Keywords: ATP; adenosine triphosphate; CBX; carbenoxolone; C-terminus; carboxyl-terminus; CNS; central nervous system; EL; extracellular loop; Gly0; core glycosylation; Gly1; high mannose glycosylation; Gly2; complex glycosylation; ICL; intracellular loop; N2a; Neu
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Keywords: ATP; Vascular injury; P2X7R; Subfailure stretch; p38 MAPK;
Keywords: ADP; adenosine diphosphate; AMP; adenosine monophosphate; ATP; adenosine triphosphate; [Ca2+]i; intracellular calcium concentration; CaM; calmodulin; CaMKII; Ca2+/calmodulin-dependent kinase II; cAMP; cyclic adenosine monophosphate; COX-2; cyclooxygenase-
Keywords: OS; oxidative stress; CNS; central nervous system; ROS; reactive oxygen species; SOD; superoxide dismutase; CAT; catalase; Cu; copper; Zn; zinc; Mn; manganese; Fe; iron; Ni; nickel; DA; dopamine; PHOX; NADPH oxidase; Nrf2; nuclear factor erythroid 2-relat
Keywords: TNAP; Development; Neurodegenerative diseases; Pyridoxal phosphate; ATP; P2X7R
Keywords: ADX; adrenalectomized; ASD; autism spectrum disorders; BD; bipolar disorder; CSF; cerebrospinal fluid; DAMPs; damage-associated molecular patterns; FS; forced swimming; HDACi; histone deacetylase inhibitor; HSP; heat shock protein; IDO; indoleamine 2,3 di
Keywords: Annexins; Calcium; Microvesicle; Blebbing; P2X7R
SNPs in the vicinity of P2X7R, RANK/RANKL/OPG and Wnt signalling pathways and their association with bone phenotypes in academy footballers
Keywords: Genetics; RANK/RANKL/OPG; P2X7R; Wnt signalling; Exercise;
Leucodin attenuates inflammatory response in macrophages and lipid accumulation in steatotic hepatocytes via P2x7 receptor pathway: A potential role in alcoholic liver disease
Keywords: Leucodin; Alcoholic liver steatosis; Inflammation; P2x7R; NLRP3;
ATP/P2X7-NLRP3 axis of dendritic cells participates in the regulation of airway inflammation and hyper-responsiveness in asthma by mediating HMGB1 expression and secretion
Keywords: Th; type helper; IL; interleukin; AHR; hyper-responsiveness; HMGB1; high mobility protein 1; DCs; dendritic cells; BMDCs; bone marrow-derived mononuclear cells; DAMPs; damage-associated molecular patterns; PAMP; pathogen-associated molecular patterns; RAG
Down-regulated miR-187 promotes oxidative stress-induced retinal cell apoptosis through P2X7 receptor
Keywords: Glaucoma; MiR-187; P2X7R; Retinal cells; Oxidative stress; Apoptosis;
Modulation of P2X7 purinergic receptor activity by extracellular Zn2+ in cultured mouse hippocampal astroglia
Keywords: CNS; central nervous system; MDD; major depressive disorder; BzATP; 3â²-O-(4-Benzoyl) benzoyl ATP; BBG; Brilliant Blue G; OGB-1; OregonGreen Bapta-1; PI; propidium iodide; VGluT1; vesicularglutamate transporter 1; P2X7R; Hippocampus; Purinergic receptor;
Release of soluble and vesicular purine nucleoside phosphorylase from rat astrocytes and microglia induced by pro-inflammatory stimulation with extracellular ATP via P2X7 receptors
Keywords: Brain cell cultures; Extracellular purine nucleoside phosphorylase (PNP); P2X7 receptor; Mechanism of release; Lysosomal vesicles; A-CM; astrocyte derived-conditioned medium; BME; Basal Medium Eagle; Bz-ATP; 3â²-O-benzoyl-benzoyl-ATP; CGNs; cerebellar gr
Pharmacological evaluation of a novel series of urea, thiourea and guanidine derivatives as P2X7 receptor antagonists
Keywords: P2X7R; Inflammation; Cyanoguanidine; Urea; Thiourea;
Original contributionHigh expression of P2X7R is an independent postoperative indicator of poor prognosis in colorectal cancer
Keywords: P2X7R; Colorectal cancer; Prognosis; Proliferation; Metastasis;
Inflammasomes and type 2 diabetes: An updated systematic review
Keywords: AIM; Absent In Melanoma; ASC; Apoptosis-associated Speck-like protein; ATF6; Activating Transcription Factor 6; CARD; Caspase Activation and Recruitment Domain; DAMPs; Damage Associated Molecular Patterns; DIO; Diet Induced Obese; IAPP; Islet Amyloid Poly
