Keywords: آگونیست ها; Type 2 diabetes mellitus; Agonists; Fatty acids; G protein-coupled receptor; Insulin secretion;
مقالات ISI آگونیست ها (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: آگونیست ها; Nuclear receptors; Inverse docking; Agonists; Endocrine disrupting activities;
Keywords: آگونیست ها; Histamine; H1-H4 receptors; Agonists; Antagonists;
Keywords: آگونیست ها; Leptin; Leptin receptor; Leptin receptor modulators; Agonists; Antagonists; Leptin-related diseasesObR, leptin receptor; G-CSF, Granulocyte Colony-Stimulating Factor; BBB, blood–brain barrier; ER-α, estrogen receptor alpha; IGF-I, insulin-like growth fact
Keywords: آگونیست ها; Glycogen synthase kinase 3; Phosphorylation; Agonists; Signal transduction; Neutrophils;
Keywords: آگونیست ها; Antihypertensive activity; AT2 receptor; Agonists; Biphenyl-2-sulfonamide derivatives; Structure-activity relationships;
Keywords: آگونیست ها; 5-HT1A receptor; Agonists; 1,3-Dioxolane; Selectivity
Identification of novel agonists and antagonists of the ecdysone receptor by virtual screening
Keywords: آگونیست ها; Ecdysone receptor; Agonists; Antagonists; Molecular docking; Molecular dynamic simulation; Virtual screening;
Synthesis and biological activities of indolizine derivatives as alpha-7 nAChR agonists
Keywords: آگونیست ها; α7 nAChR; Indolizine; Agonists; SAR; Schizophrenia; ACh; acetylcholine; THF; tetrahydrofuran; DMSO; dimethylsulfoxide; CNS; central nervous system; HRMS; high resolution mass; DIPEA; diisopropylethylamine; AChBP; acetylcholine binding protein; SAR; struc
The discovery of potent agonists for GPR88, an orphan GPCR, for the potential treatment of CNS disorders
Keywords: آگونیست ها; GPR88; GPC; Agonists; CNS; Schizophrenia
Development of neuropeptide analogs capable of traversing the integument: A case study using diapause hormone analogs in Helicoverpa zea
Keywords: آگونیست ها; Diapause hormone; Agonists; Topical application; Diapause prevention;
Phenoxymethyl 1,3-oxazoles and 1,2,4-oxadiazoles as potent and selective agonists of free fatty acid receptor 1 (GPR40)
Keywords: آگونیست ها; Anti-diabetic agents; Hypoglycemia; Glucose-stimulated insulin secretion; Free fatty acid receptor agonists; Hit expansion; Agonists; ADME profile; Cytochrome inhibition;
Discovery and optimization of 5-(2-((1-(phenylsulfonyl)-1,2,3,4-tetrahydroquinolin-7-yl)oxy)pyridin-4-yl)-1,2,4-oxadiazoles as novel gpr119 agonists
Keywords: آگونیست ها; GPR119; Agonists; Oxadiazole; Constrain; Free fraction;
Effects of adrenoceptor compounds on larval metamorphosis of the mussel Mytilus coruscus
Keywords: آگونیست ها; Mytilus coruscus; Larval metamorphosis; Adrenoceptor; Agonists; Antagonists; Chemical cue;
Targeting integrins αvβ3 and α5β1 with new β-lactam derivatives
Keywords: آگونیست ها; Lactams; Integrins; Azetidinones; Peptidomimetics; Agonists; Cell adhesion
Ligands of the neuropeptide Y Y2 receptor
Keywords: آگونیست ها; Neuropeptide Y; Y2 receptor; Antagonists; Agonists; Structure-activity relationships; Brain-penetration; Non-peptidic;
Estrogen receptors alpha (ERα) and beta (ERβ): Subtype-selective ligands and clinical potential
Keywords: آگونیست ها; ER, estrogen receptor; ERα, estrogen receptor subtype alpha; ERβ, estrogen receptor subtype beta; LBD, ligand binding domain; RBA, relative binding affinityEstrogen receptor subtype α; Estrogen receptor subtype β; Modulators; Agonists; Antagonists; Therap
A history of the role of the hERG channel in cardiac risk assessment
Keywords: آگونیست ها; hERG; human ether-a-go-go-related gene; TdP; torsades de pointes; TQT; thorough QT trial; Agonists; Blockers; hERG; Methods; Modeling; Patch clamp; Trafficking;
Biochemical and histopathological evaluation of histamine receptors (H1R, H2R, H3R and H4R)-agonist in rabbits
Keywords: آگونیست ها; Histamine; Histamine receptors; Agonists; Toxicology; Liver; Rabbit
