Keywords: فعالیت مهاری; Trypsin; Inhibitory activity; Phenylpropanoid glycoside; Secondary structure; Phenol-protein binding;
مقالات ISI فعالیت مهاری (ترجمه نشده)
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Keywords: فعالیت مهاری; Purine nucleoside phosphorylase; Dietary flavonoids; Inhibitory activity; Binding affinity; Molecular modeling;
Keywords: فعالیت مهاری; Verbascoside; Xanthine oxidase; Inhibitory activity; Fluorescence chromatographic; Circular dichroism spectra; Molecular simulation;
Keywords: فعالیت مهاری; Daidzein; Genistein; Trypsin; Inhibitory activity; Fluorescence spectroscopy; Molecular docking
Keywords: فعالیت مهاری; Dengue protease inhibitor; NS2B/NS3 complex; Molecular docking; In vitro inhibition; Inhibitory activity;
Keywords: فعالیت مهاری; Aptamer; Saxitoxin; Mutagenesis; Truncation; Inhibitory activity; G-quadruplex;
Keywords: فعالیت مهاری; Sequential injection; Monoamine oxidase; Tyramine oxidase; MAO; TOD; Inhibitory activity;
Keywords: فعالیت مهاری; New spiro-derivatives of 1,3-thiazine; Inhibitory activity; Distribution coefficients; Lipophilicity; Permeability; Correlation structure–activityK43/21, Biological Coefficient Describing Ability to Inhibit Glu-Ca-uptake; IC50, concentration of inhibition
Keywords: فعالیت مهاری; Trypsin inhibitor; Seed; Inhibitory activity; Purification; Characterization
Two new steroidal glycosides from Anemarrhena asphodeloides rhizome, and their cytotoxic activity in vitro
Keywords: فعالیت مهاری; Anemarrhena asphodeloides; Steroid; HeLa; A549; Inhibitory activity;
Design, synthesis and biological evaluation of novel 3-substituted pyrazolopyrimidine derivatives as potent Bruton's tyrosine kinase (BTK) inhibitors
Keywords: فعالیت مهاری; BTK inhibitors; 3-Substituted pyrazolopyrimidine; Structure-based drug design; Inhibitory activity; ClogP;
An integrated computational hierarchy for identification of potent inhibitors against Shikimate Kinase enzyme from Shigella sonnei, a major cause of global dysentery
Keywords: فعالیت مهاری; ATP; adenosine triphosphate; SK; Shikimate Kinase; PDB; Protein Data Bank; GOLD; Genetic Optimization for Ligand Docking; VMD; Visual Molecular Dynamics; DS; Discovery Studio; PRDOS; Protein DisOrder prediction System; PK; pharmacokinetics; BBB; blood-bra
The investigation of α-amylase inhibitory activity of selected Pinto bean peptides via preclinical study using AR42J cell
Keywords: فعالیت مهاری; α-Amylase; AR42J cell; Diabetes treatment; Inhibitory activity; Pinto bean peptide;
Molecular characterization, expression and functional analysis of two Kazal-type serine protease inhibitors from Venerupis philippinarum
Keywords: فعالیت مهاری; Venerupis philippinarum; Serine protease inhibitor; Inhibitory activity; Bacterial challenge; Innate immunity;
Coumarin sulfonates: New alkaline phosphatase inhibitors; in vitro and in silico studies
Keywords: فعالیت مهاری; Coumarins; Sulfonates; Inhibitory activity; Alkaline phosphatase; SAR; Docking studies;
Preparation and inhibition on α-d-glucosidase of low molecular weight polysaccharide from Cordyceps militaris
Keywords: فعالیت مهاری; Cordyceps militaris; Acid hydrolysis; Inhibitory activity
Synthesis of 3-acyloxyxanthone derivatives as α-glucosidase inhibitors: A further insight into the 3-substituents' effect
Keywords: فعالیت مهاری; Xanthone derivatives; α-Glucosidase; Inhibitory activity; Inhibition kinetics;
Characterization of a novel Kazal-type serine proteinase inhibitor of Arabidopsis thaliana
Keywords: فعالیت مهاری; Kazal-type domain; Serine proteinase inhibitor; Arabidopsis thaliana; Botrytis cinerea; Inhibitory activity
Synthesis and activity evaluation of the cyclic dipeptides arylidene N-alkoxydiketopiperazines
