Keywords: هاتو; CAP; cationic antimicrobial peptide; TM; transmembrane; PPI; protein-protein interaction; Fmoc; Fluorenylmethyloxycarbonyl chloride; DMF; dimethylformamide; DCM; dichloromethane; DIEA; diisopropylethylamine; HATU; 1-[bis(dimethylamino)methylene]-1H-1,2,3-
مقالات ISI هاتو (ترجمه نشده)
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Keywords: هاتو; QPA; quaternary protoberberine alkaloid; TF; transcriptional factor; UC; ulcerative colitis; IEC-6; intestinal epithelial cell-6; XBP1; X-box-binding protein 1; MIC; minimal inhibitory concentration; SAR; structure-activity relationship; SASP; Sulfasalazi
Keywords: هاتو; SI; supporting information; NBD-Cl; 4-chloro-7-nitrobenzofurazan; NBD-OH; 4-hydroxy-7-nitrobenzofurazan; DIC; N,Nâ²-diisopropylcarbodiimide; DMAP; 4-dimethylaminopyridine; DIEA; N,N-diisopropylethylamine; HATU; 1-[bis(dimethylamino)methylene]-1H-1,2,3-tr
Keywords: هاتو; Bub1; budding uninhibited by benzimidazoles 1; Cbz; benzyloxycarbonyl; CD69; a human transmembrane C-Type lectin protein; DAST; diethylaminosulfur trifluoride; dba; dibenzylideneacetone; DIPEA; N,N-diisopropylethylamine; DMAD; dimethyl acetylenedicarboxyl
Keywords: هاتو; AA; amino acid; ABC; accelerated blood clearance; Aib; 2-aminoisobutyric acid; AIBN; azobisisobutyronitrile; Ala; alanine; AMM; activated monomer mechanism; CAC; critical aggregate concentration; Cbz; benzyloxycarbonyl; CD; circular dichroism; CL; caprola
Keywords: هاتو; AF-1; activation function-1; AF-2; activation function-2; AP-1; activator protein 1; dppp; 1,3-bis(diphenylphosphino)propane; DEX; dexamethasone; DIEA; N,N-diisopropylethylamine; FKBP5; FK506-binding protein 5; GR; glucocorticoid receptor; GRE; glucocorti
Identification of highly selective and potent orexin receptor 1 antagonists derived from a dual orexin receptor 1/2 antagonist based on the structural framework of pyrazoylethylbenzamide
Keywords: هاتو; OX1R; orexin 1 receptor; OX2R; orexin 2 receptor; DORA; dual orexin receptor antagonist; SORA; selective orexin receptor antagonist; SI; selectivity index; BBB; blood-brain barrier; CNS; central nervous system; SAR; structure-activity relationship; Boc; t
Keywords: هاتو; ADMET; adsorption distribution metabolism excretion and toxicity; CtD; complexity-to-diversity; DCC; N,Nâ²-dicyclohexylcarbodiimide; DCE; 1,2-dichloroethane; DIPEA; N,Nâ²-diisopropylethylamine; DMAP; 4-dimethylaminopyridine; DMF; N,Nâ²-dimethylformamid
Keywords: هاتو; APTES; 3-aminopropyltrimethoxysilane; AuNPs; gold nanoparticles; CA-graphene/LFP; activated graphene-encapsulated LiFePO4; CTAB; hexadecyltrimethylammonium bromide; CVD; chemical vapour deposition; DCC; (N,Nâ²-dicyclohexylcarbodiimide); DMF; dimethylform
Keywords: هاتو; RNCGDQLZIATDOU-ZDRBWGSPSA-N; ICYPJNZJUFGALC-PDTBJYIYSA-N; PDRMAVOIWIVXKH-SFUSBHMVSA-N; ISADXJRTBSLWPX-ZDRBWGSPSA-N; NLBLLPROASDPSC-QWWZWVQMSA-N; XKMIKZDBUOHHDK-ZDRBWGSPSA-N; BTURADNXKHTWGA-IJOLSIAMSA-N; UEKHRDLXBMZMPD-ZYIYBEKCSA-N; UQCLCXDOXVZEOA-JARUQAPT
