دانلود مقالات ISI درباره Hobt + ترجمه فارسی

Synthesis of photoreactive ivermectin B1a derivatives and their actions on Haemonchus and Bombyx glutamate-gated chloride channels

Keywords: AVM; avermectin; DCC; dicyclohexylcarbodiimide; DIPEA; N,N-diisopropylethylamine; DMAP; 4-(dimethylamino)pyridine; DMF; N,N-dimethylformamide; DMSO; dimethyl sulfoxide; EDC; 1-ethyl-3-(3-dimethylamino-propyl)carbodiimide; GABA; γ-aminobutyric acid; GABAC

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2015 سفارش ترجمه

Structure-activity relationship study using peptide arrays to optimize Api137 for an increased antimicrobial activity against Pseudomonas aeruginosa

Keywords: Apidaecin; Gram-negative bacterium; Proline-rich antimicrobial peptide (PrAMP); Pseudomonas aeruginosa; SPOT synthesis; AMP; antimicrobial peptide; DIC; N,N′-diisopropylcarbodiimide; DIPEA; N-ethyldiisopropylamine; DMAP; 4-dimethylaminopyridine; gu; N,N

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2015 سفارش ترجمه

A novel synthetic luteinizing hormone-releasing hormone (LHRH) analogue coupled with modified β-cyclodextrin: Insight into its intramolecular interactions

Keywords: BOP; benzotriazole-1-yl-oxy-tris-(dimethylamino)-phosphonium hexafluorophosphate; CLTR-Cl; 2-chlorotrityl chloride; DCC; N,N′-dicyclohexylcarbodiimide; DMA; dimethylacetamide; DIC; N,N′-diisopropylcarbodiimide; DIEA; diisopropylethylamine; DMF; N,N-di

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2015 سفارش ترجمه

Specificity studies on Kallikrein-related peptidase 7 (KLK7) and effects of osmolytes and glycosaminoglycans on its peptidase activity

Keywords: KLK; kallikrein-related peptidase; FRET; fluorescence resonance energy transfer; MCA; 4-methyl coumarin-7-amide; Q-EDDnp; glutaminyl-[N-(2,4-dinitrophenyl)-ethylenediamine]; Abz; ortho-amino-benzoic acid; GAGs; glycosaminoglycans; HBTU; N,N,N′,N′-Tetr

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2015 سفارش ترجمه

Synthesis and SAR studies of analogues of 4-(3,3-dimethyl-butyrylamino)-3,5-difluoro-N-thiazol-2-yl-benzamide (Lu AA41063) as adenosine A2A receptor ligands with improved aqueous solubility

Keywords: HATU; 2-(1H-7-azabenzotriazol-1-yl)-1,1,3,3-tetramethyluronium hexafluorophosphate; EDC; N-ethyl-N′-dimethylaminopropyl-carbodiimide hydrochloride; HOBt; 1-hydroxy-benzotriazole; DMAP; 4-dimethylaminopyridine; DMF; dimethylformamide; DMSO; dimethyl sulf

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2015 سفارش ترجمه

BN/CC isosterism in borazaronaphthalenes towards phosphodiesterase 10A (PDE10A) inhibitors

Keywords: cAMP; cyclic adenosine monophosphate; cGMP; cyclic guanosine monophosphate; Boc; tert-butyloxycarbonyl; THF; tetrahydrofuran; DMF; dimethylformamide; CPME; cyclopentyl methyl ether; TFA; trifluoroacetic acid; EDCI; 1-ethyl-3-(3-dimethylaminopropyl)carbodi

دانلود رایگان متن کامل مقاله ISI 16 صفحه سال انتشار : 2015 سفارش ترجمه

Structure-based design and synthesis of covalent-reversible inhibitors to overcome drug resistance in EGFR

Keywords: CRI; covalent reversible inhibitor; EDC·HCl; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide hydrochloride; HOBt; hydroxybenzotriazole; DIPEA; N,N-diisopropylethylamine; EGFR; epidermal growth factor receptor; NOE; nuclear Overhauser effect; NSCLC; non-sma

دانلود رایگان متن کامل مقاله ISI 48 صفحه سال انتشار : 2015 سفارش ترجمه

The synthesis of indolo[2,3-b]quinoline derivatives with a guanidine group: Highly selective cytotoxic agents

