Keywords: تیروزین کیناز Bruton; ABC; activated B-cell type; BCM; BCL10, CARD11, MALT complex; BCR; B-cell receptor; BTK; Bruton's tyrosine kinase; CSF; cerebrospinal fluid; GCB; germinal center B-cell type; IL; interleukin; PCNSL; primary central nervous system lymphoma; TLR; toll-lik
مقالات ISI تیروزین کیناز Bruton (ترجمه نشده)
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Keywords: تیروزین کیناز Bruton; Resistin-like molecule; Macrophage; Helminth infection; T helper type 2; Toll-like Receptor 4; ABC; ATP-binding cassette transporter; ADD1; adipocyte determination and differentiation dependent factor 1; ADSF; adipocyte secreted factor; Akt (aka PKB); pro
Keywords: تیروزین کیناز Bruton; ADA; anti-drug antibodies; AMPK; 5â² adenosine monophosphate-activated protein kinase; aHUS; atypical hemolytic uremic syndrome; AMD; age-related macular degeneration; APC; antigen presenting cells; AT; anaphylatoxin; BTK; Bruton's tyrosine kinase; C1q
Keywords: تیروزین کیناز Bruton; S/B; signal to background; PDGFR; platelet-derived growth factor receptor; BTK; Bruton's tyrosine kinase; EGFR; epidermal growth factor receptor; HER-2; human epidermal growth factor 2; AMPK; AMP activated protein kinase; BMPR; bone morphogenetic protei
Transforming growth factor-β1 impairs lymph node homing of dendritic cells by downregulating C-type lectin receptor-2 expression
Keywords: تیروزین کیناز Bruton; c-Src; C-type lectin receptor; Dendritic cell trafficking; Immunosuppressive cytokines; BMDC; bone marrow-derived dendritic cell; Btk; Bruton's tyrosine kinase; CLEC-2; C-type lectin receptor-2; DC; dendritic cell; GM-CSF; granulocyte-macrophage colony-
Conversion of carbazole carboxamide based reversible inhibitors of Bruton's tyrosine kinase (BTK) into potent, selective irreversible inhibitors in the carbazole, tetrahydrocarbazole, and a new 2,3-dimethylindole series
Keywords: تیروزین کیناز Bruton; Bruton's tyrosine kinase; BTK; Indole carboxamide; Carbazole; Irreversible inhibitor;
Design and synthesis of novel pyrimidine analogs as highly selective, non-covalent BTK inhibitors
Keywords: تیروزین کیناز Bruton; Bruton's tyrosine kinase; Kinase inhibitor; Kinase selectivity; Pyrimidine; Passive cutaneous anaphylaxis;
Optimization of permeability in a series of pyrrolotriazine inhibitors of IRAK4
Keywords: تیروزین کیناز Bruton; ABC; Activated B Cell-like; BTK; Bruton's Tyrosine Kinase; CD79; Cluster of Differentiation 79; CDK; Cyclin Dependent Kinase; CLK; CDC-Like Kinase; DCM; dichloromethane; DDQ; 2,3-Dichloro-5,6-DicyanobenzoQuinone; DIPEA; N,N-diisopropylethylamine; DLBCL;
Mitigation of reactive metabolite formation for a series of 3-amino-2-pyridone inhibitors of Bruton's tyrosine kinase (BTK)
Keywords: تیروزین کیناز Bruton; Bruton's tyrosine kinase; BTK; Reactive metabolite; Covalent binding; Glutathione adduct;
The role of chromatographic and chiroptical spectroscopic techniques and methodologies in support of drug discovery for atropisomeric drug inhibitors of Bruton's tyrosine kinase
Keywords: تیروزین کیناز Bruton; Atropisomer; Bruton's tyrosine kinase; Drug discovery; Chiral separation; Circular dichroism; Interconversion;
Imaging the pharmacology of nanomaterials by intravital microscopy: Toward understanding their biological behavior
Keywords: تیروزین کیناز Bruton; ADME; absorption distribution metabolism excretion; BODIPY; borondipyrromethene; BTK; Bruton's tyrosine kinase; CIW; cranial imaging window; DCE-MRI; dynamic contrast enhanced magnetic resonance imaging; DiO/DiI/DiD/DiR; dialkylcarbocyanine dyes; ECM; e
Bruton tyrosine kinase inhibition in chronic lymphocytic leukemia
Keywords: تیروزین کیناز Bruton; Chronic lymphocytic leukemia; B-cell receptor; Bruton's tyrosine kinase; ibrutinib;
'Turn On/Off' fluorescence probe for the screening of unactivated Bruton's tyrosine kinase
Keywords: تیروزین کیناز Bruton; Bruton's tyrosine kinase; Fluorescence probe; Kinase inhibitor; Binding assay;
Finding the perfect spot for fluorine: Improving potency up to 40-fold during a rational fluorine scan of a Bruton's Tyrosine Kinase (BTK) inhibitor scaffold
Keywords: تیروزین کیناز Bruton; Bruton's Tyrosine Kinase; BTK; Structure-based drug design; Fluorine scan; Rational fluorine scan;
Potent and selective Bruton's tyrosine kinase inhibitors: Discovery of GDC-0834
Keywords: تیروزین کیناز Bruton; Kinase inhibitor; Bruton's tyrosine kinase; Btk; Rheumatoid arthritis; GDC-0834; Amide hydrolysis; Single dose IND;
TR-FRET binding assay targeting unactivated form of Bruton's tyrosine kinase
Keywords: تیروزین کیناز Bruton; Bruton's tyrosine kinase; Kinase inhibitor; Screening; Fluorescent probe; TR-FRET;
GCN5 regulates the activation of PI3K/Akt survival pathway in B cells exposed to oxidative stress via controlling gene expressions of Syk and Btk
Keywords: تیروزین کیناز Bruton; AKT; acutely transforming retrovirus AKT8 in rodent T cell lymphoma; BCR; B cell receptor; Btk; Bruton's tyrosine kinase; ChIP; chromatin immunoprecipitation; GCN5; general control non-depressible 5; H2O2; hydrogen peroxide; HAT; histone acetyltransfera