Keywords: هاتو; BPO; benzoyl peroxide; DCM; dichloromethane; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; DMSO; dimethyl sulfoxide; FaSSIF; fasted state simulated intestinal fluid; HATU; 1-[bis(dimethylamino)methylene]-1H-1,2,3-triazolo[4,5-b]pyridinium
Keywords: هاتو; Pro-apoptotic agents; Anticancer agents; Cyclic peptides; Peptidomimetics; Nur77; Tubulin; Bcl-2; NMR studies; Molecular modeling; Confocal microscopy; FACS analysis; ADT; AutoDock Tools; COSY; correlation spectroscopy; DBU; 1,8-Diazabicyclo[5.4.0]undec-7
Keywords: هاتو; Cyclic peptides; Microwave assisted synthesis; Lactam-bridge cyclic peptides; SHU9119; MTII; MWA-SPPS; microwave-assisted solid phase peptide synthesis; MBHA; methylbenzhydryl; MCR; melanocortin receptors; NDP; [Nle4, DPhe7]-αMSH; MTII; melanotan-II; RP-
Keywords: هاتو; ATRP; atom-transfer radical-polymerisation; Brij700; polyoxyethylene (100) octadecyl ether; CHAPS; 3-((3-cholamidopropyl)dimethylammonium)-1-propanesulfonate; DBDM; n-dodecyl β-D-maltoside; DCC; N,Nâ²-dicyclohexylcarbodiimide; DLS; dynamic light scatter
Keywords: هاتو; Diversity-oriented synthesis; Imidazoheterocyclic; Groebke-Blackburn-Bienayme reaction; Fused imidazole; Lewis acid; Ugi type; Ac; acetyl; Aq; aqueous; Ar; aryl; Bn; benzyl; Boc; tert-butoxycarbonyl; BDMS; bromodimethylsulfonium bromide; CDK; cyclin-d
Keywords: هاتو; AgOTf; silver triflate; BBB; blood-brain barrier; CDMT; 2-chloro-4,6-bis[3-(perfluorohexyl)propyloxy]-1,3,5-triazine; CNS; central nervous system; DMF; dimethylformamide; EM-2; endomorphin-2; Fmoc; N-(9-fluorenylmethyloxycarbonyl); GPI assay; guinea pig
Microcystins: Synthesis and structure-activity relationship studies toward PP1 and PP2A
Keywords: هاتو; Adda; (2S,3S,8S,9S)-3-amino-9-methoxy-2,6,8-trimethyl-10-phenyldeca-4,6-dienoic acid; Amba; (2S,3S)-3-amino-2-methylbutanoic acid; Boc; tert-butoxycarbonyl; BOP; benzotriazol-1-yloxy-tris-dimethylaminophosphoniumhexafluoro phosphate; Cbz; carboxybenzyl; D
Cathepsin B inhibitors: Further exploration of the nitroxoline core
Keywords: هاتو; Abz; 2-aminobenzoyl; AMC; 7-amido-4-methylcoumarin; catB; cathepsin B; DIPEA; N,N-diisopropylethylamine; DMSO; dimethyl sulfoxide; ECM; extracellular matrix; EDC; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide; HATU; 1-[bis(dimethylamino)methylene]-1H-1,2,
Substrate-derived triazolo- and azapeptides as inhibitors of cathepsins K and S
Keywords: هاتو; Azapeptide; Bradykinin; Cathepsin; 1,2,3-triazole heterocycle; Protease; Protease inhibitor; Abz; o-aminobenzoic acid; Ahx; 6-aminohexanoic acid; AEBSF; 4-(2-aminoethyl) benzenesulfonyl fluoride hydrochloride; AMC; 7-amino-4-methyl coumarin; BK; bradykini
Synthesis and biological evaluation of cyclopeptide GG-8-6 and its analogues as anti-hepatocellular carcinoma agents