The role of nuclear receptors in controlling the fine balance between proliferation and differentiation of neural stem cells
Keywords: آگونیست ها; Orphan nuclear receptors; Agonists; Self-renewal; Neurogenesis; Astrogliogenesis; Neurodegeneration
Thieno[3,2-b]thiophene-2-carboxylic acid derivatives as GPR35 agonists
Keywords: آگونیست ها; GPR35; Thieno[3,2-b]thiophene-2-carboxylic acid; Agonists;
Small molecule tertiary amines as agonists of the nuclear hormone receptor Rev-erbα
Keywords: آگونیست ها; Nuclear hormone receptor; Agonists; Drug discovery; Medicinal chemistry; SAR;
Modulation biologique des radiations ionisantes par les agonistes des Toll-like receptors : vers une amélioration de l'index thérapeutique de la radiothérapie ?
Keywords: آگونیست ها; agonistes des TLR; flagelline; index thérapeutique; modulation de la radiosensibilité; radiothérapie; récepteurs Toll-like; Toll-like receptors; agonists; radiotherapy; therapeutic index; flagellin; radiosensitivity modulation;
Meta-analysis of the relationship between ractopamine and dietary lysine levels on carcass characteristics in pigs
Keywords: آگونیست ها; Agonists; Body composition; Meat; Metabolism; Swine; β-adrenergics
Receptor-mediated transcytosis: A mechanism for active extravascular transport of nanoparticles in solid tumors
Keywords: آگونیست ها; Nanoparticles; Melanocortin type-1 receptor (MC1R); Transcytosis; Agonists; Antagonists
Inhibition de la lactation dans le post-partum : bromocriptine versus cabergoline
Keywords: آگونیست ها; Agonistes dopaminergiques; Bromocriptine; Cabergoline; Inhibition lactation; Post-partum; Bromocriptine; Cabergoline; Agonists; D2 dopamine receptor; Puerperium;
AMPK in myocardial infarction and diabetes: the yin/yang effect
Keywords: آگونیست ها; Ischemia-reperfusion injury; Myocardial infarction; AMPK; Myocardial ischemia; Diabetes; Agonists; Glucose homeostasis
TLRs as pharmacological targets for plant-derived compounds in infectious and inflammatory diseases
Keywords: آگونیست ها; Toll like receptors; Agonists; Antagonists; Plant derived compounds;
In silico analysis of the binding of agonists and blockers to the β2-adrenergic receptor
Keywords: آگونیست ها; G protein-coupled receptor; Agonists; Blockers; Induced Fit; Docking; Linear discriminant analysis; Molecular dynamics
Selective and potent agonists for estrogen receptor beta derived from molecular refinements of salicylaldoximes
Keywords: آگونیست ها; Estrogen; Receptor binding; Agonists; Salicylaldoxime; Docking; ER; estrogen receptor; ERα; estrogen receptor subtype alpha; ERβ; estrogen receptor subtype beta; LBD; ligand binding domain; RBA; relative binding affinity; RTP; relative transcriptional p
Microwave-assisted synthesis of quinoline, isoquinoline, quinoxaline and quinazoline derivatives as CB2 receptor agonists
Keywords: آگونیست ها; Receptors; Agonists; Cannabinoid receptor 2; Quinoline; Isoquinoline; Quinoxaline; Quinazoline; Microwave irradiation
Receptor agonists of macrophage migration inhibitory factor
Keywords: آگونیست ها; MIF; Cytokine; Agonists; Structure-based design; AMPK activation; ERK phosphorylation; Click chemistry
Acetylcholine as a possible signaling molecule in embryonic stem cells: Studies on survival, proliferation and death
Keywords: آگونیست ها; Non-neuronal cholinergic; Acetylcholine; Agonists; Embryonic stem cells; Drug effects; Cell vitality
Synthesis of 7-benzyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c][2,7]naphthyridin-1-ylamine and its analogs as bombesin receptor subtype-3 agonists
Keywords: آگونیست ها; Bombesin receptor subtype-3; Agonists; Small molecule
Novel sulfamoyl benzamides as selective CB2 agonists with improved in vitro metabolic stability
Keywords: آگونیست ها; CB2; Agonists; Analgesics
Does Neoadjuvant Hormonal Therapy Improve Urinary Function When Given to Men With Large Prostates Undergoing Prostate Brachytherapy?
