Keywords: Mglu5; Fear; MTEP; CDPPB; Development; Extinction;
مقالات ISI (ترجمه نشده)
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Keywords: CHPG; (RS)-2-chloro-5-hydroxyphenylglycine; FRET; fluorescence resonance energy transfer; LPS; lipopolysaccharide; mGluR5; Group I metabotropic glutamate receptor 5; MTEP; 3-[(2-methyl-1,3-thiazol-4-yl)ethynyl]pyridine; NF-κB; nuclear factor-kappa B; PAM
Keywords: ANOVA; analysis of variance; GABA; γ-aminobutyric acid; SEM; standard error of the mean; NMDA; N-methyl-d-aspartate; AMPA; α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid; iGluRs; ionotropic glutamate receptors; mGluRs; metabotropic glutamate recep
Triptolide up-regulates metabotropic glutamate receptor 5 to inhibit microglia activation in the lipopolysaccharide-induced model of Parkinson's disease
Keywords: mGlu; Metabotropic glutamate receptor; PD; Parkinson's disease; T10; Triptolide; LPS; lipopolysaccharide; NO; nitric oxide; iNOS; inducible nitric oxide synthase; TNF; tumor necrosis factor; IL; interleukin; SN; substantia nigra; COX; cyclooxygenase; JN
Prolonged administration of antidepressant drugs leads to increased binding of [3H]MPEP to mGlu5 receptors
Keywords: [3H]MPEP; mGlu5 receptors; Homer proteins; Escitalopram; Reboxetine; Milnacipran; Moclobemide; Imipramine; MTEP;
Activation of the mTOR signaling pathway in the antidepressant-like activity of the mGlu5 antagonist MTEP and the mGlu7 agonist AMN082 in the FST in rats
Keywords: Antidepressant; AMN082; mGlu receptors; MTEP; mTOR;
Antidepressant-like effect of the mGluR5 antagonist MTEP in an astroglial degeneration model of depression
Keywords: Gliotoxin; l-AAA; Depression; mGluR5 antagonist; MTEP
Development of allosteric modulators of GPCRs for treatment of CNS disorders
Keywords: 5MPEP; 5-methyl-6-(phenylethynyl)-pyridine; 6-OHDA; 6-hydroxydopamine; 7TMR; seven transmembrane receptor; 77-LH-28-1; 1-[3-(4-butyl-1-piperidinyl)propyl]-3,4-dihydro-2(1H)-quinolinone; AC-42; 4-n-butyl-1-[4-(2-methylphenyl)-4-oxo-1-butyl]-piperidine; ACh
Potentiation of mGlu5 receptors with the novel enhancer, VU0360172, reduces spontaneous absence seizures in WAG/Rij rats
Keywords: Absence epilepsy; WAG/Rij rats; mGlu5 receptor; VU0360172; MTEP;
Is the mGlu5 receptor a possible target for new antidepressant drugs?
Keywords: antidepressant drugs; ketamine; mGlu5 receptor; MTEP; MPEP; NMDA receptor
Interactions of CB1 and mGlu5 receptor antagonists in food intake, anxiety and memory models in rats
Keywords: MTEP; 3-[(2-methyl-1,3-thiazol-4-yl)ethynyl]pridine; SIB-1757; 6-methyl-2-(phenylazo)-3-pyridinol); Rimonabant; (5-(4-Chlorophenyl)-1-(2,4-dichloro-phenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide)hydrochloride; USV; ultrasonic vocalization;
mGlu5 receptor deletion reduces relapse to food-seeking and prevents the anti-relapse effects of mGlu5 receptor blockade in mice
Keywords: mGlu5; MTEP; Food; Relapse
Positive allosteric modulation of metabotropic glutamate receptor 5 down-regulates fibrinogen-activated microglia providing neuronal protection
Keywords: BBB; blood brain barrier; CDPPB; 3-cyano-N-(1,3-diphenyl-1H-pyrazol-5-yl)benzamide; CGC; cerebellar granule cells; CNS; central nervous system; DCGIV; (2S,2â²R,3â²R)-2-(2â²,3â²-dicarboxycyclopropyl)glycine; ERK1/2; extracellular signal-regulated kinas
Behavioral consequences of the mGlu5 receptor antagonist MTEP in immature rats
Keywords: MTEP; Sensorimotor performance; Exploratory behavior; Anxiety; Learning; Immature rats;
The role of group I mGlu receptors in the expression of ethanol-induced conditioned place preference and ethanol withdrawal seizures in rats
Keywords: Ethanol; Expression of CPP; Withdrawal seizure; Group I mGlu receptors antagonist; EMQMCM; MTEP;
NMDA but not AMPA glutamatergic receptors are involved in the antidepressant-like activity of MTEP during the forced swim test in mice
Keywords: mGluR5; MTEP; forced swim test; NMDA; AMPA; ligands;
