Keywords: Biphalin; Opioid receptors; MOR/DOR/KOR agonist; Synergistic analgesic effect; Cyclic peptides; Acm; acetamidomethyl; ACN; acetonitrile; BBB; blood brain barrier; Boc; t-butyloxycarbonyl; BOP; (benzotriazol-1-yloxytris(dimethylamino)phosphonium hexafluoro
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Keywords: 1H NMR; 1H -nuclear magnetic resonance spectroscopy; 13C NMR; 13C-nuclear magnetic resonance spectroscopy; TCM; traditional Chinese medicine; HRMS; high-resolution mass spectral; HOBt; 1-hydroxy, benzotriazole, hydrate; EDCI; 1-(3-dimethylaminopropyl)-3-e
Keywords: SMP; starfish myorelaxant peptide; SAR; structure-activity relationships; PP; pedal peptide; OK; orcokinin; ACh; acetylcholine; TFA; trifluoroacetic acid; RP; reversed-phase; HOBT; 1-hydroxybenzotriazole; DIPCI; N,N-diisopropylcarbodimide; ASW; artificial
Keywords: Boc; tert-butyloxycarbonyl; DMAP; 4-dimethylaminopyridine; DCM; dichloromethane; DMF; dimethylformamide; DMSO; dimethyl sulfoxide; EDCI; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide; HIV; human immunodeficiency virus; HOBt; hydroxybenzotriazole; HR-ESI;
Keywords: HOBt; hydroxybenzotriazole; EDCl; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide; DMF; N-N-dimethyl formamide; s; singlet; 5-FU; 5-fluorouracil; P. falciparum; Plasmodium falciparum; SI; Selectivity Index; TLC; Thin Layer Chromatography; IR; infra-red; NMR
Keywords: CS; chitosan; DFT; density functional theory; FTBH; Formaldehyde tert-butyl hydrazone; HOBt; 1-Hydroxybenzotriazole hydrate; TBME; tert-Butyl methyl ether; TMSCN; Trimethylsilyl cyanide; Acetophenone (PubChem CID: 7410); Ethyl benzoylformate (PubChem CID:
Keywords: Azulene; Orexin receptor; Potentiator; Agonist; Antagonist; Sleep-wake regulation; BINAP; 2,2â²-bis(diphenylphosphino)-1,1â²-binaphthyl; CHO; Chinese hamster ovary (cells); dppf; 1,1â²-bis(diphenylphosphino)ferrocene; EDC; 1-ethyl-3-(3-dimethylaminopro
Keywords: PDT; photodynamic therapy; GSH; glutathione; ROS; reactive oxygen species; TME; tumor microenvironment; ZnPc-DTP; 2(3), 9(10), 16(17), 23(24)-Tetra-(3-(2-Pyridyldithio)propionic acid) aminophenoxy) phthalocyaninato-zinc; ZnPc-SH; 2(3), 9(10),16(17), 23(24
Keywords: HA; hyaluronic acid; Tregs; regulatory T cells; T1DM; type 1 diabetes mellitus; IBD; inflammatory bowel disease; RA; rheumatoid arthritis; MHC; major histocompatibility complex; HLA; human leukocytes antigens; TLRs; toll-loke receptors; PRRs; pattern reco
Keywords: Transglycosylase; Moenomycin; Inhibitor; Biphenyl; Phosphorylpropanoate; Amine linker; A. baumannii; Acinetobacter baumannii; Arg; arginine; Asn; asparagine; Asp; aspartic acid; ATCC; american type culture collection; DMF; N,N-dimethylformamide; DMSO; di
Synthesis, characterization, and application of a novel multifunctional stationary phase for hydrophilic interaction/reversed phase mixed-mode chromatography
Keywords: HPLC; High-Performance Liquid Chromatography; RPLC; Reversed-Phase Liquid Chromatography; HILIC; Hydrophilic Interaction Liquid Chromatography; DCC; Dicyclohexylcarbodiimide; HOBT; 1-Hydroxybenzotriazole hydrate; DCM; Dichloromethane; H; Hexane; EtOAc; Et