P2X7Rs are involved in cell death, growth and cellular signaling in primary human osteoblasts
Keywords: Calcium signaling; P2X7R; Osteoblast;
ZrCl4 as a new catalyst for ester amidation: an efficient synthesis of h-P2X7R antagonists
Keywords: ZrCl4; Aminolysis; Pyroglutamide; P2X7R; IBD; Inflammation;
Research reportEffects of naringin on learning and memory dysfunction induced by gp120 in rats
Keywords: HAD; HIV-1 associated dementia; LV; lateral ventricle; MWM; Morris water maze; P2X7R; P2X7 receptor; HIV; human immunodeficiency virus; ADC; AIDS-dementia complex; SD; Sprague-Dawley; ACSF; artificial cerebrospinal fluid; PMSF; phenylmethanesulfonyl fluor
Structure-based identification and characterisation of structurally novel human P2X7 receptor antagonists
Keywords: zfP2X4R; zebrafish P2X4 receptor; P2X7R; P2X7 receptor; hP2X7R; human P2X7R; rP2X7R; rat P2X7R; BzATP; 2,3-O-(4-benzoylbenzoyl)-ATP; PI; propidium iodide; BBG; brilliant blue G; TNP-ATP; trinitrophenyl-ATP; HEK293 cells; human embryonic kidney 293 cells;
Purinergic signalling in autoimmunity: A role for the P2X7R in systemic lupus erythematosus?
Keywords: Extracellular ATP; P2X7R; Systemic lupus erythematosus; NLRP3 inflammasome; Interleukin-1β;
P2X7R activation drives distinct IL-1 responses in dendritic cells compared to macrophages
Keywords: Interleukin-1; P2X7R; Dendritic cells; Macrophages; A-740003; ATP; adenosine triphosphate; BM; bone marrow; BMM; bone marrow-derived macrophages; DAMPs; danger associated molecular patterns; DC; dendritic cells; DMSO; dimethyl sulfoxide; EDTA; ethylene di
P2X7 receptor-mediated analgesia in cancer-induced bone pain
Keywords: BSA; Bovine Serum Albumin; HBSS; Hanks' balanced salt solution; P2X7R; P2X7 receptor; RVM; rostral ventromedial medulla; SEM; standard error of the mean; WDR; wide dynamic range; cancer-induced bone pain; P2X7R antagonism; analgesia; neuronal responses;
Substance P and the neurokinin-1 receptor regulate electroencephalogram non-rapid eye movement sleep slow-wave activity locally
Keywords: EEG; electroencephalogram; EMG; electromyogram; IL-1β; interleukin-1 beta; IL-6; interleukin-6; LPS; lipopolysaccharide; NK-1R; neurokinin-1 receptor; nNOS; neuronal nitric oxide synthase; NO; nitric oxide; NREMS; non rapid-eye movement sleep; P2X7R; pur
Structure-activity relationship studies of pyrimidine-2,4-dione derivatives as potent P2X7 receptor antagonists
Keywords: P2X7 receptor; Antagonists; KN-62; Structure-activity relationships; IL-1β; Inflammation; AcCl; acetyl chloride; ACN; acetonitrile; ATP; adenosine-5â²-triphosphate; BzATP; 2â²(3â²)-O-(4-benzoylbenzoyl)-ATP; DCM; dichloromethane; DMEM; Dulbecco's Mod
Emerging role of P2X7 receptors in CNS health and disease
Keywords: ATP; P2X7R; Neuron-glia; Neurodegenerative disorder; Central nervous system;
P2X7 Receptor Mediates Spinal Microglia Activation of Visceral Hyperalgesia in a Rat Model of Chronic Pancreatitis
Keywords: Brilliant Blue G; Chronic Visceral Pain; Purinergic Receptors; siRNA Knockdown; ANOVA; analysis of variance; ATP; adenosine triphosphate sulfonic acid; BBG; brilliant blue G; CNS; central nervous system; CP; chronic pancreatitis; GAPDH; glyceraldehyde-3-p
Regulation of the P2X7R by microRNA-216b in human breast cancer
Keywords: Apoptosis; Bcl-2; Breast cancer; Caspase-3; miR-216b; P2X7R;
P2X7 receptors mediate resistance to toxin-induced cell lysis
Keywords: HEK; human embryonic kidney 293 cells; HMC-1; human mast cell line 1; P2X7R; P2X7 receptor; RT; room temperature; SLO; streptolysin O; P2X7; Plasmalemma; Blebbing; Calcium; Lysis; Annexin;
P2X7 receptor blockade protects against cisplatin-induced nephrotoxicity in mice by decreasing the activities of inflammasome components, oxidative stress and caspase-3
Keywords: Cisplatin-induced nephrotoxicity; P2X7R; NLRP3 inflammasome; Oxidative stress; Apoptosis; Caspase-3
The P2X7 receptor: Shifting from a low- to a high-conductance channel - An enigmatic phenomenon?
