Keywords: بیوسیسترها; Dasatinib derivatives; Bioisosteres; Triazole; Oxadiazole; Colony formation; Cell migration;
مقالات ISI بیوسیسترها (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: بیوسیسترها; Antibiotics; Bioisosteres; Inhibitors; Ligases; Drug design
Synthesis and antinociceptive evaluation of bioisosteres and hybrids of naproxen, ibuprofen and paracetamol
Keywords: بیوسیسترها; Bioisosteres; Hybrids; NSAIDs; Nociception; Inflammation; Formalin test;
Scaffold-hopping from xanthines to tricyclic guanines: A case study of dipeptidyl peptidase 4 (DPP4) inhibitors
Keywords: بیوسیسترها; Bioisosteres; Tricyclic guanine; DPP4 inhibitor; FAP inhibitor;
Fluoro-substituted phenylazocarboxamides: Dopaminergic behavior and N-arylating properties for irreversible binding
Keywords: بیوسیسترها; Covalent ligands; Bioisosteres; Azocarboxamide; Dopamine; D3 receptor; GPCR
Design and synthesis of new bioisosteres of spirooxindoles (MI-63/219) as anti-breast cancer agents
Keywords: بیوسیسترها; Spirooxindoles; MDM2-p53; Bioisosteres; Breast cancer; Anticancer agents;
Oseltamivir hydroxamate and acyl sulfonamide derivatives as influenza neuraminidase inhibitors
Keywords: بیوسیسترها; Influenza; Neuraminidase inhibitor; Oseltamivir; Bioisosteres; Hydroxamate; Acyl sulfonamide;
Synthesis of new N-(arylcyclopropyl)acetamides and N-(arylvinyl)acetamides as conformationally-restricted ligands for melatonin receptors
Keywords: بیوسیسترها; Melatonin; MT1 and MT2 receptors; Bioisosteres; Constrained ligands; Agonism;
Tetrazole and triazole as bioisosteres of carboxylic acid: Discovery of diketo tetrazoles and diketo triazoles as anti-HCV agents
Keywords: بیوسیسترها; Anti-HCV activity; Diketo tetrazoles; Diketo triazoles; Bioisosteres
Design and synthesis of 3,5-disubstituted boron-containing 1,2,4-oxadiazoles as potential combretastatin A-4 (CA-4) analogs
Keywords: بیوسیسترها; 3,5-Disubstituted 1,2,4-oxadiazole; Combretastatin A-4; Bioisosteres; Vascular disrupting agent; Tubulin; Boron-containing CA4 compound;
Hepatitis C NS5B polymerase inhibitors: Functional equivalents for the benzothiadiazine moiety
Keywords: بیوسیسترها; Hepatitis C; NS5B polymerase inhibitors; Benzothiadiazine; Bioisosteres
Structure-guided design and synthesis of P1â² position 1-phenylcycloalkylamine-derived pentapeptidic BACE1 inhibitors
Keywords: بیوسیسترها; Alzheimer's disease; β-Secretase; Pentapeptides; Bioisosteres; Phenylcycloalkylamines;
Design of pentapeptidic BACE1 inhibitors with carboxylic acid bioisosteres at P1′ and P4 positions
Keywords: بیوسیسترها; Alzheimer disease; β-Secretase; Inhibitors; Bioisosteres; Structure–activity relationship
Delta agonist hydroxy bioisosteres: The discovery of 3-((1-benzylpiperidin-4-yl){4-[(diethylamino)carbonyl]phenyl}amino)benzamide with improved delta agonist activity and in vitro metabolic stability
Keywords: بیوسیسترها; Delta agonism; Bioisosteres; Metabolic stability
Phosphorous acid analogs of novel P2–P4 macrocycles as inhibitors of HCV–NS3 protease
Keywords: بیوسیسترها; Hepatitis C; HCV; NS3; Protease inhibitor; Bioisosteres; Phosphonate; MK7009
Bacterial translation inhibitors, 1-acylindazol-3-ols as anthranilic acid mimics
Keywords: بیوسیسترها; Bioisosteres; Translation inhibitors; Antibacterials; Indazol; Protein binding
Design, synthesis, and anticonvulsant activity of some sulfamides
Keywords: بیوسیسترها; Sulfamides; Anticonvulsant; Rational design; Bioisosteres; Pharmacophore
Triazolo-tetrahydrofluorenones as selective estrogen receptor beta agonists
Keywords: بیوسیسترها; Tetrahydrofluorenones; SERMs; ERβ-agonists; Bioisosteres
Synthesis and biological evaluation of carboacyclic nucleosides with (Z) and (E)-9-[4,4-bis(hydroxymethyl)]-2-butenyl side chain
Keywords: بیوسیسترها; Carboacyclic; Nucleosides; Antiviral; Bioisosteres
Ketene aminal-based lactam derivatives as a novel class of orally active FXa inhibitors
Keywords: بیوسیسترها; Serine protease; Factor Xa inhibitors; Antithrombotic agents; 2-Methylbenzofuran; Thiourea; Bioisosteres; N,N′-Disubstituted ketene aminal; 2,2-Dicyanoketene aminal; 2-Nitroketene aminal; Orally active
Design and synthesis of low molecular weight compounds with complement inhibition activity
Keywords: بیوسیسترها; Non-cytotoxic; Carbonyl compounds; Carboxylic acid; Bioisosteres; Tetrazoles; trans-Phenyl acrylic acid; Complement inhibitors; Classical pathway; Hemolysis