Keywords: UDP-گلوکورونوسیل ترانسفراز; Aβ; amyloid-β-peptide; ACh; acetylcholine; Apo; apolipoprotein; APP; amyloid precursor protein; CYP; cytochrome P-450; DYRK1; dual specificity tyrosine-phosphorylation-regulated kinase 1A; GABA; γ-aminobutyric acid; GSK; glycogen synthase- kinase; HSV-
مقالات ISI UDP-گلوکورونوسیل ترانسفراز (ترجمه نشده)
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Keywords: UDP-گلوکورونوسیل ترانسفراز; Fish; Rainbow trout; Biotransformation; Cytochrome P450; UDP-glucuronosyltransferase; Glutathione S-transferase; Allometry; Allometric scaling;
Keywords: UDP-گلوکورونوسیل ترانسفراز; AL; alantolactone; AL-GSH; glutathione conjugate of alantolactone; AL-Cys; cysteine conjugate of alantolactone; AUC; area under the concentration-time curve; Cys; cysteine; CYP450; cytochrome P450; DAD; diode array detector; GSH; glutathione; GST; glutath
Keywords: UDP-گلوکورونوسیل ترانسفراز; Bee pollen; Phytometabolites; Nutrition; Therapeutic benefits; Food safety; GC-MS; gas chromatography-mass spectrometry; LC-ESI/MS; liquid chromatography-electrospray ionization mass spectrometry; TLC; thin layer chromatography; HPLC-DAD-ESI/MS; high-pe
Keywords: UDP-گلوکورونوسیل ترانسفراز; Naringenin; Glucuronidation; UDP-Glucuronosyltransferase (UGT); Liver microsome; Intestine microsome; UGT; UDP-glucuronosyltransferase;
Keywords: UDP-گلوکورونوسیل ترانسفراز; BCRP; breast cancer resistant protein; BSEP; bile salt efflux pump; GA; gestational age; GLUT1; glucose transporter 1; MCT1; monocarboxylate transporter 1; MDR; multidrug-resistance protein; MRP; multidrug-resistance like protein; NTCP; Na+-taurocholate c
Keywords: UDP-گلوکورونوسیل ترانسفراز; AUC; area under the concentration-time curve; AST; aspartate transaminase; ALT; alanine transaminase; BCRP; breast cancer resistance protein; BEI; biliary excretion index; CL/F; oral clearance; Clbiliary; in vitro biliary clearance; ER; Efflux Ratio; LCâ
Keywords: UDP-گلوکورونوسیل ترانسفراز; ADAM; advanced dissolution, absorption, and metabolism; AED; antiepileptic drug; AUC; area-under-the-curve; B/P; blood to plasma ratio; BID; twice daily; BMI; body mass index; CBZ; carbamazepine; CLint; intrinsic clearance; CLR; renal clearance; CL; clear
Keywords: UDP-گلوکورونوسیل ترانسفراز; 2-AG; 2-arachidonoyl glycerol; 11-nor-THC-COOH; 11-nor-tetrahydrocannabinol-9-caboxylic acid; 11-OH-THC; 11-hydroxy-tetrahydrocannabinol; 8-OH-THC; 8-hydroxy-tetrahydrocannabinol; CB; cannabinoid; CB1R; Type I cannabinoid receptor; CB2R; Type II cannabino
Keywords: UDP-گلوکورونوسیل ترانسفراز; DRE; drug resistant epilepsy; PWE; patients with epilepsies; AEDs; anti-epileptic drugs; MTLE; mesial temporal lobe epilepsy; FCD; focal cortical dysplasia; BCRP; breast cancer resistance protein; MVP; major vault protein; MDT; smultidrug transporters; BB
Keywords: UDP-گلوکورونوسیل ترانسفراز; Clint; intrinsic clearance; Clint app.; apparent intrinsic clearance; DAD; diod array detector; DMSO; dimethyl sulfoxide; ER; endoplasmic reticulum; fu; unbound fraction of a drug in the microsomal incubation mixture; HPLC; high performance liquid chromat
Keywords: UDP-گلوکورونوسیل ترانسفراز; Acyl glucuronide; Drug development; Drug toxicity; In vitro screening; In vivo model; Immune activation; Protein adduct; Reactive metabolite; UDP-glucuronosyltransferase; ADR; adverse drug reaction; AG; acyl glucuronide; AGE; advanced glycation end prod