A unique red-emitting two-photon fluorescent probe with tumor-specificity for imaging in living cells and tissues
Keywords: HOBT; 1-hydroxybenzotriazole; EDC; N-(3-dimethylaminopropyl)-N'-ethylcarbod-iimide hydrochloride; DIEA; ethyldiisopropylamine; DMF; dimethylformamide; Red-emitting two-photon fluorescent probe; High-definition three-dimensional imaging; Tumor-specific ima
Synthesis of readily available fluorophenylalanine derivatives and investigation of their biological activity
Keywords: AChE; acetylcholinesterase; BAC; bacitracin; BChE; butyrylcholinesterase; ChE; cholinesterases; DMAP; 4-(dimethylamino)pyridine; EDC; N-(3-dimethylaminopropyl)-Nâ²-ethylcarbodiimide hydrochloride; ESBL; extended-spectrum β-lactamase; FLU; fluconazole; m
Keywords: BBB; blood brain barrier; BK; bradykinin; Boc; t-butyloxycarbonyl; BR; bradykinin receptor; CNS; central nervous system; DALKD; [des-Arg10, Leu9]-kallidin; DIPEA; diisopropylethylamine; DMF; N,N-dimethylformamide; Dyn A; dynorphin A; Fmoc; fluorenylmethyl
Keywords: RNCGDQLZIATDOU-ZDRBWGSPSA-N; ICYPJNZJUFGALC-PDTBJYIYSA-N; PDRMAVOIWIVXKH-SFUSBHMVSA-N; ISADXJRTBSLWPX-ZDRBWGSPSA-N; NLBLLPROASDPSC-QWWZWVQMSA-N; XKMIKZDBUOHHDK-ZDRBWGSPSA-N; BTURADNXKHTWGA-IJOLSIAMSA-N; UEKHRDLXBMZMPD-ZYIYBEKCSA-N; UQCLCXDOXVZEOA-JARUQAPT
Keywords: CD; circular dichroism; CPE; cytopathic effect; DMF; dimethylformamide; FBS; fetal bovine serum; Fmoc; 9-fluorenylmethoxycarbonyl; HBTU; O-benzotriazole-N,N,Nâ²,Nâ²-tetramethyl-uronium-hexafluorophosphate; HOBt; N-hydroxybenzotriazole; HPLC; high perfor
Keywords: AA; amino acid; AcOH; acetic acid; 6-Cl-HOBt; 6-chloro-1-hydroxybenzotriazole; DCM; dichloromethane; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; Fmoc; 9-fluorenylmethoxycarbonyl; h; hour; HOBt; 1-hydroxybenzotriazole hydrate; HPLC; high-
Keywords: ABTS; 2,2â²-azino-bis-(3-ethylbenzothiazoline-6-sulfonate; AS; acetosyringone; BC; bacterial cellulose; BC-NFs; bacterial cellulose nanofibers; CA; coniferyl aldehyde; FF; furfural; FESEM; field emission scanning electron microscopy; FTIR; fourier transf
Keywords: Antisense oligonucleotides; PEGylation; Disulfide bioconjugates; Solid phase synthesis; Gene silencing; ON; oligonucleotide; PEG; polyethylene glycol; CPG; controlled pore glass; LCAA; long chain amino alkyl; TCEP; tris(2-carboxyethyl)phosphin; TBP; tri-n
Keywords: Sulfatase; Enzyme; Inhibitor; Estrogen; Cancer; SERM; ALP; alkaline phosphatase; DEA; diethylamine; DHEA; dehydroepiandrosterone; DHEAS; dehydroepiandrosterone sulfate; 5-diol; 5-androstene-3β,17β-diol; DIPEA; diisopropylamine; E1; estrone; E1S; estrone
Keywords: Boc; t-butyloxycarbonyl; Boc-Lys(Boc)-Osu; Nα,Nε-di-Boc-l-lysine hydroxysuccinimide ester; BSA; bovine serum albumin; Cbz; carboxybenzyl; CLRs; C-type lectin receptors; CRD; carbohydrate-recognition domain; Con A; Concanavaline A; DBU; 1,8-diazabicyclo[
