Synthesis and SAR studies of analogues of 4-(3,3-dimethyl-butyrylamino)-3,5-difluoro-N-thiazol-2-yl-benzamide (Lu AA41063) as adenosine A2A receptor ligands with improved aqueous solubility

Synthesis and SAR studies of analogues of 4-(3,3-dimethyl-butyrylamino)-3,5-difluoro-N-thiazol-2-yl-benzamide (Lu AA41063) as adenosine A2A receptor ligands with improved aqueous solubility

Database: Elsevier - ScienceDirect (ساینس دایرکت)
Journal: Bioorganic & Medicinal Chemistry Letters - Volume 25, Issue 6, 15 March 2015, Pages 1212-1216

Gitte Kobberøe Mikkelsen, Morten Langgård, Tenna Juul Schrøder, Mads Kreilgaard, Erling B. Jørgensen, Guillaume Brandt, Yann Griffon, Ray Boffey, Benny Bang-Andersen,