Keywords: هاتو; HCC; hepatocellular carcinoma; MDP; muramyl dipeptide; SAR; structure and activity relationship; SPPS; solid phase peptide synthesis; MeOH; methanol; MTT; 3-(4,5-dimethyl-2-thiazolyl)-2,5-diphenyl-2-H-tetrazolium bromide; PI; propidium iodide; VP-16; etop
Design, synthesis, and evaluation of carboxyl-modified oseltamivir derivatives with improved lipophilicity as neuraminidase inhibitors
Keywords: هاتو; NA; neuraminidase; OS; oseltamivir; OC; oseltamivir carboxylate; TFA; trifluor-oacetic acid; HATU; 1-[bis(dimethylamino)methylene]-1H-1,2,3-triazolo[4,5-b]pyr-idinium 3-oxid hexafluorophosphate; DIPEA; N,N-diisopropylethylamine; PDB; protein data bank; In
Evaluation of a novel GRPR antagonist for prostate cancer PET imaging: [64Cu]-DOTHA2-PEG-RM26
Keywords: هاتو; BBN; bombesin; BFCs; bifunctional chelates; BSA; bovine serum albumin; CB-TE2A; 4,11-bis(carboxymethyl)-1,4,8,11-tetraazabicyclo[6.6.2]hexadecane; CH3CN; acetonitrile; C-NE3TA; 4-carboxymethyl-7-[2-(carboxymethyl-amino)-3-(4-nitro-phenyl)-propyl]-[1,4,7]t
N-Thiazolylamide-based free fatty-acid 2 receptor agonists: Discovery, lead optimization and demonstration of off-target effect in a diabetes model
Keywords: هاتو; AUCu; unbound area-under-the-curve; (S)-BINAP; (S)-(-)-(1,1â²-binaphthalene-2,2â²-diyl)bis(diphenylphosphine); CLu; unbound systemic clearance rate; Compd; compound; DIEA; N,N-diisopropyl ethylamine, EtOAc, ethyl acetate; FFA2 receptor; free fatty acid-
Phenylglycine racemization in Fmoc-based solid-phase peptide synthesis: Stereochemical stability is achieved by choice of reaction conditions
Keywords: هاتو; COMU; (1-cyano-2-ethoxy-2-oxoethylidenaminooxy)dimethylaminomorpholinocarbenium hexafluorophosphate; DBU; 1,8-diazabicyclo[5.4.0]undec-7-ene; DEPBT; 3-diethoxyphosphoryloxy)-1,2,3-benzotriazin-4(3H)-one; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethyl
Formation of platinum (II) as a six member ring for sustained polymeric delivery
Keywords: هاتو; Hyaluronic acid; Cisplatin chemotherapy; Lysine; Homo-lysine; Five-membered ring; Six-membered ring; HA; hyaluronic acid; PPG; photoremovable protecting group; pHP; p-hydroxyphenacyl; Fmoc; fluorenylmethoxy-carbonyl; HATU; 2-(1H-7-azabenzotriazol-1-yl)-1,
Activity cliff for 7-substituted pyrrolo-pyrimidine inhibitors of HCK explained in terms of predicted basicity of the amine nitrogen
Keywords: هاتو; EDCI; 1-(3-dimethylaminopropyl)-3-ethylcarbodiimide; HATU; 1-[bis(dimethylamino)methylene]-1H-1,2,3-triazolo[4,5-b]pyridinium 3-oxid hexafluorophosphate; HCK; hematopoietic cell kinase; HOBt; hydroxybenzotriazole; NABH(OAc)3; sodium triacetoxyborohydride;
Coating lanthanide nanoparticles with carbohydrate ligands elicits affinity for HeLa and RAW264.7 cells, enhancing their photodamaging effect
Keywords: هاتو; DIC; 1,3-diisopropylcarbodiimide; DIPEA; N,N-diisopropylethylamine; DLS; dynamic light scattering; DMAP; N,N-dimethyl-4-aminopyridine; DMF; N,N-dimethylformamide; DMEM; Dulbecco's Modified Eagle Medium; EPR effect; enhanced permeability and retention ef