Keywords: Neocryptolepine; Antiproliferative activity; Antifungal activity; Biofilm; Guanidine group; Mechanism of action; Apoptosis; Hemolytic activity; Boc; tert-butyloxycarbonyl group; BSTU; N,N′-bis-Boc-thiourea; DIPEA; N,N-diisopropylethylamine; DMF; dimethy

دانلود رایگان متن کامل مقاله ISI 50 صفحه سال انتشار : 2015 سفارش ترجمه

Implications of N-capped urea/thiourea and C-capped 3-(1-piperazinyl)-1,2-benzisothiazole with bridging Gly-Val/Phe-Gly-Val-Pro as therapeutic targets

Keywords: Peptides; Conjugation; Antimicrobial; Antiglycation; Urease inhibition; H+/K+-ATPase activity; ANSA; 1-amino-2-naphthol-4-sulphonic acid; Bis-PNPC; bis(4-nitrophenyl)carbonate; Boc; tert-butyloxycarbonyl; DCM; dichloromethane; EGTA; ethylene glycol tetraa

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2014 سفارش ترجمه

[Dmt1]DALDA analogues with enhanced μ opioid agonist potency and with a mixed μ/κ opioid activity profile

Keywords: Boc; tert-butyloxycarbonyl; DAMGO; H-Tyr-d-Ala-Gly-Phe(NMe)-Gly-ol; Dmp; 2′,6′-dimethylphenylalanine; Dmt; 2′,6′-dimethyltyrosine; [Dmt1]DALDA; H-Dmt-d-Arg-Phe-Lys-NH2; DSLET; H-Tyr-d-Ser-Gly-Phe-Leu-Thr-OH; EDT; 1,2-ethanediol; Emp; 2′-ethyl-6â

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2014 سفارش ترجمه

N-methylthioacetylation of RYYRIK-NH2 with enhanced specific binding affinity and high antagonist activity for nociceptin ORL1 receptor

Keywords: DTT; dithiothreitol; Fmoc; 9-fluorenylmethoxycarbonyl; GPCR; G protein-coupled receptor; HBTU; 2-(1H-benzotriazole-1-yl)-1,1,3,3-tetramethyluronium hexafluorophosphate; HOBt; 1-hydroxybenzotriazole; MALDI-TOF; matrix-assisted laser desorption ionization t

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2014 سفارش ترجمه

Synthetically modified l-histidine-rich peptidomimetics exhibit potent activity against Cryptococcus neoformans

Keywords: AA; amino acid; Boc; tert-butoxycarbonyl; DIC; 1,3-diisopropylcarbodiimide; DIEA; N,N-diisopropylethylamine; EYPC; egg yolk l-a-phosphatidylcholine; DMF; N,N-dimethylformamide; EYPG; egg yolk l-a-phosphatidyl-dl-glycerol; TBTU; O-(benzotriazol-1-yl)-N,N,N

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2014 سفارش ترجمه

A total synthesis of a highly N-methylated cyclodepsipeptide [2S,3S-Hmp]-aureobasidin L using solid-phase methods

Keywords: Aureobasidin; N-Methylated cyclodepsipeptide; Depsidipeptide; Fmoc-based solid-phase peptide synthesis; Boc; tert-butyloxycarbonyl; BTC; bis-(trichloromethyl)-carbonate; 13C NMR; carbon-13 nuclear magnetic resonance; COSY; correlation spectroscopy; DBU; 1

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2014 سفارش ترجمه

Tritium-labelled isovaleryl-RYYRIK-NH2 as potential antagonist probe for ORL1 nociceptin receptor

Keywords: Boc; butoxycarbonyl; Bmax; receptor density; DMEM; Dulbecco's Modified Eagle's Medium; DMF; N,N-dimethylformamide; FBS; fetal bovine serum; GPCR; G protein-coupled receptor; HBTU; 2-(1H-benzotriazole-1-yl)-1,1,3,3-tetramethyluronium hexafluorophosphat

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2014 سفارش ترجمه

Peptides that activate the 20S proteasome by gate opening increased oxidized protein removal and reduced protein aggregation

Keywords: ALS; amyotrophic lateral sclerosis; AMC; 7-amido-4-methylcoumarin; z-ARR-AMC; z-Ala-Arg-Arg-amido-4-methylcoumarin; ChT-L; chymotrypsin-like proteasomal activity; DMF; N,N-dimethyl formamide; DMSO; dimethyl sulfoxide; DNPH; 2,4-dinitrophenylhydrazine; DTT

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2014 سفارش ترجمه

G-quadruplex DNA recognition by nucleophosmin: New insights from protein dissection