Keywords: فعالیت مهاری; Arylidene N-alkoxydiketopiperazines; Synthesis; Caspase-3; Antitumor activities; Inhibitory activity; Molecular docking;
Synthesis and potent inhibitory activities of carboxybenzyl-substituted 8-(3-(R)-aminopiperidin-1-yl)-7-(2-chloro/cyanobenzyl)-3-methyl-3,7-dihydro-purine-2,6-diones as dipeptidyl peptidase IV (DPP-IV) inhibitors
Keywords: فعالیت مهاری; Diabetes; Dipeptidyl peptidase IV inhibitor; 3-Methyl-3,7-dihydro-purine-2,6-dione; Synthesis; Inhibitory activity
Steroidal glycosides from Marsdenia tenacissima
Keywords: فعالیت مهاری; Marsdenia tenacissi; Tenacigenin B; Nitric oxide; Inhibitory activity;
Silk gland-specific proteinase inhibitor serpin16 from the Bombyx mori shows cysteine proteinase inhibitory activity
Keywords: فعالیت مهاری; Serpin (serine proteinase inhibitor); Bombyx mori; Silk gland-specific; Inhibitory activity; Structure
Synthesis and biological evaluation of open-chain analogs of cyclic peptides as inhibitors of cellular Shp2 activity
Keywords: فعالیت مهاری; Chain peptides; Synthesis; SHP2; Inhibitory activity; Molecular docking;
A Kazal-type serine proteinase inhibitor from Cyclina sinensis is involved in immune response and signal pathway initiation
Keywords: فعالیت مهاری; Cyclina sinensis; Kazal-type serine protease inhibitor; RNA interference; Inhibitory activity; Innate immunity;
4-Hydroxybenzyl-substituted amino acid derivatives from Gastrodia elata
Keywords: فعالیت مهاری; Gastrodia elata Blume; Orchidaceae; 4-Hydroxybenzyl- substituted amino acid derivatives; Pyroglutamate deriva tives; Inhibitory activity
Synthesis and biological evaluation of novel 7-substituted 3-(4-phenoxyphenyl)thieno[3,2-c]pyridin-4-amines as potent Bruton’s tyrosine kinase (BTK) inhibitors
Keywords: فعالیت مهاری; BTK inhibitors; Thieno[3,2-c]pyrid-4-amine; Inhibitory activity; Kinase selectivity
Involvement of a Serpin serine protease inhibitor (OoSerpin) from mollusc Octopus ocellatus in antibacterial response
Keywords: فعالیت مهاری; Octopus ocellatus; Serpin; Immune response; Inhibitory activity; Bactericide;
Discovery of thieno[3,2-c]pyridin-4-amines as novel Bruton's tyrosine kinase (BTK) inhibitors
Keywords: فعالیت مهاری; BTK inhibitors; Thieno[3,2-c]pyridin-4-amine; Inhibitory activity; Kinase selectivity;
Design, synthesis, and SAR of embelin analogues as the inhibitors of PAI-1 (plasminogen activator inhibitor-1)
Keywords: فعالیت مهاری; Embelin; Natural product; PAI-1; Inhibitory activity; SAR study
Biphenyls from aerial parts of Ribes takare
Keywords: فعالیت مهاری; Biphenyl; Ribes takare D. Don; α-Glycosidase; Inhibitory activity
Unified flexible total synthesis of chlorofusin and artificial Click mimics as antagonists against p53-HDM2 interactions
Keywords: فعالیت مهاری; Chlorofusin; Artificial mimic; Total synthesis; p53-MDM2 interaction; Inhibitory activity;
Molecular characterization, expression and function analysis of a five-domain Kazal-type serine proteinase inhibitor from pearl oyster Pinctada fucata
Keywords: فعالیت مهاری; Pinctada fucata; Serine proteinase inhibitor; Microbial challenge; Quantitative real-time PCR; Inhibitory activity;
Evaluation of fungicides enestroburin and SYP1620 on their inhibitory activities to fungi and oomycetes and systemic translocation in plants
Keywords: فعالیت مهاری; Quinone outer inhibitors; Inhibitory activity; Preventive activity; Systemic translocation
Screening for potential new probiotic based on probiotic properties and α-glucosidase inhibitory activity
Keywords: فعالیت مهاری; Lactic acid bacteria; Antioxidative; α-Glucosidase; Inhibitory activity; Caco-2 cells;
A mu class glutathione S-transferase from Manila clam Ruditapes philippinarum (RpGSTμ): Cloning, mRNA expression, and conjugation assays
Keywords: فعالیت مهاری; Mu class glutathione S-transferase; Ruditapes philippinarum; Catalytic activity; Inhibitory activity; Immune response