Keywords: Nicotinic acetylcholine receptor; α4β2 subtypes; α7 subtypes; Two-electrode voltage clamp; Calcium imaging; EDC HCl; N-(3-dimethylaminopropyl)-Nâ²-ethylcarbodiimide hydrochloride; HOBt; 1-hydroxybenzotriazole hydrate; PEPPSIâ¢-IPr; [1,3-bis(2,6-diiso
Keywords: Monobactam; Siderophore; Structure-activity relationship; Antibacterial activity; Click chemistry; AZN; Aztreonam; MDR; multidrug-resistant; SAR; structureâactivity relationship; PIH; pyridoxal isonicotinoyl hydrazone; Trt; triphenylmethyl; Boc; t-but
Keywords: Pro-apoptotic agents; Anticancer agents; Cyclic peptides; Peptidomimetics; Nur77; Tubulin; Bcl-2; NMR studies; Molecular modeling; Confocal microscopy; FACS analysis; ADT; AutoDock Tools; COSY; correlation spectroscopy; DBU; 1,8-Diazabicyclo[5.4.0]undec-7
Keywords: SPPS; solid phase peptide synthesis; DMF; dimethyl formamide; DIPEA; diisopropylethylamine; DIPC; diisopropylcarbodiimide; HOBt; 1-hydroxybenzotriazole; Fmoc; 9-fluorenylmethyloxycarbonyl; HFIP; 1,1,1,3,3,3-hexafluoropropan-2-ol; TFA; trifluoroacetic acid
Keywords: MeCN; acetonitrile; CL; clearance; Dess-Martin periodinane; 1,1,1-tris(acetyloxy)-1,1-dihydro-1,2-benziodoxol-3-(1H)-one; DIBALH; diisobutylaluminum hydride; DMF; N,N-dimethylformamide; EtOAc; ethyl acetate; HBTU; N,N,Nâ²,Nâ²-tetramethyl-O-(1H-benzotr
Keywords: BBB; blood-brain barrier; Boc; tert-butyloxycarbonyl; cAMP; cyclic adenosine monophosphate; CNS; central nervous system; DAMGO; H-Tyr-d-Ala-Gly-NMePhe-Gly-ol; DCM; dichloromethane; DIEA; N,N-diisopropylethylamine; DOR; δ-opioid receptor; DPDPE; Tyr-c(d
Keywords: MCF 7; HeLa; EDCI; HOBt; Diamide
Keywords: Cyclic peptides; Microwave assisted synthesis; Lactam-bridge cyclic peptides; SHU9119; MTII; MWA-SPPS; microwave-assisted solid phase peptide synthesis; MBHA; methylbenzhydryl; MCR; melanocortin receptors; NDP; [Nle4, DPhe7]-αMSH; MTII; melanotan-II; RP-
Keywords: Abz; ortho-aminobenzoic acid; EDDnp; N-(2,4-dinitrophenyl)-ethylenediamine; FRET; fluorescence resonance energy transfer; hMIP; human mitochondrial intermediate peptidase; HOBt; hydroxybenzotriazole; TBTU; O-(benzotriazol-1-yl)-N,N,Nâ²,Nâ²-tetramethylur
Keywords: Betulonic acid derivatives; Synthesis; Antitumor; Apoptosis; Mitochondrial pathway; ADM; adriamycin; AO/EB; acridine orange/ethidium bromide; BetA; betulonic acid; 13C NMR; 13C Nuclear Magnetic Resonance; DMF; N, N-dimethylformamide; DMSO; dimethyl sulfox
Keywords: Obesity; Diabetes; DGAT1; Inhibitor; Adamantane; DGAT; acyl CoA:diacylglycerol acyltransferase; TG; triglyceride; DIPEA; N,N-diisopropylethylamine; OLTT; oral lipid tolerance test; DIO; diet-induced obesity; EDCI; 1-ethyl-3-(3-dimethylaminopropyl)carbodii
Keywords: Ac; acetyl; ACTH; adrenocorticotropic hormone; Alloc; allyloxycarbonyl; Boc; t-butoxycarbonyl; BSA; bovine serum albumin; DIC; N,Nâ²,-diisopropylcarbodiimide; DIEA; diisopropylethylamine; DMEM; Dulbecco's Modified Eagle Medium; DMF; N,N-dimethylformami
Keywords: αCD44; anti-CD44 antibody; bTyr-NSP; biotinylated tyrosine-derived nanospheres; bTyr-NSP-PTX; biotinylated tyrosine-derived nanospheres loaded with paclitaxel; CTAB; cetyltrimethylammonium bromide; ESA; epithelial-specific antigen; DCC; N,Nâ²-dicyclohex
