Keywords: مقررات آلوستریک; AC-42; 4-(4-Butyl-1-piperidinyl)-1-(2-methylphenyl)-1-butanone hydrochloride; ACh; acetylcholine; AM; allosteric modulator; BQCA; Benzyl quinolone carboxylic acid; ECL; extracellular loop; FRET; Förster resonance energy transfer; F-V curve; Function -
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Keywords: مقررات آلوستریک; DC; decoding center; PTC; peptidyl transferase center; EF; elongation factor; tRNA; transfer RNA; mRNA; messenger RNA; rRNA; ribosomal RNA; A; aminoacyl; P; peptidyl; E; exit; RF; release factor; Allosteric regulation; Bacterial ribosome; Coarse-graining;
Keywords: مقررات آلوستریک; metabolic engineering; protein engineering; regulation; metabolism; allosteric regulation; control;
Keywords: مقررات آلوستریک; Allosteric regulation; Allosteric pathway; Cooperativity; Enzyme kinetics; Methylglyoxal synthase; Oligomeric protein;
Keywords: مقررات آلوستریک; Glucocorticoid receptor; Glucocorticoid evolution; Allosteric regulation; Alligator; Xenopus; Chicken
Keywords: مقررات آلوستریک; Metabolic control analysis; Allosteric regulation; Metabolic networks; Kinetic models; Kinetic modeling; Prediction performance; Systems metabolic engineering;
Keywords: مقررات آلوستریک; Oryza sativa; Gramineae; Allosteric regulation; Enzyme activation; Fructose-1,6-biphosphate; Glucose-6-phosphate; Oxalate oxidase; Substrate inhibition (of enzymes);
Keywords: مقررات آلوستریک; SAXS, small-angle X-ray scattering; SIC, selected-ion chromatogramDNA methylation; DNMT1; epigenetics; allosteric regulation; autoinhibition
Keywords: مقررات آلوستریک; Homeopathy; High-dilutions; Hormesis; Cell biology; Systems biology; Similia rule; Energy landscape; Allosteric regulation; Pharmacodynamics; Receptors;
Keywords: مقررات آلوستریک; Conformational selection; Induced fit; Single enzyme; Allosteric regulation; In silico drug design; De novo protein synthesis;
Keywords: مقررات آلوستریک; BTP; 1,3-bis[tris(hydroxymethyl)methylamino]propane; DAH7P; 3-deoxy-d-arabino-heptulosonate 7-phosphate; DAH7PS; 3-deoxy-d-arabino-heptulosonate 7-phosphate synthase; E4P; d-erythrose 4-phosphate; PDB; protein data bank; PEG; polyethylene glycol; SAXS; sm
Keywords: مقررات آلوستریک; PK; pyruvate kinase; ITC; isothermal titration calorimetry; NADH; β-Nicotinamide adenine dinucleotide reduced disodium salt hydrate; LDH type II; L-Lactic Dehydrogenase from rabbit muscle; ADP; adenosine diphosphate; PEP; phosphoenolpyruvate; Phe; phenyl
Increased transcript levels and kinetic function of pyruvate kinase during severe dehydration in aestivating African clawed frogs, Xenopus laevis
Keywords: مقررات آلوستریک; Allosteric regulation; Anaerobiosis; Gluconeogenesis; Glycolysis; Metabolism; Reversible protein phosphorylation;
Development of a phosphorylated Momordica charantia protein system for inhibiting susceptible dose-dependent C. albicans to available antimycotics: An allosteric regulation of protein
Keywords: مقررات آلوستریک; Antimycotic-susceptible C. albicans; Fungal growth inhibition; Phosphorylated Momordica charantia protein; Circular dichroism spectroscopy; Allosteric regulation;
Magnesium and calcium ions differentially affect human serine racemase activity and modulate its quaternary equilibrium toward a tetrameric form
Keywords: مقررات آلوستریک; ATP; adenosine triphosphate; ADP; adenosine diphosphate; AMP; adenosine monophosphate; hSR; human serine racemase; AMw; apparent molecular weight; TEA; triethanolamine; LDH; lactate dehydrogenase; Serine racemase; Allosteric regulation; Metal-protein inte
Structural insights into the activation mechanisms of human HtrA serine proteases
Keywords: مقررات آلوستریک; HtrA proteins; Serine proteases; Allosteric regulation; PDZ domain;
Gating role of His 72 in TmPurL enzyme uncovered by structural analyses and molecular dynamics simulations
Keywords: مقررات آلوستریک; TmPurL; PurL from Thermotoga maritima; StPurL; PurL from Salmonella typhimurium; FGAR; formylglycinamide ribonucleotide; IGP; imidazole glycerol phosphate; GMP; guanosine monophosphate; Glutamine amidotransferases; Wing gate; Ammonia channel; Molecular dy
A highly active bile salt hydrolase from Enterococcus faecalis shows positive cooperative kinetics
Keywords: مقررات آلوستریک; Bile salt hydrolase; Gut organism; Bile acids; Allosteric regulation; Penicillin V acylase; Enzyme kinetics;
