Keywords: فعالیت ضد انعقادی; Mice; Valproic acid; Anticonvulsant activity; Seizure intensity; Circadian rhythm;
مقالات ISI فعالیت ضد انعقادی (ترجمه نشده)
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Synthesis and anticonvulsant activity of some 2-pyrazolines derived from chalcones
Keywords: فعالیت ضد انعقادی; Chalcones; 2-Pyrazolines; Carbothioamide; Carboxyamide; Anticonvulsant activity;
Keywords: فعالیت ضد انعقادی; Epilepsy; Behavior; Anticonvulsant activity; Rosmarinic acid; Anxiolytic activity; Comorbidities;
Keywords: فعالیت ضد انعقادی; Succinimides; Anticonvulsant activity; Antinociceptive properties; Anesthetic activity; Ion channels
Keywords: فعالیت ضد انعقادی; Anticonvulsant activity; Formalin; Oxaliplatin; Motor coordination; Ion channel binding; Pyrrolidine-2; 5-dione
Keywords: فعالیت ضد انعقادی; Pyrrolidine-2,5-dione; Succinimide; Anticonvulsant activity; In vivo studies; MES test; scPTZ test; Six-Hertz (6 Hz) test; Hybrid compounds
Keywords: فعالیت ضد انعقادی; 2,3-Dioxoindolin-1-acetamide; Synthesis; Anticonvulsant activity; Antidepressant activity; Pentylenetetrazole
Keywords: فعالیت ضد انعقادی; Anticonvulsant activity; Antinociceptive properties; Succinimides; In vivo and in vitro studies; Mutagenicity and antimutagenicity studies;
Keywords: فعالیت ضد انعقادی; Epilepsy; Anticonvulsant activity; Pyrrolidin-2-one derivatives
Keywords: فعالیت ضد انعقادی; Benzisoxazole; Pyrrolidine-2, 5-dione; Anticonvulsant activity; Quantification studiesOTVYFOWEWOAQAW-UHFFFAOYSA-N; VSRWWPQVUDBNNU-UHFFFAOYSA-N
Keywords: فعالیت ضد انعقادی; Histamine; GPCR; H3 receptor; Pharmacophore elements; Epilepsy; Anticonvulsant activity; Convulsion; Phenytoin
Keywords: فعالیت ضد انعقادی; Indazole; 1,3,4-Thiadiazoles; Anticonvulsant activity; Neurotoxicity;
Keywords: فعالیت ضد انعقادی; Pyrrolidine-2,5-dione; Anticonvulsant activity; In vivo studies
Keywords: فعالیت ضد انعقادی; Anxiolytic activity; Anticonvulsant activity; Rota rod; Sodium pentobarbital-induced sleeping time
Evaluation of anticonvulsant and analgesic activity of new hybrid compounds derived from N-phenyl-2-(2,5-dioxopyrrolidin-1-yl)-propanamides and -butanamides
Keywords: فعالیت ضد انعقادی; Anticonvulsant activity; Six-herz (6 Hz) test; Pain models; Binding; Hybrid compounds; Pyrrolidine-2,5-dione;
5,6-Dihydropyrimidine-1(2H)-carbothioamides: Synthesis, in vitro GABA-AT screening, anticonvulsant activity and molecular modelling study
Keywords: فعالیت ضد انعقادی; Pyrimidine; Carbothioamides; GABA-AT; Anticonvulsant activity; In vitro;
Synthesis and evaluation of anticonvulsant properties of new N-Mannich bases derived from pyrrolidine-2,5-dione and its 3-methyl-, 3-isopropyl, and 3-benzhydryl analogs
Keywords: فعالیت ضد انعقادی; Pyrrolidine-2,5-dione; N-Mannich bases; Anticonvulsant activity;
Early preclinical evaluation of dihydropyrimidin(thi)ones as potential anticonvulsant drug candidates
Keywords: فعالیت ضد انعقادی; Anticonvulsant activity; Dihydropyrimidin(thi)ones; Epilepsy; Toxicity;
