Keywords: دی کلرواساتات; Observer-reported outcome measure; Clinical trial; Rare disease; Dichloroacetate; Pyruvate dehydrogenase complex;
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Keywords: دی کلرواساتات; BG; Blood Glucose; DCA; Dichloroacetate; ECG; Electrocardiography; EGFR; Estimated Glomerular Filtration Rate; FDG; Fluorodeoxyglucose; GKI; Glucose-Ketone Index; GKIC; Glucose-Ketone Index Calculator; HGCM; Highly Glycolytic Cancers and Metastases; KD-R;
Keywords: دی کلرواساتات; AMPK; AMP-activated protein kinase; DCA; Dichloroacetate; FACD; Fatty acyl CoA dehydrogenase; G-6-Pase; Glucose-6-phosphatase; HFD; High-fat diet; HGP; Hepatic glucose production; KCT; β-ketoacyl CoA thiolase; LDH; Lactate dehydrogenase; MPC; Mitochondri
Keywords: دی کلرواساتات; ACSVL3; acyl-coA synthetase VL3; ALDH1; aldehyde dehydrogenase; ALDOA; aldolase A; ALDOC; aldolase C; AMPK; 5â² AMP-activated protein kinase; ASNS; asparagine synthetase; BTICs; brain tumor initiating cells; 3-BrOP; 3-bromo-2-oxopropionate-1-propyl ester
Keywords: دی کلرواساتات; 56MESS; (1S2S-diaminocyclohexane)platinum(II)] dichloride; AIBN; 2,2â²-azobisisobutyronitrile; Apt; aptamer; AUC; area under curve; BBR3464; (trans,trans,trans)-bis-mu-(hexane-16-diamine)-mu-[diammineplatinum(II)]bis[diammine(chloro)platinum(II)] tetrani
Keywords: دی کلرواساتات; DCA; dichloroacetate; FAO; fatty acid oxidation; GO; glucose oxidation; HIF-1; hypoxia-inducible factor 1; CaL channels; L-type calcium channels; NFATs; nuclear factor of activated T cells; NO; nitric oxide; MCT-PAH; monocrotaline-induced PAH; PAH; pulmon
Keywords: دی کلرواساتات; Dichloroacetate; leiomyoma; oxidative stress; apoptosis; myometrium;
Keywords: دی کلرواساتات; CI; Complex I; DCA; dichloroacetate; 2-DG; 2-deoxy-glucose; GDH; glutamate dehydrogenase; GLS; glutaminase; HK; hexokinase; LICs; Leukemia Initiating Cells; MDR; multidrug resistance; mtDNA; mitochondrial DNA; MSCs; mesenchymal stem cells; nDNA; nuclear D
Keywords: دی کلرواساتات; Dichloroacetate; Pyruvate dehydrogenase kinase; GSTZ1; Pharmacogenetics; Pharmacokinetics; Inhibition of metabolism;
Keywords: دی کلرواساتات; DCA; Dichloroacetate; ECAR; extra cellular acidification rate; JC-1; 5,5â²,6,6â²-tetrachloro-1,1â²,3,3â²-tetraethylbenzimidazolycarbocyanine; MMP; ÎÏm, mitochondrial membrane potential; NAD+; Â nicotinamide adenine dinucleotide; NADH; reduced nicoti
Keywords: دی کلرواساتات; AGO; adrenal gland oncocytoma; BHDS; Birt-Hogg-Dubée syndrome; CCRCC; clear cell renal cell carcinoma; CD; mtDNA common deletion; DAP3; death-associated protein 3; DCA; dichloroacetate; ERRα; estrogen-related receptor alpha; ETC; electron transport chai
Keywords: دی کلرواساتات; AAT; aspartate aminotransferase; Ala; alanine; AlaT; alanine aminotransferase; ALD; aldolase; AOA; aminooxyacetate; Asp; aspartate; CS; citrate synthase; 2-DOG; 2-deoxyglucose; DCA; dichloroacetate; DHAP; dihydroxyacetone phosphate; ENO; enolase; Ery4P; e
Keywords: دی کلرواساتات; Metabolic modulation; Pyruvate dehydrogenase kinase; Warburg effect; Dichloroacetate;
Keywords: دی کلرواساتات; M-CSF; macrophage colony-stimulating factor; IFN-γ; interferon-gamma; M-MÏ; macrophage differentiated from CD14 positive monocytes in the presence of M-CSF; Mγ-MÏ; macrophage differentiated from CD14 positive monocytes in the presence of M-CSF and IFN
Keywords: دی کلرواساتات; Measles virus; Persistent infection; Mitochondria; Dichloroacetate
Keywords: دی کلرواساتات; Dichloroacetate; postoperative adhesions; oxidative stress; apoptosis