Membrane and inhibitor interactions of intracellular phospholipases A2
Keywords: مقررات آلوستریک; Phospholipase A2; PAPC; Catalytic cycle; Allosteric regulation; Eicosanoid pathway; Molecular dynamics simulations; DXMS;
Structure of γ-tubulin small complex based on a cryo-EM map, chemical cross-links, and a remotely related structure
Keywords: مقررات آلوستریک; Microtubule nucleation; Allosteric regulation; Integrative modeling; Computational structure prediction; Comparative models;
A conserved two-step binding for the UAF1 regulator to the USP12 deubiquitinating enzyme
Keywords: مقررات آلوستریک; Deubiquitinating enzyme; Allosteric regulation; Protein structure; Small angle X-ray scattering (SAXS); Surface Plasmon Resonance (SPR); Enzyme catalysis;
Regulatory network of the allosteric ATP inhibition of E. coli phosphofructokinase-2 studied by hybrid dimers
Keywords: مقررات آلوستریک; Allosteric regulation; Subunits interactions; Hybrid enzyme dimers; Phosphofructokinase-2; Allosteric communication;
Discovery of novel nonpeptide allosteric inhibitors interrupting the interaction of CDK2/cyclin A3 by virtual screening and bioassays
Keywords: مقررات آلوستریک; Cell cycle; Allosteric regulation; CDK2 allosteric inhibitors; Virtual screening;
Intracellular Ca2+ oscillations generated via the extracellular Ca2+-sensing receptor (CaSR) in response to extracellular Ca2+ or l-phenylalanine: Impact of the highly conservative mutation Ser170Thr
Keywords: مقررات آلوستریک; Ca2+ oscillations; Amino acid signaling; CaSR mutant S170T; Allosteric regulation
Systematic discovery of molecular probes targeting multiple non-orthosteric and spatially distinct sites in the botulinum neurotoxin subtype A (BoNT/A)
Keywords: مقررات آلوستریک; Molecular probes; Non-orthosteric binding; Botulinum toxin; Molecular docking; Biomarkers; Allosteric regulation; Holistic binding
Structural and evolutionary divergence of cyclic nucleotide binding domains in eukaryotic pathogens: Implications for drug design
Keywords: مقررات آلوستریک; Cyclic nucleotide signaling; Allosteric regulation; Phylogeny; Bioinformatics; Evolution; Pathogenic variation
Subunit interfaces contribute differently to activation and allosteric modulation of neuronal nicotinic acetylcholine receptors
Keywords: مقررات آلوستریک; Nicotinic acetylcholine receptors; Allosteric regulation; Mutagenesis site specific; Cysteine-mediating cross-linking; Interface; Oocyte; Cys-loop receptors; nAChR; nicotinic acetylcholine receptor; Mor; morantel; Oxa; oxantel; OR2; oocyte Ringer's; DTT;
Distinct structural features of Rex-family repressors to sense redox levels in anaerobes and aerobes
Keywords: مقررات آلوستریک; Transcription regulation; Anaerobic fermentation; DNA binding protein; Rossmann fold; Winged helix domain; Allosteric regulation;
Mapping the UDP-N-acetylglucosamine regulatory site of human glucosamine-6P synthase by saturation-transfer difference NMR and site-directed mutagenesis
Keywords: مقررات آلوستریک; Glucosamine-6-phosphate synthase; UDPGlcNAc binding site; Glutamine amidotransferase; STD-NMR; Allosteric regulation; Transferred NOE; Fru6P; d-fructose-6-phosphate; Glc6P; d-glucose-6-phosphate; GlcN6P; d-glucosamine-6-phosphate; hGfat; human l-glutamine
Dimerization-induced allostery in protein kinase regulation
Keywords: مقررات آلوستریک; dimerization; allosteric regulation; protein kinases; pseudokinase
An alternative allosteric regulation mechanism of an acidophilic l-lactate dehydrogenase from Enterococcus mundtii 15-1A
Keywords: مقررات آلوستریک; B.; Bacillus; Bf.; Bifidobacterium; CD; circular dichroism; FBP; fluctose-1,6-bisphosphate; Ec.; Enterococcus; E.; Escherichia; LDH; lactate dehydrogenase; LAB; lactic acid bacteria; Lb.; Lactobacillus; Lc.; Lactococcus; rms; root mean square; VUV; vacuum
Structure of N-acetyl-l-glutamate synthase/kinase from Maricaulis maris with the allosteric inhibitor l-arginine bound
Keywords: مقررات آلوستریک; AAK; amino acid kinase; GNAT; GCN5-related acetyltransferase; mmNAGS/K; Maricaulis maris N-acetyl-l-glutamate synthase/kinase; mmNAGS/K-Arg; mmNAGS/K bound with l-arginine; mmNAGS/K-CoA; mmNAGS/K bound with CoA; NAG; N-acetyl-l-glutamate; NAGK; N-acetyl-l
PAOPA, a potent dopamine D2 receptor allosteric modulator, prevents and reverses behavioral and biochemical abnormalities in an amphetamine-sensitized preclinical animal model of schizophrenia