2-Aminomethylthieno[3,2-d]pyrimidin-4(3H)-ones bearing 3-methylpyrazole hinge binding moiety: Highly potent, selective, and time-dependent inhibitors of Cdc7 kinase
Keywords: هاتو; CPME; cyclopentyl methyl ether; DCM; dichloromethane; DMA; N,N-dimethylacetamide; DMAP; 4-dimethylaminopyridine; DME; 1,2-dimethoxyethane; DMF; N,N-dimethylformamide; DMSO; dimethyl sulfoxide; EDCI; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide hydrochlor
Discovery of spiro[indole-3,2â²-pyrrolidin]-2(1H)-one based inhibitors targeting Brr2, a core component of the U5 snRNP
Keywords: هاتو; CDCl3; deuterated chloroform; DHX29; DEAH-Box helicase 29 (an ATP-dependent RNA helicase); DIPEA; N,Nâ²-diisopropylethylamine; DMSO-d6; dimethyl sulfoxide-d6; EDC·HCl; 1-(3-(dimethylamino)propyl)-3-ethylcarbodiimide hydrochloride; eIF4A1; eukaryotic ini
Studies of CDK 8/19 inhibitors: Discovery of novel and selective CDK8/19 dual inhibitors and elimination of their CYP3A4 time-dependent inhibition potential
Keywords: هاتو; ADME; absorption, distribution, metabolism, and excretion; AML; acute myelogenous leukemia; AUC; area under the blood concentration time curve; b.i.d.; twice a day; CDK; Cyclin-dependent kinase; CLtotal; clearance; Cmax; maximum drug concentration; CRC; c
New amphiphilic neamine conjugates bearing a metal binding motif active against MDR E. aerogenes Gram-negative bacteria
Keywords: هاتو; Antibacterial activity; Gram-negative bacteria; Metal-binding groups; Membrane permeability; Multidrug resistant bacteria; Neamine derivatives; HOAt; 1-hydroxy-7azabenzotriazole; HATU; 1-[Bis(dimethylamino)methylene]-1H-1,2,3-triazolo[4,5-b]pyridinium-3-o
Anorexigenic effects induced by RVD-hemopressin(α) administration
Keywords: هاتو; ACN; acetonitrile; AgRP; agouti related peptide; ARC; arcuate nucleus; BAT; brown adipose tissue; CART; cocaine and amphetamine-regulated transcript; CRH; corticotrophin releasing hormone; DA; dopamine; DCM; dichloromethane; DIPEA; N,N-Diisopropylethylami
Ser422 phosphorylation blocks human Tau cleavage by caspase-3: Biochemical implications to Alzheimer's Disease
Keywords: هاتو; Aa; amino acid; ACN; acetonitrile; AUFS; absorbance units full scale; CHCA; 1-Cyano 4-Hydroxy Cinnamic Acid; Da; Dalton; DHB; 2,5-dihydroxy benzoic acid; DMF; N,Nâ²-dimethyl formamide; EDT; ethane dithiol; h; human; HATU; 1-[Bis(dimethylamino)methylene]-
Facile synthesis of indole-pyrimidine hybrids and evaluation of their anticancer and antimicrobial activity
Keywords: هاتو; Indole; Pyrimidine; HATU; Claisen-Schmidt condensation; Anticancer activity; Antimicrobial studies;
Design and synthesis of fused bicyclic inhibitors targeting the L5 loop site of centromere-associated protein E
Keywords: هاتو; DIPEA; N,N-diisopropylethylamine; HATU; hexafluorophosphate O-(7-azabenzotriazol-1-yl)-N,N,Nâ²,Nâ²-tetramethyluronium; PD; pharmacodynamic; CENP-E; Electrostatic potential map (EPM); 2,3-Dihydro-1-benzothiophene 1,1-dioxide derivatives; Anti-cancer agen