α-Glucosidase inhibitors isolated from medicinal plants
Keywords: فعالیت مهاری; α-Glucosidase inhibitor; Inhibitory activity; Medicinal plants
Design and syntheses of novel Nâ²-((4-oxo-4H-chromen-3-yl)methylene)benzohydrazide as inhibitors of cyanobacterial fructose-1,6-/sedoheptulose-1,7-bisphosphatase
Keywords: فعالیت مهاری; Cyanobacteria harmful algal blooms; Benzohydrazone; Chromone; Inhibitory activity;
Diversity of Streptococcus thermophilus in bacteriocin production; inhibitory spectrum and occurrence of thermophilin genes
Keywords: فعالیت مهاری; Streptococcus thermophilus; Inhibitory activity; Bacteriocins; Thermophilin genes; Bioprotective features; Natural cultures
Inhibition of acetylcholinesterases of the pinewood nematode, Bursaphelenchus xylophilus, by phytochemicals from plant essential oils
Keywords: فعالیت مهاری; Bursaphelenchus xylophilus; Acetylcholinesterase; Phytochemicals of plant essential oils; Inhibitory activity
Synthesis of kifunensine thioanalogs and their inhibitory activities against HIV-RT and α-mannosidase
Keywords: فعالیت مهاری; Kifunensine; Thiokifunensine; Staudinger/aza-Wittig/cyclization; Pummerer rearrangement; Inhibitory activity
Synthesis of 1,5-diarylhaloimidazole analogs and their inhibitory activities against PGE2 production from LPS-treated RAW 264.7 cells
Keywords: فعالیت مهاری; Halogenated 1,5-diarylimidazoles; COX-2; Inhibitory activity; PGE2 production; Anti-inflammation;
Purification and characterization of angiotensin I-converting enzyme inhibitory peptide from enzymatic hydrolysates of Styela clava flesh tissue
Keywords: فعالیت مهاری; Styela clava; Angiotensin I-converting enzyme (ACE); Enzymatic hydrolysate; Inhibitory activity
Sequential injection spectrophotometric system for evaluation of mushroom tyrosinase-inhibitory activity
Keywords: فعالیت مهاری; Sequential injection analysis; Spectrophotometry; Mushroom tyrosinase; Inhibitory activity;
A four-domain Kunitz-type proteinase inhibitor from Solen grandis is implicated in immune response
Keywords: فعالیت مهاری; Solen grandis; Kunitz-type proteinase inhibitor; Innate immunity; Real-time PCR; Inhibitory activity;
Chiral β-arylalkyl-1H-1,2,4-triazoles as demethylase inhibitors: Biological evaluation and its stereoselective interaction with sterol 14α-demethylase from Penicillium digitatum
Keywords: فعالیت مهاری; Chiral triazole; P. digitatum; Inhibitory activity; Binding constant; Molecular docking;
In vitro antibacterial activity of three medicinal plants-Boswellia (Luban) species
Keywords: فعالیت مهاری; Antibacterial activity; Plant extracts; Luban; Boswellia frereana; Boswellia sacra; Yemen; Oman; Dhofar; Somalia; Antifungal activity; Boswellia; Inhibitory activity; Bacterial strain; Bacteriostatic activity; Bactericidal activity; Antimicrobial activity
Potent antiprotozoal activity of a novel semi-synthetic berberine derivative
Keywords: فعالیت مهاری; Berberine; 5,6-Didehydro-8,8-diethyl-13-oxodihydroberberine chloride; African trypanosomiasis; Leishmaniasis; Malaria; Inhibitory activity
Identification, structural properties and chelating capacity of miltipolone as a broad-spectrum inhibitor to cancer cells
Keywords: فعالیت مهاری; Danshen; Miltipolone; Inhibitory activity; Tautomeric effect; Metal ion chelator
Synthesis and biological activity of new bispyridinium salts of 4,4â²-bispyridyl-5,5â²-perfluoroalkyl-2,2â²-bisoxazoles
Keywords: فعالیت مهاری; Bisoxazol; Bispyridinium; Antiproliferative; Choline kinase; Inhibitory activity;
Toward potent α-glucosidase inhibitors based on xanthones: A closer look into the structure–activity correlations
Keywords: فعالیت مهاری; Xanthone derivatives; α-glucosidase; Inhibitory activity; Inhibition kinetics