Design, synthesis, anticonvulsant evaluation and docking study of 2-[(6-substituted benzo[d]thiazol-2-ylcarbamoyl)methyl]-1-(4-substituted phenyl)isothioureas
Keywords: فعالیت ضد انعقادی; Benzothiazoles; Anticonvulsant activity; GABA-A; Toxicity; Molecular docking; Structure-activity relationship;
p-TSA-catalyzed one-pot synthesis and docking studies of some 5H-indeno[1,2-b]quinoline-9,11(6H,10H)-dione derivatives as anticonvulsant agents
Keywords: فعالیت ضد انعقادی; 5H-Indeno[1,2-b]quinoline; One pot; p-toluene sulfonic acid (p-TSA); Anticonvulsant activity; Molecular docking
Synthesis, characterization and pharmacological screening of novel benzimidazole derivatives
Keywords: فعالیت ضد انعقادی; Benzimidazole; Anticonvulsant activity; Pharmacological screening;
Design, synthesis and anticonvulsant activity of new hybrid compounds derived from N-phenyl-2-(2,5-dioxopyrrolidin-1-yl)-propanamides and -butanamides
Keywords: فعالیت ضد انعقادی; Pyrrolidine-2,5-dione; Hybrid compounds; Anticonvulsant activity; In vivo studies; In vitro studies
Anticonvulsant activity, crystal structures, and preliminary safety evaluation of N-trans-cinnamoyl derivatives of selected (un)modified aminoalkanols
Keywords: فعالیت ضد انعقادی; Anticonvulsant activity; Cinnamamide; Crystal structure; Mutagenicity; Hepatotoxicity; VGKGECXRGHIYEU-BQYQJAHWSA-N; GJPZZIANRWWLDZ-ZHACJKMWSA-N; VFXFJIKUTQKGSR-CMDGGOBGSA-N; BEAPCLFCORNJAQ-VOTSOKGWSA-N; WAGNUSGHQMACQN-BQYQJAHWSA-N; KSQWDMMEWCUHHC-VAWYXSNF
Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy)alkyl]- and N-{2-[2-(phenoxy)ethoxy]ethyl}aminoalkanols as anticonvulsant agents
Keywords: فعالیت ضد انعقادی; VGGMLGZQRUZPAC-HQKYYOGZSA-N; SORDYQMTTXQNIQ-CQSZACIVSA-NAminoalkanols; Anticonvulsant activity; Seizures; Sigma receptors; 5-HT; MES; Metabolic stability; Mutagenicity; Vibrio harveyi; Pharmacokinetics
Antinociceptive properties of N-Mannich bases derived from 3-substituted pyrrolidine-2,5-dione in the formalin model of persistent pain in mice
Keywords: فعالیت ضد انعقادی; Pyrrolidine-2,5-dione; Anticonvulsant activity; Central sensitization of pain; Formalin model of tonic pain; Licking response
Synthesis, anticonvulsant activity and molecular modeling study of some new hydrazinecarbothioamide, benzenesulfonohydrazide, and phenacylacetohydrazide analogues of 4(3H)-quinazolinone
Keywords: فعالیت ضد انعقادی; Synthesis; 4(3H)-Quinazolinones; Anticonvulsant activity; Molecular modeling study
Design, synthesis and biological evaluation of new hybrid anticonvulsants derived from N-benzyl-2-(2,5-dioxopyrrolidin-1-yl)propanamide and 2-(2,5-dioxopyrrolidin-1-yl)butanamide derivatives
Keywords: فعالیت ضد انعقادی; Pyrrolidine-2,5-dione; Hybrid compounds; Anticonvulsant activity; In vivo studies; In vitro studies; Metabolic stability;
N-[(2,6-Dimethylphenoxy)alkyl]aminoalkanols-their physicochemical and anticonvulsant properties
Keywords: فعالیت ضد انعقادی; IAUIETVLERVGPI-VEKYKZPFSA-N; 6Â Hz; Ames test; Aminoalkanols; Anticonvulsant activity; Crystal structure; DSC; MES; Mutagenicity; Rotarod; Seizures; TG; TOX;