Keywords: TIS; Triisopropylsilane; TFA; Trifluoroacetic acid; DMF; Dimethylformamide; DCM; Dichloromethane; HBTU; 1-H-Benzotriazolium, 1-[bis(dimethylamino)methylene]-hexafluorophosphate(1-), 3 oxide; HOBt; N-hydroxybenzotriazole; DIEA; Di-isopropylethylamine; Fmoc

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2014 سفارش ترجمه

Structure-based design, synthesis and biological testing of etoposide analog epipodophyllotoxin-N-mustard hybrid compounds designed to covalently bind to topoisomerase II and DNA

Keywords: Boc2O; di-tert-butyl dicarbonate; CHO; Chinese hamster ovary; Et3N; triethylamine; EtOAc; ethyl acetate; HOBt; (1-hydroxybenzotriazole); ICE; immunodetection of complexes of enzyme-to-DNA; K562 cells; human erythroleukemic cells; kDNA; catenated DNA; MTS;

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2014 سفارش ترجمه

Gadolinium-based contrast agents targeted to amyloid aggregates for the early diagnosis of Alzheimer's disease by MRI

Keywords: Alzheimer's disease; Amyloid; Gadolinium; DOTA; Pyridine containing TriAza (PCTA); Magnetic resonance imaging (MRI); BAT; bis-amine-bis-thiol; BTA; 2-(4-N-methylaminophenyl)benzothiazole; CA; contrast agent; CMC; critic micelle concentration; CV; cone vol

دانلود رایگان متن کامل مقاله ISI 19 صفحه سال انتشار : 2014 سفارش ترجمه

Affinity-based screening of MDM2/MDMX-p53 interaction inhibitors by chemical array: Identification of novel peptidic inhibitors

Keywords: FAM; carboxyfluorescein; FP; fluorescence polarization; HBTU; O-(1H-benzotriazol-1-yl)-N,N,N′,N′-tetramethyluronium hexafluorophosphate; HOBt; 1-hydroxy-1H-benzotriazole; MDM2; mouse double minute 2 homolog; MDMX; mouse double minute X homolog; TAMRA;

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2013 سفارش ترجمه

Triphenylphosphonium salts of 1,2,4-benzothiadiazine 1,1-dioxides related to diazoxide targeting mitochondrial ATP-sensitive potassium channels

Keywords: ATP; adenosine triphosphate; SUR; sulfonylurea receptor; Kir; inwardly rectifying potassium channel; mitoKATP channel; mitochondrial ATP-sensitive potassium channel; DCC; N,N′-dicyclohexylcarbodiimide; NHS; N-hydroxysuccinimide; HOBt; hydroxybenzotriazo

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2013 سفارش ترجمه

A new class of aggregation inhibitor of amyloid-β peptide based on an O-acyl isopeptide

Keywords: Aβ; amyloid β peptide; AD; Alzheimer's disease; DIC; N,N′-diisopropylcarbodiimide; DMF; N,N-dimethylformamide; DMSO; dimethyl sulfoxide; FAM; carboxyfluorescein; HOBt; N-hydroxybenzotriazole; HPLC; high-performance liquid chromatography; kDa; kiloda

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2013 سفارش ترجمه

Design of a novel LOX-1 receptor antagonist mimicking the natural substrate

Keywords: CTLD; C-type lectin-like domain; DiI; 1,1′-dioctadecyl-3,3,3′,3′-tetramethyllindocarbocyanine perchlorate; HOBt; 1-hydroxybenzotriazole; LDL; low-density lipoprotein; LOX-1; lectin-like oxidized low-density lipoprotein receptor-1; ox-LDL; oxidized l

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2013 سفارش ترجمه

Potency optimization of Huwentoxin-IV on hNav1.7: A neurotoxin TTX-S sodium-channel antagonist from the venom of the Chinese bird-eating spider Selenocosmia huwena

Keywords: ACF; animal-component free; BSA; bovine serum albumin; CaCl2; calcium chloride; CD; circular dichroism spectroscopy; CHO; Chinese hamster ovary; CNS; central nervous system; CO2; carbon dioxide; CsF; cesium fluoride; CsOH; cesium hydroxide; DIC; diisoprop

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2013 سفارش ترجمه

Synthetic tripeptides as alternate substrates of murein peptide ligase (Mpl)

