Triazole pyrimidine nucleosides as inhibitors of Ribonuclease A. Synthesis, biochemical, and structural evaluation
Keywords: نیاسینهای تریازول; RNase A, bovine pancreatic Ribonuclease A; PEG, poly(ethylene glycol); U5P, deoxyuridine 5′-phosphate; ppA-3′-p, 5′-diphosphoadenosine 3′-phosphateRibonuclease A; Inhibition; X-ray crystallography; Triazole nucleosides; Structure-assisted inhibitor design