Keywords: مطالعه داکینگ; Ionic liquids; Pyridazinone-vanillyl; Characterization; Antimicrobial; Docking study;
مقالات ISI مطالعه داکینگ (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: مطالعه داکینگ; Coumarin dimer; Chemically engineered extract; TDDFT calculation; Tyrosinase; Docking study;
Keywords: مطالعه داکینگ; GCGR; glucagon receptor; cAMP; cyclic-adenosine monophosphate; T2DM; type 2 diabetes mellitus; SGLT-2; sodium-glucose cotransporter-2; HGP; hepatic glucose production; GPCRs; G-protein coupled receptors; SAR; structure-activity relationship; Ser; Serine;
Keywords: مطالعه داکینگ; Docking study; Molecular dynamics; Pharmacology;
Keywords: مطالعه داکینگ; Dihydrazones; H+/K+-ATPase; Anti-inflammatory activity; Antioxidants; Docking study;
Keywords: مطالعه داکینگ; Butyrylcholinesterase; Alzheimer's disease; Docking study; Carbazole; In-vitro and In-vivo assay;
Keywords: مطالعه داکینگ; Anti-inflammatory; COX-2 inhibitors; COX-1/COX-2 inhibition; Cyclocoumarol; Cyclooxygenase; Docking study;
Keywords: مطالعه داکینگ; Furan; Thiophene; Carbohydrazides; Carboxamides; Anti-tubercular activity; MABA assay; Docking study;
Keywords: مطالعه داکینگ; Acetamides; Antimicrobial screening; Docking study; Lipophilicity; Molecular interaction; EGFR;
Synthesis of novel chromenones linked to 1,2,3-triazole ring system: Investigation of biological activities against Alzheimer's disease
Keywords: مطالعه داکینگ; Alzheimer's disease; Anti-cholinesterase; Chromenones; Docking study; Neuroprotective activity; β-Secretase inhibitory activity; 1,2,3-Triazole;
Keywords: مطالعه داکینگ; Dimethylaminocurcumin; Antioxidant; Anti-inflammatory; Antibacterial; Docking study
Keywords: مطالعه داکینگ; ADME prediction; Antifungal; Antioxidant; Docking study; 1,2,3-Triazole
Keywords: مطالعه داکینگ; Adamantyl nitroxide; Superoxide scavenging activity; Anticancer; Docking study
Keywords: مطالعه داکینگ; Imidazole derivatives; Antimicrobial activity; Docking study;
Keywords: مطالعه داکینگ; 1,2,3-Triazole; Antitubercular; Antioxidant; Docking study; ADME prediction;
Keywords: مطالعه داکینگ; Acridine-chromenone; Alzheimer’s disease; Anti-cholinesterase; Docking study; Neuroprotective activity; Quinoline-chromenone; β-Secretase inhibitor
Keywords: مطالعه داکینگ; Anticonvulsant agents; Acridone; Benzodiazepine (BZD) receptors; Docking study; 1,2,4-Oxadiazole;
Keywords: مطالعه داکینگ; Acridone; Acetylcholinesterase; Antioxidant activity; Docking study;
Keywords: مطالعه داکینگ; Alzheimer's disease; Acetylcholinesterase; Acridone-1,2,3-triazole; Docking study
Keywords: مطالعه داکینگ; Acetylcholinesterase; Alzheimer's disease; Chroman-4-one; Docking study; Homoisoflavonoids;
Keywords: مطالعه داکینگ; Curcumin; Eudragit EPO; Spray drying; Solid dispersion; Docking study
Keywords: مطالعه داکینگ; Acetylcholinesterase; Alzheimer's disease; Benzofuran; Docking study; Pyridinium;
Keywords: مطالعه داکینگ; Alzheimer's disease; Acetylcholinesterase; Indolinone; Oxindole; Docking study
Keywords: مطالعه داکینگ; Alzheimer's disease; Acetylcholinesterase; Coumarins; Docking study
Keywords: مطالعه داکینگ; Factor Xa; Anticoagulant; Conjugation; Docking study;
Keywords: مطالعه داکینگ; Azides; Strain-promoted cycloaddition; Papain inhibitors; Biosensors; Docking study
Keywords: مطالعه داکینگ; Alzheimer's disease; Acetylcholinesterase; Coumarins; Docking study;
Keywords: مطالعه داکینگ; Salvia syriaca; Acetylcholinesterase; Alzheimer's disease; Docking study; β-sitosterol; Daucosterol
Keywords: مطالعه داکینگ; AhR; TCDD; Homology modeling; Docking study; Pig
Keywords: مطالعه داکینگ; Acetylcholinesterase; Alzheimer's disease; Benzofuran; Docking study; Pyridinium
Keywords: مطالعه داکینگ; 4-anilinoquinoline-3-carboxamide; EGFR-TK inhibitors; Pharmacophore; Docking study; Binding energy; Anti-proliferative activity;
A cascade synthesis, in vitro cholinesterases inhibitory activity and docking studies of novel Tacrine-pyranopyrazole derivatives
Keywords: مطالعه داکینگ; Multicomponent reaction; Tacrine-pyranopyrazole derivatives; Cholinesterase inhibition; Alzheimer's disease; Docking study;
Design, synthesis, biological evaluation, homology modeling and docking studies of (E)-3-(benzo[d][1,3]dioxol-5-ylmethylene) pyrrolidin-2-one derivatives as potent anticonvulsant agents
Keywords: مطالعه داکینگ; (E)-3-(Benzo[d][1,3]dioxol-5-ylmethylene)pyrrolidin-2-one; Design; Synthesis; Anticonvulsant; Homology modeling; Docking study;