Keywords: Escherichia coli; Mpl; Murein peptide ligase; Peptidoglycan recycling; Tripeptide substrates; Abu; 2-aminobutyric acid; AcOH; acetic acid; Apm; 2-aminopimelic acid; A2pm; 2,6-diaminopimelic acid; Bn; benzyl; Boc; t-butyloxycarbonyl; DCC; N,N′-dicyclohex

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2013 سفارش ترجمه

Design, synthesis and evaluation of antimicrobial activity of N-terminal modified Leucocin A analogues

Keywords: AMP; antimicrobial peptide; CD; circular dichroism; DIC; 1,3-diisopropylcarbodiimide; Fmoc; 9-fluorenylmethyloxycarbonyl; HOBt; N-hydroxybenzotriazole; RP-HPLC; reversed phase high performance liquid chromatography; LAB; lactic acid bacteria; LeuA; Leucoc

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2013 سفارش ترجمه

Differences in the inhibition of coagulation factor XIII-A from animal species revealed by Michael Acceptor- and thioimidazol based blockers

Keywords: Abz; ortho-aminobenzoic acid; CAD; cadaverine; DNP; 2,4-dinitrophenyl; tBu; tert-butyl ester; Trt; trityl; Fmoc; Fluorenylmethyloxycarbonyl; DMF; Dimethylformamide; TBTU; O-(Benzotriazol-1-yl)-N,N,N',N'-tetramethyluronium tetrafluoroborate; HOBt; Hydroxyb

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2013 سفارش ترجمه

Radiochemical and radiobiological assessment of a pyridyl-S-cysteine functionalized bombesin derivative labeled with the 99mTc(CO)3+ core

Keywords: Boc; t-butyloxycarbonyl; BSA; bovine serum albumin; Cys; cysteine; DIEA; N,N-diisopropylethylamine; DIC; diisopropylcarbamide; DMEM; Dulbecco's modified Eagle medium; DMF; dimethylformamide; EDTA; ethylenediaminetetraacetic acid; ESI-MS; electrospray io

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2013 سفارش ترجمه

The pro-apoptotic action of new analogs of the insect gonadoinhibiting peptide Neb-colloostatin: Synthesis and structure-activity studies

Keywords: Ach; 1-aminocyclohexane-1-carboxylic acid; Acp; 1-aminocyclopentane-1-carboxylic acid; CD; circular dichroism; DMF; dimethylformamide; EDT; 1,2-ethanedithiol; Fmoc; 9-fluorenylmethoxycarbonyl; HBTU; O-benzotriazole-N,N,N′,N′-tetramethyl-uronium-hexafl

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2013 سفارش ترجمه

New generation of efficient peptide-based vectors, NickFects, for the delivery of nucleic acids

Keywords: CPP; cell-penetrating peptide; CR; charge ratio; DLS; dynamic light scattering; DIEA; diisopropylethylamine; EGFP; enhanced green fluorescent protein; HBTU; O-benzotriazole-N,N,N′,N′-tetramethyl-uronium-hexafluoro-phosphate; HOBT; hydroxybenzotriazole

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2013 سفارش ترجمه

Backbone cyclic helix mimetic of chemokine (C-C motif) receptor 2: A rational approach for inhibiting dimerization of G protein-coupled receptors

Keywords: ACN; acetonitrile allocallyloxycarbonyl; BBB; blood brain barrier; Boc; t-butyloxycarbonyl; BTC; bis(trichloromethyl)carbonate; CCR2; chemokine (C-C motif) receptor 2; CCR5; chemokine (C-C motif) receptor 5; CNS; central nervous system; DIPEA; diisopr

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2013 سفارش ترجمه

Discovery of pyrazole as C-terminus of selective BACE1 inhibitors

Keywords: Alzheimer's disease; BACE1; C-terminus; Click chemistry; In situ screening assay; Pyrazole; EDCl; N-(3-dimethylaminopropyl)-N′-ethylcarbodiimide hydrochloride; HOBt; N-hydroxybenzotriazole; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; E

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2013 سفارش ترجمه

Design, synthesis, and biological activities of novel hexahydropyrazino[1,2-a]indole derivatives as potent inhibitors of apoptosis (IAP) proteins antagonists with improved membrane permeability across MDR1 expressing cells

Keywords: HATU; O-(7-azabenzotriazol-1-yl)-N,N,N′,N′-tetramethyluronium hexafluorophosphate; DIPEA; N-ethyldiisopropylamine; Ac; acetyl; CDCl3; deuteratedchloroform; DMF; N,N-dimethylformamide; DMSO; dimethyl sulfoxide; DMT-MM; 4-(4,6-dimethoxy-1,3,5-triazin-2-