Keywords: دی کلرواساتات; CRC; colorectal cancer; DCA; dichloroacetate; PDH; pyruvate dehydrogenase; PDK; pyruvate dehydrogenase kinase; MA; mitochondrial activity.; Dichloroacetate; Pyruvate dehydrogenase kinase; Anoxia; Mitochondrial function; Colorectal cancer;
Keywords: دی کلرواساتات; 2-DG; 2-deoxy-D-glucose; CoA; coenzyme A; COX; cytochrome c oxidase; DCA; Dichloroacetate; EMT; epithelial-to-mesenchymal transition; ERR; estrogen-related receptor; ETC; electron transport chain; F1; 6BP, fructose 1,6-bisphosphate; F2; 6BP, fructose-2,6-
Keywords: دی کلرواساتات; 2DG; 2-deoxy-glucose; 6-AN; aminocicotinamide; ABC; ATP-binding cassette transporter; CSCs; cancer stem cells; DCA; dichloroacetate; G6PD; glucose-6-phosphate dehydrogenase; GLUT; glucose transporter; HIF; hypoxia-inducible factors; HK2; hexokinase 2; Kra
Keywords: دی کلرواساتات; HE; hepatic encephalopathy; MHE; minimal hepatic encephalopathy; CLD; chronic liver disease; TCA cycle; tricarboxylic acid cycle; NMR; nuclear magnetic resonance; BDL; bile-duct ligation; DCA; dichloroacetate; PDH; pyruvate dehydrogenase; PC; pyruvate car
Keywords: دی کلرواساتات; Gastric neoplasm; 5-Flurouracil; Hypoxia; Chemoresistance; Pyruvate dehydrogenase kinase; Dichloroacetate
Keywords: دی کلرواساتات; A2870; ovarian cancer cells; A2870cis; cisplatin resistant ovarian cancer cells; A549; lung cancer cells; ABRs; auditory brainstem responses; AUC; area under the curve; AuNP; gold nanoparticles; CDDP or cisplatin; cis-diamminedichloroplatinum(II); Cis-(ch
Keywords: دی کلرواساتات; CSF; cerebrospinal fluid; DCA; dichloroacetate; EDTA; ethylenediaminetetraacetic acid; GSTZ1; glutathione transferase zeta 1; MA; maleylacetone; MAAI; maleylacetoacetate isomerase; MELAS; mitochondrial encephalomyopathy, lactic acidosis and stroke-like ep
Keywords: دی کلرواساتات; APM; antigen processing machinery; BMI; body mass index; CTLs; cytotoxic T-cells; DC; dendritic cells; DCA; dichloroacetate; ERK; extracellular signal-regulated kinases; GTN; glyceryl trinitrate; HAT; histone acetyltransferases; HLA; human leukocyte antig
Novel approaches in the treatment of diabetic cardiomyopathy
Keywords: دی کلرواساتات; ACE; angiotensin convertase enzyme; ACEi; angiotensin convertase enzyme inhibitor; ADP; adenosine di phosphate; AGE; advanced glycation end products; AM; adrenomedullin; AMP; adenosine mono phosphate; ARB; angiotensin receptor blocker; ATP; adenosine tri
Treating patients suffering from myalgic encephalopathy/chronic fatigue syndrome (ME/CFS) with sodium dichloroacetate: An open-label, proof-of-principle pilot trial
Keywords: دی کلرواساتات; Myalgic encephalitis; Chronic fatigue syndrome; Nutriceutical; Dichloroacetate; Fatigue severity scale; Treatment;
Anticancer effects of some novel dichloroacetophenones through the inhibition of pyruvate dehydrogenase kinase 1
Keywords: دی کلرواساتات; PDK; pyruvate dehydrogenase kinase; PDC; pyruvate dehydrogenase complex; MMP; mitochondrial membrane potential; ROS; reactive oxygen species; OXPHOS; oxidative phosphorylation; TCA; tricarboxylic acid; PDPs; pyruvate dehydrogenase phosphatases; DCA; dichl
Glycolysis regulates LPS-induced cytokine production in M2 polarized human macrophages
Keywords: دی کلرواساتات; a.u.; arbitrary unit; C/EBP; CCAAT-enhancer-binding protein; ChIP; chromatin immunoprecipitation; DCA; dichloroacetate; ECAR; extracellular acidification rate; ERK; extracellular signal-regulated kinase; ETO; etomoxir; FAO; fatty acid oxidation; IFNγ; in