Keywords: BSA; bovine serum albumin; Cl-HOBt; 6-chloro-1-hydroxybenzotriazole; CuAAC; copper(I)-catalyzed azide-alkyne cycloaddition; DCM; dichloromethane; DIC; diisopropyl carbodiimide; DIEA; diisopropylethylamine; DMEM; Dulbecco's Modified Eagle Medium; DMF; N,
Keywords: AMPs; antimicrobial peptides; ATCC; American type culture collection; CD; circular dichroism; CFU; colony forming units; CLSI; Clinical and Laboratory Standards Institute; DIPEA; N,N-diisopropylethylamine; DMEM; Dulbecco's modified eagle's medium; DMF; N,
Keywords: Peptidomimetic boronates; Proteasome inhibitors; Docking studies; ChT-L; chymotrypsin-like; T-L; trypsin-like; PGPH; post-glutamyl peptide hydrolyzing; DMSO; dimethyl sulfoxide; DMF; dimethylformamide; Pd2(dba)3; tris(benzylideneacetone)dipalladium; EDC;
Antiobesity and emetic effects of a short-length peptide YY analog and its PEGylated and alkylated derivatives
Keywords: Ac; acetyl; Aib; 2-aminoisobutyric acid; tBu; tert-butyl; Cha; 3-cyclohexylalanine; CHAPS; 3-[(3-cholamidopropyl)dimethylammonio]-1-propanesulfonate; DIO; diet-induced obese; DIPCDI; N,Nâ²-diisopropylcarbodiimide; DMF; N,N-dimethylformamide; DMSO; dimeth
Design, synthesis, in vitro and in vivo evaluation, and structure-activity relationship (SAR) discussion of novel dipeptidyl boronic acid proteasome inhibitors as orally available anti-cancer agents for the treatment of multiple myeloma and mechanism stud
Keywords: SAR; structureactivity relationship; UPP; ubiquitinproteasome pathway; FDA; Food and Drug Administration; ATP; Adenosine triphosphate; CP; core particle; RP; regulatory proteasome; C-L; caspase-like; T-L; trypsin-like; CT-L; chymotrypsin-like; EDCI; 1-eth
Nano-peroxidase fabrication on cation exchanger nanocomposite: Augmenting catalytic efficiency and stability for the decolorization and detoxification of Methyl Violet 6B dye
Keywords: Peroxidase; Polypyrrole-zirconium(IV)selenoiodate cation exchanger nanocomposite; Immobilization; Methyl Violet 6B; Oxidative degradation; Detoxification; HOBT; 1-hydroxybenzotriazole; GP; ginger peroxidase; MV 6B; Methyl Violet 6B; TEM; transmission elec
Microcystins: Synthesis and structure-activity relationship studies toward PP1 and PP2A
Keywords: Adda; (2S,3S,8S,9S)-3-amino-9-methoxy-2,6,8-trimethyl-10-phenyldeca-4,6-dienoic acid; Amba; (2S,3S)-3-amino-2-methylbutanoic acid; Boc; tert-butoxycarbonyl; BOP; benzotriazol-1-yloxy-tris-dimethylaminophosphoniumhexafluoro phosphate; Cbz; carboxybenzyl; D
Cathepsin B inhibitors: Further exploration of the nitroxoline core
Keywords: Abz; 2-aminobenzoyl; AMC; 7-amido-4-methylcoumarin; catB; cathepsin B; DIPEA; N,N-diisopropylethylamine; DMSO; dimethyl sulfoxide; ECM; extracellular matrix; EDC; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide; HATU; 1-[bis(dimethylamino)methylene]-1H-1,2,
Synthesis and in vitro characterization of a P2X7 radioligand [123I]TZ6019 and its response to neuroinflammation in a mouse model of Alzheimer disease