Keywords: UDP-گلوکورونوسیل ترانسفراز; ADMET; absorption, distribution, metabolism, excretion, toxicity; AHR; aryl hydrocarbon receptor; AUC; area under the curve; BVU; (E)-5-(2-bromovinyl) uracil; CAR; constitutive androstane receptor; cMOAT; Canalicular multispecific organic anion transporte
Keywords: UDP-گلوکورونوسیل ترانسفراز; PAPS; 3â²-Phosphoadenosine 5â²-phosphosulfate; DTNB; 5,5â²-Dithiobis(2-nitrobenzoic acid); APAP; Acetaminophen; ALT; Alanine aminotrasferase; BSA; Bovine serum albumin; CCl4; Carbon tetrachloride; Ccr2; C-C chemokine receptor 2; CFB; Clofibrate; CD;
Keywords: UDP-گلوکورونوسیل ترانسفراز; Mycophenolic acid; Inosine-5ʹ-monophosphate dehydrogenase; Nagase analbuminemic rat; Nonlinear mixed effects modeling; UDP-Glucuronosyltransferase
Keywords: UDP-گلوکورونوسیل ترانسفراز; UDP-glucuronosyltransferase; Glucuronidation; In vitro–in vivo extrapolation; Liver; Intestine; Availability; Clearance; Prediction
Keywords: UDP-گلوکورونوسیل ترانسفراز; CYP; cytochrome P-450; GSH-transferase; glutathione-S-transferase; UDP-glucuronosyltransferase; uridine 5â²-diphospho-glucuronosyltransferase; EGb761®; Ginkgo biloba extract, CAS 122933-57-7; AhR; aryl hydrocarbon receptor; PXR; pregnane X receptor; CAR
Keywords: UDP-گلوکورونوسیل ترانسفراز; CYP; cytochrome P450; 3-D; three-dimensional; APAP; acetaminophen; NAPQI; N-acetyl-p-benzoquinone imine; GSH; glutathione; ROS; reactive oxygen species; UGT; UDP-glucuronosyltransferase; SULT; sulfotransferase; ABT; 1-aminobenzotriazole; mBCl; monochlorob
Keywords: UDP-گلوکورونوسیل ترانسفراز; AhR; aryl hydrocarbon receptor; ARE; antioxidant response element; BT; black tea; CYP; cytochrome P450; DME; drug-metabolizing enzymes; DR4; direct repeat with 4Â bp spacer; DRE; dioxin response elements; GT; green tea beverage; EC; epicatechin; EGC; epig
Keywords: UDP-گلوکورونوسیل ترانسفراز; Aβ; amyloid-β-peptide; AD; Alzheimer's disease; BR; bilirubin; BV; biliverdin; BVR; biliverdin reductase; CAT; catalase; CCNA2; gene encoding for cyclin-A2; CCNB1; gene encoding for G2/mitotic-specific cyclin-B1; CEP2; centrosomal protein 2; Cmax; pea
Keywords: UDP-گلوکورونوسیل ترانسفراز; ABC transporter; ATP-binding cassette transporter; CD; conjugated dienes; CDEPA; 2-chloro-N-(2,6-diethylphenyl)acetamide; CMEPA; 2-chloro-N-(2-methyl-6 ethylphenyl)acetamide; DEA; 2,6-diethylaniline; GSH; glutathion; GST; glutathione-S-transferase; LPO; l
Species differences in drug glucuronidation: Humanized UDP-glucuronosyltransferase 1 mice and their application for predicting drug glucuronidation and drug-induced toxicity in humans
Keywords: UDP-گلوکورونوسیل ترانسفراز; UDP-glucuronosyltransferase; Glucuronidation; Species difference; Humanized mice; Drug metabolism; Toxicity;
New insights into the metabolism and toxicity of bisphenol A on marine fish under long-term exposure
Keywords: UDP-گلوکورونوسیل ترانسفراز; Bisphenol A glucuronide; UDP-Glucuronosyltransferase; Oryzias melastigma; Chorion; Reproductive toxicity;
Significance of A-to-I RNA editing of transcripts modulating pharmacokinetics and pharmacodynamics
