Practical one-pot protocol for the syntheses of 2-chloro-pyrrolo[3,2-d]pyrimidines

A novel one-pot protocol for the syntheses of 2-chloro-pyrrolo[3,2-d]pyrimidines was described. A series of 2-chloro-pyrrolo[3,2-d]pyrimidines were prepared from readily available starting materials in moderate to good yields using this methodology.

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