Keywords: ACN; Acetonitrile; AD; Alzheimer's disease; AMF; ammonium formate; ATP; adenosine-triphosphate; BzATP; 3â²-O-(4-Benzoyl)benzoyl ATP, strong agonist for P2X7 receptor; CNS; central nervous system; DMEM; Dulbecco's Modified Eagle's Medium; DMF; dimethylfor
Design, synthesis and pharmacological evaluation of N-(5-chloro-2,4-dihydroxybenzoyl)-(R)-N-arylmethyl-1,2,3,4-tetrahydro-3-isoquinolinecarboxamides as potent Hsp90 inhibitors
Keywords: Hsp90 inhibitors; CETSA; Molecular dynamics simulation; Apoptosis; IKK; (R)-Tic; (R)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid; GA; geldanamycin; BnBr; Benzyl bromide; CETSA; cellular thermal shift assay; DMEM; Dulbecco's modified Eagle's medium; R
Design and synthesis of aminoester heterodimers containing flavone or chromone moieties as modulators of P-glycoprotein-based multidrug resistance (MDR)
Keywords: P-gp; P-glycoprotein; SAR; Structure-activity relationships; DOX; Doxorubicin; EDCI; 1-(3-dimethylaminopropyl)-3-ethylcarbodiimmide hydrochloride; HOBt; 1-Hydroxybenzotriazole hydrate; DMAP; 4-dimethylaminopyridine; P-gp modulators; MDR reversers; Heterod
The dominant role of side chains in supramolecular double helical organisation in synthetic tripeptides
Keywords: Self-assembly; Double helices; Side chain interactions; Supramolecular heterogeneity; Aib; α-aminoisobutyric acid; Boc; tertiary butyloxy carbonyl; DCC; dicyclohexyl-carbodiimide; 4F-Phe; 4-Fluoro phenylalanine; HOBt; 1-hydroxy benzotriazole; OMe; methox
Development of potent and proteolytically stable human neuromedin U receptor agonists
Keywords: Neuromedin U (NMU); NMU-8; Neuromedin U receptor agonists; Plasma stability; 1â²Nal; 1â²-naphtylalanine; 2â²Nal; 2â²-naphtylalanine; 7-OH-Tic; 7-hydroxy-L-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid; ACN; acetonitrile; AUC; area under the curve;
The 4-N-acyl and 4-N-alkyl gemcitabine analogues with silicon-fluoride-acceptor: Application to 18F-Radiolabeling
Keywords: dFdC; 2â²,2â²-difluoro-2â²-deoxycytidine (Gemcitabine); hENT1; human equilibrative nucleoside transport protein 1; dCK; deoxycytidine kinase; dFdU; 2â²,2â²-difluorouridine; CDA; cytidine deaminase; [18F]FAC; 1-(2-deoxy-2-[18F]fluoro-β-d-arabinofuran
Synthesis and biological evaluation of a library of hybrid derivatives as inhibitors of influenza virus PA-PB1 interaction
Keywords: Anti-Influenza; PA-PB1; RdRp; Amino acid coupling; SPPS; Diphenyl-pyridine; AcOEt; Ethyl acetate; CC50; Half maximal cytotoxic concentration; cRNA; complementar RNA; DCM; dichloromethane; DDQ; 2,3-Dichloro-5,6-dicyano-1,4-benzoquinone; DIPEA; N,N-Diisopro
Synthesis and evaluation of a novel urea-based 68Ga-complex for imaging PSMA binding in tumor
Keywords: SPECT; single photon emission computer tomography; PET; positron emission tomography; HPLC; High performance liquid chromatography; HRMS; High-resolution mass spectrometry; PBS; phosphate buffered saline; SPE; solid-phase extraction; GMP; good manufacturi