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2013 سفارش ترجمه

Linear and cyclic glycopeptide as HIV protease inhibitors

Keywords: HIV-1 protease; Linear and cyclic glycopeptides; Solid and solution peptide synthesis; Molecular docking; AIDS; acquired immunodeficiency syndrome; CTC; 2-chlorotrityl chloride; DCM; dichloromethane; DIPEA; N,N-diisopropyl ethylamine; DMF; N,N-dimethylfor

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2013 سفارش ترجمه

Anthelmintic PF1022A: stepwise solid-phase synthesis of a cyclodepsipeptide containing N-methyl amino acids

Keywords: ACN; acetonitrile; Boc; tert-butyloxycarbonyl; BOPCl; N,N′-bis(2-oxo-3-oxazolidinyl)phosphinic chloride; DCM; dichloromethane; DEAD; diethylazodicarboxylate; DHP; 3,4-dihydro-2H-pyrane; DIC; N,N′-diisopropylcarbodiimide; DIEA; diisopropylethylamine; D

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2012 سفارش ترجمه

Identification of a novel Smoothened antagonist that potently suppresses Hedgehog signaling

Keywords: Smo; smoothened; Hh; hedgehog; Ptc; patched; Shh; sonic hedgehog; β arr2; β-arrestin2; β arr2-GFP; β-arrestin2-green fluorescent protein chimera; Gli; glioma-associated oncogene; GPCR; G-protein-coupled receptor; V2R; vasopressin2 receptor; HTS; high-

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2012 سفارش ترجمه

Proteasome inhibitors for cancer therapy

Keywords: BOP; (benzotriazol-1-yloxy)tris(dimethylamino)phosphonium hexafluorophosphate; DMSO; dimethyl sulfoxide; HMPA; hexamethyl phosphoramide; HOBt; 1-hydroxybenzotriazole; NMM; N-methylmorpholine; DMF; N,N-dimethyformamide; LDA; lithium diisopropylamide; THF;

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2012 سفارش ترجمه

Inhibitors of specific ceramide synthases

Keywords: Ceramide synthase; Ceramide; Inhibitor; Ceramide synthase activity assay; BSA; bovine serum albumin; Cer; ceramide; dhCer; dihydroceramide; CerS; (dihydro)ceramide synthase; DES; dihydroceramide desaturase; EDC; 1-ethyl-3-[3-dimethylaminopropyl]carbodiimi

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2012 سفارش ترجمه

Macroporous methacrylate-based monoliths as platforms for DNA microarrays

Keywords: GMA; glycidyl methacrylate; EDMA; ethylene dimethacrylate; HEMA; 2-hydroxyethyl methacrylate; CEMA; 2-cyanoethyl methacrylate; GDMA; glycerol dimethacrylate; 2-D and 3-D; two and three-dimensional, respectively; DMAP; 4-(dimethylamino)pyridine; CDI; 1,1-c

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2012 سفارش ترجمه

Synthesis and comparative assessment of a labeled RGD peptide bearing two different 99mTc-tricarbonyl chelators for potential use as targeted radiopharmaceutical

Keywords: Arg/R; arginine; Asp/D; aspartic acid; Boc; t-butyloxycarbonyl; BSA; bovine serum albumin; CPA; 3-l-cysteine propionic acid; Cys; cysteine; d-Phe/f; d-phenylalanine; DIEA; N,N-diisopropylethylamine; DIPC; diisopropylcarbamide; DMEM; Dulbecco's modified

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2012 سفارش ترجمه

7-Substituted-pyrrolo[3,2-d]pyrimidine-2,4-dione derivatives as antagonists of the transient receptor potential ankyrin 1 (TRPA1) channel: A promising approach for treating pain and inflammation

Keywords: AITC; allyl isothiocyanate; BSA; bovine serum albumin; CA; cinnamaldehyde; CHO; Chinese hamster ovary cells; COPD; chronic obstructive pulmonary disease; DMEM; Dulbecco's modified eagle medium; DRG; dorsal root ganglia; EDAC; N-ethyl-N′-(3-dimethylami

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2012 سفارش ترجمه

The role of endocytosis on the uptake kinetics of luciferin-conjugated cell-penetrating peptides

Keywords: CPP; Cell-penetrating peptide; siRNA; Short interfering ribonucleic acid; EGF; Epidermal growth factor; EGFR; Epidermal growth factor receptor; CME; Clathrin-mediated endocytosis; SPPS; Solid phase peptide synthesis; t-Boc; tert-Butyloxycarbonyl; HOBt; Hy