Keywords: UDP-گلوکورونوسیل ترانسفراز; ABC; ATP-binding cassette transporter; ADAR; adenosine deaminase acting on RNA; ADH; alcohol dehydrogenase; AhR; aryl hydrocarbon receptor; AKR; aldo-keto reductase; ALS; amyotrophic lateral sclerosis; AZIN1; antizyme inhibitor 1; AMPA; α-amino-3-hydroxy
Safety assessment of Oryeong-san, a traditional herbal formula: Study of subacute toxicity and influence of cytochrome P450s and UDP-glucuronosyltransferases
Keywords: UDP-گلوکورونوسیل ترانسفراز; Herbal formula; Oryeong-san; Subacute toxicity; Cytochrome P450s; UDP-glucuronosyltransferase;
In vitrometabolic mapping of neobavaisoflavone in human cytochromes P450 and UDP-glucuronosyltransferase enzymes by ultra high-performance liquid chromatography coupled with quadrupole time-of-flight tandem mass spectrometry
Keywords: UDP-گلوکورونوسیل ترانسفراز; Neobavaisoflavone; Cytochromes P450; UDP-glucuronosyltransferase; Species difference; Metabolic pathway;
Targeting NLRP3 inflammasome via acetylsalicylic acid: Role in suppressing hepatic dysfunction and insulin resistance induced by atorvastatin in naïve versus alcoholic liver in rats
Keywords: UDP-گلوکورونوسیل ترانسفراز; AFL; alcoholic fatty liver; ALD; alcoholic liver disease; ALK; alkaline phosphatase; ALT; alaninetransaminase; ASA; acetylsalicylic acid; AST; aspartate transaminase; Bcl2; B cell lymphoma type 2; BSP; bromsulphthalein; COX-I; cyclooxygenase I; GSH; gluta
From TCDD-mediated toxicity to searches of physiologic AHR functions
Keywords: UDP-گلوکورونوسیل ترانسفراز; AHR; aryl hydrocarbon receptor; CAR; constitutive androstane receptor; PXR; pregnane-X-receptor; CYP; cytochrome P450; IDO1; indoleamine-2,3-dioxygenase; UDP; UDP-glucuronosyltransferase; FICZ; 6-formylindolo[3,2-b]carbazole; ICZ; indolo[3,2-b]carbazole;
Improving oral bioavailability of resveratrol by a UDP-glucuronosyltransferase inhibitory excipient-based self-microemulsion
Keywords: UDP-گلوکورونوسیل ترانسفراز; ACN; acetonitrile; AP; apical; BL; basolateral; CYP450; cytochrome P450 proteins; FBS; fetal bovine serum; IC50; half-inhibitory concentration; MEM; minimum essential medium; MTT; 3-(40,50-dimethylthiazol-20-yl)-2,5-diphenyltetrazolium bromide; NEAA; none
Effect of UGT2B7*2 and CYP2C8*4 polymorphisms on diclofenac metabolism
Keywords: UDP-گلوکورونوسیل ترانسفراز; CYP; cytochrome P450; CYP-reductase; NADPH cytochrome P450 reductase; DCF-AG; diclofenac acyl glucuronide; DCF-SG; diclofenac glutathione conjugate; DILI; drug-induced liver injury; ESI; electrospray ionization; GST; glutathione S-transferase; GWAS; genom
Metabolic profiling of corylin in vivo and in vitro
Keywords: UDP-گلوکورونوسیل ترانسفراز; Corylin; Metabolites profile; Cytochromes P450; UDP-glucuronosyltransferase; Species differences;
Identification and characterization of in vitro inhibitors against UDP-glucuronosyltransferase 1A1 in uva-ursi extracts and evaluation of in vivo uva-ursi-drug interactions
Keywords: UDP-گلوکورونوسیل ترانسفراز; Uva-ursi extract; In vitro UGT1A1 inhibition; Gallotannin; 1,2,3,6-Tetragalloylglucose; In vivo herbâdrug interaction; UGT; UDP-glucuronosyltransferase; TeGG; 1,2,3,6-tetragalloylglucose; 4-MU; 4-methylumbelliferone; UDPGA; uridine 5â²-diphosphoglucuro
Activation of Nrf2 signaling by natural products-can it alleviate diabetes?