Anticonvulsant activity of Morusin isolated from Morus alba: Modulation of GABA receptor
Keywords: فعالیت ضد انعقادی; Anticonvulsant activity; Morusin; Isoniazid; Maximum electroshock; GABA
Synthesis and anticonvulsant activity of some new pyrazolo[3,4-b]pyrazines and related heterocycles
Keywords: فعالیت ضد انعقادی; Pyrazolo[3,4-b]pyrazines; Oxadiazoles; Thiadiazoles; Imidazothiadiazoles; Thiazolidinones; Anticonvulsant activity;
Prediction of potent therapeutic anticonvulsant ligands to N-methyl-d-aspartate receptors among substituted 4,6-dichloroindole-2-carboxylic acids: Molecular modeling approach
Keywords: فعالیت ضد انعقادی; 4,6-Dichloroindole-2-carboxylic acids; QSAR; Pharmacophore; NMDA receptor; Anticonvulsant activity
Neuropharmacological screening of essential oil from oleo gum resin of Gardenia lucida Roxb
Keywords: فعالیت ضد انعقادی; Gardenia lucida; Rubiaceae; Essential oil; Anticonvulsant activity; CNS depressant activity;
New imidazo[1,2-a]pyridines carrying active pharmacophores: Synthesis and anticonvulsant studies
Keywords: فعالیت ضد انعقادی; Imidazo[1,2-a]pyridine; Anticonvulsant activity; Toxicology;
Synthesis and evaluation of pharmacological properties of some new xanthone derivatives with piperazine moiety
Keywords: فعالیت ضد انعقادی; 5-HT; Adrenergic receptors; Anticonvulsant activity; Epilepsy; 1,4-Piperazine derivatives; MES; Serotoninergic receptors; Xanthone;
Design, synthesis and anticonvulsant properties of new N-Mannich bases derived from 3-phenylpyrrolidine-2,5-diones
Keywords: فعالیت ضد انعقادی; N-Mannich bases; 3-Phenylpyrrolidine-2,5-diones; Succinimides; Anticonvulsant activity; In vivo studies; In vitro studies; Epilepsy;
Augmentation of GABAergic neurotransmission by novel N-(substituted)-2-[4-(substituted)benzylidene]hydrazinecarbothioamides-A potential anticonvulsant approach
Keywords: فعالیت ضد انعقادی; Hydrazinecarbothioamides; Anticonvulsant activity; Neurotoxicity; Docking; GABA assay;
Novel limonene and citral based 2,5-disubstituted-1,3,4-oxadiazoles: A natural product coupled approach to semicarbazones for antiepileptic activity
Keywords: فعالیت ضد انعقادی; 1,3,4-Oxadiazoles; Semicarbazones; Limonene; Citral; Anticonvulsant activity
Structure–activity relationships of the aromatic site in novel anticonvulsant pyrrolo[1,2-a]pyrazine derivatives
Keywords: فعالیت ضد انعقادی; 2,6-Diketopiperazine; 2,6-Piperazinedione; Pyrrolo[1,2-a]pyrazine; Anticonvulsant activity; Multicomponent reactions; Ugi reaction
Synthesis and anticonvulsant activity of new phenytoin derivatives
Keywords: فعالیت ضد انعقادی; Phenytoin; Oxadiazole; Thiadiazole; Triazole; Anticonvulsant activity
Design, synthesis and evaluation of dialkyl 4-(benzo[d][1,3]dioxol-6-yl)-1,4-dihydro-2,6-dimethyl-1-substituted pyridine-3,5-dicarboxylates as potential anticonvulsants and their molecular properties prediction