Effect of the metabotropic glutamate receptor type 5 antagonists MPEP and MTEP in parkinsonian monkeys
Keywords: mGluR5; Dyskinesia; Levodopa; MPTP monkey; MPEP; MTEP;
Effects of the mGlu2/3 Agonist LY379268 and the mGlu5 Antagonist MTEP on Ethanol Seeking and Reinforcement Are Differentially Altered in Rats with a History of Ethanol Dependence
Keywords: Ethanol dependence; LY379268; metabotropic glutamate receptor; MTEP; relapse; self-administration
Metabotropic glutamate receptor subtype 5 antagonism in learning and memory
Keywords: Metabotropic glutamate receptor 5; Spatial learning; Fear conditioning; Avoidance learning; MPEP; MTEP; Locomotion; (Rat); (Mouse)
Structure–activity relationships in a novel series of 7-substituted-aryl quinolines and 5-substituted-aryl benzothiazoles at the metabotropic glutamate receptor subtype 5
Keywords: mGluR, metabotropic glutamate receptor; iGluR, ionotropic glutamate receptor; MPEP, 2-methyl-6-(phenylethynyl)pyridine; MTEP, 3-((2-methyl-4-thiazolyl)ethynyl)pyridineMetabotropic glutamate receptor subtype 5; mGluR5; MPEP; MTEP; Drug abuse
Physical and crystallographic characterisation of the mGlu5 antagonist MTEP and its monohydrochloride
Keywords: 3-[(2-methyl-1,3-thiazol-4-yl)ethynyl]pyridine; MTEP; MTEP hydrochloride; crystal structure; Hirshfeld surface analysis; synthesis; acid dissociation constant; solubility; physicochemical properties; NMR spectroscopy;
Metabotropic glutamate receptor 5 (mGluR5) antagonists attenuate cocaine priming- and cue-induced reinstatement of cocaine seeking
Keywords: Relapse; Addiction; Psychostimulant; Glutamate; Metabotropic; mGluR5; MPEP; MTEP
Metabotropic Glutamate Receptors as Targets for Multipotential Treatment of Neurological Disorders
Keywords: Astrocytes; inflammation; metabotropic glutamate receptors; microglia; neuron; neuroprotection; 4CPG; (S)-4-carboxyphenylglycine; 6-OHDA; 6-hydroxydopamine; Aβ; β-amyloid; AIDA; 1-aminoindan-1, 5-dicarboxylic acid; ALS; amyotrophic lateral sclerosis; AM
mGlu5 receptor deletion does not confer seizure protection to mice
Keywords: mGlu5 receptors; MTEP; Seizures; Epilepsy; Mice
The influence of various glutamate receptors antagonists on anxiety-like effect of ethanol withdrawal in a plus-maze test in rats
Keywords: Ethanol withdrawal; Anxiety; Elevated plus-maze; Memantine; Acamprosate; MTEP; EMQMCM; NMDA; mGlu receptor; Behavior
Anxiolytic-like action of MTEP expressed in the conflict drinking Vogel test in rats is serotonin dependent
Keywords: Anxiety; 5-HT1 receptors; 5-HT2 receptors; 5-HT release; mGlu5 receptors; MTEP; Conflict drinking Vogel test; Rat
In vitro metabolic studies on the selective metabotropic glutamate receptor sub-type 5 (mGluR5) antagonist 3-[(2-methyl-1,3-thiazol-4-yl) ethynyl]-pyridine (MTEP)
Keywords: Metabotropic glutamate receptor; Drug metabolism; CYP1A2; CYP2C; MPEP; MTEP
Antidepressant-like and anxiolytic-like actions of the mGlu5 receptor antagonist MTEP, microinjected into lateral septal nuclei of male Wistar rats
Keywords: DRL-72 s, differential reinforcement of the low-rate 72 s; IRT, inter-response time.Antidepressant-like; Anxiolytic-like; DRL-72 s; Elevated plus-maze; Lateral Septum; MTEP; NMDA
Estrus variation in anticonflict-like effects of the mGlu5 receptor antagonist MTEP, microinjected into lateral septal nuclei of female Wistar rats
Keywords: Conflict behavior; Estrous cycle; Lateral Septum; MTEP; NMDA
Potential antidepressant-like effect of MTEP, a potent and highly selective mGluR5 antagonist
Keywords: mGluR5; MTEP; Depression; Olfactory bulbectomy; Tail suspension test; Forced swimming test;
Inhibition of Transient Lower Esophageal Sphincter Relaxation and Gastroesophageal Reflux by Metabotropic Glutamate Receptor Ligands
Keywords: GABA; γ-aminobutyric acid; GERD; gastroesophageal reflux disease; L-AP4; L-(+)-2-amino-4-phosphonobutyric acid; mGluR; metabotropic glutamate receptor; MPEP; 2-methyl-6-(phenylethynyl)-pyridine; MTEP; 3-([2-methyl-1,3-thiazol-4-yl)ethynyl]pyridine; NMDA;