Keywords: مقررات آلوستریک; PAOPA; Allosteric regulation; Dopamine D2 receptor; Schizophrenia; Amphetamine; Animal models;
Deciphering the kinetic mechanisms controlling selected plant ADP-glucose pyrophosphorylases
Keywords: مقررات آلوستریک; Maize; ADP-glucose pyrophosphorylase; Enzyme kinetics; Allosteric regulation; Mechanism;
The potato tuber, maize endosperm and a chimeric maize-potato ADP-glucose pyrophosphorylase exhibit fundamental differences in Pi inhibition
Keywords: مقررات آلوستریک; ADP-glucose pyrophosphorylase; Phosphate inhibition; Mechanism; Allosteric regulation
Allosteric Controls of Nuclear Receptor Function in the Regulation of Transcription
Keywords: مقررات آلوستریک; DBD, DNA binding domain; LBD, ligand binding domain; RE, response element; RID, receptor interacting domain; GRE, GR binding sitenuclear receptors; allosteric regulation
Reciprocal enzyme regulation as a source of bistability in covalent modification cycles
Keywords: مقررات آلوستریک; Allosteric regulation; Post-translational modification; Total quasi-steady state approximation; Symmetry; Modularity
Nucleotide allosteric regulation of the glutamate dehydrogenases of Teladorsagia circumcincta and Haemonchus contortus
Keywords: مقررات آلوستریک; Haemonchus contortus; Teladorsagia (Ostertagia) circumcincta; Glutamate dehydrogenase (E.C. 1.4.1.3); Allosteric regulation; Nucleotides
Ligand binding and structural changes associated with allostery in yeast NAD+-specific isocitrate dehydrogenase
Keywords: مقررات آلوستریک; Isocitrate dehydrogenase; Tricarboxylic acid cycle; Allosteric regulation; Half-site ligand binding; Disulfide bond
Structural and functional characterization of α-isopropylmalate synthase and citramalate synthase, members of the LeuA dimer superfamily
Keywords: مقررات آلوستریک; Allosteric regulation; Branched chain amino acid biosynthesis; Isopropylmalate synthase; Citramalate synthase; Hydrogen/deuterium exchange; LeuA dimer domain
Novel mutator mutants of E. coli nrdAB ribonucleotide reductase: Insight into allosteric regulation and control of mutation rates
Keywords: مقررات آلوستریک; Ribonucleotide reductase; dNTP pools; DNA replication fidelity; Allosteric regulation;
Toward understanding the molecular basis for chemical allosteric modulator design
Keywords: مقررات آلوستریک; Allosteric regulation; Allosteric modulators; Structural rigidity; “Allosteric-like” rule
Acidic pH promotes oligomerization and membrane insertion of the BclXL apoptotic repressor
Keywords: مقررات آلوستریک; Protein oligomerization; Molten globule; Membrane insertion; Ligand binding; Allosteric regulation;
Regulation of the structure and activity of pyruvate carboxylase by acetyl CoA
Keywords: مقررات آلوستریک; Acetyl CoA; Pyruvate carboxylase; Allosteric regulation; Biotin
A marriage full of surprises; forty-five years living with glutamate dehydrogenase
Keywords: مقررات آلوستریک; Glutamate dehydrogenase; Kinetic mechanism; Allosteric regulation; Homotropic effectors; Negative cooperativity; Subunit asymmetry; Protein engineering; Hybrid hexamers
Inverse agonist-like action of cadmium on G-protein-gated inward-rectifier K+ channels
Keywords: مقررات آلوستریک; Allosteric regulation; Crystallography; Electrophysiology; G-protein; Inward rectifier K+ channel
Integrating molecular dynamics and co-evolutionary analysis for reliable target prediction and deregulation of the allosteric inhibition of aspartokinase for amino acid production
Keywords: مقررات آلوستریک; Aspartokinase; Allosteric regulation; Molecular dynamics simulation; Statistical coupling analysis
UMP kinase from Mycobacterium tuberculosis: Mode of action and allosteric interactions, and their likely role in pyrimidine metabolism regulation
Keywords: مقررات آلوستریک; UMPK; Cooperative kinetics; Allosteric regulation; Pyrimidine metabolism; Thermodynamic binding parameters; Antitubercular drug target;
Disruption of quaternary structure in Escherichia coli dihydrodipicolinate synthase (DHDPS) generates a functional monomer that is no longer inhibited by lysine
Keywords: مقررات آلوستریک; Dihydrodipicolinate synthase; Protein stability; Enzyme kinetics; Allosteric regulation; Lysine biosynthesis; Oligomerization
The interaction of azurin and C-terminal domain of p53 is mediated by nucleic acids
Keywords: مقررات آلوستریک; Azurin; p53; Nucleic acid; Allosteric regulation; Anticancer