Keywords: فعالیت ضد انعقادی; Benzofurazanyl; Benzo[d][1,3]dioxo-6-yl; 1,4-Dihydropyridine; Anticonvulsant activity; Antinociceptive activityBNQLHFJUQIIXHT-UHFFFAOYSA-N; QWUKZVHTUUICOM-UHFFFAOYSA-N; MPQJJXRGOXYEOP-UHFFFAOYSA-N
Synthesis and biological properties of new N-Mannich bases derived from 3-methyl-3-phenyl- and 3,3-dimethyl-succinimides. Part V
Keywords: فعالیت ضد انعقادی; Anticonvulsant activity; Mannich bases; Succinimides; 3,3-Disubstituted-pyrrolidine-2,5-diones; In vivo studies; In vitro studies; Sodium channels; Vibrio harveyi assay
Design, synthesis and anticonvulsant evaluation of N-(benzo[d]thiazol-2-ylcarbamoyl)-2-methyl-4-oxoquinazoline-3(4H)-carbothioamide derivatives: A hybrid pharmacophore approach
Keywords: فعالیت ضد انعقادی; Benzothiazole; 4-Oxoquinazoline-3(4H)-carbothioamide; Anticonvulsant activity; Neuroprotection; AMPA induced seizureDHANPQHXXULONF-UHFFFAOYSA-N; QABFTVHENPQHIO-UHFFFAOYSA-N
Synthesis, anticonvulsant and neurotoxicity evaluation of some new pyrimidine-5-carbonitrile derivatives
Keywords: فعالیت ضد انعقادی; Cyanopyrimidine; Schiff’s base; Anticonvulsant activity; Neurotoxicity; Lipophilicity
Synthesis and anticonvulsant activity of novel 2,6-diketopiperazine derivatives. Part 2: Perhydropyrido[1,2-a]pyrazines
Keywords: فعالیت ضد انعقادی; 2,6-diketopiperazine; 2,6-piperazinedione; Pyrido[1,2-a]pyrazine; Anticonvulsant activity; Chirality
Synthesis and anticonvulsant activity of ethyl 1-(2-arylhydrazinecarboxamido)-2,2-dimethylcyclopropanecarboxylate derivatives
Keywords: فعالیت ضد انعقادی; 1-(2-Arylhydrazinecarboxamido)-2,2-dimethylcyclopropanecarboxylate; Anticonvulsant activity; MES test; scPTZ test;
Synthesis of some novel 1-(2-naphthyl)-2-(imidazol-1-yl)ethanone oxime ester derivatives and evaluation of their anticonvulsant activity
Keywords: فعالیت ضد انعقادی; Oxime ester; (arylalkyl)imidazole; Azole derivatives; Anticonvulsant activity; E/Z isomers;
Synthesis and anticonvulsant evaluation of dimethylethanolamine analogues of valproic acid and its tetramethylcyclopropyl analogue
Keywords: فعالیت ضد انعقادی; Valproic acid esteric and amide deraivatives; Anticonvulsant activity; Maximal electroshock seizure test; Subcutaneous metrazol seizure test; Pharmacokinetic-pharmacodynamic correlation;
Synthesis and anticonvulsant activity of 1-(8-(benzyloxy)quinolin-2-yl)-6-substituted-4,6-diazaspiro[2,4]heptane-5,7-diones
Keywords: فعالیت ضد انعقادی; 1-(8-(Benzyloxy)quinolin-2-yl-6-substituted-4,6-diazaspiro[2,4]heptane-5,7-diones; Anticonvulsant activity; MES test; scPTZ test
Synthesis and anticonvulsant activity of new N-Mannich bases derived from 3-(2-fluorophenyl)- and 3-(2-bromophenyl)-pyrrolidine-2,5-diones. Part II
Keywords: فعالیت ضد انعقادی; N-Mannich bases; 3-Phenyl-pyrrolidine-2,5-diones; Succinimides; Anticonvulsant activity
Synthesis, anticonvulsant activity and 5-HT1A/5-HT7 receptors affinity of 1-[(4-arylpiperazin-1-yl)-propyl]-succinimides
Keywords: فعالیت ضد انعقادی; anticonvulsant activity; 5-HT1A/5-HT7 receptor ligands; 3,3-disubstituted pyrrolidine-2,5-diones; arylpiperazines