Alloc; allyloxycarbonyl; Boc; t-butoxycarbonyl; BSA; bovine serum albumin; DIC; N,Nâ²,-diisopropylcarbodiimide; DIEA; diisopropylethylamine; DMEM; Dulbecco's Modified Eagle Medium; DMF; N,N-dimethylformami
Keywords: Fumagillin; Biotinylated fumagillin; Angiogenesis; Cell permeability; Endothelial cell; Cancer cell; HUVEC; human umbilical vein endothelial cells; MetAP2; eukaryotic methionine aminopeptidase type II; HRP; horseradish peroxidase; DPPA; diphenylphosphoryl
A PEGylated analog of short-length Neuromedin U with potent anorectic and anti-obesity effects
Keywords: Neuromedin U (NMU); NMU-8; Polyethylene glycol (PEG); Diabetes; Obesity; NMU; neuromedin U; PEG; polyethyleneglycol; PipAc; 2-(piperazin-1-yl)acetic acid; CNS; central nervous system; DIO; diet-induced obesity; EMCS; N-(6-maleimidocaproyloxy)succinimide;
Synthesis and evaluation of novel ureido/thioureido derivatives of amino acid conjugated 2,3-dichlorophenyl piperazine as highly potent antiglycating agents
Keywords: AGE; advanced glycation end products; Boc; t-butoxycarbonyl; BSA; bovine serum albumin; EDCI; 1-(3-dimethylaminopropyl)-3-ethyl-carbodiimide·HCl; HOBt; 1-hydroxybenzotriazole; NMM; N-methyl morpholine; PBS; phosphate buffer saline; PZN; 1-(2,3-dichloroph
Novel type of plasmin inhibitors: Providing insight into P4 moiety and alternative scaffold to pyrrolopyrimidine
Keywords: MMP; matrix metalloproteinase; UK; urokinase; pNA; para-nitroanilide; MCA; 7-amino-4-methyl-coumarin amide; Boc; t-butoxycarbonyl; Pyr; pyroglutamic acid; Plasmin inhibitors; Benzimidazole; Scaffold; Pyrrolopyrimidine; P4 moiety; Structure-activity rela
REDOR solid-state NMR as a probe of the membrane locations of membrane-associated peptides and proteins
Keywords: δ; chemical shift; γ; buildup rate; Ï; REDOR dephasing time; A; buildup extent; Chol; cholesterol; Chol_d6; cholesterol-2,2,3,4,4,6-d6; Chol_d7; cholesterol-25,26,26,26,27,27,27-d7; CP; cross-polarization; d; dipolar coupling; Fmoc; 9-fluorenylmethoxyc
Tetrahedron report number 994β-Elimination competitions leading to CC bonds from alkylpalladium intermediates
Keywords: Palladium; Elimination; Heterocyclisation; Heck reaction; Wacker reaction; Aza-Wacker reaction; Selectivity; Atm; atmosphere; Boc; t-butoxycarbonyl; cat; catalytic; COD; 1,5-cyclooctadiene; Cy; cyclohexyl; dba; dibenzylidene acetone; DMA; N,N-dimethylacet
High content analysis to determine cytotoxicity of the antimicrobial peptide, melittin and selected structural analogs
Keywords: HBTU; O-benzotriazole-N,N,Nâ²,Nâ²-tetramethyl-uronium-hexafluoro-phosphate; PyBOPb; enzotriazole-1-yl-oxy-tris-pyrrolidino-phosphonium hexafluorophosphate; HOBt; N-hydroxybenzotriazole; DIEA; N,Nâ²-diisopropylethylamine; MBHA; 4-methylbenzhydrylamine;
Rational conversion of noncontinuous active region in proteins into a small orally bioavailable macrocyclic drug-like molecule: The HIV-1 CD4:gp120 paradigm
Keywords: AcOH; acetic acid; Alloc; allyloxycarbonyl; Boc; t-butoxycarbonyl; BTC; bis(trichloromethyl)carbonate; DBU; 1,8-diazabicyclo[5.4.0]undec-7-ene; DCM; methylene chloride; DIC; N,Nâ²-diisopropylcarbodiimide; DIPEA; diisopropylethylamine; DMAP; dimethylamino
Application of hydrolytic kinetic resolution (HKR) in the synthesis of bioactive compounds
Keywords: Hydrolytic kinetic resolution; Terminal epoxides; Bis-epoxides; meso-Epoxides; Natural products; Synthesis; Biological activity; Ac; acetyl; AD; asymmetric dihydroxylation; AE; asymmetric epoxidation; Bn; benzyl; NBS; N-bromosuccinimide; Boc; t-butoxycarb
Solid-phase synthesis of backbone-cyclized β-helical peptides
Keywords: Alkanesulfonamide; Safety-catch linker; Cyclic peptide; Solid-phase peptide synthesis; β-Hairpin; β-Turn; β-Helix; HPLC; Gel-permeation chromatography; AS-SLC; alkanesulfonamide safety-catch linker; CBC; cleavage-by-cyclization; Boc; t-butoxycarbonyl;
Recent approaches to the construction of 1-azaspiro[4.5]decanes and related 1-azaspirocycles
Keywords: Azaspirocyclic ring systems; Spirocycles; 3° Carbon center; Ac; acetyl; AIBN; azobisisobutyronitrile(2,2â²-azo(2-methylpropionitrile)); Ar; aryl; Bn; benzyl; Boc; t-butoxycarbonyl; Bu; butyl; Cbz; benzyloxycarbonyl; Cy; cyclohexyl; DBB; di-t-butylbiphen
A synthon approach to spiro compounds
Keywords: Photochromism; Synthon; Spiro compounds; BINAP; 2,2â²-bis(diphenylphospospiro)-1,1â²-binaphthalene; Boc; t-butoxycarbonyl; CTAB; cetyltrimethylammonium bromide; DEAD; diethylazodicarboxylate; 4-DMAP; 4-(dimethylamino)pyridine; Fmoc; 9-fluorenylmethoxyca
Recent advances in ether dealkylation
Keywords: O-Dealkylation; Deprotection; Debenzylation; Review; Ac; acetyl; Alloc/Aloc; allyloxycarbonyl; BMIM; 1-n-butyl-3-imidazolium; Bn; benzyl; Boc; t-butoxycarbonyl; BOM; benzyloxymethyl; Bz; benzoyl; CAN; ceric ammonium nitrate; Cbz; benzyloxycarbonyl; CSI; c
Sulfide- and selenide-based linkers in phase tag-assisted synthesis
Keywords: Solid phase; Linkers; Sulfur; Selenium; AIBN; 2,2â²-azobis(2-methylpropionitrile); Alloc; allyloxycarbonyl; Boc; t-butoxycarbonyl; Cbz; benzyloxycarbonyl; CSA; 10-camphorsulfonic acid; DABCO; diazabicyclo[2.2.2]octane; DAST; diethylaminosulfur trifluorid