Design, synthesis, docking study, α-glucosidase inhibition, and cytotoxic activities of acridine linked to thioacetamides as novel agents in treatment of type 2 diabetes
Keywords: مطالعه داکینگ; α-Glucosidase; Type 2 diabetes; Acridine; Thioacetamide; Docking study;
Design and synthesis of novel coumarin-pyridinium hybrids: In vitro cholinesterase inhibitory activity
Keywords: مطالعه داکینگ; Cholinesterases; Coumarins; Docking study; Kinetic study; Pyridinium salts; β-secretase (BACE1);
Amelioration of postmenopausal osteoporosis and anticancer properties of an antioxidant enriched fraction from Hygrophila spinosa T. Anders
Keywords: مطالعه داکینگ; Antiosteoporotic activity; Antioxidant enriched fraction; Docking study; Hygrophila spinosa; Ovariectomy;
Treatment of cadmium(II) and zinc(II) with N2-donor linkages in presence of β-diketone ligand; supported by structural, spectral, theoretical and docking studies
Keywords: مطالعه داکینگ; Cadmium(II); Nitrogen donor linker; DFT study; Docking study; Coordination polymer;
Discovery of thinopyrimidine-triazole conjugates as c-Met targeting and apoptosis inducing agents
Keywords: مطالعه داکینگ; N-methylpicolinamide; Thienopyrimidine; Triazole; c-Met; Antitumor activity; Docking study; Apoptosis;
Ridaifen-F conjugated with cell-penetrating peptides inhibits intracellular proteasome activities and induces drug-resistant cell death
Keywords: مطالعه داکینگ; Proteasome inhibitor; Tamoxifen derivative; Cell-penetrating peptide; Docking study;
Microwave-assisted synthesis of novel 5-substituted benzylidene amino-2-butyl benzofuran-3-yl-4-methoxyphenyl methanones as antileishmanial and antioxidant agents
Keywords: مطالعه داکینگ; Benzofuran derivatives; Antileishmanial activity; Antioxidant activity; Docking study; ADME properties;
Synthesis and antimycobacterial activity of 1-(β-d-Ribofuranosyl)-4-coumarinyloxymethyl- / -coumarinyl-1,2,3-triazole
Keywords: مطالعه داکینگ; Antimycobacterial; Click chemistry; 1,2,3-Triazole; Cytotoxicity; In silico pharmacokinetics; Docking study;
Novel tetrahydrocarbazole benzyl pyridine hybrids as potent and selective butryl cholinesterase inhibitors with neuroprotective and β-secretase inhibition activities
Keywords: مطالعه داکینگ; Alzheimer's disease; Butyrylcholinesterase; Docking study; 2,3,4,9-Tetrahydro-1H-carbazole; In-vitro assay;
Design and synthesis of BPR1K653 derivatives targeting the back pocket of Aurora kinases for selective isoform inhibition
Keywords: مطالعه داکینگ; Aurora kinase inhibitor; Anticancer agents; Docking study; SAC; spindle assembly checkpoint; CPC; chromosomal passenger complex; pHH3Ser10; phosphorylation on serine 10 of histone H3; MI; mitotic index;
Discovery of anilino-furo[2,3-d]pyrimidine derivatives as dual inhibitors of EGFR/HER2 tyrosine kinase and their anticancer activity
Keywords: مطالعه داکینگ; Furopyrimidine; EGFR/HER2 kinase; In-vivo activity; Flow cytometry; Docking study;
In vivo and in silico sedative-hypnotic like activity of 7-methyljuglone isolated from Diospyros lotus L.
Keywords: مطالعه داکینگ; Medicinal plants; Diospyros lotus L.; 7-methyljuglone; Gaba; Sedative-hypnotic activity; Docking study;
Synthesis and molecular docking study of some 5,6-dichloro-2-cyclopropyl-1H-benzimidazole derivatives bearing triazole, oxadiazole, and imine functionalities as potent inhibitors of urease
Keywords: مطالعه داکینگ; Benzimidazole; 1,2,4-Triazole; Schiff base; Docking study; Antiurease activity;
Discovery of novel cyclic peptide inhibitors of dengue virus NS2B-NS3 protease with antiviral activity
Keywords: مطالعه داکینگ; Dengue virus; Protease inhibitor; Cyclic peptide; Docking study; Antiviral activity;
Isolation and identification of cytotoxic compounds from a fruticose lichen Roccella montagnei, and it's in silico docking study against CDK-10
Keywords: مطالعه داکینگ; Docking study; Roccellic acid; Everninic acid; Cytotoxic activity;
3,4-Dimethoxybenzohydrazide derivatives as antiulcer: Molecular modeling and density functional studies
Keywords: مطالعه داکینگ; Synthesis; 3,4-Dimethoxybenzohydrazide; Urease inhibition; Docking study; Cytotoxicity; DFT; X-rays analysis;
Synthesis, SAR and molecular docking studies of benzo[d]thiazole-hydrazones as potential antibacterial and antifungal agents
Keywords: مطالعه داکینگ; Benzo[d]thiaozole; SAR; Antimicrobial; Docking study;