Pharmacological synergism of 2,2-dichloroacetophenone and EGFR-TKi to overcome TKi-induced resistance in NSCLC cells
Keywords: دی کلرواساتات; Erlotinib (PubChem CID: 176870); Gefitinib (PubChem CID: 123631); Sodium dichloroacetate (PubChem CID: 517326); 2,2-dichloroacetophenone (PubChem CID: 72870); Synergism; Dichloroacetophenone; Dichloroacetate; EGFR; Apoptosis; Acquired resistance;
Defects in mitochondrial energetic function compels Fanconi Anaemia cells to glycolytic metabolism
Keywords: دی کلرواساتات; AML; acute myeloid leukaemia; AMPK; Adenosine Monophosphate-Activated Protein Kinase; Antimyc; antimycin A; BMF; bone marrow failure; DCA; dichloroacetate; H2DCF; 2â²,7â²-dichlorofluorescein; H2DCFDA; 2â²,7â²-dichlorodihydrofluorescein diacetate; HSC;
Original ArticleAP1G1 is involved in cetuximab-mediated downregulation of ASCT2-EGFR complex and sensitization of human head and neck squamous cell carcinoma cells to ROS-induced apoptosis
Keywords: دی کلرواساتات; AP1G1; ASCT2; EGFR; Endocytosis; Cetuximab; AP1G1; adaptor-related protein complex 1 gamma 1 subunit; ASCT2; alanine-serine-cysteine transporter 2; ATP; adenosine triphosphate; DCA; dichloroacetate; EGFR; epidermal growth factor receptor; GFP; Green fluor
Sensitization of breast cancer cells to paclitaxel by dichloroacetate through inhibiting autophagy
Keywords: دی کلرواساتات; Dichloroacetate; Breast cancer; Autophagy; Chemotherapy;
Deficiencies in mitochondrial dynamics sensitize Caenorhabditis elegans to arsenite and other mitochondrial toxicants by reducing mitochondrial adaptability
Keywords: دی کلرواساتات; OMM; outer mitochondrial membrane; DRP1; dynamin-related protein-1; MFN1; mitofusin 1; MFN2; mitofusin 2; mtDNA; mitochondrial DNA; PINK1; PTEN-induced putative kinase 1; PARK2; parkin; DOA; dominant optic atrophy; CMT2A; Charcot-Marie-Tooth neuropathy ty
Targeting HIF-1α is a prerequisite for cell sensitivity to dichloroacetate (DCA) and metformin
Keywords: دی کلرواساتات; Cancer metabolism; Dichloroacetate; Glycolytic enzymes; HIF-1α; Metformin;
Activation of mitochondrial oxidation by PDK2 inhibition reverses cisplatin resistance in head and neck cancer
Keywords: دی کلرواساتات; HNC; head and neck cancer; DCA; dichloroacetate; CDDP; cisplatin; OXPHOS; oxidative phosphorylation; PDK2; pyruvate dehydrogenase kinase 2; PDHE1α; pyruvate dehydrogenase isoform E1α; ROS; reactive oxygen species; ÎΨm; mitochondrial membrane potential
Anti-cancer synergy of dichloroacetate and EGFR tyrosine kinase inhibitors in NSCLC cell lines
Keywords: دی کلرواساتات; Pyruvate dehydrogenase kinase; Dichloroacetate; Epidermal growth factor Receptor; Erlotinib; Gefitinib; Drug combination
Time-programmed DCA and oxaliplatin release by multilayered nanofiber mats in prevention of local cancer recurrence following surgery
Keywords: دی کلرواساتات; Local cancer recurrence; Local treatment; Multilayered electrospun nanofibers; Time-programmed release; Dichloroacetate; Oxaliplatin;
GSTZ1 expression and chloride concentrations modulate sensitivity of cancer cells to dichloroacetate
Keywords: دی کلرواساتات; [Clâ]; chloride concentration; DCA; dichloroacetate; ERK; extracellular signal-regulated kinase; GSTZ1; glutathione transferase Z1; HER2; human epidermal growth factor receptor 2; PDC; pyruvate dehydrogenase complex; PDK; pyruvate dehydrogenase kinase;
Design, synthesis and anticancer activity of diam(m)ine platinum(II) complexes bearing a small-molecular cell apoptosis inducer dichloroacetate