Keywords: آگونیست ها; prostate; urinary retention; brachytherapy; agonists; organ sizeHT, hormone therapy; I-PSS, International Prostate Symptom Score; NHT, neoadjuvant HT; PSA, prostate specific antigen; PV, prostate volume; TURP, transurethral resection of the prostate; UD30
SERMs and SARMs: Detection of their activities with yeast based bioassays
Keywords: آگونیست ها; Agonists; Antagonists; In vitro bioassays; Androgenic activity; Estrogenic activity; Metabolism
Synthesis and structure-activity relationships of N-aryl-piperidine derivatives as potent (partial) agonists for human histamine H3 receptor
Keywords: آگونیست ها; Histamine H3 receptor; Agonists;
Synthesis and dual PPARα/δ agonist effects of 1,4-disubstituted 1,2,3-triazole analogues of GW 501516
Keywords: آگونیست ها; Triazoles; GW 501516; Agonists; PPARα; PPARδ; Multiwell assay
2-Amino-9-aryl-3-cyano-4-methyl-7-oxo-6,7,8,9-tetrahydropyrido[2′,3′:4,5]thieno[2,3-b]pyridine derivatives as selective progesterone receptor agonists
Keywords: آگونیست ها; Progesterone; Progesterone receptor; Agonists; Selective agonists; Nuclear receptor; Endometriosis
Selective, potent PPARγ agonists with cyclopentenone core structure
Keywords: آگونیست ها; Nuclear receptors; PPARs; Agonists; Cyclopentenones; Prostaglandins
Morpholine containing CB2 selective agonists
Keywords: آگونیست ها; Cannabinoid receptor; Anti-inflammatory; CB1; CB2; Agonists; Selectivity
Molecular orbital differentiation of agonist and antagonist activity in the GlycineB-iGluR-NMDA receptor
Keywords: آگونیست ها; HOMO; LUMO; Agonists; Antagonist; GlycineB-iGluR-NMDA; Activity
Altered peptide ligands can modify the Th2 T cell response to the immunodominant 161-175 peptide of LACK (Leishmania homolog for the receptor of activated C kinase)
Keywords: آگونیست ها; LACK; Leishmania; Flanking residues; Core determinant; Altered peptide ligands; Agonists; I-Ad; T cell receptor; Th1/Th2
Synthesis and biological evaluation of p-carborane bisphenols and their derivatives: Structure–activity relationship for estrogenic activity
Keywords: آگونیست ها; Estrogen receptor; Agonists; Carborane; Phenols; Structure–activity relationship
Novel and potent small-molecule urotensin II receptor agonists
Keywords: آگونیست ها; Urotensin II; Agonists; SAR; R-SAT; Parallel synthesis
Novel delta opioid receptor agonists exhibit differential stimulation of signaling pathways
Keywords: آگونیست ها; Delta opioid receptor; Agonists; Differential stimulation; Selectivity
Endothelial permeability is controlled by spatially defined cytoskeletal mechanics: Atomic force microscopy force mapping of pulmonary endothelial monolayer
Keywords: آگونیست ها; Pulmonary endothelium; Permeability; Agonists; Actin cytoskeleton; Force mapping
Kainate receptors: Pharmacology, function and therapeutic potential
Keywords: آگونیست ها; Kainate receptors; Agonists; Antagonists; LTP; Synaptic plasticity; Therapeutic potential;
Arylsulfonamide CB2 receptor agonists: SAR and optimization of CB2 selectivity
Keywords: آگونیست ها; Arylsulfonamide; Cannabinoid receptor; CB1; CB2; Agonists; Selectivity