Keywords: UDP-گلوکورونوسیل ترانسفراز; Nrf2; type 2 diabetes; natural products; hyperglycemia; cellular stress; insulin sensitivity; β-cell function; vascular complications; AGE; advanced glycation end products; AhR; arylhydrocarbon receptor; AMPK; AMP-activated kinase; ARE; antioxidant respo
Inhibition of UDP-glucuronosyltransferase (UGT)-mediated glycyrrhetinic acid 3-O-glucuronidation by polyphenols and triterpenoids
Keywords: UDP-گلوکورونوسیل ترانسفراز; UDP-Glucuronosyltransferase; UGT; Licorice; Glycyrrhetinic acid; Glycyrrhizin; Glucuronidation; Glucuronide; Natural medicine; Adverse reaction; Pseudohyperaldosteronism; DMSO; dimethyl sulfoxide; GA; Glycyrrhetinic acid; HPLC; high-performance liquid chr
Identification and expression patterns of UDP-glycosyltransferase (UGT) genes from insect pest Athetis lepigone (Lepidoptera: Noctuidae)
Keywords: UDP-گلوکورونوسیل ترانسفراز; UDP-glucuronosyltransferase; Athetis lepigone; Phylogenetic analysis; Expression pattern; Diverse functions;
Prevalence of UDP-glucuronosyltransferase polymorphisms (UGT1A6â2, 1A7â12, 1A8â3, 1A9â3, 2B7â2, and 2B15â2) in a Saudi population
Keywords: UDP-گلوکورونوسیل ترانسفراز; Glucuronidation; UDP-glucuronosyltransferase; UGT1A; UGT2B; Saudi gene polymorphism;
Pharmacogenomics: Precision Medicine and Drug Response
Keywords: UDP-گلوکورونوسیل ترانسفراز; CYP; cytochrome P450; EHR; electronic health record; eMERGE; Electronic Medical Records and Genomics; GWAS; genome-wide association study; NGS; next-generation sequencing; NIH; National Institutes of Health; ns; nonsynonymous; PGRN; Pharmacogenomics Resea
Identification and validation of microRNAs directly regulating the UDP-glucuronosyltransferase 1A subfamily enzymes by a functional genomics approach
Keywords: UDP-گلوکورونوسیل ترانسفراز; UGT; UDP-glucuronosyltransferase; 3â²-UTR; 3â²-untranslated region; SNP; single nucleotide polymorphism; miRNA; microRNA; UDPGA; uridine diphosphate glucuronic acid; qPCR; quantitative real-time PCR; MRE; miRNA response element; Ez-Glu; ezetimibe glucur
Simultaneous quantification of estrogens, their precursors and conjugated metabolites in human breast cancer cells by LC-HRMS without derivatization
Keywords: UDP-گلوکورونوسیل ترانسفراز; 3β-HSD; 3β-hydroxysteroiddehydrogenase; 17β-HSD; 17β-hydroxysteroiddehydrogenase; AD; androstenedione; DHEA; dehydroepiandrosterone; DHEA-S; dehydroepiandrosterone-3-sulfate; DMEM; Dulbecco's Modified Eagle Medium F-12; DMSO; dimethylsulfoxide; DPBS;
Effects of diclofenac on the expression of Nrf2 and its downstream target genes in mosquito fish (Gambusia affinis)
Keywords: UDP-گلوکورونوسیل ترانسفراز; PPCPs; pharmaceuticals and personal care products; DCF; diclofenac; tBHQ; tert-butylhydroquinone; Nrf2; NF-E2-related factor 2; NQO-1; NADPH quinine oxidoreductase 1; GCLC; r-glutamylcysteine ligase catalytic subunit; GSTA; alpha-glutathione S-transferase
N-glucuronidation catalyzed by UGT1A4 and UGT2B10 in human liver microsomes: Assay optimization and substrate identification
Keywords: UDP-گلوکورونوسیل ترانسفراز; HLM; human liver microsomes; MS; mass spectroscopy; NNAL; 4-(methylnitrosamino)-1-(3-pyridyl)-1-butanol; QTOF; quadrupole time-of-flight; UDPGA; uridine diphosphoglucuronic acid; UGT; UDP-glucuronosyltransferase; UPLC; ultra performance liquid chromatogra
Comparison of the Predictability of Human Hepatic Clearance for Organic Anion Transporting Polypeptide Substrate Drugs Between Different In Vitro-In Vivo Extrapolation Approaches