Fragment-wise design of inhibitors to 3C proteinase from enterovirus 71
Keywords: هاتو; HFMD; hand, foot and mouth disease; 3Cpro; 3C proteinase; EV71; enterovirus 71; HRV; human rhinovirus; NMR; nuclear magnetic resonance; RP-HPLC; reverse phase-high pressure liquid chromatography; TFA; trifluoroacetic acid; LC; liquid chromatography; MS; m
Synthesis and biological activities of indolizine derivatives as alpha-7 nAChR agonists
Keywords: هاتو; α7 nAChR; Indolizine; Agonists; SAR; Schizophrenia; ACh; acetylcholine; THF; tetrahydrofuran; DMSO; dimethylsulfoxide; CNS; central nervous system; HRMS; high resolution mass; DIPEA; diisopropylethylamine; AChBP; acetylcholine binding protein; SAR; struc
Two fluid sources and genetic implications for the Hatu gold deposit, Xinjiang, China
Keywords: هاتو; Fluid inclusions; Stable isotopes; Noble gas isotopes; Gold deposit; Hatu; Xinjiang
Discovery of antitumor anthra[2,3-b]furan-3-carboxamides: Optimization of synthesis and evaluation of antitumor properties
Keywords: هاتو; Anthra[2,3-b]furan-3-carboxamides; DNA ligands; Topoisomerase inhibitors; Protein kinase inhibitors; Cytotoxicity; Circumvention of multidrug resistance; Antitumor activity; CDI; 1,1â²-carbonyldiimidazole; DCC; N,Nâ²-dicyclohexylcarbodiimide; EDC; 1-eth
Design and synthesis of new potent anticancer benzothiazole amides and ureas featuring pyridylamide moiety and possessing dual B-RafV600E and C-Raf kinase inhibitory activities
Keywords: هاتو; Anticancer activity; Benzothiazole; Urea; Amide; Pyridylamide; B-RafV600E; C-Raf; ATCC; American tissue culture collection; CDI; 1,1'-carbonyldiimidazole; CLogP; Calculated LogP (Partition coefficient); DIPEA; N,N-diisopropylethylamine; DTT; Dithiothreito
Definition of an 18-mer Synthetic Peptide Derived from the GB virus C E1 Protein as a New HIV-1 Entry Inhibitor
Keywords: هاتو; Acm; acetamidomethyl; ACN; acetonitrile; Dbz; diaminobenzoyl; DHB; 2,5-dihydroxybenzoic acid; DIPEA; diisopropylethylamine; FP; fusion peptide; GBV-C; GB virus C; HAART; highly active antiretroviral therapy; HATU; 2-(1H-7-azabenzotriazole-1-yl)-1,1,3,3-te
Synthesis and biological evaluation of the [d-MeAla11]-epimer of coibamide A
Keywords: هاتو; Hva; α-hydroxyisovaleric acid; HATU; O-(7-azabenzotriazol-1-yl)-1,1,3,3-tetramethyluronium hexafluorophosphate; BTC; bis(trichloromethyl) carbonate; DIC; 1,3-diisopropylcarbodiimide; HOBt; 1-hydroxybenzotriazole; HOAt; 1-hydroxy-7-azabenzotriazole; TFA;
Design and synthesis of novel bivalent ligands (MOR and DOR) by conjugation of enkephalin analogues with 4-anilidopiperidine derivatives
Keywords: هاتو; ACN; Acetonitrile; Boc; tert-butyloxycarbonyl; CHO; Chinese hamster ovary; DCM; Dichloromethane; DIPEA; N,N-Diisopropylethylamine; DALEA; [D-Ala2, Leu5] enkephalin amide; DAMGO; [D-Ala2,NMePhe4,Gly5-ol]enkephalin; Dmt; 2,6-dimethyltyrosine; DPDPE; c[D-Pen