Keywords: دی کلرواساتات; Platinum complexes; Anticancer activity; Drug resistance; Dichloroacetate
Functional classification and biochemical characterization of a novel rho class glutathione S-transferase in Synechocystis PCC 6803
Keywords: دی کلرواساتات; GST, glutathione S-transferase; GSH, reduced glutathione; DCA, dichloroacetate; CDNB, 1-chloro-2,4-dinitrobenzene; GSTZ, glutathione S-transferase zetaCyanobacteria; Detoxification; Glutathione; Dichloroacetate; Water pollutant; Bioremediation
Dichloroacetate alters Warburg metabolism, inhibits cell growth, and increases the X-ray sensitivity of human A549 and H1299 NSC lung cancer cells
Keywords: دی کلرواساتات; DCA; dichloroacetate; PI; propidium iodide; NSCLC; non-small-cell lung cancer; SBRT; stereotactic body radiation therapy; Dichloroacetate (DCA); Fractionated/split-dose; Non-small cell lung cancer (NSCLC); Double-strand DNA break repair; Warburg effect;
1H NMR metabolomics analysis of the effect of dichloroacetate and allopurinol on breast cancers
Keywords: دی کلرواساتات; Cancer NMR metabolomics; Dichloroacetate; Allopurinol; Pyruvate dehydrogenase kinase Xanthine oxidase;
Dichloroacetate and cancer: New home for an orphan drug?
Keywords: دی کلرواساتات; Dichloroacetate; Cancer; Mitochondria; Pyruvate dehydrogenase complex; Hypoxia inducible factor-1 alpha; Warburg effect;
The Xenopus oocyte: A model for studying the metabolic regulation of cancer cell death
Keywords: دی کلرواساتات; ACC; acetyl CoA carboxylase; DCA; dichloroacetate; FAS; fatty acid synthase; G6P; glucose-6-phosphate; PDH; pyruvate dehydrogenase; PEP; phosphoenolpyruvate; PK; pyruvate kinase; PPP; pentose phosphate pathway; TIGAR; TP53-induced glycolysis and apoptosis
Necrosis of cervical carcinoma by dichloroacetate released from electrospun polylactide mats
Keywords: دی کلرواساتات; Dichloroacetate; Electrospun mats; Metabolism target; ATP depletion; Necrosis;
Spectrum of neurological and survival outcomes in pyruvate dehydrogenase complex (PDC) deficiency: Lack of correlation with genotype
Keywords: دی کلرواساتات; CIDEM; Center for Inherited Disorders of Energy Metabolism; CQ; cognitive quotient; DCA; dichloroacetate; MELAS; mitochondrial encephalomyopathy with lactic acidosis and stroke-like episodes; PDC; pyruvate dehydrogenase complex; TPP; thiamine pyrophosphat
The spectrum of pyruvate dehydrogenase complex deficiency: Clinical, biochemical and genetic features in 371 patients
Keywords: دی کلرواساتات; Congenital lactic acidosis; Dichloroacetate; Neuroimaging; Ketogenic diet; Pyruvate dehydrogenase complex; Thiamine;
The spectrum of pyruvate dehydrogenase complex deficiency: Clinical, biochemical and genetic features in 371 patients
Keywords: دی کلرواساتات; Congenital lactic acidosis; Dichloroacetate; Neuroimaging; Ketogenic diet; Pyruvate dehydrogenase complex; Thiamine;
Prediction of death in the SMNÎ7 mouse model of spinal muscular atrophy: Insight into disease stage and progression
Keywords: دی کلرواساتات; Tissue lactate level; Respiratory rate; Prediction of death; Dichloroacetate; Neonate oral gavages; Motor function; Modeling body weight; Moribund;
Cannabinoid receptor trafficking in peripheral cells is dynamically regulated by a binary biochemical switch
Keywords: دی کلرواساتات; ATTC; American type culture collection; AMAM; anilino-monoindolylmaleimide; CB1; cannabinoid receptor type-1; CB2; cannabinoid receptor type-2; CDx; cluster of differentiation x; CHO; Chinese hamster ovary-K1; CM; cell membrane; CNR1; CB1 receptor gene; C