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2012 سفارش ترجمه

TAT-mediated photochemical internalization results in cell killing by causing the release of calcium into the cytosol of cells

Keywords: TMR; carboxytetramethylrhodamine; CPP; cell-penetrating peptide; TAT; trans-activator of transcription; TM-PCI; TMR-TAT mediated photochemical internalization; RBC; red blood cell; PDT; photodynamic therapy; DMF; dimethylformamide; DCM; dichloromethane; T

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2012 سفارش ترجمه

The discovery and synthesis of JNJ 31020028, a small molecule antagonist of the Neuropeptide Y Y2 receptor

Keywords: DCM; dichloromethane; HOBt; 1-hydroxy-benzotriazole; EDCI; 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide; BOC; butoxycarbonyl; MeOH; methanol; K2CO3; potassium carbonate; Na2CO3; sodium carbonate; DMF; dimethylformamide; Et3N; triethylamine; Et2O; ether;

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2011 سفارش ترجمه

Capturing of the free cysteine residue in the ligand-binding site by affinity labeling of the ORL1 nociceptin receptor

Keywords: Ac-RYYRIK-NH2; the one-letter amino acid code denotes Ac-Arg-Tyr-Tyr-Arg-Ile-Lys-NH2; BSA; bovine serum albumin; DMEM; Dulbecco's modified Eagle's medium; DMF; N,N-dimethylformamide; EC50; the concentration for the half maximal effective concentration

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2011 سفارش ترجمه

Effects of positively charged arginine residues on membrane pore forming activity of Rev-NIS peptide in bacterial cells

Keywords: CD; circular dichroism; diSC35; 3,3′-dipropylthiadicarbocyanine iodide; FITC; fluorescein isothiocyanate; FD; FITC-dextran; AMP; antimicrobial peptide; NIS; nuclear entry inhibitory signal; TFE; 2,2,2-trifluoroethanol; SDS; sodium dodecyl sulfate; MIC;

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2011 سفارش ترجمه

Biological and conformational evaluation of angiotensin II lactam bridge containing analogues

Keywords: AAA; Amino acid analysis; ACN; Acetonitrile; AII; angiotensin II; BOP; (Benzotriazol-1-yl-oxy)tris(dimethylamino)phosphonium hexafluorophosphate; BSA; bovine serum albumin; CD; Circular Dichroism; CE; Capillary Electrophoresis; CHO; Chinese hamster ovary;

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2011 سفارش ترجمه

Active immunization against IL-23p19 improves experimental arthritis

Keywords: BDB; bis-diazo-benzidine; CFA; complete Freund adjuvant; CIA; collagen-induced arthritis; CIIb; bovine type II collagen; DIEA; diisopropyethylamine; DMF; dimethylformamide; EAE; experimental allergic encephalomyelitis; G-CSF; granulocyte-colony-stimulatin

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2011 سفارش ترجمه

Synthesis and evaluation of bidentate ligands designed to interact with PDZ domains

Keywords: CDI; carbonyldiimidazole; Cyc; cyclohexane; DABCO; diazabicyclooctane; DCM; dichloromethane; DIEA; diisopropylethylamine; DMAP; 4-dimethylaminopyridine; DMF; N,N-dimethylformamide; EDC; 1-ethyl-3-(3-dimethylamino propyl)carbodiimide; EtOAc; ethylacetate;

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2011 سفارش ترجمه

A sucrose-derived scaffold for multimerization of bioactive peptides

Keywords: Boc; tert-butoxycarbonyl; BSA; bovine serum albumin; CCK2R; cholecystokinin 2 receptor; CCK4; Trp-Met-Asp-Phe-NH2; Cl-HOBt; 6-chloro-1-hydroxybenzotriazole; CuAAC; copper(I)-catalyzed azide-alkyne cycloaddition; DCM; dichloromethane; DIC; diisopropyl carb

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2011 سفارش ترجمه

Hydrophilic methacrylate monoliths as platforms for protein microarray

Keywords: Macroporous hydrophilic monoliths; Photo-initiated polymerization; Polymer porogens; GMA; glycidyl methacrylate; HEMA; 2-hydroxyethyl methacrylate; GDMA; glycerol dimethacrylate; EDMA; ethylene dimethacrylate; DHPMA; 2,3-dihydroxypropyl methacrylate; DoOH

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2011 سفارش ترجمه