Keywords: UDP-گلوکورونوسیل ترانسفراز; active transport; cytochrome P450; glucuronosyltransferase (UGT); hepatic clearance; hepatic transport; hepatocytes; membrane transport/transporters; organic anion transporting polypeptide transporters; transporters; AUC; area under the plasma concentrati
Effects of diammonium glycyrrhizinate on hepatic and intestinal UDP-Glucuronosyltransferases in rats: Implication in herb-drug interactions
Keywords: UDP-گلوکورونوسیل ترانسفراز; Diammonium glycyrrhizinate; UDP-glucuronosyltransferase; Sprague-Dawley rat; Drug-drug interactionGLN, diammonium glycyrrhizinate; GA, glycyrrhetinic acid; DDI, drug-drug interaction; CYPs, cytochrome P450s; UGTs, UDP-glucuronosyltransferases; MMF, mycoph
Homodimerization of UDP-glucuronosyltransferase 2B7 (UGT2B7) and identification of a putative dimerization domain by protein homology modeling
Keywords: UDP-گلوکورونوسیل ترانسفراز; UDP-glucuronosyltransferase; UGT2B7; Homology model; Dimerization; Enzyme kinetics; Glucuronidation
Efavirenz biotransformation as an up-stream event of mood changes in HIV-infected patients
Keywords: UDP-گلوکورونوسیل ترانسفراز; EFV; efavirenz; cART; combined antiretroviral therapy; CNS; central nervous system; CSF; cerebrospinal fluid; CYP; cytochrome P450; UGT; UDP-glucuronosyltransferase; 8-OH-EFV; 8-hydroxy-efavirenz; 7-OH-EFV; 7-hydroxy-efavirenz; 8,14-diOH-EFV; , 8,14-dihyd
The UGT2B28 Sex-steroid Inactivation Pathway Is a Regulator of Steroidogenesis and Modifies the Risk of Prostate Cancer Progression
Keywords: UDP-گلوکورونوسیل ترانسفراز; UDP-glucuronosyltransferase; Prostate cancer prognosis; Disease aggressiveness; Steroid metabolism; Circulating hormone levels;
Transcriptome association analysis identifies miR-375 as a major determinant of variable acetaminophen glucuronidation by human liver
Keywords: UDP-گلوکورونوسیل ترانسفراز; ALF; acute liver failure; NAPQI; N-acetyl-p-benzoquinone imine; UGT; UDP-glucuronosyltransferase; SULT; sulfotransferase; CYP; cytochrome P450; 3â²-UTR; 3â²-untranslated region; SNP; single nucleotide polymorphism; miRNA; microRNA; UDPGA; uridine diphos
Reduction of p53 by Knockdown of the UGT1 Locus in Colon Epithelial Cells Causes an Increase in Tumorigenesis
Keywords: UDP-گلوکورونوسیل ترانسفراز; Apoptosis; Colon Cancer; ER Stress; UGT1A; AOM; azoxymethane; CRC; colorectal cancer; DSS; dextran sodium sulfate; ER; endoplasmic reticulum; IEC; intestinal epithelial cells; IL; interleukin; MTT; 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium brom
Chenodeoxycholic acid significantly impacts the expression of miRNAs and genes involved in lipid, bile acid and drug metabolism in human hepatocytes
Keywords: UDP-گلوکورونوسیل ترانسفراز; ABC; ATP-binding cassette transporter; AGPAT2; 1-acylglycerol-3-phosphate O-acyltransferase; AhR; arylhydrocarbon receptor; AKR1C1; aldo-keto reductase 1C1; APO; apolipoprotein; ASBT; apical sodium dependent bile acid transporter; BAs; bile acids; BSEP; b
CommentaryRoles of human UDP-glucuronosyltransferases in clearance and homeostasis of endogenous substrates, and functional implications
Keywords: UDP-گلوکورونوسیل ترانسفراز; UDP-glucuronosyltransferase; Bilirubin; Serotonin; 20-HETE; Vitamins A and D; AhR; aryl hydrocarbon receptor; CAR; constitutive androstane receptor; HETE; hydroxyeicosatetraenoic acid; LTB4; leucotriene B4; PPAR; peroxisome proliferator-activated receptor