Keywords: P2X7R; Ion channel activity; Patch-clamp; Calcium; Second messenger;
Pharmacological blockage and P2X7 deletion hinder aversive memories: Reversion in an enriched environment
Keywords: ANOVA; analysis of variance; BBG; Brilliant Blue G; EE; enriched environment; FC; fear-conditioning; KO; knockout; LTM; long-term memory; LTP; long-term potentiation; MWM; Morris water maze; NE; non-enriched environment; P2X7R; P2X7 receptor; RM; repeated
Mechanical vibration inhibits osteoclast formation by reducing DC-STAMP receptor expression in osteoclast precursor cells
Keywords: Mechanical vibration; Osteoclasts; DC-STAMP; P2X7R; RANKL;
Assessment of mercury chloride-induced toxicity and the relevance of P2X7 receptor activation in zebrafish larvae
Keywords: P2X7R; Mercury; Zebrafish larvae; Oxidative stress;
Aloe vera downregulates LPS-induced inflammatory cytokine production and expression of NLRP3 inflammasome in human macrophages
Keywords: ATP; adenosine-5â²-triphosphate; ASC; apoptosis-associated speck-like protein containing a caspase recruitment domain; ELISA; enzyme-linked immunosorbent assay; ERK; extracellular-signal-regulated kinase; GM-CSF; granulocyte-macrophage colony stimulating
Oxidative stress induced by P2X7 receptor stimulation in murine macrophages is mediated by c-Src/Pyk2 and ERK1/2
Keywords: P2X7R; P2X7 receptor channels; LPS; lipopolysaccharide; IL-1β; interleukin-1β; TNFα; tumor necrosis factor α; ROS; reactive oxygen species; JNK; c-Jun N-terminal kinase; ERK1/2; extracellular regulated kinases 1 and 2; MAPKs; mitogen-activated protein
Research ReportThe anti-apoptotic and neuro-protective effects of human umbilical cord blood mesenchymal stem cells (hUCB-MSCs) on acute optic nerve injury is transient
Keywords: Axonal regeneration; Hucb-MSCs; Optic nerve injury; Fluorogold retrograde tracing; GAP43; P2X7R;
Regulation of lung surfactant secretion by microRNA-150
Keywords: P2X7R; miR-150; Surfactant secretion;
Calmidazolium selectively inhibits exocytotic glutamate release evoked by P2X7 receptor activation
Keywords: A-438079; 3-(5-(2,3-dichlorophenyl)-1H-tetrazol-1-yl)-methyl pyridine; BzATP; 2â²-3â²-O-(benzoylbenzoyl)ATP; [Ca2+]i; intracellular Ca2+ concentration; P2X7R; P2X7 receptor; ROI; region of interest; VOCCs; voltage operated calcium channels; Glutamate re
Regional changes in purines and selected purinergic receptors in immature rat brain exposed to lead
Keywords: ATP; P2X7R; Connexin 43; Adenosine; Lead toxicity
Characterization of the molecular interaction between caveolin-1 and the P2X receptors 4 and 7 in E10 mouse lung alveolar epithelial cells
Keywords: Caveolin-1; P2X4R; P2X7R; Alveolar epithelium; Mouse lung