Design, synthesis and evaluation of a gonadotropin releasing hormone-based subunit vaccine in rams (Ovis aries)
Keywords: هاتو; AcOH; acetic acid; Ac2O; acetic anhydride; ANOVA; analysis of variance; BSA; bovine serum albumin; BW; body weight; C16; 2-amino-d,l-hexadecanoic acids; DCM; dichloromethane; DMF; dimethyl formamide; DIPEA; N,N-diisopropylethylamine; EDTA; ethylenediamine
Design, synthesis, pharmacological characterization of a fluorescent agonist of the P2Y14 receptor
Keywords: هاتو; DXQJLXWZLNCEJX-VBCGWZPHSA-N; BODIPY; boron-dipyrromethene; cAMP; 3â²,5â²-cyclic adenosine monophosphate; CHO; Chinese hamster ovary; COMU; [[(Z)-(1-cyano-2-ethoxy-2-oxoethylidene)amino]oxy-morpholin-4-ylmethylidene]-dimethylazanium hexafluorophosphate;
Synthesis, structural characterization and effect on human granulocyte intracellular cAMP levels of abscisic acid analogs
Keywords: هاتو; ABA; abscisic acid; [cAMP]i; intracellular cAMP concentration; [cADPR]i; intracellular cADPR concentration; HATU; O-(7-azabenzotriazol-1-yl)-1,1,3,3 tetramethyluroniumhexafluorophosphate; NaBH4; sodiumborohydride; DIBAL; diisobutylaluminium hydride; Absci
Specific in vitro binding of a new 99mTc-radiolabeled derivative of the C-terminal decapeptide of prothymosin alpha on human neutrophils
Keywords: هاتو; Aca; aminocaproic acid (6 amino-hexanoic acid); AcS; acetylated serine; dmGly; dimethylglycine; EDT; ethanedithiol; FC; flow cytometry; fMLP; N-formyl-methionine-leucine-phenylalanine; HATU; 1-[Bis(dimethylamino)methylene]-1H-1,2,3-triazolo[4,5-b]pyridini
Synthesis and SAR studies of analogues of 4-(3,3-dimethyl-butyrylamino)-3,5-difluoro-N-thiazol-2-yl-benzamide (Lu AA41063) as adenosine A2A receptor ligands with improved aqueous solubility
Keywords: هاتو; HATU; 2-(1H-7-azabenzotriazol-1-yl)-1,1,3,3-tetramethyluronium hexafluorophosphate; EDC; N-ethyl-Nâ²-dimethylaminopropyl-carbodiimide hydrochloride; HOBt; 1-hydroxy-benzotriazole; DMAP; 4-dimethylaminopyridine; DMF; dimethylformamide; DMSO; dimethyl sulf
The importance of the 6- and 7-positions of tetrahydroisoquinolines as selective antagonists for the orexin 1 receptor
Keywords: هاتو; BOP; (benzotriazol-1-yloxy)tris(dimethylamino)phosphonium hexafluorophosphate; HATU; 1-[bis(dimethylamino)methylene]-1H-1,2,3-triazolo[4,5-b]pyridinium 3-oxid hexafluorophosphate; HPLC; high performance liquid chromatography; OX1; orexin 1 receptor; OX2;
Discovery of benzothiazoles as antimycobacterial agents: Synthesis, structure-activity relationships and binding studies with Mycobacterium tuberculosis decaprenylphosphoryl-β-d-ribose 2â²-oxidase
Keywords: هاتو; TB; tuberculosis; Mtb; Mycobacterium tuberculosis; MIC; minimal inhibitory concentration; CYP; cytochrome P450; SAR; structure-activity relationships; MMIC; mammalian cytotoxicity; DprE1; decaprenylphosphoryl-β-d-ribose 2â²-oxidase; TEA; triethylamine